专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明授权

US08211924B2 1-(azolin-2-yl)amino-1,2-diphenylethane compounds for combating animal pests 有权
公开(公告)号：US08211924B2
公开(公告)日：2012-07-03
申请号：US12667299
申请日：2008-07-02
申请人： Markus Kordes , Christopher Koradin , Ronan Le Vezouet , Ernst Baumann , Deborah L. Culbertson , Douglas D. Anspaugh , Hassan Oloumi-Sadeghi , Cecille Ebuenga
发明人： Markus Kordes , Christopher Koradin , Ronan Le Vezouet , Ernst Baumann , Deborah L. Culbertson , Douglas D. Anspaugh , Hassan Oloumi-Sadeghi , Cecille Ebuenga
IPC分类号： A01N43/78 , A01N43/76 , A61K31/425 , A61K31/42 , C07D277/00 , C07D263/00
CPC分类号： C07D263/28 , A01N43/50 , A01N43/76 , A01N43/78 , A01N47/12 , A01N47/16 , C07D233/48 , C07D277/18 , C07D417/06 , C07D417/12
摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, —C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.

2. 发明申请

US20100280078A1 1-(Azolin-2-yl)amino-1,2-diphenylethane compounds for combating animal pests 有权
公开(公告)号：US20100280078A1
公开(公告)日：2010-11-04
申请号：US12667299
申请日：2008-07-02
申请人： Markus Kordes , Christopher Koradin , Ronan Le Vezouet , Ernst Baumann , Deborah L. Culbertson , Douglas D. Anspaugh , Hassan Oloumi-Sadeghi , Cecile Ebuenga
发明人： Markus Kordes , Christopher Koradin , Ronan Le Vezouet , Ernst Baumann , Deborah L. Culbertson , Douglas D. Anspaugh , Hassan Oloumi-Sadeghi , Cecile Ebuenga
IPC分类号： A01N43/78 , C07D277/18 , A61K31/426 , C07D417/12 , C07D417/14 , A61K31/427 , C07D263/28 , A01N43/76 , A61K31/421 , A61K31/4439 , A61P33/00 , A01P7/00 , A01P7/02 , A01P7/04 , A01P5/00
CPC分类号： C07D263/28 , A01N43/50 , A01N43/76 , A01N43/78 , A01N47/12 , A01N47/16 , C07D233/48 , C07D277/18 , C07D417/06 , C07D417/12
摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds. wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NRX, R1 is selected from the group consisting of —ORA, —NRB1RB2, C(═O)—RC, —C(═O)—ORD, —C(═O)—SRE, —C(═O)—NRB1RB2′, —C(═S)—RC′, —C(═S)—ORD′, —C(═S)—SRE′, —C(═S)—NRB1RB2, —C(═NR1a)—RC′, —C(═NR1b)—ORD′, —C(═NR1c)—SRE′, —C(═NR1d)—NRB1RB2, —S(═O)—RF, —S(═O)2—RG, —S(═O)2—NRB1RB2′, —P(═O)RH1RH2, —P(═S)RH1RH2, —B—C(═O)—RI, —B—O—C(═O)—RI, —B—S—C(═O)—RI, —B—N(RJ)—C(═O)—RK, —B—C(═S)—RK, —B—O—C(═S)—RK, —B—S—C(═S)—RK, —B—N(RJ)—C(═S)—RK, C1-C8-alkenyl, C1-C8-alkynyl, C3-C8-cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R1e, naphthyl, which is unsubstituted or may carry 1 to 4 substituents R1f, a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R1g, hetaryl, which is unsubstituted or may carry 1 to 4 substituents R1h, and C1-C6-alkyl, which carries a radical selected from the group consisting of —NR1iR1j, C1-C4-alkoxycarbonyl, C3-C8-cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R2, R3, R4, R5, R6 and R7 are each independently hydrogen, halogen, OH, SH, NH2, SO3H, COOH, cyano, nitro, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylamino etc.

3. 发明授权

US07563921B2 2-cyano-3(halo)alkoxy-benzenesulfonamide compounds for combating animal pests 失效
标题翻译：用于对抗动物害虫的2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物
公开(公告)号：US07563921B2
公开(公告)日：2009-07-21
申请号：US12137624
申请日：2008-06-12
申请人： Wolfgang von Deyn , Henricus Maria Martinus Bastiaans , Matthias Pohlman , Michael Rack , Ernst Baumann , Michael Puhl , Michael Hofmann , Livio Tedeschi , Markus Kordes , Christopher Koradin , Douglas D. Anspaugh , Deborah L. Culbertson , Henry van Tuyl Cotter , Hassan Oloumi-Sadeghi
发明人： Wolfgang von Deyn , Henricus Maria Martinus Bastiaans , Matthias Pohlman , Michael Rack , Ernst Baumann , Michael Puhl , Michael Hofmann , Livio Tedeschi , Markus Kordes , Christopher Koradin , Douglas D. Anspaugh , Deborah L. Culbertson , Henry van Tuyl Cotter , Hassan Oloumi-Sadeghi
IPC分类号： C07C319/20 , C07C323/32 , C07C311/15 , A01N25/00 , A01N25/26 , A01P17/00 , A61K31/18
CPC分类号： C07C319/20 , A01N41/06 , C07C311/29 , C07C323/62
摘要： The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula I.
摘要翻译：本发明涉及2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物I，其中变量Alk和R1至R5如权利要求1所定义，和/或其农业上有用的盐。此外，本发明涉及化合物I和/或其盐对抗动物害虫的用途; 包含至少一种式I化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物，其具有杀虫作用，如果需要，至少一种表面活性剂; 以及一种对抗动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，材料或环境，或材料，植物，防止动物攻击或侵染的种子，土壤，表面或空间，其中农药有效量的至少一种式I的2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物和/或至少一种农业上可接受的的盐。包括从土壤和叶面昆虫中保护种子免受土壤昆虫和所得植物的根和芽的方法，包括在种子播种前和/或后发芽后将种子与2-氰基-3-（卤代）烷氧基 - 苯磺酰胺通式Ⅰ的化合物

4. 发明申请

US20080306297A1 NOVEL 2-CYANO-3(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS 失效
标题翻译：新型2-氰基-3（HALO）烷氧基苯甲酰胺化合物，用于组合动物饲料
公开(公告)号：US20080306297A1
公开(公告)日：2008-12-11
申请号：US12137624
申请日：2008-06-12
申请人： Wolfgang von Deyn , Henricus Maria Martinus Bastiaans , Matthias Pohlman , Michael Rack , Ernst Baumann , Michael Puhl , Michael Hofmann , Livio Tedeschi , Markus Kordes , Christopher Koradin , Douglas D. Anspaugh , Deborah L. Culbertson , Henry van Tuyl Cotter , Hassan Oloumi-Sadeghi
发明人： Wolfgang von Deyn , Henricus Maria Martinus Bastiaans , Matthias Pohlman , Michael Rack , Ernst Baumann , Michael Puhl , Michael Hofmann , Livio Tedeschi , Markus Kordes , Christopher Koradin , Douglas D. Anspaugh , Deborah L. Culbertson , Henry van Tuyl Cotter , Hassan Oloumi-Sadeghi
IPC分类号： C07C255/53
CPC分类号： C07C319/20 , A01N41/06 , C07C311/29 , C07C323/62
摘要： Novel 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds for combating animal pestsThe invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts.Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxybenzenesulfonamide compound of the general formula I
摘要翻译：用于对抗动物害虫的新型2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物本发明涉及2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物I，其中变量Alk和R1至R5如权利要求1中所定义，和/或其农业上有用的盐。此外，本发明涉及化合物I和/或其盐对抗动物害虫的用途; 包含至少一种式I化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物，其具有杀虫作用，如果需要，至少一种表面活性剂; 以及一种对抗动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，材料或环境，或材料，植物，防止动物攻击或侵染的种子，土壤，表面或空间，其中农药有效量的至少一种式I的2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物和/或至少一种农业上可接受的的盐。包括从土壤和叶面昆虫中保护种子免受土壤昆虫和所得植物的根和芽的方法，包括在种子播种前和/或后发芽之前将种子与2-氰基-3-（卤代）烷氧基苯磺酰胺化合物接触通式I

5. 发明授权

US07544637B2 2-cyano-3(halo)alkoxy-benzenesulfonamide compounds for combating animal pests 失效
标题翻译：用于对抗动物害虫的2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物
公开(公告)号：US07544637B2
公开(公告)日：2009-06-09
申请号：US11791398
申请日：2005-11-24
申请人： Wolfgang von Deyn , Henricus Maria Martinus Bastiaans , Matthias Pohlman , Michael Rack , Ernst Baumann , Michael Puhl , Michael Hofmann , Livio Tedeschi , Markus Kordes , Christopher Koradin , Douglas D. Anspaugh , Deborah L. Culbertson , Henry van Tuyl Cotter , Hassan Oloumi-Sadeghi
发明人： Wolfgang von Deyn , Henricus Maria Martinus Bastiaans , Matthias Pohlman , Michael Rack , Ernst Baumann , Michael Puhl , Michael Hofmann , Livio Tedeschi , Markus Kordes , Christopher Koradin , Douglas D. Anspaugh , Deborah L. Culbertson , Henry van Tuyl Cotter , Hassan Oloumi-Sadeghi
IPC分类号： C07C311/15 , A01N25/00 , A01N25/26 , A01P17/00 , A61K31/18
CPC分类号： C07C319/20 , A01N41/06 , C07C311/29 , C07C323/62
摘要： The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula I
摘要翻译：本发明涉及2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物I，其中变量Alk和R1至R5如权利要求1所定义，和/或其农业上有用的盐。此外，本发明涉及化合物I和/或其盐对抗动物害虫的用途; 包含至少一种式I化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物，其具有杀虫作用，如果需要，至少一种表面活性剂; 以及一种对抗动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，材料或环境，或材料，植物，防止动物攻击或侵染的种子，土壤，表面或空间与杀虫有效量的式I的至少一个2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物和/或至少一种农业上可接受的盐其中。包括从土壤和叶面昆虫中保护种子免受土壤昆虫和所得植物的根和芽的方法，包括在种子播种前和/或后发芽后将种子与2-氰基-3-（卤代）烷氧基 - 苯磺酰胺通式I的化合物

6. 发明申请

US20110224075A1 Pesticidal Active Mixtures Comprising Aminothiazoline Compounds 失效
标题翻译：包括氨基噻唑啉化合物的杀虫活性混合物
公开(公告)号：US20110224075A1
公开(公告)日：2011-09-15
申请号：US12934461
申请日：2009-03-24
申请人： Markus Kordes , Ronan Le Vezouet , Jurgen Langewald , Ralph Paulini , Deborah L. Culbertson , Douglas D. Anspaugh , Luiz Antonio Jose , Hassan Oloumi-Sadeghi
发明人： Markus Kordes , Ronan Le Vezouet , Jurgen Langewald , Ralph Paulini , Deborah L. Culbertson , Douglas D. Anspaugh , Luiz Antonio Jose , Hassan Oloumi-Sadeghi
IPC分类号： A01N25/26 , A01N43/78 , A61K31/427 , A61K31/426 , A01N43/42 , A61K31/4709 , A61K31/4725 , A01N43/40 , A61K31/4439 , A01N43/16 , A61K31/7016 , A01N43/56 , A61K31/415 , A01N43/88 , A61K31/5395 , A61K31/44 , A01N37/34 , A61K31/277 , A01N43/38 , A61K31/403 , A01N43/58 , A61K31/50 , A61P33/00 , A01P7/02 , A01P7/04
CPC分类号： A01N43/78 , A01N43/08 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/707 , A01N43/88 , A01N43/90 , A01N47/02 , A01N47/06 , A01N47/30 , A01N47/34 , A01N47/40 , A01N51/00 , A01N53/00 , A01N2300/00
摘要： The present invention relates to pesticidal mixtures comprising as active compounds 1) at least one aminothiazoline compound I of formula I: wherein R1 is selected from hydrogen, COCH3, COCH2CH3 or COCH2C(CH3)3; R2 and R3 together with the carbon atoms of the phenyl ring to which they are attached form a ring which, depending on the tautomeric formula I a) or b) is depicted as: a benzene ring, a saturated 5-, 6-, or 7-membered carbocycle, a partially unsaturated 5-, 6-, or 7-membered carbocycle, a 5-, 6-, or 7-membered saturated heterocycle, a partially unsaturated 5-, 6-, or 7-membered heterocycle, which heterocycles contain 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and a 5- or 6-membered heteroaromatic ring which contains 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and wherein the ring is unsubstituted or may carry any combination of 1, 2, 3, or 4 radicals selected from the group consisting of halogen, CH3, CH2CH3, CF3, CH3O, cyano and (═O) (oxo); R4 is selected from hydrogen, fluoro, chloro, bromo, CF3, CH3O or CH3; R5, R6 are selected from hydrogen, chloro, fluoro, bromo, CH3, CH3O or CF3, wherein at least one of R5 or R6 is not hydrogen; with the proviso that R2 and R3 together do not form a —OCH2—O— or a —OCF2O-group; or the tautomers, enantiomers, diastereomers or salts thereof, and 2) at least one active compound II selected from group A as defined in the description, use of these mixtures for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using these mixtures.
摘要翻译：本发明涉及包含作为活性化合物的杀虫混合物1）至少一种式I的氨基噻唑啉化合物I：其中R 1选自氢，COCH 3，COCH 2 CH 3或COCH 2 C（CH 3）3; R2和R3与它们所连接的苯环的碳原子一起形成环，其取决于互变异构体式a a）或b）被描述为：苯环，饱和的5-，6-或 7元碳环，部分不饱和5-，6-或7-元碳环，5-，6-或7-元饱和杂环，部分不饱和5-，6-或7-元杂环，其中杂环含有选自O，S和N作为环成员的1,2或3个杂原子，以及含有1,2或3个选自O，S和N作为环成员的杂原子的5或6元杂芳环，并且其中所述环是未取代的或可以携带选自卤素，CH 3，CH 2 CH 3，CF 3，CH 3 O，氰基和（= O）（氧代）的1,2,3或4个基团的任何组合。 R4选自氢，氟，氯，溴，CF 3，CH 3 O或CH 3; R5，R6选自氢，氯，氟，溴，CH3，CH3O或CF3，其中R5或R6中的至少一个不是氢; 条件是R2和R3一起不形成-OCH2-O-或-OCF2O-基团; 或其互变异构体，对映异构体，非对映异构体或其盐，以及2）选自如说明书中定义的组A的至少一种活性化合物II，这些混合物用于防治昆虫，螨虫或线虫的用途，以及治疗，控制，防止或保护动物免受使用这些混合物的寄生虫的感染或感染。

7. 发明申请

US20100167925A1 Substituted Azolin-2-yl-Amino Compounds 审中-公开
标题翻译：取代的唑啉-2-基氨基化合物
公开(公告)号：US20100167925A1
公开(公告)日：2010-07-01
申请号：US12376455
申请日：2007-08-06
申请人： Christopher Koradin , Markus Kordes , Ronan Le Vezouet , Deborah L. Culbertson , Douglas D. Anspaugh
发明人： Christopher Koradin , Markus Kordes , Ronan Le Vezouet , Deborah L. Culbertson , Douglas D. Anspaugh
IPC分类号： A01C1/06 , A01N43/78 , C07D417/02
CPC分类号： C07D417/12 , A01N43/50 , A01N43/76 , A01N43/78 , C07D277/18
摘要： The present invention relates to azolin-2-yl-amino compounds of formulae (I. a) and (1.b) and their salts which are useful for combating animal pest, in particular arthropod and nematodes. The present invention also relates to a method for combating such pests and for protecting crops against infestation or infection by such pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests. Formula (I.a), formula (I.b) wherein n is 0 to 4; X is S, O or NR5; A is —C(R6a)(R6b)—, O, NR7, S, S(O) or S(O)2; B is a bond Or CH2; R1 is H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R2a, R2b are H, CN, C1-C6-alkyl, C2-C6-alkenyl, C1-C6-alkylcarbonyl, (C1-C6-alkyl)-thiocarbonyl, C(O)NRaRb, C(S)NRaRb, (SO2)NRaRb, phenyl, benzyl, 5 or 6 membered heterocyclic ring etc.; or R1 together with R2a is C3-C5-alkandiyl; or R1 together with R2 are C(O); R3a, R3b, R3c, R3d are H, halogen, CN, C1-C6-alkyl, C1-C6-alkylamino, C3-C6-cycloalkyl, phenyl, benzyl, etc.; R4a, R4b are H, halogen, C1-C6-alkyl, C2-C6-alkenyl, phenyl, benzyl, 5 or 6 membered hetaryl; or R4a together with Rb may also be ═O, ═NRC or ═CRdRe; or R2a together with R4a may form a bridging bivalent radical.
摘要翻译：本发明涉及用于对抗动物害虫，特别是节肢动物和线虫的式（Ⅰa）和（Ⅰb）的唑啉-2-基氨基化合物及其盐。本发明还涉及一种防治这种害虫并防止作物抵抗这种害虫侵染或感染的方法。此外，本发明涉及用于对抗动物害虫的兽用组合物。式（Ⅰa），式（Ⅰb）其中n为0-4; X是S，O或NR5; A是-C（R6a）（R6b） - ，O，NR7，S，S（O）或S（O） B是键或CH2; R1是H，CN，C1-C6-烷基，C2-C6-烯基，C1-C6-烷基羰基，C3-C6-环烷基，苯基，苄基等; R2a，R2b是H，CN，C1-C6-烷基，C2-C6-烯基，C1-C6-烷基羰基，（C1-C6-烷基） - 硫代羰基，C（O）NRaRb，C（S）NRaRb，（SO2 ）NRaRb，苯基，苄基，5或6元杂环等; 或R 1与R 2a一起为C 3 -C 5 - 烷二基; 或R 1与R 2一起为C（O）; R3a，R3b，R3c，R3d是H，卤素，CN，C1-C6-烷基，C1-C6-烷基氨基，C3-C6-环烷基，苯基，苄基等; R4a，R4b是H，卤素，C1-C6-烷基，C2-C6-烯基，苯基，苄基，5或6元杂芳基; 或R 4a与R b一起也可以是= O，= NRC或= CRdRe; 或R 2a与R 4a一起形成桥连二价基团。

8. 发明申请

US20100010058A1 Azoline Compounds for Combating Arthropod Pests 审中-公开
标题翻译：用于防治节肢动物害虫的唑啉化合物
公开(公告)号：US20100010058A1
公开(公告)日：2010-01-14
申请号：US12305267
申请日：2007-05-25
申请人： Christopher Koradin , Markus Kordes , Ronan Le Vezouet , Deborah L. Culbertson , Douglas D. Anspaugh , Henry Van Tuyl Cotter
发明人： Christopher Koradin , Markus Kordes , Ronan Le Vezouet , Deborah L. Culbertson , Douglas D. Anspaugh , Henry Van Tuyl Cotter
IPC分类号： A01N43/78 , C07D277/18 , A01P5/00 , A01P7/00
CPC分类号： C07D277/18
摘要： The present invention relates to azoline compounds and their salts which are useful for combating arthropod pests. The present invention also relates to a method for combating arthropod pests and to agricultural compositions for combating said pests. It has been found that these objectives can be achieved by azoline compounds of the general formulae Ia or Ib, wherein X is S, O or NR4; Ar is phenyl or a 5 or 6 membered heteroaromatic ring; R1 is H, C1-C6-alkyl, C2-C6-alkenyl, phenyl, a heteroaromatic ring etc.; R2a, R2b are H, CN, C1-C6-alkyl etc.; R1 together with R2a may also form a linear C2-C4-alkandiyl; R3a-d are H, halogen, C1-C6-alkyl etc.
摘要翻译：本发明涉及可用于防治节肢动物害虫的唑啉化合物及其盐。本发明还涉及一种防治节肢动物害虫的方法和用于对抗所述害虫的农业组合物。已经发现，这些目的可以通过通式Ia或Ib的唑啉化合物来实现，其中X是S，O或NR 4; Ar是苯基或5或6元杂芳环; R1是H，C1-C6-烷基，C2-C6-烯基，苯基，杂芳环等; R2a，R2b是H，CN，C1-C6-烷基等; R1与R2a一起也可以形成直链C 2 -C 4 - 烷二基; R3a-d为H，卤素，C1-C6烷基等。

9. 发明申请

US20080176826A1 Pyridine Compounds For Combating Arthropod Pests and Nematodes 审中-公开
标题翻译：用于防治节肢动物害虫和线虫的吡啶化合物
公开(公告)号：US20080176826A1
公开(公告)日：2008-07-24
申请号：US11914996
申请日：2006-05-24
申请人： Michael Puhl , Michael Rack , Thomas Schmidt , Michael Hofmann , Ernst Baumann , Markus Kordes , Wolfgang Von Deyn , David G. Kuhn , Deborah L. Culbertson , Douglas D. Anspaugh , Henry Van Tuyl Cotter , Hassan Oloumi-Sadeghi , Tony Bucci , Henricus Maria Martinus Bastiaans
发明人： Michael Puhl , Michael Rack , Thomas Schmidt , Michael Hofmann , Ernst Baumann , Markus Kordes , Wolfgang Von Deyn , David G. Kuhn , Deborah L. Culbertson , Douglas D. Anspaugh , Henry Van Tuyl Cotter , Hassan Oloumi-Sadeghi , Tony Bucci , Henricus Maria Martinus Bastiaans
IPC分类号： A01N43/44 , C07D401/12 , A01P7/00 , A01N43/40
CPC分类号： A01N43/40 , C07D401/12
摘要： The present invention relates to new pyridine compounds which are useful for combating animal pests, in particular insects, arachnids and nematodes. The invention also relates to a method for combating insects, nematodes and arachnids.The pyridine compounds have the formula I as defined below. Likewise, compounds of the formula II are suitable for combating pests. In formulae I and II n is 1 or 2, and R1, R2, R3, R4 and R5 are as defined in the claims and in the specification.
摘要翻译：本发明涉及可用于对抗动物害虫，特别是昆虫，蜘蛛和线虫的新的吡啶化合物。本发明还涉及一种防治昆虫，线虫和蜘蛛的方法。吡啶化合物具有如下定义的式I。同样，式II化合物适用于防治害虫。在式I和II中，n为1或2，R 1，R 2，R 3，R 4， >和R＆gt; 5如权利要求书和说明书中所定义。

10. 发明授权

US08173675B2 Substituted amino-thiourea compounds for combating animal pests 失效
标题翻译：用于对抗动物害虫的取代氨基 - 硫脲化合物
公开(公告)号：US08173675B2
公开(公告)日：2012-05-08
申请号：US12601017
申请日：2008-05-13
申请人： Christopher Koradin , Markus Kordes , Ernst Baumann , Ronan Le Vezouet , Deborah L. Culbertson
发明人： Christopher Koradin , Markus Kordes , Ernst Baumann , Ronan Le Vezouet , Deborah L. Culbertson
IPC分类号： A61K31/47 , C07D215/14
CPC分类号： A01N47/36 , A01N47/32 , C07C335/14 , C07C2602/08 , C07C2602/10 , C07D307/82 , C07D333/66
摘要： The invention relates to substituted amino-thiourea compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amino-thiourea compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such compounds. The substituted amino-thiourea compounds are defined by the following formula (I): wherein A, B, R1, R2, R3, R4, R5.1, R5.2 and R6 are defined as in the description.
摘要翻译：本发明涉及式（I）的取代的氨基 - 硫脲化合物，其涉及其对映体，非对映异构体和盐以及包含这些化合物的组合物。本发明还涉及取代的氨基 - 硫脲化合物，其盐或包含它们的组合物用于对抗动物害虫的用途。此外，本发明还涉及应用这些化合物的方法。取代的氨基 - 硫脲化合物由下式（I）定义：其中A，B，R1，R2，R3，R4，R5.1，R5.2和R6如说明书所定义。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式