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1. 发明申请

US20060041883A1 System and method for configuring computer for operation 有权
公开(公告)号：US20060041883A1
公开(公告)日：2006-02-23
申请号：US10922264
申请日：2004-08-19
申请人： Howell Chambers , Kevin Henegar , David Karner , Andrew Mueller
发明人： Howell Chambers , Kevin Henegar , David Karner , Andrew Mueller
IPC分类号： G06F9/445
CPC分类号： G06F9/4411
摘要： A method for deploying software in a computer system includes providing a deployment maintenance mechanism (DMM) which includes drivers for hardware. A deployment mechanism which includes an image with drivers for hardware and which identifies hardware associated with the computer, along with a native operating system, are also provided. For hardware detected by the deployment mechanism and not having an associated driver in the image, a driver from the DMM is copied into the deployment mechanism using the native operating system. The native operating system is then re-booted to deploy drivers for hardware associated with the computer.

2. 发明申请

US20050187388A1 Method for the preparation of aryl ethers 审中-公开
标题翻译：芳基醚的制备方法
公开(公告)号：US20050187388A1
公开(公告)日：2005-08-25
申请号：US11059895
申请日：2005-02-17
申请人： Mateusz Cebula , Kevin Henegar
发明人： Mateusz Cebula , Kevin Henegar
IPC分类号： C07D265/30 , C07D265/32
CPC分类号： C07D265/30
摘要： The invention provides a method of preparing a compound of formula (I): wherein R, R1, n and m are as defined herein, or a pharmaceutically acceptable salt thereof.
摘要翻译：本发明提供制备式（I）化合物的方法：其中R 1，R 1，n和m如本文所定义，或其药学上可接受的盐。

3. 发明申请

US20050124668A1 Amino acids with affinity for the alpha2delta-protein 审中-公开
标题翻译：对α2delta蛋白具有亲和力的氨基酸
公开(公告)号：US20050124668A1
公开(公告)日：2005-06-09
申请号：US10949908
申请日：2004-09-24
申请人： Christopher Deur , Kevin Henegar , Christine Kolz , Jonathan Miller , Augastine Osuma , Mark Plummer , Brian Samas , Jacob Schwarz , Andrew Thorpe , David Wustrow
发明人： Christopher Deur , Kevin Henegar , Christine Kolz , Jonathan Miller , Augastine Osuma , Mark Plummer , Brian Samas , Jacob Schwarz , Andrew Thorpe , David Wustrow
IPC分类号： A61P23/00 , C07C227/32 , C07C229/08 , C07C229/28 , C07C229/34 , C07D263/26 , A61K31/44 , A61K31/198 , A61K31/277 , C07D213/55
CPC分类号： C07C229/08 , C07B2200/07 , C07C227/32 , C07C229/28 , C07C229/34 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14 , C07D263/26 , Y02P20/582
摘要： Certain β-amino acids that bind to the alpha-2-delta (α2δ) subunit of a calcium channel are disclosed. These compounds and their pharmaceutically acceptable salts are useful in the treatment of a variety of psychiatric, pain and other disorders.
摘要翻译：公开了结合钙通道的α-2-δ（α2delta）亚基的某些β-氨基酸。这些化合物及其药学上可接受的盐可用于治疗各种精神病，疼痛和其它疾病。

4. 发明申请

US20050038123A1 Process and intermediates to prepare latanoprost 审中-公开
标题翻译：制备拉坦前列素的方法和中间体
公开(公告)号：US20050038123A1
公开(公告)日：2005-02-17
申请号：US10920567
申请日：2004-08-18
申请人： Kevin Henegar
发明人： Kevin Henegar
IPC分类号： C07C59/54 , C07C59/72 , C07C405/00 , C07D307/935 , A61K31/557 , A61K31/19
CPC分类号： C07D307/935 , C07C59/54 , C07C59/72 , C07C405/0016
摘要： The present invention is a novel intermediate, compound of the formula (VI) and salts thereof. In addition, the invention includes a process for the preparation of a prostaglandin intermediates compounds (IV) and (XVIII) which comprises (1) contacting a the corresponding enone with (−)-chlorodiisopinocampheylborane while maintaining the reaction mixture temperature in the range of from about −50° to about 0° and (2) contacting the reaction mixture of step (1) with a boron complexing agent.
摘要翻译：本发明是一种新的中间体式（Ⅵ）化合物及其盐。另外，本发明包括制备前列腺素中间体化合物（Ⅳ）和（ⅩⅧ）的方法，其包括（1）使相应的烯酮与（ - ） - 氯二异蒎烷yl基硼烷接触，同时保持反应混合物的温度在约-50°至约0°，和（2）使步骤（1）的反应混合物与硼络合剂接触。

5. 发明申请

US20070129550A1 AMINO ACIDS WITH AFFINITY FOR THE ALPHA-2-DELTA-PROTEIN 失效
标题翻译：具有ALPHA-2-DELTA-PROTEIN的亲和力的氨基酸
公开(公告)号：US20070129550A1
公开(公告)日：2007-06-07
申请号：US11567878
申请日：2006-12-07
申请人： Peter Blazecka , Joseph Bozelak , Norman Colbry , Timothy Curran , Annise Goodman , Kevin Henegar , Garrett Hoge , Paul Johnson , Augustine Osuma , Mark Plummer , Jacob Schwarz , Derek Vrieze , Ji Zhang
发明人： Peter Blazecka , Joseph Bozelak , Norman Colbry , Timothy Curran , Annise Goodman , Kevin Henegar , Garrett Hoge , Paul Johnson , Augustine Osuma , Mark Plummer , Jacob Schwarz , Derek Vrieze , Ji Zhang
IPC分类号： A61K31/44 , C07D413/02 , C07D213/55 , C07C255/45 , C07C229/14
CPC分类号： C07C229/08 , C07B2200/07 , C07C227/32 , C07C229/28 , C07C229/34 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14 , C07D263/26 , Y02P20/582
摘要： Certain β-amino acids that bind to the alpha-2-delta (α2δ) subunit of a calcium channel are disclosed. These compounds and their pharmaceutically acceptable salts are useful in the treatment of a variety of psychiatric, pain and other disorders. Also disclosed are methods of making the β-amino acids.
摘要翻译：公开了结合钙通道的α-2-δ（α2delta）亚基的某些β-氨基酸。这些化合物及其药学上可接受的盐可用于治疗各种精神病，疼痛和其它疾病。还公开了制备β-氨基酸的方法。

6. 发明申请

US20060287309A1 [1,8]NAPHTHYRIDIN-2-ONES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA 审中-公开
公开(公告)号：US20060287309A1
公开(公告)日：2006-12-21
申请号：US11466822
申请日：2006-08-24
申请人： Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
发明人： Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
IPC分类号： A61K31/5383 , A61K31/519 , A61K31/525 , A61K31/496 , A61K31/4745 , C07D491/02 , C07D487/02
CPC分类号： C07D471/04
摘要： This invention relates to compounds of the formula 1 wherein G, D, A, Z, Q, X, Y, R1, and R4 through R7 are defined as in the specification, processes for preparing the same and intermediates used in making the same, and pharmaceutical compositions containing such compounds and their use in the treatment of central nervous system disorders and other disorders.

7. 发明申请

US20050187399A1 Method for the preparation of aryl ethers 审中-公开
标题翻译：芳基醚的制备方法
公开(公告)号：US20050187399A1
公开(公告)日：2005-08-25
申请号：US11060172
申请日：2005-02-17
申请人： Mateusz Cebula , Kevin Henegar
发明人： Mateusz Cebula , Kevin Henegar
IPC分类号： C07C41/03 , C07C43/23 , C07C217/28 , C07C217/34 , C07F7/08 , C07F7/18
CPC分类号： C07C41/03 , C07B2200/07 , C07C43/23 , C07C217/34 , C07F7/1804 , Y02P20/55
摘要： The invention comprises an enantioselective method of preparing a compound of formula (IV): wherein n, m, R and R1 are as defined herein. Use of the compounds of formula (IV) in a method of preparing compounds of formula (IX) and novel intermediates useful in the method are also described.
摘要翻译：本发明包括制备式（IV）化合物的对映选择性方法：其中n，m，R和R 1如本文所定义。还描述了在制备式（IX）化合物的方法中使用式（Ⅳ）化合物和在该方法中有用的新中间体。

8. 发明申请

US20060287310A1 [1,8]NAPHTHYRIDIN-2-ONES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA 审中-公开
标题翻译： [1,8]萘啶-2-酮及相关化合物治疗苦参碱
公开(公告)号：US20060287310A1
公开(公告)日：2006-12-21
申请号：US11466828
申请日：2006-08-24
申请人： Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
发明人： Jerry Clark , Jamie Davis , David Favor , Lorraine Fay , Lloyd Franklin , Kevin Henegar , Douglas Johnson , Brian Nichelson , Ligong Ou , Joseph Repine , Michael Walters , Andrew White , Zhijian Zhu
IPC分类号： A61K31/5383 , A61K31/519 , A61K31/496 , A61K31/4745 , C07D471/02 , C07D491/02 , C07D487/02
CPC分类号： C07D471/04
摘要： This invention relates to compounds of the formula 1 wherein G, D, A, Z, Q, X, Y, R1, and R4 through R7 are defined as in the specification, processes for preparing the same and intermediates used in making the same, and pharmaceutical compositions containing such compounds and their use in the treatment of central nervous system disorders and other disorders.
摘要翻译：本发明涉及式1的化合物，其中G，D，A，Z，Q，X，Y，R 1和R 4至R 7 在说明书中定义，其制备方法和用于制备其的中间体，以及含有这些化合物的药物组合物及其在治疗中枢神经系统疾病和其它疾病中的用途。

9. 发明申请

US20050197355A1 COMPOUNDS USEFUL IN PREPARING CAMPTOTHECIN DERIVATIVES 审中-公开
标题翻译：化合物可用于制备CAMPTOTHECIN衍生物
公开(公告)号：US20050197355A1
公开(公告)日：2005-09-08
申请号：US10791198
申请日：2004-03-02
申请人： Kevin Henegar
发明人： Kevin Henegar
IPC分类号： A61K31/4545 , A61K31/4745
CPC分类号： A61K31/4745 , A61K31/4545 , A61K2300/00
摘要： Novel compounds are provided having the formula and salts thereof, where R1 is hydrogen, an alkyl, aralkyl, hydroxymethyl, carboxymethyl, acyloxymethyl or trialkylsilyl group, or a group —CH2NR3R4 where N is a linking nitrogen atom and where (a) R3 and R4 are independently selected from hydrogen and alkyl, alkenyl, hydroxyalkyl and alkoxyalkyl groups; (b) R3 is hydrogen or an alkyl, alkenyl, hydroxyalkyl or alkoxyalkyl group, and R4 is —COR5 where R5 is hydrogen or an alkyl, alkenyl, hydroxyalkyl or alkoxyalkyl group; or (c) R3 and R4 taken together with the linking nitrogen atom form a saturated 3- to 7-member heterocyclic group. These compounds are useful intermediates in a process to prepare camptothecin derivatives including the anti-cancer drug irinotecan.
摘要翻译：提供了具有式及其盐的新化合物，其中R 1是氢，烷基，芳烷基，羟甲基，羧甲基，酰氧基甲基或三烷基甲硅烷基或基团-CH 2 其中N为连接氮原子，其中（a）R 3和R 4为H，独立地选自氢和烷基，烯基，羟基烷基和烷氧基烷基; （b）R 3是氢或烷基，烯基，羟基烷基或烷氧基烷基，R 4是-COR 5，其中R SUP > 5是氢或烷基，烯基，羟基烷基或烷氧基烷基; 或（c）R 3和R 4与连接氮原子一起形成饱和的3-至7-元杂环基。这些化合物在制备喜树碱衍生物的方法中是有用的中间体，包括抗癌药物伊立替康。

10. 发明申请

US20050101643A1 Amino acids with affinity for the alpha2delta-protein 失效
标题翻译：对α2delta蛋白具有亲和力的氨基酸
公开(公告)号：US20050101643A1
公开(公告)日：2005-05-12
申请号：US10949907
申请日：2004-09-24
申请人： Peter Blazecka , Joseph Bozelak , Norman Colbry , Timothy Curran , Annise Goodman , Kevin Henegar , Garrett Hoge , Paul Johnson , Augustine Osuma , Mark Plummer , Jacob Schwarz , Derek Vrieze , Ji Zhang
发明人： Peter Blazecka , Joseph Bozelak , Norman Colbry , Timothy Curran , Annise Goodman , Kevin Henegar , Garrett Hoge , Paul Johnson , Augustine Osuma , Mark Plummer , Jacob Schwarz , Derek Vrieze , Ji Zhang
IPC分类号： A61P23/00 , C07C227/32 , C07C229/08 , C07C229/28 , C07C229/34 , C07D263/26 , A61K31/44 , A61K31/198 , C07C227/18
CPC分类号： C07C229/08 , C07B2200/07 , C07C227/32 , C07C229/28 , C07C229/34 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14 , C07D263/26 , Y02P20/582
摘要： Certain β-amino acids that bind to the alpha-2-delta (α2δ) subunit of a calcium channel are disclosed. These compounds and their pharmaceutically acceptable salts are useful in the treatment of a variety of psychiatric, pain and other disorders. Also disclosed are methods of making the β-amino acids.
摘要翻译：公开了结合钙通道的α-2-δ（α2delta）亚基的某些β-氨基酸。这些化合物及其药学上可接受的盐可用于治疗各种精神病，疼痛和其它疾病。还公开了制备β-氨基酸的方法。

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