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1. 发明授权

US4556737A Sulfonium compounds, processes for preparing the compounds and pharmacological composiitons containing the same 失效
标题翻译：锍化合物，制备化合物的方法和含有该化合物的药物组合物
公开(公告)号：US4556737A
公开(公告)日：1985-12-03
申请号：US583674
申请日：1984-02-27
申请人： Akihide Koda , Mikio Hori , Naosuke Matsuura , Mitsugi Yasumoto , Ichiro Yamawaki , Shuichi Ueda , Yukio Tada
发明人： Akihide Koda , Mikio Hori , Naosuke Matsuura , Mitsugi Yasumoto , Ichiro Yamawaki , Shuichi Ueda , Yukio Tada
IPC分类号： A61K31/095 , A61K31/10 , A61K31/13 , A61K31/18 , A61K31/205 , C07C381/12 , C07D307/12 , C07D309/06 , C07C103/12 , C07C41/18 , C07C43/20 , C07C148/00
CPC分类号： C07D307/12 , C07C309/30 , C07C381/12
摘要： This invention provides novel sulfonium compounds, processes for the preparation of the sulfonium compounds, and pharmacological composition containing the sulfonium compound. The compounds of this invention are useful for treating allergy.
摘要翻译：本发明提供新的锍化合物，锍化合物的制备方法和含有锍化合物的药物组合物。本发明的化合物可用于治疗过敏。

2. 发明授权

US4670583A Amide compounds 失效
标题翻译：酰胺化合物
公开(公告)号：US4670583A
公开(公告)日：1987-06-02
申请号：US772857
申请日：1985-09-05
申请人： Akihide Koda , Mikio Hori , Mitsugi Yasumoto , Naosuke Matsuura , Ichiro Yamawaki , Yukio Tada
发明人： Akihide Koda , Mikio Hori , Mitsugi Yasumoto , Naosuke Matsuura , Ichiro Yamawaki , Yukio Tada
IPC分类号： A61K31/165 , A61K31/195 , A61P37/08 , C07C67/00 , C07C233/16 , C07C233/27 , C07C313/00 , C07C317/44 , C07C323/60 , C07C149/40 , C07C103/38 , C07C103/58
CPC分类号： A61K31/165 , C07C233/16
摘要： This invention provides an amide compound represented by the formula ##STR1## wherein R.sub.1 is vinyl, 2-(methylsulfinyl)ethyl, 2-(methylsulfonyl)ethyl, 2-(2-acetylamino-2-carboxyethylthio)ethyl or 2-[2-(4-amino-4-carboxybutyrylamino)-2-(carboxymethylcarbamoyl)ethylthio]ethyl and R.sub.2 is hydrogen or lower alkyl, process for the preparation thereof, and antiallergic compositions cotaining the amide compound.
摘要翻译：本发明提供由式（I）表示的酰胺化合物，其中R 1是乙烯基，2-（甲基亚磺酰基）乙基，2-（甲基磺酰基）乙基，2-（2-乙酰基氨基-2-羧乙硫基）乙基或2- [2-（4-氨基-4-羧基丁酰氨基）-2-（羧甲基氨基甲酰基）乙基]乙基，R2是氢或低级烷基，其制备方法和与酰胺化合物接触的抗过敏组合物。

3. 发明授权

US4340543A Sulfonium compounds 失效
标题翻译：锍化合物
公开(公告)号：US4340543A
公开(公告)日：1982-07-20
申请号：US231126
申请日：1981-02-03
申请人： Akihide Koda , Mikio Hori , Mitsugi Yasumoto , Ichiro Yamawaki , Yuji Yamada , Katsuo Takikawa
发明人： Akihide Koda , Mikio Hori , Mitsugi Yasumoto , Ichiro Yamawaki , Yuji Yamada , Katsuo Takikawa
IPC分类号： A61K31/34 , A61K31/341 , A61K31/35 , A61K31/351 , A61P35/00 , A61P37/04 , C07D307/10 , C07D309/04
CPC分类号： C07D307/10 , C07D309/04 , Y10S514/96 , Y10S514/962 , Y10S514/966
摘要： Sulfonium compounds represented by the formula ##STR1## have anticancer activity, immunostimulant activity and the like, and useful as the active components of drugs and agricultural chemicals.
摘要翻译：由式（I）表示的锍化合物具有抗癌活性，免疫刺激活性等，可用作药物和农药的活性成分。

4. 发明授权

US4581372A Sulfonium compounds 失效
标题翻译：锍化合物
公开(公告)号：US4581372A
公开(公告)日：1986-04-08
申请号：US541799
申请日：1983-10-14
申请人： Akihide Koda , Mikio Hori , Mitsugi Yasumoto , Ichiro Yamawaki , Yuji Yamada , Katsuo Takikawa
发明人： Akihide Koda , Mikio Hori , Mitsugi Yasumoto , Ichiro Yamawaki , Yuji Yamada , Katsuo Takikawa
IPC分类号： A61K31/34 , A61K31/341 , A61K31/35 , A61K31/351 , A61P35/00 , A61P37/04 , C07D307/10 , C07D309/04
CPC分类号： C07D307/10 , C07D309/04
摘要： Sulfonium compounds represented by the formula ##STR1## having immunostimulant activity and useful as the active components of drugs and agricultural chemicals.
摘要翻译：由式（I）表示的具有免疫刺激活性并可用作药物和农药活性成分的锍化合物。

5. 发明授权

US4696929A Derivative of piperazine having anti-allergic and anti-inflammatory action 失效
标题翻译：具有抗过敏和抗炎作用的哌嗪衍生物
公开(公告)号：US4696929A
公开(公告)日：1987-09-29
申请号：US809876
申请日：1985-12-17
申请人： Ichiro Yamawaki , Kazuo Ogawa , Naohiko Ono , Takaji Honna , Sekio Nagayama , Mitsugi Yasumoto
发明人： Ichiro Yamawaki , Kazuo Ogawa , Naohiko Ono , Takaji Honna , Sekio Nagayama , Mitsugi Yasumoto
IPC分类号： C07D405/12 , A61K31/495 , A61P29/00 , A61P37/08 , A61P43/00 , C07D209/28 , C07D403/12 , C07F7/18 , C12N9/99
CPC分类号： C07D209/28 , Y02P20/55
摘要： A piperazine derivative represented by the formula (I) below ##STR1## wherein R.sup.1 is lower alkyl or phenyl, R.sup.2 is hydrogen or lower alkyl, n is an integer of 2 to 10, is useful as an effective component of anti-inflammatory agent or antiallergic agent.
摘要翻译：由下式（I）表示的哌嗪衍生物，其中R 1为低级烷基或苯基，R 2为氢或低级烷基，n为2至10的整数，可用作抗 - 抗炎剂或抗过敏剂。

6. 发明授权

US4092313A Preparation of 5-fluoropyrimidin-4-one derivatives 失效
标题翻译： 5-氟嘧啶-4-酮衍生物的制备
公开(公告)号：US4092313A
公开(公告)日：1978-05-30
申请号：US729980
申请日：1976-10-06
申请人： Mitugi Yasumoto , Junichi Yamashita , Ichiro Yamawaki , Norio Unemi , Kenji Kitazato , Sadao Hashimoto , Setsuro Fujii
发明人： Mitugi Yasumoto , Junichi Yamashita , Ichiro Yamawaki , Norio Unemi , Kenji Kitazato , Sadao Hashimoto , Setsuro Fujii
IPC分类号： C07D239/52 , C07D239/36
CPC分类号： C07D239/52
摘要： A 5-fluoropyrimidin-4-one derivative represented by the formula ##STR1## wherein R is straight-chain or branched-chain alkyl having 4 to 18 carbon atoms, straight-chain or branched-chain alkenyl having 2 to 18 carbon atoms, alkylene oxido having 3 to 10 carbon atoms, aryl or aralkyl;Processes for preparing the derivative;An anti-tumor composition containing the derivative as an effective component and an excipient.
摘要翻译：其中R为具有4至18个碳原子的直链或支链烷基，具有2至18个碳原子的直链或支链烯基，亚烷基具有3至10个碳原子的氧化物，芳基或芳烷基; 制备衍生物的方法; 包含衍生物作为有效成分和特殊物质的抗肿瘤组合物。

7. 发明授权

US6134133A Piezoelectric transformer inverter 有权
标题翻译：压电变压器
公开(公告)号：US6134133A
公开(公告)日：2000-10-17
申请号：US389286
申请日：1999-09-02
申请人： Takashi Noma , Ichiro Yamawaki , Yasuyuki Morishima
发明人： Takashi Noma , Ichiro Yamawaki , Yasuyuki Morishima
IPC分类号： H02M7/48 , H02M7/538 , H02M7/539 , H05B41/24
CPC分类号： H02M7/53806
摘要： A piezoelectric transformer inverter includes an inverter unit and a step-down chopper unit. The inverter unit includes a ceramic piezoelectric transformer whose secondary terminal is to be connected to a fluorescent tube, a drive unit which is connected to a primary terminal of the ceramic piezoelectric transformer, and an inverter control circuit for controlling luminance of the fluorescent tube to a desired value. The step-down chopper unit includes a switching device which is disposed on the side where the voltage of the inverter unit is input, a free wheeling device connected between the switching device and a reference potential, and a PWM feedback control circuit for providing a feedback control to maintain an average voltage of the rectangular-wave voltage of the switching device constant. In the piezoelectric transformer inverter, even when the feedback control by the PWM feedback control circuit is impossible, the on-duty of the chopper unit is restricted so that it is not greater than a given amount.
摘要翻译：压电变压器逆变器包括逆变器单元和降压斩波单元。逆变器单元包括将二次端子连接到荧光管的陶瓷压电变压器，连接到陶瓷压电变压器的初级端子的驱动单元和用于将荧光管的亮度控制为所需值。降压斩波器单元包括设置在输入逆变器单元的电压的一侧的开关装置，连接在开关装置和参考电位之间的续流装置，以及用于提供反馈的PWM反馈控制电路控制以保持开关装置的矩形波电压的平均电压恒定。在压电变压器逆变器中，即使不能通过PWM反馈控制电路进行反馈控制，限制了斩波器单元的占空比，使其不大于给定量。

8. 发明授权

US4080455A 5-Fluoropyrimidin-4-one compositions 失效
标题翻译： 5-氟嘧啶-4-酮组合物
公开(公告)号：US4080455A
公开(公告)日：1978-03-21
申请号：US701216
申请日：1976-06-30
申请人： Mitugi Yasumoto , Junichi Yamashita , Ichiro Yamawaki , Norio Unemi , Kenji Kitazato , Sadao Hashimoto , Setsuro Fujii
发明人： Mitugi Yasumoto , Junichi Yamashita , Ichiro Yamawaki , Norio Unemi , Kenji Kitazato , Sadao Hashimoto , Setsuro Fujii
IPC分类号： C07D239/52 , A61K31/505
CPC分类号： C07D239/52
摘要： A 5-fluoropyrimidin-4-one derivative represented by the formula ##STR1## wherein R is straight-chain or branched-chain alkyl having 4 to 18 carbon atoms, straight-chain or branched-chain alkenyl having 2 to 18 carbon atoms, alkylene oxido having 3 to 10 carbon atoms, aryl or aralkyl;Processes for preparing the derivative;An anti-tumor composition containing the derivative as an effective component and an excipient.
摘要翻译：其中R为具有4至18个碳原子的直链或支链烷基，具有2至18个碳原子的直链或支链烯基，亚烷基具有3至10个碳原子的氧化物，芳基或芳烷基; 制备衍生物的方法; 包含衍生物作为有效成分和特殊物质的抗肿瘤组合物。

9. 发明授权

US6159987A Bicyclolactam compounds, use thereof and intermediates for preparing thereof 失效
标题翻译：双环内酰胺化合物，其用途及其制备中间体
公开(公告)号：US6159987A
公开(公告)日：2000-12-12
申请号：US432115
申请日：1999-11-02
申请人： Junji Yamamoto , Takashi Arima , Nobuo Kasahara , Masato Nanri , Kazuo Ogawa , Ichiro Yamawaki , Manabu Kaneda
发明人： Junji Yamamoto , Takashi Arima , Nobuo Kasahara , Masato Nanri , Kazuo Ogawa , Ichiro Yamawaki , Manabu Kaneda
IPC分类号： A61K31/40 , A61K31/445 , A61K31/47 , A61K31/55 , A61P25/22 , C07D215/22 , C07D215/227 , C07D221/16 , C07D221/04 , A01K31/4353
CPC分类号： C07D215/227 , A61K31/40 , A61K31/445 , A61K31/47 , A61K31/55 , C07D221/16
摘要： A bicyclolactam compound of the formula (1) is disclosed, which has an excellent anxiolytic effect, is high in safety, and is useful as an effective component of medicinals which are greatly diminished in side effects such as hypnotic, muscle relaxant and sedative effects ##STR1## A bicyclolactam derivative represented by the following formula (1) is also disclosed, and is useful as an effective component of an anxiolytic agent ##STR2##
摘要翻译：公开了式（1）的双环内酰胺化合物，其具有优异的抗焦虑作用，安全性高，可用作药物的有效成分，其在副作用如催眠，肌肉松弛剂和镇静作用A中大大降低还公开了由下式（1）表示的双环内酰胺衍生物，可用作抗焦虑剂的有效成分

10. 发明授权

US4814449A Substance 4181-2 失效
标题翻译：物质4181-2
公开(公告)号：US4814449A
公开(公告)日：1989-03-21
申请号：US48297
申请日：1987-05-11
申请人： Qi Chang-qing , Tian Jie , Teruyoshi Marunaka , Yuji Yamada , Ichiro Yamawaki , Toshio Ohtani , Yoshinori Minami , Hitoshi Saito
发明人： Qi Chang-qing , Tian Jie , Teruyoshi Marunaka , Yuji Yamada , Ichiro Yamawaki , Toshio Ohtani , Yoshinori Minami , Hitoshi Saito
IPC分类号： C07D498/14 , C12P17/18 , C07D498/12 , A61K31/33 , A61K31/445
CPC分类号： C07D498/14 , C12P17/188 , C12R1/465 , Y10S514/908
摘要： Disclosed are a compound of the general formula ##STR1## wherein R.sub.1 and R.sub.2 are the same or different and each represents a hydrogen atom, an alkyl group or an acyl group, process for the production thereof and use thereof. The compounds have an antitumor activity, and those wherein both of R.sub.1 and R.sub.2 represent a hydrogen atom or an acyl group are novel compounds.
摘要翻译：公开了通式（II）的化合物，其中R 1和R 2相同或不同，各自表示氢原子，烷基或酰基，其制备方法和用途。这些化合物具有抗肿瘤活性，其中R1和R2都表示氢原子或酰基的化合物是新化合物。

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