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1. 发明授权

US4352752A Process for the preparation of dipeptides 失效
标题翻译：制备二肽的方法
公开(公告)号：US4352752A
公开(公告)日：1982-10-05
申请号：US240983
申请日：1981-03-05
申请人： Iwao Ojima , Shigemi Suga
发明人： Iwao Ojima , Shigemi Suga
IPC分类号： B01J23/00 , C07B61/00 , C07C67/00 , C07C231/00 , C07C231/10 , C07C235/34 , C07C237/12 , C07C237/20 , C07C237/22 , C07D205/08 , C07D205/085 , C07K1/113 , C07K1/12 , C07K5/06 , C07C103/52 , C07C101/30 , C07C101/72
CPC分类号： C07K1/12 , C07D205/08 , C07D205/085
摘要： There is provided a novel process for the preparation of a dipeptide represented by the formula: ##STR1## wherein Ar represents an aromatic group; R.sup.1 represents a hydrogen atom, an alkyl group or an aryl group; R.sup.2 represents a hydrogen atom, an alkyl group or an aromatic group; Y represents a hydroxy group, an amino group or an acylamino group, which comprises subjecting a .beta.-lactam compound represented by the formula: ##STR2## wherein Ar, R.sup.1 and R.sup.2 have the same meanings as defined above, and X represents a hydroxy group, an amino group or an acylamino group, an azido group or a benzyloxy group, to hydrogenolysis in the presence of a catalyst. The process can be practiced without any complicated procedure as seen in the conventional processes for the preparation of peptides.
摘要翻译：提供了制备由下式表示的二肽的新方法：其中Ar表示芳族基团; R1表示氢原子，烷基或芳基; R2表示氢原子，烷基或芳基; Y表示羟基，氨基或酰氨基，其包括使由下式表示的β-内酰胺化合物：其中Ar，R 1和R 2具有与上述相同的含义，X表示羟基，氨基或酰氨基，叠氮基或苄氧基，在催化剂存在下氢解。该方法可以在没有任何复杂的程序的情况下进行，如在用于制备肽的常规方法中所见。

2. 发明授权

US5228898A Substituted bicycloheptandione derivatives 失效
标题翻译：取代的双环蛋白衍生物
公开(公告)号：US5228898A
公开(公告)日：1993-07-20
申请号：US651266
申请日：1992-02-03
申请人： Akiyoshi Ueda , Shigemi Suga , Hiroyuki Adachi , Toshio Aihara , Kazuyuki Tomida , Hideki Yamagishi , Hideo Hosaka
发明人： Akiyoshi Ueda , Shigemi Suga , Hiroyuki Adachi , Toshio Aihara , Kazuyuki Tomida , Hideki Yamagishi , Hideo Hosaka
IPC分类号： C07D239/26 , A01N31/06 , A01N35/06 , A01N37/18 , A01N37/34 , A01N37/42 , A01N41/06 , A01N41/08 , A01N41/10 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/76 , A01N43/78 , C07C20060101 , C07C45/67 , C07C49/323 , C07C49/433 , C07C49/477 , C07C49/517 , C07C49/733 , C07C49/747 , C07C49/792 , C07C49/813 , C07C49/83 , C07C49/84 , C07C65/36 , C07C67/30 , C07C69/76 , C07C201/12 , C07C205/45 , C07C205/46 , C07C253/30 , C07C255/56 , C07C309/86 , C07C317/24 , C07C317/44 , C07C323/22 , C07C323/52 , C07D213/50 , C07D213/61 , C07D213/70 , C07D231/16 , C07D239/34 , C07D239/38 , C07D239/52 , C07D239/56 , C07D239/58 , C07D277/24 , C07D277/34 , C07D521/00
CPC分类号： C07D213/70 , A01N35/06 , A01N37/18 , A01N37/42 , A01N41/06 , A01N41/10 , A01N43/40 , A01N43/56 , A01N43/78 , C07C205/45 , C07C255/56 , C07C317/24 , C07C45/673 , C07C45/676 , C07C49/433 , C07C49/477 , C07C49/517 , C07C49/733 , C07C49/747 , C07C49/792 , C07C49/813 , C07C49/84 , C07C65/36 , C07C69/76 , C07D213/50 , C07D213/61 , C07D231/16 , C07D277/34 , C07C2102/20
摘要： This invention relates to substituted bicycloheptadione derivatives with high herbicidal activity which are represented by general formula (I) ##STR1## (where R.sup.1 is a lower alkyl group, a phenyl group which may be substituted, an aralkyl group which may be substituted, or a heterocyclic group which may be substituted;R.sup.2 is, same or different, a halogen, an alkoxy group, an alkylthio group, an alkylsulfonyl group, an alkyl group, an alkoxyalkyl group, or an alkoxylcarbonyl group, and n is 0 to 4;R.sup.3 and R.sup.4 are, same or different, hydrogen or a lower alkyl group).
摘要翻译： PCT No.PCT / JP90 / 00850 Sec。一九九二年二月三日 102（e）日期1993年2月3日PCT Filed 1990年6月29日PCT公布。公开号WO91 / 00260 PCT 1991年1月10日。本发明涉及通式（I）表示的具有高除草活性的取代二环庚二酮衍生物（Ⅰ）（其中R1是低级烷基，可被取代的苯基，可被取代的芳烷基或可被取代的杂环基; R 2相同或不同，为卤素，烷氧基，烷硫基，烷基磺酰基，烷基，烷氧基烷基或烷氧基羰基基团，n为0至4; R 3和R 4相同或不同，为氢或低级烷基）。

3. 发明授权

US5792861A Process for the production of 4-substituted azetidinone derivative 失效
标题翻译：用于制备4-取代的氮杂环丁酮衍生物的方法
公开(公告)号：US5792861A
公开(公告)日：1998-08-11
申请号：US743327
申请日：1996-11-04
申请人： Tamio Hara , Yuuki Nakagawa , Nobuo Matsui , Shigemi Suga
发明人： Tamio Hara , Yuuki Nakagawa , Nobuo Matsui , Shigemi Suga
IPC分类号： C07D413/06 , C07F7/18 , C07D205/08 , C07D403/06 , C07D417/06
CPC分类号： C07D413/06 , C07F7/1892 , Y02P20/55
摘要： The present invention provides a process for the production of a 4-substituted azetidinone. The process comprises reacting ##STR1## wherein R represents a hydrogen atom or a protecting group for N, R.sup.1 represents an alkyl which may be a substituent having an unprotected or protected hydroxyl group; and Z represents a leaving group; with ##STR2## wherein R.sup.2 represents hydrogen or alkyl, R.sup.3 and R.sup.4 each represent hydrogen, alkyl, alkenyl, alkynyl, phenyl, cycloalkyl, or naphthyl, or R.sup.3 and R.sup.4, together with the carbon atom to which they are bonded, form a ring system; X and Y each represent oxygen, sulfur or N-r.sup.1, wherein r.sup.1 represents a hydrogen atom or lower alkyl; A, B, D and E each represent nitrogen or C-r.sup.2, wherein r.sup.2 represents hydrogen, halogen, lower alkyl or lower alkoxy, provided that at least two of A, B, D and E are C-r.sup.2 ; and a ring involving G, J and K has two carbon/carbon double bonds therein and one of G, J and K represents oxygen, sulfur or N-r.sup.1 while the remaining two represent C-r.sup.2 ; in the presence of M(Hal).sub.n (R.sup.5).sub.m (V) wherein M represents a metal atom; Hal represents halogen; R.sup.5 represents lower alkyl, lower alkoxy, phenoxy, substituted phenoxy or cyclopentadienyl; and n and m are each 0, 1, 2, 3, 4 or 5, provided that n+m stands for the valence of M; and a base to thereby give: ##STR3##
摘要翻译：本发明提供了制备4-取代的氮杂环丁酮的方法。该方法包括使其中R表示氢原子或N为保护基的化合物（III）反应，R 1表示可以是具有未被保护或被保护的羟基的取代基的烷基; Z表示离去基团; 代表氢或烷基，R3和R4各自表示氢，烷基，烯基，炔基，苯基，环烷基或萘基，或R3和R4与它们所键合的碳原子一起形成环系; X和Y各自表示氧，硫或N-r1，其中r1表示氢原子或低级烷基; A，B，D和E各自表示氮或C-R 2，其中R 2表示氢，卤素，低级烷基或低级烷氧基，条件是A，B，D和E中的至少两个为C-R 2; 涉及G，J和K的环在其中具有两个碳/碳双键，G，J和K之一表示氧，硫或N-r1，其余两个表示C-r2; 在M（Hal）n（R5）m（V）的存在下，其中M表示金属原子; 卤代表卤素; R5表示低级烷基，低级烷氧基，苯氧基，取代的苯氧基或环戊二烯基; n和m分别为0,1,2,3,4或5，条件是n + m代表M的化合价; （II-1）或（II-2）所示的基础，从而得到：

4. 发明授权

US5739078A Fluoran compounds, intermediates and color forming recording materials 失效
标题翻译：氟化合物，中间体和成色记录材料
公开(公告)号：US5739078A
公开(公告)日：1998-04-14
申请号：US663135
申请日：1996-08-22
申请人： Mitsuhiro Yanagita , Takehiro Sato , Shigemi Suga , Tomoya Hidaka , Toru Kawabe , Mamoru Aizawa , Shinichi Sato , Izuo Aoki
发明人： Mitsuhiro Yanagita , Takehiro Sato , Shigemi Suga , Tomoya Hidaka , Toru Kawabe , Mamoru Aizawa , Shinichi Sato , Izuo Aoki
IPC分类号： B41M5/145 , B41M5/327 , C07C217/92 , C07D493/10 , C09B11/24 , C09B11/28
CPC分类号： C09B11/28 , B41M5/1455 , B41M5/3275 , C07C217/92 , C07D493/10 , C09B11/24
摘要： By using the fluoran compound represented by the following general formula (I); ##STR1## wherein R.sup.1 is alkyl containing 1 to 4 carbon atoms, R.sup.3 is alkyl containing 1 to 8 carbon atoms, R.sup.4 is hydrogen or alkyl containing 1 to 8 carbon atoms, or R.sup.3 and R.sup.4 may bond with each other to form a ring together with a N atom, R.sup.2 is alkyl containing 1 to 4 carbon atoms, and n denotes 0, 1 or 2, however, the substituents represented by R.sup.2 may be different with each other when n is 2, as a color former for color forming recording materials, recording materials which have excellent properties in whiteness of the background of the material under light and in photostability of color-formed images on the materials as well as in sufficient color forming capability of the material even after having exposed them to light, can be provided.
摘要翻译： PCT No.PCT / JP95 / 02096 Sec。 371日期：1996年8月22日 102（e）日期1996年8月22日PCT提交1995年10月13日PCT公布。 WO96 / 11986 PCT公开号日期：1996年4月25日利用下述通式（I）表示的荧蒽化合物。（I）其中R 1是含有1至4个碳原子的烷基，R 3是含有1至8个碳原子的烷基，R 4是氢或含有1至8个碳原子的烷基，或者R 3和R 4可以彼此键合形成与N原子一起形成的环，R2是含有1〜4个碳原子的烷基，n表示0,1或2，但是，当n为2时，由R 2表示的取代基可以相互不同，作为用于成色记录材料，即使在将其暴露于光之后，在材料上的颜色形成图像的光的背景的白色度以及颜色形成图像的光稳定性以及材料的充分的颜色形成能力方面具有优异的性能的记录材料，可以提供。

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