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1. 发明授权

US06362212B1 Oxime derivative and bactericide containing the same as active ingredient 失效
标题翻译：含有与活性成分相同的肟衍生物和杀菌剂
公开(公告)号：US06362212B1
公开(公告)日：2002-03-26
申请号：US09728321
申请日：2000-12-04
申请人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Tsuneo Iwakawa , Kazuo Ueda , Michio Masuko
发明人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Tsuneo Iwakawa , Kazuo Ueda , Michio Masuko
IPC分类号： A61K31415
CPC分类号： C07D231/06 , A01N43/50 , C07D231/12 , C07D233/64 , C07D249/08 , C07D257/04 , C07D261/08 , C07D263/10 , C07D263/32 , C07D271/06 , C07D271/10 , C07D277/10 , C07D285/06
摘要： A compound represented by general formula (I) or a salt thereof, a process for producing the same, an intermediate for the production thereof, and a bactericide (fungicide) containing the same as the active ingredient wherein R1 represent optionally substituted aryl, optionally substituted heterocycle, mono- or di-substituted methyleneamino, optionally substituted (substituted imino)methyl, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, substituted carbonyl or substituted sulfonyl; R2 represents alkyl, alkenyl, alkynyl or cycloalkyl; R3 represents optionally substituted heterocycle; R4 represents hydrogen, alkyl, alkoxy, halogen, nitro, cyano or haloalkyl; M represents oxygen, S(O)i (i being 0, 1 or 2), NR16 (R16 being hydrogen, alkyl or acyl) or a single bond; n represents 0 or 1, provided n represent 1 when R3 represents imidazol-1-yl or 1H-1, 2, 4-triazol-1-yl; and the symbol˜represents the E form, Z form or a mixture thereof.
摘要翻译：由通式（I）表示的化合物或其盐，其制备方法，其制备中间体和含有该活性成分的杀菌剂（杀真菌剂），其中R 1表示任选取代的芳基，任选取代的取代的亚氨基甲基，任选取代的烷基，任选取代的烯基，任选取代的炔基，取代的羰基或取代的磺酰基; R2代表烷基，烯基，炔基或环烷基; R3表示任选取代的杂环; R4代表氢，烷基，烷氧基，卤素，硝基，氰基或卤代烷基; M表示氧，S（O）i（i为0,1或2），NR 16（R 16为氢，烷基或酰基）或单键; 当R 3表示咪唑-1-基或1H-1,2,4-三唑-1-基时，n表示0或1，条件是n表示1。符号〜表示E形式，Z形式或其混合物。

2. 发明授权

US6096741A Oxime derivatives, hydrazone derivatives and use thereof 失效
标题翻译：肟衍生物，腙衍生物及其用途
公开(公告)号：US6096741A
公开(公告)日：2000-08-01
申请号：US284239
申请日：1999-04-14
申请人： Moriyasu Masui , Norihiko Tanimoto , Kuniyoshi Nishida
发明人： Moriyasu Masui , Norihiko Tanimoto , Kuniyoshi Nishida
IPC分类号： A01N37/50 , A01N41/06 , A01N41/10 , A01N43/40 , A01N43/46 , A01N43/80 , A01N47/16 , C07C251/36 , C07C251/48 , C07C251/52 , C07C251/54 , C07C251/74 , C07C259/06 , C07D207/12 , C07D211/42 , C07D211/46 , C07D211/58 , C07D211/72 , C07D213/30 , C07D243/08 , C07D261/02 , C07D295/185 , C07D295/26 , C07D333/16 , C07D401/12 , C07D413/12 , A61K31/535
CPC分类号： C07D213/30 , A01N37/50 , A01N41/06 , A01N41/10 , A01N43/40 , A01N43/46 , A01N43/80 , A01N47/16 , C07C251/36 , C07C251/48 , C07C251/52 , C07C251/54 , C07C251/74 , C07C259/06 , C07D207/12 , C07D211/42 , C07D211/46 , C07D211/58 , C07D211/72 , C07D243/08 , C07D261/02 , C07D295/185 , C07D295/26 , C07D333/16 , C07D401/12
摘要： Compounds having fungicidal activities and represented by general formula (I) and salts and hydrates thereof ##STR1## wherein R.sup.1 represents an optionally substituted aryl, an optionally substituted alkl or the like; R.sup.2 represents an optionally substituted al,y an optionally substituted alkenyl, an optionally substituted alyyl, an optionally substituted aryl, an optionally substituted heterocyclic group or the like; R.sup.3 represents an optionally substituted alkl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted arylsulfonyl, an optionally substituted heterocyclic group or the like; R.sup.4 and R.sup.5, which may be the same or different, represent each a hydrogen atom, an optionally substituted al,y or an optionally substituted allkoxy, or R.sup.4 and R.sup.5 may form together with the adjacent nitrogen atom an optionally substituted monocycle or polycycle; X and Y, which may be the same or different, represents each an oxygen atom or NR.sup.6 wherein R.sup.6 represents a hydrogen atom, an optionally substituted alkyl an optionally substituted aryl, an optionally substituted alkanoyl, or an optionally substituted aroyl; Z represents an oxygen atom or a sulfur atom; and a wavy line (.about.) represents the configuration of an E isomer, a Z isomer, or a mixtue thereof.
摘要翻译： PCT No.PCT / JP97 / 03585第 371 1999年4月14日第 102（e）1999年4月14日PCT PCT 1997年10月7日PCT公布。第WO98 / 16499号公报日期：1998年4月23日具有杀真菌活性并由通式（I）表示的化合物及其盐和水合物，其中R1表示任选取代的芳基，任选取代的烷基等; R 2表示任选取代的芳基，任选取代的烯基，任选取代的芳基，任选取代的芳基，任选取代的杂环基等; R3表示任选取代的烷基，任选取代的烯基，任选取代的炔基，任选取代的芳基磺酰基，任选取代的杂环基团等; R 4和R 5可以相同或不同，表示氢原子，任选被取代的烷基，y或任选取代的全烷氧基，或者R 4和R 5可以与相邻的氮原子一起形成任选取代的单环或多环; X和Y可以相同或不同，表示每个氧原子或NR 6，其中R 6表示氢原子，任选取代的烷基，任选取代的芳基，任选取代的烷酰基或任选取代的芳酰基; Z表示氧原子或硫原子; 和波浪线（DIFFERENCE）表示E异构体，Z异构体或其混合物的构型。

3. 发明授权

US5650539A Process for producing alkoxyiminoacetamide compounds and intermediates 失效
标题翻译：制备烷氧基亚氨基乙酰胺化合物和中间体的方法
公开(公告)号：US5650539A
公开(公告)日：1997-07-22
申请号：US563297
申请日：1995-11-28
申请人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Shoji Shinomoto , Masahiko Nagai
发明人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Shoji Shinomoto , Masahiko Nagai
IPC分类号： C07C249/12 , C07C251/48 , C07C255/64 , H04L12/56 , C07C231/02
CPC分类号： C07C255/64 , C07C249/12 , C07C251/48
摘要： A compound of the formula [I] ##STR1## wherein X is hydrogen, lower alkyl, lower alkoxy or halogen; R is lower alkyl; and .about. is any configuration of E-isomer, Z-isomer or a mixture thereof is produced by reacting a compound of the formula ##STR2## wherein X and .about. are defined above, W is --CN or --COOR; and R is a lower alkyl, with methylamine in the presence of methanol. The compound [I] is useful for an agricultural fungicide. An intermediate used for producing the compound [I] is also disclosed.
摘要翻译：式I化合物其中X是氢，低级烷基，低级烷氧基或卤素; R为低级烷基; 并且差异是E-异构体，Z-异构体或其混合物的任何构型是通过使下式定义的式（II）化合物与其中X和DIFFERENCE的定义相同，W是-CN或-COOR; 在甲醇存在下，R为低级烷基，甲胺。化合物[I]可用于农药杀菌剂。还公开了用于制备化合物[I]的中间体。

4. 发明授权

US5627284A Process for producing (E)-alkoxyimino or hydroxyiminoacetamide compounds and intermediates therefor 失效
标题翻译：（E） - 烷氧基亚氨基或羟基亚氨基乙酰胺化合物及其中间体的制备方法
公开(公告)号：US5627284A
公开(公告)日：1997-05-06
申请号：US433931
申请日：1995-05-02
申请人： Akira Takase , Hiroyuki Kai , Moriyasu Masui , Kuniyoshi Nishida
发明人： Akira Takase , Hiroyuki Kai , Moriyasu Masui , Kuniyoshi Nishida
IPC分类号： C07C41/16 , C07C43/225 , C07C249/06 , C07C249/12 , C07C255/37 , C07C255/38 , C07C255/64 , C07D213/64 , C07D213/62
CPC分类号： C07D213/64 , C07C249/06 , C07C249/12 , C07C255/37 , C07C255/38 , C07C255/64 , C07C41/16
摘要： The present invention relates to a process for producing (E)-alkoxyiminoacetamide compounds useful as agricultural fungicides and a process for producing (E)-hydroxyiminoacetamide compounds useful as intermediates for producing them. The present invention also relates to an industrial process for producing (E)-methoxyiminoacetamide compounds useful as agricultural fungicides. This process is advantageous in terms of the cost, safety and the like.
摘要翻译：本发明涉及可用作农业杀真菌剂的（E） - 烷氧基亚氨基乙酰胺化合物的制备方法和用于生产（E） - 羟基亚氨基乙酰胺化合物的方法。本发明还涉及用于生产用作农业杀真菌剂的（E） - 甲氧基亚氨基乙酰胺化合物的工业方法。该方法在成本，安全性等方面是有利的。

5. 发明授权

US5693859A Process of producing intermediates for use in production of alkoxyiminoacetamides and intermediates to be used therein 失效
标题翻译：制备用于生产烷氧基亚氨基乙酰胺的中间体及其中使用的中间体的方法
公开(公告)号：US5693859A
公开(公告)日：1997-12-02
申请号：US578029
申请日：1995-12-26
申请人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Moriyasu Masui
发明人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Moriyasu Masui
IPC分类号： C07D215/12 , C07C51/58 , C07C59/84 , C07C59/88 , C07C59/90 , C07C227/02 , C07C229/42 , C07C231/02 , C07C233/56 , C07C235/72 , C07C235/78 , C07C237/20 , C07C249/08 , C07C319/12 , C07C319/20 , C07C323/62 , C07D215/20 , C07D215/36 , C07D239/26 , C07D239/34 , C07D239/38 , C07D239/42 , C07D261/08 , C07D261/10 , C07D261/12 , C07D261/14 , C07D263/32 , C07D263/36 , C07D263/46 , C07D263/48 , C07D263/56 , C07D263/58 , C07D277/62 , C07D303/38 , C07D413/04 , C07C233/05
CPC分类号： C07C59/84 , C07C231/02 , C07C249/08
摘要： There is disclosed a process of producing an .alpha.-ketamide as an intermediate for use in the production of various alkoxyiminoacetamide compounds which are useful as fungicides. Also disclosed is an intermediate to be used in this process.
摘要翻译：公开了一种制备用作生产可用作杀真菌剂的各种烷氧基亚氨基乙酰胺化合物的中间体的α-甲酰胺的方法。还公开了在该方法中使用的中间体。

6. 发明授权

US5488159A Process for producing methoxyiminoacetamide compounds and intermediates 失效
标题翻译：制备甲氧基亚氨基乙酰胺化合物和中间体的方法
公开(公告)号：US5488159A
公开(公告)日：1996-01-30
申请号：US295458
申请日：1994-08-25
申请人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Shoji Shinomoto , Masahiko Nagai
发明人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Shoji Shinomoto , Masahiko Nagai
IPC分类号： C07C249/12 , C07C251/48 , C07C255/64 , C07C239/20
CPC分类号： C07C251/48 , C07C249/12 , C07C255/64
摘要： A compound of the formula [I]: ##STR1## wherein X is hydrogen, lower alkyl, lower alkoxy or halogen; .about. is any configuration of E-isomer, Z-isomer or a mixture thereof is produced by reacting a compound of the formula [II] ##STR2## wherein X and .about. are as defined above; W is --CN or --COOR; and R is a lower alkyl, with methylamine in the presence of methanol. The compound [I] is useful for an agricultural fungicide. An intermediate used for producing the compound [I] is also disclosed.
摘要翻译：式[I]的化合物：其中X是氢，低级烷基，低级烷氧基或卤素; 差异是E-异构体，Z-异构体或其混合物的任何构型是通过使式[II]化合物[II]化合物或其混合物与其中X和DIFFERENCE如上定义反应而制备的。 W是-CN或-COOR; 在甲醇存在下，R为低级烷基，甲胺。化合物[I]可用于农药杀菌剂。还公开了用于制备化合物[I]的中间体。

7. 发明授权

US5442063A Process for producing (E)-alkoxyimino or hydroxyimino-acetamide compounds and intermediates therefor 失效
标题翻译：（E） - 烷氧基亚氨基或羟基亚氨基 - 乙酰胺化合物及其中间体的制备方法
公开(公告)号：US5442063A
公开(公告)日：1995-08-15
申请号：US144425
申请日：1993-11-02
申请人： Akira Takase , Hiroyuki Kai , Moriyasu Masui , Kuniyoshi Nishida
发明人： Akira Takase , Hiroyuki Kai , Moriyasu Masui , Kuniyoshi Nishida
IPC分类号： C07C43/225 , A01N37/50 , C07C20060101 , C07C249/06 , C07C249/12 , C07C251/48 , C07C251/60 , C07C255/37 , C07C255/38 , C07C255/62 , C07C255/64 , C07C317/48 , C07C323/57 , C07C323/63 , C07D213/64 , C07D401/08 , C07F7/02
CPC分类号： C07C249/12 , C07C249/06 , C07C255/38 , C07C255/64 , C07C43/225
摘要： The present invention relates to a process for producing (E)-alkoxyiminoacetamide compounds useful as agricultural fungicides and a process for producing (E)-hydroxyiminoacetamide compounds useful as intermediates for producing them. The present invention also relates to an industrial process for producing (E)-methoxyiminoacetamide compounds useful as agricultural fungicides. This process is advantageous in terms of the cost, safety and the like.
摘要翻译：本发明涉及可用作农业杀真菌剂的（E） - 烷氧基亚氨基乙酰胺化合物的制备方法和用于生产（E） - 羟基亚氨基乙酰胺化合物的方法。本发明还涉及用于生产用作农业杀真菌剂的（E） - 甲氧基亚氨基乙酰胺化合物的工业方法。该方法在成本，安全性等方面是有利的。

8. 发明授权

US5387714A Process of producing intermediates for use in production of alkoxyiminoacetamides and intermediates to be used therein 失效
标题翻译：制备用于生产烷氧基亚氨基乙酰胺的中间体及其中使用的中间体的方法
公开(公告)号：US5387714A
公开(公告)日：1995-02-07
申请号：US953884
申请日：1992-09-30
申请人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Moriyasu Masui
发明人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Moriyasu Masui
IPC分类号： C07D215/12 , C07C51/58 , C07C59/84 , C07C59/88 , C07C59/90 , C07C227/02 , C07C229/42 , C07C231/02 , C07C233/56 , C07C235/72 , C07C235/78 , C07C237/20 , C07C249/08 , C07C319/12 , C07C319/20 , C07C323/62 , C07D215/20 , C07D215/36 , C07D239/26 , C07D239/34 , C07D239/38 , C07D239/42 , C07D261/08 , C07D261/10 , C07D261/12 , C07D261/14 , C07D263/32 , C07D263/36 , C07D263/46 , C07D263/48 , C07D263/56 , C07D263/58 , C07D277/62 , C07D303/38 , C07D413/04 , C07C55/38 , C07C59/21
CPC分类号： C07C59/84 , C07C231/02 , C07C249/08
摘要： There is disclosed a process of producing an .alpha.-ketamide as an intermediate for use in the production of various alkoxyiminoacetamide compounds which are useful as fungicides. Also disclosed is an intermediate to be used in this process.
摘要翻译：公开了一种制备用作生产可用作杀真菌剂的各种烷氧基亚氨基乙酰胺化合物的中间体的α-甲酰胺的方法。还公开了在该方法中使用的中间体。

9. 发明授权

US06268312B1 Oxime derivative and bactericide containing the same as active ingredient 失效
标题翻译：含有与活性成分相同的肟衍生物和杀菌剂
公开(公告)号：US06268312B1
公开(公告)日：2001-07-31
申请号：US09370255
申请日：1999-08-09
申请人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Tsuneo Iwakawa , Kazuo Ueda , Michio Masuko
发明人： Akira Takase , Hiroyuki Kai , Kuniyoshi Nishida , Tsuneo Iwakawa , Kazuo Ueda , Michio Masuko
IPC分类号： A01N4348
CPC分类号： C07D231/06 , A01N43/50 , C07D231/12 , C07D233/64 , C07D249/08 , C07D257/04 , C07D261/08 , C07D263/10 , C07D263/32 , C07D271/06 , C07D271/10 , C07D277/10 , C07D285/06
摘要： A compound represented by general formula (I) or a salt thereof, a process for producing the same, an intermediate for the production thereof, and a bactericide (fungicide) containing the same as the active ingredient wherein R1 represent optionally substituted aryl, optionally substituted heterocycle, mono- or di-substituted methyleneamino, optionally substituted (substituted imino)methyl, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, substituted carbonyl or substituted sulfonyl; R2 represents alkyl, alkenyl, alkynyl or cycloalkyl; R3 represents optionally substituted heterocycle; R4 represents hydrogen, alkyl, alkoxy, halogen, nitro, cyano or haloalkyl; M represents oxygen, S(O)i (i being 0, 1 or 2), NR16 (R16 being hydrogen, alkyl or acyl) or a single bond; n represents 0 or 1, provided n represent 1 when R3 represents imidazol-1-yl or 1H-1,2,4-triazol-1-yl; and the symbol˜represents the E form, Z form or a mixture thereof.
摘要翻译：由通式（I）表示的化合物或其盐，其制备方法，其制备中间体和含有该活性成分的杀菌剂（杀真菌剂），其中R 1表示任选取代的芳基，任选取代的取代的亚氨基甲基，任选取代的烷基，任选取代的烯基，任选取代的炔基，取代的羰基或取代的磺酰基; R2代表烷基，烯基，炔基或环烷基; R3表示任选取代的杂环; R4代表氢，烷基，烷氧基，卤素，硝基，氰基或卤代烷基; M表示氧，S（O）i（i为0,1或2），NR 16（R 16为氢，烷基或酰基）或单键; 当R 3表示咪唑-1-基或1H-1,2,4-三唑-1-基时，n表示0或1，条件是n表示1。符号〜表示E形式，Z形式或其混合物。

10. 发明授权

US06251949B1 Oxime derivatives, hydrazone derivatives and use thereof 失效
标题翻译：肟衍生物，腙衍生物及其用途
公开(公告)号：US06251949B1
公开(公告)日：2001-06-26
申请号：US09457672
申请日：1999-12-09
申请人： Moriyasu Masui , Norihiko Tanimoto , Kuniyoshi Nishida
发明人： Moriyasu Masui , Norihiko Tanimoto , Kuniyoshi Nishida
IPC分类号： A61K3115
CPC分类号： C07D213/30 , A01N37/50 , A01N41/06 , A01N41/10 , A01N43/40 , A01N43/46 , A01N43/80 , A01N47/16 , C07C251/36 , C07C251/48 , C07C251/52 , C07C251/54 , C07C251/74 , C07C259/06 , C07D207/12 , C07D211/42 , C07D211/46 , C07D211/58 , C07D211/72 , C07D243/08 , C07D261/02 , C07D295/185 , C07D295/26 , C07D333/16 , C07D401/12
摘要： Compounds having fungicidal activities and represented by general formula (I) and salts and hydrates thereof wherein R1 represents an optionally substituted aryl, an optionally substituted alkyl or the like; R2 represents an optionally substituted alkyl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted aryl, an optionally substituted heterocyclic group or the like; R3 represents an optionally substituted alkyl, an optionally substituted alkenyl, an optionally substituted alkynyl, an optionally substituted arylsulfonyl, an optionally substituted heterocyclic group or the like; R4 and R5, which may be the same or different, represent each a hydrogen atom, an optionally substituted alkyl, or an optionally substituted alkoxy, or R4 and R5 may form together with the adjacent nitrogen atom an optionally substituted monocycle or polycycle; X and Y, which may be the same or different, represents each an oxygen atom or NR6 wherein R6 represents a hydrogen atom, an optionally substituted alkyl, an optionally substituted aryl, an optionally substituted alkanoyl, or an optionally substituted aroyl; Z represents an oxygen atom or a sulfur atom; and a wavy line (˜) represents the configuration of an E isomer, a Z isomer, or a mixture thereof.
摘要翻译：具有杀真菌活性并由通式（I）表示的化合物及其盐和水合物，其中R 1表示任选取代的芳基，任选取代的烷基等; R 2表示任选取代的烷基，任选取代的烯基，任选取代的炔基，任选取代的芳基，任选取代的杂环基等; R 3表示任选取代的烷基，任选取代的烯基，任选取代的炔基，任选取代的芳基磺酰基，任选取代的杂环基团等; R 4和R 5可以相同或不同，表示氢原子，任选取代的烷基或任选取代的烷氧基，或者R 4和R 5可以与相邻的氮原子一起形成任选取代的单环或多环; X和Y可以相同或不同，表示每个氧原子或NR 6，其中R 6表示氢原子，任选取代的烷基，任选取代的芳基，任选取代的烷酰基或任选取代的芳酰基; Z表示氧原子或硫原子; 波浪线（〜）表示E异构体，Z异构体或其混合物的构型。

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