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1. 发明申请

US20060293318A1 Stereospecifically substituted benzo[1,3]dioxolyl derivatives 审中-公开
标题翻译：立体选择性取代的苯并[1,3]二氧杂环戊烯基衍生物
公开(公告)号：US20060293318A1
公开(公告)日：2006-12-28
申请号：US11452026
申请日：2006-06-13
申请人： Beat Frei , Jean-Marc Plancher , Stephan Roever , Daniel Zimmerli
发明人： Beat Frei , Jean-Marc Plancher , Stephan Roever , Daniel Zimmerli
IPC分类号： A61K31/5377 , C07D413/02
CPC分类号： C07D317/46
摘要： The present invention relates to compounds of formula (I) wherein R1 and R2 are as defined in the description and claims, and pharmaceutically acceptable salts thereof, for use as therapeutically active substances. The compounds are useful for the treatment and/or prophylaxis of diseases which are associated with the modulation of CB1 receptors.
摘要翻译：本发明涉及式（I）化合物，其中R 1和R 2 2如说明书和权利要求及其药学上可接受的盐所定义，用于治疗活性物质。该化合物可用于治疗和/或预防与调节CB1受体相关的疾病。

2. 发明授权

US5520864A Controlled mixture formation 失效
标题翻译：控制混合物形成
公开(公告)号：US5520864A
公开(公告)日：1996-05-28
申请号：US387807
申请日：1995-02-21
申请人： Beat Frei
发明人： Beat Frei
IPC分类号： F02B1/04 , F02B75/02 , F02D35/00 , F02M17/16 , F02M69/06
CPC分类号： F02M17/16 , F02D35/0046 , F02M69/06 , F02B1/04 , F02B2075/027
摘要： Controlled mixture formation. This invention pertains to the generation of homogenous mixtures having a freely selectable composition and is produced by using a rotary distribution cup driven by its own motor, with metered quantities of fuel being supplied to the pre-chamber of a rotary fuel distribution cup via a feed pipe extending through a metering valve in such a manner that the composition of the mixture produced in each case can be adjusted, irrespective of the amount of the air, over the entire operating range of the internal combustion engine, with the fuel being radially distributed by centrifugal force, very finely divided and mixed with air in a mixing chamber wherein the quantity and composition of the mixture are adjusted by means of the metering valve in conjunction with a control valve in such a way that the production of the mixture and its conveyance take place at approximately ambient pressure, with a motor performance graph establishing the optimum setting for the metering and regulating valves for mixture production at approximately ambient pressure while improving fuel consumption and the exhaust gas quality, with the invention, in connection with the noted control system being especially suitable for the best possible operation of four-stroke engines with lean fuel mixtures at lambda values of at least 1.5.
摘要翻译： PCT No.PCT / EP92 / 01922 Sec。 371日期1995年2月21日 102（e）日期1995年2月21日PCT提交1992年8月21日PCT公布。出版物WO94 / 0481200 日期1994年3月3日。控制混合物形成。本发明涉及产生具有可自由选择的组合物的均质混合物，并且通过使用由其自身的电动机驱动的旋转分配杯来制造，其中计量的燃料经由进料供应到旋转燃料分配杯的预制室管道延伸通过计量阀，使得在各种情况下生产的混合物的组成可以在内燃机的整个工作范围内调节，而不管空气的量，而燃料由径向分布在内燃机的整个工作范围内离心力，非常精细地分配并与混合室中的空气混合，其中混合物的数量和组成通过计量阀与控制阀一起调节，使得混合物的产生及其输送在大约环境压力下，电机性能图确定了计量和调节阀的最佳设置在大气环境压力下进行混合生产，同时改善燃料消耗和废气质量，本发明结合所提出的控制系统特别适用于具有稀释燃料混合物的四冲程发动机在λ值为至少1.5。

3. 发明申请

US20100056513A1 STEREOSPECIFICALLY SUBSTITUTED BENZO[1,3]DIOXOLYL DERIVATIVES 审中-公开
标题翻译：立体取代苯并[1,3]二氧化物衍生物
公开(公告)号：US20100056513A1
公开(公告)日：2010-03-04
申请号：US12614461
申请日：2009-11-09
申请人： Beat Frei , Jean-Marc Plancher , Stephan Roever , Daniel Zimmerli
发明人： Beat Frei , Jean-Marc Plancher , Stephan Roever , Daniel Zimmerli
IPC分类号： A61K31/5377 , C07D413/10
CPC分类号： C07D317/46
摘要： The present invention relates to compounds of formula (I) wherein R1 and R2 are as defined in the description and claims, and pharmaceutically acceptable salts thereof, for use as therapeutically active substances. The compounds are useful for the treatment and/or prophylaxis of diseases which are associated with the modulation of CB1 receptors.
摘要翻译：本发明涉及式（I）化合物，其中R 1和R 2如说明书和权利要求中所定义，及其药学上可接受的盐，用作治疗活性物质。该化合物可用于治疗和/或预防与调节CB1受体相关的疾病。

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