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1. 发明授权

US08242161B2 Topical formulations comprising 1-N-arylpyrazole derivatives and amitraz 有权
标题翻译：包含1-N-芳基吡唑衍生物和氨基拉唑的局部制剂
公开(公告)号：US08242161B2
公开(公告)日：2012-08-14
申请号：US12420325
申请日：2009-04-08
申请人： Albert Boeckh , Luiz Gustavo Cramer , Mark D. Soll
发明人： Albert Boeckh , Luiz Gustavo Cramer , Mark D. Soll
IPC分类号： A01N43/56
CPC分类号： A01N43/56 , A01N47/02 , A01N2300/00 , A01N37/52
摘要： The present invention provides for, inter alia, novel topical formulations comprising at least one 1-N-arypyrazole derivative and amitraz and to methods for treating, controlling, or preventing parasite infestations on mammals or birds The inventive formulations include spot-on, pour-on or spray formulations and may include a further ectoparasiticide, such as an IGR compound, an avermectin or milbemycin derivative, or a pyrethroid insecticides, and anthelmintics, such as benzimidazoles and imidazothiazoles. The inventive formulation provides a larger duration of parasite control at a faster rate of control. The inventive formula remains effective up to three months from the first application. Moreover, the inventive formulations prevent tick attachment to the animal, thereby providing protection against tick borne diseases. The ectoparasites which may be controlled, treated or prevented by the present invention includes ticks, fleas, mites, mange, lice, mosquitoes, flies and cattle grubs.
摘要翻译：本发明特别提供了包含至少一种1-N-阿吡唑衍生物和氨喋啶的新型局部制剂，以及用于治疗，控制或预防哺乳动物或鸟类寄生虫侵袭的方法。本发明的制剂包括点状，可以包括另外的外寄生物杀虫剂，例如IGR化合物，除虫菌素或米尔倍霉素衍生物，拟除虫菊酯杀虫剂，以及驱肠虫药如苯并咪唑和咪唑并噻唑。本发明的配方以更快的控制速率提供更大的寄生虫控制持续时间。本发明的公式从第一次申请至多三个月仍然有效。此外，本发明的制剂防止蜱附着于动物，从而提供防止蜱携带疾病的保护。本发明可以控制，治疗或预防的外寄生虫包括蜱，跳蚤，螨虫，虱子，虱子，蚊子，苍蝇和牛。。。

2. 发明申请

US20090192207A1 Topical Formulations Comprising 1-N-Arylpyrazole Derivatives and Amitraz 有权
标题翻译：包含1-N-Arylpyrazole衍生物和Amitraz的局部制剂
公开(公告)号：US20090192207A1
公开(公告)日：2009-07-30
申请号：US12420325
申请日：2009-04-08
申请人： Albert Boeckh , Luiz Gustavo Cramer , Mark D. Soll
发明人： Albert Boeckh , Luiz Gustavo Cramer , Mark D. Soll
IPC分类号： A01N43/56
CPC分类号： A01N43/56 , A01N47/02 , A01N2300/00 , A01N37/52
摘要： The present invention provides for, inter alia, novel topical formulations comprising at least one 1-N-arypyrazole derivative and amitraz and to methods for treating, controlling, or preventing parasite infestations on mammals or birds The inventive formulations include spot-on, pour-on or spray formulations and may include a further ectoparasiticide, such as an IGR compound, an avermectin or milbemycin derivative, or a pyrethroid insecticides, and anthelmintics, such as benzimidazoles and imidazothiazoles. The inventive formulation provides a larger duration of parasite control at a faster rate of control. The inventive formula remains effective up to three months from the first application. Moreover, the inventive formulations prevent tick attachment to the animal, thereby providing protection against tick borne diseases. The ectoparasites which may be controlled, treated or prevented by the present invention includes ticks, fleas, mites, mange, lice, mosquitoes, flies and cattle grubs.
摘要翻译：本发明特别提供了包含至少一种1-N-阿吡唑衍生物和氨喋啶的新型局部制剂，以及用于治疗，控制或预防哺乳动物或鸟类寄生虫侵袭的方法。本发明的制剂包括点状，可以包括另外的外寄生物杀虫剂，例如IGR化合物，除虫菌素或米尔倍霉素衍生物，拟除虫菊酯杀虫剂，以及驱肠虫药如苯并咪唑和咪唑并噻唑。本发明的配方以更快的控制速率提供更大的寄生虫控制持续时间。本发明的公式从第一次申请至多三个月仍然有效。此外，本发明的制剂防止蜱附着于动物，从而提供防止蜱携带疾病的保护。本发明可以控制，治疗或预防的外寄生虫包括蜱，跳蚤，螨虫，虱子，虱子，蚊子，苍蝇和牛。。。

3. 发明申请

US20080160067A1 Novel soft chewable, tablet, and long-acting injectable veterinary antibiotic formulations 审中-公开
标题翻译：新型软咀嚼片，片剂和长效注射用兽药抗生素配方
公开(公告)号：US20080160067A1
公开(公告)日：2008-07-03
申请号：US11899282
申请日：2007-09-05
申请人： Albert Boeckh , Mark D. Soll , Monica Tejwani-Motwani , Robert P. Waranis , Fangjun Wu
发明人： Albert Boeckh , Mark D. Soll , Monica Tejwani-Motwani , Robert P. Waranis , Fangjun Wu
IPC分类号： A61K9/68 , A61K31/40
CPC分类号： A61K9/0056 , A61K9/0019 , A61K9/2013 , A61K9/2018 , A61K47/10
摘要： This document relates to formulations for combating bacterial infections in animals which provide for improved long-acting oral and injectable formulations for systemic delivery of antibiotics, which are designed to achieve high bioavailability.
摘要翻译：本文件涉及用于对抗动物细菌感染的制剂，其提供改进的用于系统递送抗生素的长效口服和可注射制剂，其被设计为实现高生物利用度。

4. 发明申请

US20080003282A1 Antiparasitical agents and methods for treating, preventing and controlling external parasites in animals 审中-公开
标题翻译：抗真菌药物和治疗，预防和控制动物外部寄生虫的方法
公开(公告)号：US20080003282A1
公开(公告)日：2008-01-03
申请号：US11580731
申请日：2006-10-13
申请人： Mark Soll , Albert Boeckh , Krishan Kumar , Natalya Shub
发明人： Mark Soll , Albert Boeckh , Krishan Kumar , Natalya Shub
IPC分类号： A01N25/34 , A01N43/56 , A01P15/00 , C07D231/02
CPC分类号： C07D231/44 , A01N43/56 , A01N47/02 , A23K20/137 , A23K50/40
摘要： This invention provides for antiparasitical agents and methods for treating, preventing and controlling external parasites in animals.
摘要翻译：本发明提供了用于治疗，预防和控制动物外部寄生虫的抗惊厥剂和方法。

5. 发明申请

US20060046988A1 Methoprene formulations for the control of tick infestations 审中-公开
标题翻译：用于控制蜱虫侵袭的甲基杀螨剂配方
公开(公告)号：US20060046988A1
公开(公告)日：2006-03-02
申请号：US10929176
申请日：2004-08-30
申请人： Albert Boeckh , Mark Soll , Luiz Cramer
发明人： Albert Boeckh , Mark Soll , Luiz Cramer
IPC分类号： A01N43/40 , A01N53/00 , A01N43/58 , A01N43/60
CPC分类号： A01N49/00 , A01N2300/00
摘要： The present invention relates to a composition and process, in particular for controlling ticks on animals, characterized in that the composition includes, on the one hand, at least one compound of IGR (insect growth regulator) type, in doses and proportions which are parasiticidally effective on ticks, in a fluid vehicle which is acceptable for the animal and convenient for local application to the skin, preferably localized over a small surface area.
摘要翻译：本发明涉及一种组合物和方法，特别是用于控制动物的蜱，其特征在于该组合物一方面包含至少一种IGR（昆虫生长调节剂）类型的化合物，其剂量和比例为寄生虫螨在蜱上有效，在动物中可接受的流体媒介物，并且方便局部施用于皮肤，优选地定位在小的表面积上。

6. 发明申请

US20050234119A1 Antiparasitical agents and methods for treating, preventing and controlling external parasites in animals 审中-公开
标题翻译：抗真菌药物和治疗，预防和控制动物外部寄生虫的方法
公开(公告)号：US20050234119A1
公开(公告)日：2005-10-20
申请号：US10826105
申请日：2004-04-16
申请人： Mark Soll , Albert Boeckh , Krishan Kumar , Natalya Shub
发明人： Mark Soll , Albert Boeckh , Krishan Kumar , Natalya Shub
IPC分类号： A01N43/56 , A01N47/02 , A61K31/415 , A61K31/416
CPC分类号： A61K31/415 , A01N43/56 , A01N47/02 , A61K31/416 , A01N25/02 , A01N25/00 , A01N2300/00
摘要： This invention provides for antiparasitical agents and methods for treating, preventing and controlling external parasites in animals.
摘要翻译：本发明提供了用于治疗，预防和控制动物外部寄生虫的抗惊厥剂和方法。

7. 发明申请

US20070293446A1 Compositions comprising C-13 alkoxyether macrolide compounds and phenylpyrazole compounds 有权
标题翻译：包含C-13烷氧基醚大环内酯化合物和苯基吡唑化合物的组合物
公开(公告)号：US20070293446A1
公开(公告)日：2007-12-20
申请号：US11799796
申请日：2007-05-03
申请人： Mark Soll , Albert Boeckh , Natalya Shub
发明人： Mark Soll , Albert Boeckh , Natalya Shub
IPC分类号： A61K31/70 , A61P33/00 , C07H17/04
CPC分类号： A61K45/06 , A01N43/56 , A01N47/02 , A61K31/415 , A61K31/4439 , A61K31/70 , C07D493/22 , A01N43/90 , A01N2300/00 , A61K2300/00
摘要： Provided is a novel ivermectin derivative and compositions for the treatment or prophylaxis of parasite infestations in mammals or birds which comprise: (A) a pharmaceutically effective amount of a 1-N-phenylpyrazole compound; (B) a pharmaceutically effective amount of an ivermectin derivative of formula (II) wherein: R14 represents —(CH2)sO—Z wherein, s is 1 or 2; Y represents —CH(OR15)—, —C(═O)— or —C(═NOR15); R15 represents hydrogen, alkyl or phenyl; and R16 represents —CH3 or —CH2CH3; Z is alkyl, alkenyl, alkynyl, acyl, alkylalkoxy, aryl, alkanoyloxy, alkoxycarbonyl, alkenoyl, alkynoyl, or aroyl.
摘要翻译：提供了一种新颖的伊维菌素衍生物和用于治疗或预防哺乳动物或鸟类中寄生虫侵袭的组合物，其包含：（A）药学有效量的1-N-苯基吡唑化合物; （B）药学有效量的式（II）的伊维菌素衍生物，其中：R 14表示 - （CH 2）n OZ其中 s为1或2; Y表示-CH（OR 15） - ， - C（-O） - 或-C（-NOR 15）。 R 15表示氢，烷基或苯基; 并且R 16表示-CH 3或-CH 2 CH 3; Z是烷基，烯基，炔基，酰基，烷基烷氧基，芳基，烷酰氧基，烷氧基羰基，烯酰基，炔酰基或芳酰基。

8. 发明授权

US07262214B2 1-N-arylpyrazole derivatives in prevention of arthropod-borne and mosquito-borne diseases 有权
标题翻译： 1-N-芳基吡唑衍生物预防节肢动物和蚊子传播疾病
公开(公告)号：US07262214B2
公开(公告)日：2007-08-28
申请号：US10374627
申请日：2003-02-26
申请人： Mark Soll , Albert Boeckh
发明人： Mark Soll , Albert Boeckh
IPC分类号： A01N43/56
CPC分类号： A01N25/002 , A61K31/4439 , A01N43/56
摘要： This invention provides for a method for preventing or interrupting the transmission of anthropod and mosquito-borne diseases from a first actual or putative amplifying or incipient host to a second actual or putative amplifying or incipient host, which comprises applying or administering a formulation comprising an effective amount of at least one 1-N-arylpyrazole to said first actual or putative amplifying host and/or actual or putative amplifying or incipient host. This invention also provides for a method of using a bait placed in a bird station, the bait comprises an affective amount of at least one 1-N-arylpyrazole either alone or in combination with an antiparasitic, antihelmintic, or insecticidal agents. This invention also provides for an apparatus for delivering an effective amount of a formulation according to the present invention to a bird or animal in an environment where it resides.
摘要翻译：本发明提供了一种预防或阻止从第一实际或推定的放大或初始宿主向第二实际或推定的放大或初始宿主传播节肢动物和蚊子传播疾病的方法，其包括施用或施用包含有效至少一个1-N-芳基吡唑的量与所述第一实际或推定的放大宿主和/或实际或推定的放大或初始宿主。本发明还提供了使用放置在鸟站中的诱饵的方法，该诱饵单独包含至少一种1-N-芳基吡唑的情感量，或与抗寄生虫，抗耳蜗或杀虫剂组合。本发明还提供了一种用于将有效量的根据本发明的制剂递送到其所在环境中的鸟或动物的装置。

9. 发明授权

US06998131B2 Spot-on formulations for combating parasites 有权
标题翻译：用于防治寄生虫的现货配方
公开(公告)号：US06998131B2
公开(公告)日：2006-02-14
申请号：US10279356
申请日：2002-10-24
申请人： Mark D. Soll , Albert Boeckh
发明人： Mark D. Soll , Albert Boeckh
IPC分类号： A01N25/32
CPC分类号： A01N43/56 , A01N47/02 , A61K31/70 , A01N2300/00 , A61K2300/00
摘要： In particular this invention provides for spot-on compositions for the treatment or prophylaxis of parasite infestations in mammals or birds which comprise: (1) a composition comprising (A) an effective amount of a 1-phenylpyrazole derivative; and (B) an effective amount of emamectin; (2) an acceptable liquid carrier vehicle; and (3) optionally, a crystallization inhibitor. The invention also provides for a method of treating parasitic infestations or for the prophylaxis of parasite infestations in mammals or birds which comprises topically applying to said mammal treating parasitic infestations or for the prophylaxis of parasite infestations in mammals or birds which comprises topically applying to said mammal or bird an effective amount of a composition according to the present invention.
摘要翻译：特别地，本发明提供了用于治疗或预防哺乳动物或鸟类中的寄生虫感染的斑点组合物，其包括

10. 发明申请

US20050192319A1 Spot-on formulations for combating parasites 审中-公开
标题翻译：用于防治寄生虫的现货配方
公开(公告)号：US20050192319A1
公开(公告)日：2005-09-01
申请号：US11055234
申请日：2005-05-16
申请人： Albert Boeckh , Mark Soll , Philippe Jeannin
发明人： Albert Boeckh , Mark Soll , Philippe Jeannin
IPC分类号： A01N43/56 , A01N47/02 , A61K31/4439 , A61K31/415 , A61K31/4178
CPC分类号： A61K9/0017 , A01N43/56 , A01N47/02 , A61K31/415 , A61K31/70 , A61K45/06 , A01N2300/00 , A61K2300/00
摘要： In particular this invention provides for spot-on compositions for the treatment or prophylaxis of parasite infestations in mammals or birds which comprise: (1) a composition comprising (A) an effective amount of a 1-phenylpyrazole derivative; and (B) an effective amount of emamectin, latidectin or lepimectin; (2) an acceptable liquid carrier vehicle; and (3) optionally, a crystallization inhibitor. The invention also provides for a method of treating parasitic infestations or for the prophylaxis of parasite infestations in mammals or birds which comprises topically applying to said mammal treating parasitic infestations or for the prophylaxis of parasite infestations in mammals or birds which comprises topically applying to said mammal or bird an effective amount of a composition according to the present invention.
摘要翻译：特别地，本发明提供了用于治疗或预防哺乳动物或鸟类寄生虫侵袭的斑点组合物，其包括：（1）包含（A）有效量的1-苯基吡唑衍生物的组合物; 和（B）有效量的阿维菌素，赖氨酸或莱匹维林; （2）可接受的液体载体载体; 和（3）任选的结晶抑制剂。本发明还提供了一种治疗寄生虫侵袭或预防哺乳动物或鸟类中的寄生虫侵袭的方法，其包括局部施用于所述哺乳动物治疗寄生虫侵袭或预防哺乳动物或鸟类中的寄生虫侵袭，其包括局部施用于所述哺乳动物或鸟类有效量的根据本发明的组合物。

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