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41. 发明授权

US4399139A 5,6-Dihydro-11-alkylene-morphanthridin-6-ones, their pharmaceutical compositions and method of use 失效
标题翻译： 5,6-二氢-11-亚烷基 - 异佛尔酮-6-酮，其药物组合物和使用方法
公开(公告)号：US4399139A
公开(公告)日：1983-08-16
申请号：US359936
申请日：1982-03-19
申请人： Gerd Steiner , Ludwig Friedrich , Dieter Lenke
发明人： Gerd Steiner , Ludwig Friedrich , Dieter Lenke
IPC分类号： A61K31/00 , A61K31/55 , A61P1/04 , C07D223/20 , C07F9/59 , C07D403/06
CPC分类号： C07F9/591 , C07D223/20 , Y10S514/926
摘要： Novel 5,6-dihydro-11-alkylene-morphanthridin-6-ones of the formula ##STR1## where R.sup.1, R.sup.2, R.sup.3 and R.sup.4 have the meanings given in the description, their preparation and their use.The novel compounds are particularly useful in the treatment of gastric and duodenal ulcers.
摘要翻译：其中R 1，R 2，R 3和R 4具有本说明书中给出的含义及其制备方法及其用途的新颖的5,6-二氢-11-亚烷基 - 异恶唑-6-酮。新型化合物特别可用于治疗胃和十二指肠溃疡。

42. 发明授权

US08268815B2 Pyrimidine compounds and use thereof 失效
标题翻译：嘧啶化合物及其用途
公开(公告)号：US08268815B2
公开(公告)日：2012-09-18
申请号：US12842776
申请日：2010-07-23
申请人： Hervè Geneste , Andreas Haupt , Wilfried Braje , Wilfried Lubisch , Gerd Steiner
发明人： Hervè Geneste , Andreas Haupt , Wilfried Braje , Wilfried Lubisch , Gerd Steiner
IPC分类号： C07D401/12 , C07D413/12 , C07D417/12 , A61K31/506 , A61P25/36
CPC分类号： C07D417/12 , C07D401/12 , C07D413/12
摘要： The invention relates to compounds of formula (I) and the use of these compounds.
摘要翻译：本发明涉及式（I）化合物和这些化合物的用途。

43. 发明授权

US07491729B2 3-Substituted 3,4-dihydro-thieno[2,3-d]pyrimidin-4-one derivatives, production and use thereof 有权
标题翻译： 3-取代的3,4-二氢 - 噻吩并[2,3-d]嘧啶-4-酮衍生物，的制备和用途
公开(公告)号：US07491729B2
公开(公告)日：2009-02-17
申请号：US10539708
申请日：2003-12-17
申请人： Margaretha Bakker , Wilfried Hornberger , Andreas Kling , Udo Lange , Helmut Mack , Achim Moeller , Reinhold Mueller , Kurt Schellhaas , Martin Schmidt , Gerd Steiner , Karsten Wicke
发明人： Margaretha Bakker , Wilfried Hornberger , Andreas Kling , Udo Lange , Helmut Mack , Achim Moeller , Reinhold Mueller , Kurt Schellhaas , Martin Schmidt , Gerd Steiner , Karsten Wicke
IPC分类号： A01N43/54 , A61K31/505 , C07D239/00 , C07D471/00 , C07D487/00 , C07D491/00
CPC分类号： C07D495/14
摘要： 3-Substituted 3,4-dihydrothieno[2,3-d]pyrimidin-4-one derivatives, production and use thereof. The invention relates to 3,4-dihydrothieno[2,3-d]pyrimidin-4-one derivatives which are substituted in position 3 by 5-membered heteroaryl which may be fused to an aryl or heteroaryl radical, where the heteroaryl and, if appropriate, the fused aryl or heteroaryl radical may have 1, 2 or 3 substituents selected independently of one another from C1-5-alkyl, C1-5-alkoxy, C1-5-alkylthio, halogen, CN, halo-C1-5-alkyl, halo-C1-5-alkoxy, hydroxy, —NH2, —N(R6)2, —NH(R6), aryl, aryloxy, aralkyl, aralkyloxy and heteroaryl, where the substituents aryl, aryloxy, aralkyl, aralkyloxy and heteroaryl may have 1, 2 or 3 substituents selected independently of one another from C1-5-alkyl, C1-5-alkoxy, C1-5-alkylthio, halogen, CN, halo-C1-5-alkyl, halo-C1-5-alkoxy, hydroxy, —NH2, —N(R6)2 and —NH(R6). The preparation and use of these derivatives, especially for therapeutic purposes, e.g. for the treatment of depressions, are likewise described.
摘要翻译： 3-取代的3,4-二氢噻吩并[2,3-d]嘧啶-4-酮衍生物，的制备和用途。本发明涉及在3位被5位杂芳基取代的3,4-二氢噻吩并[2,3-d]嘧啶-4-酮衍生物，其可以与芳基或杂芳基稠合，其中杂芳基和稠合的芳基或杂芳基可以具有1,2或3个彼此独立地选自C 1-5 - 烷基，C 1-5 - 烷氧基，C 1-5 - 烷硫基，卤素，CN，卤代-C 1-5 - 烷基，卤代C 1-5 - 烷氧基，羟基，-NH 2，-N（R 6）2，-NH（R 6），芳基，芳氧基，芳烷基，芳烷氧基和杂芳基，其中芳基，芳氧基，芳烷基，芳烷氧基和杂芳基可以具有1,2或3个彼此独立地选自C 1-5 - 烷基，C 1-5 - 烷氧基，C 1-5 - 烷硫基，卤素，CN，卤代C 1-5 - 烷基，卤代-C 1-5 - 烷氧基，羟基，-NH 2，-N（R 6）2和-NH（R 6）。这些衍生物的制备和使用，特别是用于治疗目的，例如为了处理凹陷，同样地描述。

44. 发明申请

US20060166984A1 Amino substituted benzo(hetero)cyclic derivatives 审中-公开
公开(公告)号：US20060166984A1
公开(公告)日：2006-07-27
申请号：US10547914
申请日：2004-02-20
申请人： Gerd Steiner , Thomas Schmidt , Markus Kordes , Wolfgang Von Deyn , Michael Hofmann , Ernst Baumann , Michael Puhl , Gain Heffernan , Deborah Culbertson , Michael Treacy
发明人： Gerd Steiner , Thomas Schmidt , Markus Kordes , Wolfgang Von Deyn , Michael Hofmann , Ernst Baumann , Michael Puhl , Gain Heffernan , Deborah Culbertson , Michael Treacy
IPC分类号： A01N43/84
CPC分类号： A01N43/72 , A01N43/60
摘要： Use of compounds Formula (I), A=a 5- to 7-membered ring which may contain 1-3 heteroatoms and which may be saturated or partially or completely unsaturated; R1═OH, SH, NH2, CN, NO2, halogen, C1-C6-alkyl, C1-C6-haloalkyl; C1-C6-alkoxy, C1-C6-haloalkoxy, C1-C6-alkylthio, C1-C6-haloalkylthio, C2-C6-alkenyl, C2-C6alkenyloxy, C2-C6-alkenylthio, C2-C6-alkynyl, C2-C6-alkynyloxy, C2-C6-alkynylthio, C1-C6-alkylsulfonyl, C1-C6-alkylsulfoxyl, C2-C6-alkenylsulfonyl, C2-C6-alkylsulfoxyl, C1-C6-alkylcarbonyl, C1-C6-alkoxycarbonyl, C1-C6-aklylcarbonyloxy; R2═C1-C6-alkyl or a mono- or bicyclic 5- to 10-membered aromatic ringsystem which may contain 1 to 4 heteroatoms and which is either bonded directly or through an O, S, C1-C6-alkylene or C1-C6-alkyleneoxy linkage to A or fused to A and which may be substituted; R3, R4═H, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkyl-amino, C1-C6-alkoxy, C3-C6-cycloalkyl, or R3 and R4 together with the nitrogen atom to which they are attached form a saturated or partially saturated mono- or bicyclic 5- to 10-membered ring system containing 1 to 3 heteroatoms or a 5-membered hetaryl containing 1 to 4 nitrogen atoms, wherein the carbon and/or nitrogen atoms in the ring systems may be substituted or phenyl or benzyl which may be substituted; or R3 and R4 together form the chains —(CH2)2N+(O—)(CH2)2— or —(CH2)3N+(O−)(CH2)2—; m=0 to 4; n is 0 to 4; and the enantiomers, diastereomers, cis/trans isomers or salts thereof for combatting insects, arachnids or nematodes, methods for the control of these pests and of protecting growing plants attack or infestation by these pests by applying a pesticidally effective amount of a compound of formula (I), processes for preparing them, and compositions comprising them.

45. 发明申请

US20060014805A1 Pesticidal fluoroalkene derivatives 审中-公开
公开(公告)号：US20060014805A1
公开(公告)日：2006-01-19
申请号：US10523325
申请日：2003-07-30
申请人： Markus Kordes , Wolfgang Deyn , Thomas Schmidt , Gerd Steiner , David Kuhn , Yulin Hu , Henry Cotter , Deborah Culbertson , David Kuhn , Yulin Hu , Henry Cotter , Deborah Culbertson
发明人： Markus Kordes , Wolfgang Deyn , Thomas Schmidt , Gerd Steiner , David Kuhn , Yulin Hu , Henry Cotter , Deborah Culbertson , David Kuhn , Yulin Hu , Henry Cotter , Deborah Culbertson
IPC分类号： A01N43/40 , A01N43/78 , A01N43/76 , A01N43/64 , A01N43/50
CPC分类号： A01N43/90 , A01N43/74 , C07D277/36 , C07D277/74
摘要： Pesticidal fluoroalkene derivatives (I) wherein A is oxygen, NRa; Ra is hydrogen; optionally halogenated alkyl, alkenyl, alkynyl; X is hydrogen, halogen; optionally halogenated alkyl or phenyl; R1,R2 are hydrogen, halogen, hydroxyl, cyano, nitro, mercapto, amino; alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkylthio, alkylamino, dialkylamino, alkoxycarbonyl, alkylcarbonyloxy, optionally halogenated or substituted by 1 to 3 Rb groups: Rb is cyano, nitro, halogen, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl; optionally halogenated alkyl, haloalkyl, alkenyl, alkenyloxy, alkynyl, alkoxy, haloalkoxy, alkylthio, alkylamino, dialkylamino, formyl, alkylcarbonyl, alkylsulfonyl, alkoxysulfonyl, alkylsulfonyloxy, alkoxycarbonyl, alkylcarbonyloxy, alkylaminocarbonyl, dialkylaminocarbonyl, alkylaminothiocarbonyl, dialkylaminothiocarbonyl, alkylenedioxy or cycloalkyl; Het is a monocyclic or bicyclic 3- to 10-membered heteroaromatic ring system containing 1 to 5 heteroatoms selected from oxygen, sulfur and nitrogen, optionally halogenated or substituted by 1 to 4 Rc groups: Rc is Rb, alkoxyalkyl, alkylsulfinyl, alkylaminosulfonyl, di-alkylaminosulfonyl, alkylcarbonylamino, optionally substituted by halogen or 1 to 3 cyano, hydroxy, mercapto, amino, C1-C6-alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, C1-C6-alkoxycarbonyl, C1-C6-alkylcarbonyloxy or nitro groups; cycloalkyl, cycloalkoxy, saturated or partially unsaturated heterocyclyl, heterocyclyloxy, aryl, aryloxy, arylthio, arylalkoxy, arylalkyl, hetaryl, hetaryloxy, hetarylthio, optionally substituted; m is 0-2; n is 0-3; p is 0-6, methods for the preparation of compounds I, compositions and methods comprising the compounds and compositions for the control of nematodes, insects, arachnids, harmful fungi and unwanted plants, and for treating, controlling, preventing and protecting warm-blodded animals, fish and humans against infestation and infection by helminths, arachnids and arthropod endo- and ectoparasites.

46. 发明授权

US06414157B1 3-Substituted tetrahydropyridopyrimidinone derivatives, method for producing the same, and their use 有权
标题翻译： 3-取代的四氢吡啶并嘧啶酮衍生物，其制备方法及其用途
公开(公告)号：US06414157B1
公开(公告)日：2002-07-02
申请号：US09529231
申请日：2000-04-10
申请人： Wilfried Lubisch , Uta Dullweber , Dorothea Starck , Gerd Steiner , Alfred Bach , Franz Emling , Xavier Garcia-Ladona , Hans-Jürgen Teschendorf , Karsten Wicke
发明人： Wilfried Lubisch , Uta Dullweber , Dorothea Starck , Gerd Steiner , Alfred Bach , Franz Emling , Xavier Garcia-Ladona , Hans-Jürgen Teschendorf , Karsten Wicke
IPC分类号： C07D47100
CPC分类号： C07D471/04
摘要： 3-substituted tetrahydropyridopyrimidinone derivatives of the formula (I) wherein the radicals have the meanings given in the Description, to a method for producing said derivatives and, to their use for producing active ingredients for drugs.
摘要翻译：式（I）的3-取代四氢吡啶并嘧啶酮衍生物，其中基团具有说明书中给出的含义，所述衍生物的制备方法及其制备用于药物的活性成分的用途。

47. 发明授权

US06300354B1 N-substituted azabicycloheptane derivatives, production and use thereof 失效
标题翻译： N-取代的氮杂双环庚烷衍生物，其制备和应用
公开(公告)号：US06300354B1
公开(公告)日：2001-10-09
申请号：US09744405
申请日：2001-01-24
申请人： Gerd Steiner , Thomas Höger , Liliane Unger , Hans-Jürgen Teschendorf , Frieder Juchelka
发明人： Gerd Steiner , Thomas Höger , Liliane Unger , Hans-Jürgen Teschendorf , Frieder Juchelka
IPC分类号： A61K31428
CPC分类号： C07D417/06
摘要： Compounds of the formula I: in which R1, R2, R3 and R4 have the meanings stated in the description, are described. The novel compounds are suitable for controlling diseases.
摘要翻译：描述了其中R1，R2，R3和R4具有说明书所述含义的式I化合物：新化合物适用于控制疾病。

48. 发明授权

US06222034B1 3-substituted pyrido[4′,3′:4,5]thieno[2,3-d]pyrimidine derivatives, their preparation and their use 有权
标题翻译： 3-取代的吡啶并[4'，3'：4,5]噻吩并[2,3-d]嘧啶衍生物，其制备及其用途
公开(公告)号：US06222034B1
公开(公告)日：2001-04-24
申请号：US09254449
申请日：1999-03-10
申请人： Gerd Steiner , Wilfried Lubisch , Alfred Bach , Franz Emling , Karsten Wicke , Hans-Jürgen Teschendorf , Berthold Behl , Sharon Cheetham , Frank Kerrrigan
发明人： Gerd Steiner , Wilfried Lubisch , Alfred Bach , Franz Emling , Karsten Wicke , Hans-Jürgen Teschendorf , Berthold Behl , Sharon Cheetham , Frank Kerrrigan
IPC分类号： C07D49514
CPC分类号： C07D495/14
摘要： A 3-substituted 3,4,5,6,7,8-hexahydropyrido[4′,3′:4,5]thieno[2,3-d]pyrimidine compound of formula I wherein R1 is hydrogen, C1-C4-alkyl, acetyl or benzoyl, optionally substituted phenyl-C1-C4-alkyl, naphthyl-C1-C3-alkyl, phenyl-C2-C3-alkanone or a phenylcarbamoyl-C2-alkyl, R2 is optionally substituted phenyl, pyridyl, pyrimidyl or pyrazinyl, or an optionally substituted bicyclus wherein one of the two fused rings is a phenyl, a pyridyl, a pyrimidyl or a pyrazinyl ring, A is NH or oxygen, B is hydrogen or methyl, C is hydrogen, methyl or hydroxyl, X is nitrogen, Y is CH2, CH2—C2, CH2—C2—CH2 or CH2—CH, Z is nitrogen, C or CH, and the linkage between Y and Z is a single or a double bond, and n is 2, 3 or 4, or a physiologically tolerated salt thereof, and compositions comprising them and their use as antagonists of 5HT1B and 5HT1A and for the treatment of depression and related disorders.
摘要翻译：式I的3-取代的3,4,5,6,7,8-六氢吡啶并[4'，3'：4,5]噻吩并[2,3-d]嘧啶化合物，其中R1为氢，C1-C4-烷基，乙酰基或苯甲酰基，任选取代的苯基-C 1 -C 4 - 烷基，萘基-C 1 -C 3 - 烷基，苯基-C 2 -C 3 - 烷酮或苯基氨基甲酰基-C 2 - 烷基，R 2是任选取代的苯基，吡啶基，嘧啶基或吡嗪基，或任选取代的双环，其中两个稠合环之一为苯基，吡啶基，嘧啶基或吡嗪基，A为NH或氧，B为氢或甲基，C为氢，甲基或羟基，X为氮，Y 是CH2，CH2-C2，CH2-C2-CH2或CH2-CH，Z是氮，C或CH，Y和Z之间的键是单键或双键，并且是2,3或4，或生理上耐受的盐，以及包含它们的组合物及其作为5HT1B和5HT1A的拮抗剂的用途以及用于治疗抑郁症和相关疾病的用途。

49. 发明授权

US6159981A 3-substituted pyrido [3',4':4,5] Thieno [2,3-d] pyrimidine derivatives, and production and use of the same 有权
标题翻译： 3-取代的吡啶并[3'，4'：4,5]噻吩并[2,3-d]嘧啶衍生物及其制备和使用
公开(公告)号：US6159981A
公开(公告)日：2000-12-12
申请号：US445178
申请日：1999-12-08
申请人： Gerd Steiner , Uta Dullweber , Dorothea Starck , Alfred Bach , Karsten Wicke , Hans-Jurgen Teschendorf , Francisco-Javier Garcia-Ladona , Franz Emling
发明人： Gerd Steiner , Uta Dullweber , Dorothea Starck , Alfred Bach , Karsten Wicke , Hans-Jurgen Teschendorf , Francisco-Javier Garcia-Ladona , Franz Emling
IPC分类号： A61K31/519 , A61P25/00 , A61P25/24 , A61P43/00 , C07D495/14 , A61K31/495 , A61K31/505
CPC分类号： C07D495/14
摘要： 3-Substituted 3,4,5,6,7,8-hexahydropyrido [3',4':4,5]-thieno[2,3-d]pyrimidine derivatives of the formula I ##STR1## where R.sup.1 is a hydrogen atom, a C.sub.1 -C.sub.4 -alkyl group, an acetyl group, a phenylalkyl C.sub.1 -C.sub.4 radical, the aromatic system being unsubstituted or substituted by halogen, C.sub.1 -C.sub.4 -alkyl, trifluoromethyl, hydroxyl, C.sub.1 -C.sub.4 -alkoxy, amino, cyano or nitro groups, or is a phenylalkanone radical, it being possible for the phenyl group to be substituted by halogen,R.sup.2 is a phenyl, pyridyl, pyrimidinyl or pyrazinyl group which is unsubstituted or mono- or disubstituted by halogen atoms, C.sub.1 -C.sub.4 -alkyl, trifluoromethyl, trifluoromethoxy, hydroxyl, C.sub.1 -C.sub.4 -alkoxy, amino, monomethylamino, dimethylamino, cyano or nitro groups and which may be fused to a benzene nucleus which can be unsubstituted or mono- or disubstituted by halogen atoms, C.sub.1 -C.sub.4 -alkyl, hydroxyl, trifluoromethyl, C.sub.1 -C.sub.4 -alkoxy, amino, cyano or nitro groups and may contain 1 nitrogen atom, or to a 5- or 6-membered ring which may contain 1-2 oxygen atoms,A is NH or an oxygen atom,Y is CH.sub.2, CH.sub.2 --CH.sub.2, CH.sub.2 --CH.sub.2 --CH.sub.2 or CH.sub.2 --CH,Z is a nitrogen atom, carbon atom or CH, it also being possible for the linkage between Y and Z to be a double bond,and n is 2, 3 or 4, and the physiologically tolerated salts thereof.
摘要翻译： PCT No.PCT / EP98 / 03231 Sec。 371 1999年12月8日第 102（e）日期1999年12月8日PCT提交1998年5月29日PCT公布。第WO98 / 56793号公报日期：19983年12月17日 - 取代式I的3,4,5,6,7,8-六氢吡啶并[3'，4'：4,5] - 噻吩并[2,3-d]嘧啶衍生物，其中R1是一个氢原子，一个C 1 -C 4烷基，一个乙酰基，一个苯基烷基C 1 -C 4基团，该芳族体系是未被取代的或被卤素，C 1 -C 4烷基，三氟甲基，羟基，C 1 -C 4烷氧基，氨基氰基或硝基，或者是苯基烷酮基，苯基可以被卤素取代，R2是苯基，吡啶基，嘧啶基或吡嗪基，其是未被取代的或被卤原子单取代或被C1- C4-烷基，三氟甲基，三氟甲氧基，羟基，C 1 -C 4 - 烷氧基，氨基，一甲基氨基，二甲基氨基，氰基或硝基，并且它们可以与苯核稠合，苯核可被未被取代或被卤素原子， C 4 - 烷基，羟基，三氟甲基，C 1 -C 4 - 烷氧基，氨基，氰基或硝基，并且可以含有1个氮原子，或可以含有5或6元环，含有1-2个氧原子，A是NH或氧原子，Y是CH 2，CH 2 -CH 2，CH 2 -CH 2 -CH 2或CH 2 -CH，Z是氮原子，碳原子或CH，也可以是 Y与Z之间的连接为双键，n为2,3或4，以及其生理上耐受的盐。

50. 发明授权

US5258357A Carboxamides, their preparation and their use as herbicides 失效
标题翻译：羧甲酰胺，它们的制备及其作为除草剂的用途
公开(公告)号：US5258357A
公开(公告)日：1993-11-02
申请号：US947538
申请日：1992-09-21
申请人： Peter Muenster , Gerd Steiner , Wolfgang Freund , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Peter Muenster , Gerd Steiner , Wolfgang Freund , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/08 , A01N43/10 , A01N43/28 , C07D307/68 , C07D333/38 , C07D407/12 , C07D409/12 , C07D417/12 , A01N57/08 , C07D307/38
CPC分类号： C07D407/12 , A01N43/08 , A01N43/10 , A01N43/28 , C07D307/68 , C07D333/38 , C07D409/12 , C07D417/12
摘要： Carboxamides of the formulae Ia to Ic ##STR1## where X is oxygen or sulfur;R.sup.1 is hydrogen or substituted or unsubstituted cycloalkyl or alkyl;R.sup.2 is hydroxy, alkoxy, cyanoalkyl, substituted or unsubstituted alkenyl, alkynyl, phenyl or naphthyl, a substituted or unsubstituted 5- to 6-membered heterocyclic structure or one of the groups stated for R.sup.1, orR.sup.1 and R.sup.2 together are a 4- to 7-membered chain which contains, in addition to methylene groups, one of the following groups as ring member: oxygen, sulfur, N-methyl or carbonyl;R.sup.3 and R.sup.4 are each nitro, cyano, halogen, substituted or unsubstituted amino, alkoxy, alkylthio, a substituted or unsubstituted 5- to 6 -membered heterocyclic structure, substituted or unsubstituted alkenyl, alkynyl, phenyl, phenoxy or phenylthio, or one of the groups stated for R.sup.1 ;R.sup.5 is formyl, 4,5-dihydrooxazol-2-yl or COYR.sup.6 (Y=O,S);R.sup.6 is hydrogen, cycloalkyl, substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkenyl or phenyl,a 5- to 6-membered heterocyclic structure, phthalimido, tetrahydrophthalimido, succinimido, maleimido, benzotriazolyl ora group --N.dbd.CR.sup.7 R.sup.8, whereR.sup.7 and R.sup.8 are hydrogen or alkyl, and R.sup.8 may also be cycloalkyl, phenyl, furyl or R.sup.7 and R.sup.8 together form a 4- to 7 -membered alkylene chain; and if R.sup.5 is carboxyl, methoxycarbonyl or ethoxycarbonyl and R.sup.2 is hydrogen, R.sup.3 is not hydrogen and R.sup.4 is not hydrogen or methyl, and if R.sup.5 is carboxyl, methoxycarbonyl or ethoxycarbonyl and R.sup.4 is hydrogen, R.sup.3 is not hydrogen or R.sup.2 is not one of the following groups: hydrogen; C.sub.1 -C.sub.4 -alkyl, phenyl; 2-(3,4-dimethoxyphenyl)ethyl or 2,5 -dichlorothien-3-yl;processes for the manufacture of compounds I and herbicidal agents containing them.
摘要翻译：式Ia至Ic的酰胺酰胺其中X是氧或硫; R1是氢或取代或未取代的环烷基或烷基; R 2是羟基，烷氧基，氰基烷基，取代或未取代的烯基，炔基，苯基或萘基，取代或未取代的5至6元杂环结构或对于R1表示的基团之一，或R 1和R 2一起为4- 除了亚甲基之外，还含有以下基团之一的环元素：氧，硫，N-甲基或羰基的7-元链; R 3和R 4各自为硝基，氰基，卤素，取代或未取代的氨基，烷氧基，烷硫基，取代或未取代的5-至6-元杂环结构，取代或未取代的烯基，炔基，苯基，苯氧基或苯硫基， R1表示的组; R5是甲酰基，4,5-二氢恶唑-2-基或COYR 6（Y = O，S）; R 6是氢，环烷基，取代或未取代的烷基，烯基，炔基，环烯基或苯基，5-至6-元杂环结构，邻苯二甲酰亚氨基，四氢邻苯二甲酰亚胺基，琥珀酰亚胺基，马来酰亚胺基，苯并三唑基或基团-N = CR 7 R 8，其中R 7和R 8 R 8也可以是环烷基，苯基，呋喃基，或者R 7和R 8一起形成4-7个亚烷基链; 如果R5是羧基，甲氧基羰基或乙氧基羰基，R2是氢，R3不是氢，R4不是氢或甲基，如果R5是羧基，甲氧基羰基或乙氧基羰基，R4是氢，R3不是氢或R2不是以下组：氢; C 1 -C 4 - 烷基，苯基; 2-（3,4-二甲氧基苯基）乙基或2,5-二氯噻吩-3-基; 制备化合物I和含有它们的除草剂的方法。

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