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21. 发明授权

US5292911A Monocyclic terpene derivatives 失效
标题翻译：单环萜烯衍生物
公开(公告)号：US5292911A
公开(公告)日：1994-03-08
申请号：US849576
申请日：1992-03-10
申请人： Hisao Takayanagi , Yasunori Kitano , Yasuhiro Morinaka
发明人： Hisao Takayanagi , Yasunori Kitano , Yasuhiro Morinaka
IPC分类号： C07C33/42 , C07C45/29 , C07C45/51 , C07C47/24 , C07C49/587 , C07C69/65 , C07C255/16 , C07C255/46 , C07F7/18 , C07F7/10 , C07C69/52
CPC分类号： C07F7/1856 , C07C255/16 , C07C255/46 , C07C33/423 , C07C45/298 , C07C45/511 , C07C45/512 , C07C47/24 , C07C49/587 , C07C69/65 , C07F7/1852 , C07C2101/18
摘要： Novel monocyclic terpene derivative of the formula: ##STR1## wherein R is hydrogen atom, trimethylsilyl group or 1-ethoxyethyl group, and novel intermediates therefor. The terpene derivative (I) is a useful intermediate for preparing Sarcophytol A having an anti-carcinogenesis promoter activity and an antitumor activity.
摘要翻译：下式的新型单环萜衍生物：其中R是氢原子，三甲基甲硅烷基或1-乙氧基乙基，及其新颖的中间体。萜烯衍生物（I）是制备具有抗致癌作用启动子活性和抗肿瘤活性的Sarcophytol A的有用中间体。

22. 发明授权

US5149843A Conjugated diene compounds 失效
标题翻译：连接二烯化合物
公开(公告)号：US5149843A
公开(公告)日：1992-09-22
申请号：US712043
申请日：1991-06-07
申请人： Hisao Takayanagi , Yasunori Kitano , Yasuhiro Morinaka
发明人： Hisao Takayanagi , Yasunori Kitano , Yasuhiro Morinaka
IPC分类号： C07D303/12 , C07C33/02 , C07C43/15 , C07C43/178 , C07C45/29 , C07C45/51 , C07C47/24 , C07C47/263 , C07C47/277 , C07C49/24 , C07C49/255 , C07C49/587 , C07C69/007 , C07C69/63 , C07C69/732 , C07C69/78 , C07C309/65 , C07C309/73 , C07D303/14 , C07F7/02 , C07F7/08 , C07F7/18
CPC分类号： C07F7/1856 , C07C33/02 , C07C43/15 , C07C43/178 , C07C45/298 , C07C45/516 , C07C47/24 , C07C47/263 , C07C47/277 , C07C49/24 , C07C49/255 , C07C49/587 , C07C69/007 , C07C69/732 , C07D303/14 , C07F7/1852 , C07C2101/18
摘要： Conjugated diene compounds of the general formula: ##STR1## which are industrially advantageous intermediates for preparing sarcophytol A useful as an anticarcinogenic promotor or antitumor agent are provided.

23. 发明授权

US5116858A 4-imidazoline derivatives 失效
标题翻译： 4-咪唑啉衍生物
公开(公告)号：US5116858A
公开(公告)日：1992-05-26
申请号：US514832
申请日：1990-04-26
申请人： Yoshio Hayashi , Yasuhiro Morinaka , Masaki Shinoda , Hiroyoshi Nishi , Kazutoshi Watanabe , Nobuko Fukushima
发明人： Yoshio Hayashi , Yasuhiro Morinaka , Masaki Shinoda , Hiroyoshi Nishi , Kazutoshi Watanabe , Nobuko Fukushima
IPC分类号： A61K31/415 , A61P25/28 , A61P43/00 , C07D233/70
CPC分类号： C07D233/70
摘要： 4-Imidazoline derivatives represented by the formula (I) and/or formula (II): ##STR1## wherein R.sup.1 represents C.sub.1 -C.sub.8 alkyl, C.sub.3 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 alkynyl, C.sub.3 -C.sub.8 cycloalkyl, or optionally substituted aralkyl; R.sup.2 and R.sup.3 independently represent hydrogen, C.sub.3 -C.sub.20 alkyl, C.sub.3 -C.sub.20 alkenyl, C.sub.3 -C.sub.20 alkynyl, C.sub.3 -C.sub.20 alkoxy, C.sub.3 -C.sub.20 alkenyloxy, C.sub.3 -C.sub.20 alkynyloxy, C.sub.3 -C.sub.8 cyloalkyl, C.sub.1 -C.sub.10 alkylthio, or optionally substituted aralkyl or aralkyloxy; R.sup.4 represents C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.8 cycloalkyl, or optionally substituted aralkyl; provided that R.sup.2 and R.sup.3 cannot be hydrogen at the same time, and pharmaceutically acceptable salts thereof. A pharmaceutical formulation containing the compound is also provided.

24. 发明授权

US07148926B2 Image sensing apparatus and signal processing method therefor 失效
标题翻译：图像传感装置及其信号处理方法
公开(公告)号：US07148926B2
公开(公告)日：2006-12-12
申请号：US10311672
申请日：2002-05-09
申请人： Yasuhiro Morinaka , Hiroyoshi Komobuchi , Akito Kidera , Toshiya Fujii
发明人： Yasuhiro Morinaka , Hiroyoshi Komobuchi , Akito Kidera , Toshiya Fujii
IPC分类号： H04N3/14
CPC分类号： H04N9/045 , H04N5/347 , H04N5/3728
摘要： A color filter arrangement (11) is used, in which a plurality of filter units are each made of 2×2 arrangements of red (R), green (G), green (G) and blue (B) color elements. First, signal charges are added up for all pixels belonging to each of a plurality of pixel blocks made of quadratic arrangements of 3×3 of pixels, which are larger than the filter units (2×2 arrangement). Then, compressed color information for each of the pixel blocks is obtained from a result of the addition for each pixel block, taking the 2×2 arrangements of pixel blocks as large filter units.
摘要翻译：使用滤色器装置（11），其中多个滤色器单元分别由红（R），绿（G），绿（G）和蓝（B）色元素的2×2布置构成。首先，对于属于大于滤波器单元（2x2排列）的3×3像素的二次排列构成的多个像素块中的每一个像素块的所有像素，相加信号电荷。然后，以每个像素块的加法结果，以像素块的2×2布置为大的滤波器单位，获得每个像素块的压缩颜色信息。

25. 发明授权

US5118827A Monocyclic terpene derivatives 失效
标题翻译：单克隆衍生物
公开(公告)号：US5118827A
公开(公告)日：1992-06-02
申请号：US555999
申请日：1990-07-16
申请人： Hisao Takayanagi , Yasunori Kitano , Yasuhiro Morinaka
发明人： Hisao Takayanagi , Yasunori Kitano , Yasuhiro Morinaka
IPC分类号： C07C33/42 , C07C45/29 , C07C45/51 , C07C47/24 , C07C49/587 , C07C69/65 , C07C255/16 , C07C255/46 , C07F7/18
CPC分类号： C07F7/1856 , C07C255/16 , C07C255/46 , C07C33/423 , C07C45/298 , C07C45/511 , C07C45/512 , C07C47/24 , C07C49/587 , C07C69/65 , C07F7/1852 , C07C2101/18
摘要： Novel monocyclic terpene derivative of the formula: ##STR1## wherein R is hydrogen atom, trimethylsilyl group or 1-ethoxyethyl group, and novel intermediate therefor. The terpene derivative (I) is a useful intermediate for preparing Sarcophytol A having an anti-carcinogenesis promoter activity and an antitumor activity.

26. 发明授权

US4857542A Prophylactic and therapeutic composition for circulatory disorders and method of treatment 失效
标题翻译：循环障碍的预防和治疗组合物及治疗方法
公开(公告)号：US4857542A
公开(公告)日：1989-08-15
申请号：US122516
申请日：1987-11-19
申请人： Hiroyoshi Nishi , Toshiaki Watanabe , Satoshi Yuki , Yasuhiro Morinaka , Katsuhiko Iseki , Hiroko Sakurai
发明人： Hiroyoshi Nishi , Toshiaki Watanabe , Satoshi Yuki , Yasuhiro Morinaka , Katsuhiko Iseki , Hiroko Sakurai
IPC分类号： C07D231/20 , C07D231/22 , C07D231/26 , C07D231/28 , C07D231/56
CPC分类号： C07D231/56 , C07D231/20 , C07D231/22 , C07D231/26 , C07D231/28
摘要： A prophylactic and therapeutic agent for circulatory disorders, comprising a pyrazolone derivative of the formula: ##STR1## wherein R.sub.1 represents a hydrogen atom, an aryl group, an alkyl group having 1 to 5 carbon atoms or an alkoxycarbonylalkyl group having a total carbon number of 3 to 6; R.sub.2 represents a hydrogen atom, an aryloxy group, an arylmercapto group, an alkyl group having 1 to 5 carbon atoms or hydroxyalkyl group having 1 to 3 carbon atoms; or R.sub.1 and R.sub.2 taken together represent an alkylene group having 3 to 5 carbon atoms; R.sub.3 represents a hydrogen atom, an alkyl group having 1 to 5 carbon atoms, a cycloalkyl group having 5 to 7 carbon atoms, a hydroxyalkyl group having 1 to 3 carbon atoms, a benzyl group, a naphthyl group, or a phenyl group which is unsubstituted or substituted with 1 to 3 substituents which are the same or different selected from the group consisting of alkyl groups having 1 to 5 carbon atoms, alkoxy groups having 1 to 5 carbon atoms, hydroxyalkyl groups having 1 to 3 carbon atoms, alkoxycarbonyl groups having total carbon number of 2 to 5, alkylmercapto groups having 1 to 3 carbon atoms, alkylamino groups having 1 to 4 carbon atoms, dialkylamino groups having total carbon number of 2 to 8, halogen atoms, trifluoromethyl group, carboxyl group, cyano group, hydroxyl group, nitro group, amino group and acetamide group,or a pharmaceutically acceptable salt thereof as an acitve ingredient.The agent of the present invention is useful as a prophylactic and therapeutic agent for circulatory disorders, particularly as an inhibitor agaisnt lipid peroxidation and/or an agent for normalizing cerebral dysfunctions.
摘要翻译：一种循环系统疾病的预防和治疗剂，其包含下式的吡唑啉酮衍生物：其中R 1表示氢原子，芳基，具有1至5个碳原子的烷基或具有总碳数的烷氧基羰基烷基 3至6; R2表示氢原子，芳氧基，芳基巯基，碳原子数1〜5的烷基或碳原子数1〜3的羟烷基。或R 1和R 2一起表示具有3至5个碳原子的亚烷基; R3表示氢原子，碳原子数1〜5的烷基，碳原子数5〜7的环烷基，碳原子数1〜3的羟烷基，苄基，萘基或苯基，未取代或被1〜3个选自碳原子数1〜5的烷基，碳原子数为1〜5的烷氧基，碳原子数1〜3的烷氧基，碳原子数1〜3的烷氧基，烷氧基羰基，总碳数为2至5，具有1至3个碳原子的烷基巯基，具有1至4个碳原子的烷基氨基，总碳数为2至8的二烷基氨基，卤素原子，三氟甲基，羧基，氰基，羟基基团，硝基，氨基和乙酰胺基，或其药学上可接受的盐作为acitve成分。本发明的药剂可用作循环障碍的预防和治疗剂，特别是作为抑制剂脂质过氧化作用的抑制剂和/或用于使脑功能障碍正常化的药剂。

27. 发明授权

US4613613A .gamma.-butyrolactone derivatives, process for preparing the same and immunomodulating compositions containing the same as active ingredients 失效
标题翻译： γ-丁内酯衍生物，其制备方法和含有该活性成分的免疫调节组合物
公开(公告)号：US4613613A
公开(公告)日：1986-09-23
申请号：US647979
申请日：1984-09-06
申请人： Tomei Oguri , Yasuhiro Morinaka , Shuichiro Kadowaki
发明人： Tomei Oguri , Yasuhiro Morinaka , Shuichiro Kadowaki
IPC分类号： A61K31/365 , A61P29/00 , C07D307/33 , C07D307/58 , C07D307/94 , A61K31/34 , C07D307/10 , C07D307/26
CPC分类号： C07D307/33 , C07D307/58 , C07D307/94
摘要： A .gamma.-butyrolactone derivative represented by the following formula: ##STR1## wherein R.sup.1 represents a hydrogen atom, a straight or branched alkyl group having 1-8 carbon atoms, a phenyl group; R.sup.2 and R.sup.3 may be the same or different and each represents a hydrogen atom, a straight or branched alkyl group having 1-8 carbon atoms, a cycloalkyl group having 3-10 carbon atoms, a benzyl group, a phenyl group, a phenyl group substituted with a substituent selected from the group consisting of a halogen atom, an alkoxy group, a nitro group, an amino group, an alkyl group having 1-4 carbon atoms, a nitrile group and an alkoxycarbonyl group; R.sup.2 and R.sup.3 may be linked to form an alkylene group having 4-6 carbon atoms; X represents a hydrogen atom, a straight or branched alkyl group having 1-8 carbon atoms, a cycloalkyl group having 3-10 carbon atoms, a benzyl group or a substituent represented by the formula ##STR2## (wherein R.sup.4 represents a straight or branched alkyl group having 1-8 carbon atoms, a cycloalkyl group having 3-10 carbon atoms, a benzyl group, a phenyl group or a phenyl group substituted with a substituent selected from the group consisting of a halogen atom, an alkoxy group, a nitro group, an alkylthio group, a nitrile group, an alkoxycarbonyl group and an alkyl group having 1-4 carbon atoms) or a salt thereof. The invention also provides an immunomodulating composition wherein the aforedescribed compound is the active component.
摘要翻译：由下式表示的γ-丁内酯衍生物：其中R1表示氢原子，具有1-8个碳原子的直链或支链烷基，苯基; R2和R3可以相同或不同，各自表示氢原子，具有1-8个碳原子的直链或支链烷基，具有3-10个碳原子的环烷基，苄基，苯基，苯基被选自卤素原子，烷氧基，硝基，氨基，具有1-4个碳原子的烷基，腈基和烷氧羰基组成的组中的取代基取代; R2和R3可以连接形成具有4-6个碳原子的亚烷基; X表示氢原子，具有1-8个碳原子的直链或支链烷基，具有3-10个碳原子的环烷基，苄基或由式“IMAGE”表示的取代基（其中R4表示直链或支链具有1-8个碳原子的烷基，具有3-10个碳原子的环烷基，苄基，苯基或被选自卤素原子，烷氧基，硝基的取代基取代的苯基基团，烷硫基，腈基，烷氧基羰基和具有1-4个碳原子的烷基）或其盐。本发明还提供一种免疫调节组合物，其中上述化合物是活性成分。

28. 发明授权

US4086349A Quinolopyran-4-one-2-carboxylic acid derivatives and salts thereof as novel compounds and as medicines for treatment of allergic asthma 失效
标题翻译：喹诺酮-4-酮-2-羧酸衍生物及其盐作为新化合物和用作治疗过敏性哮喘的药物
公开(公告)号：US4086349A
公开(公告)日：1978-04-25
申请号：US709779
申请日：1976-07-29
申请人： Yasuhiro Morinaka , Kazuo Takahashi
发明人： Yasuhiro Morinaka , Kazuo Takahashi
IPC分类号： C07D491/04 , C07D491/052 , A61K31/47
CPC分类号： C07D491/04 , Y10S514/826
摘要： Quinolopyran-4-one-2-carboxylic acid derivatives and salts thereof are provided as novel compounds and as medicines for treatment of allergic asthma, each of the derivatives being represented by the general formula ##STR1## wherein X designates a member selected from the group consisting of alkyl groups having 1 to 5 carbon atoms, alkoxy groups having 1 to 5 carbon atoms, halogen atoms, aryl-substituted alkoxy groups having 7 to 10 total carbon atoms, alkoxycarbonyl groups having 2 to 6 total carbon atoms, and aryl groups having 6 to 10 carbon atoms, and n is any one of the integers 1 through 4, X being the same group or different groups in the case where n is at least 2.
摘要翻译：提供了喹诺酮-4-酮-2-羧酸衍生物及其盐作为新化合物和用作治疗过敏性哮喘的药物，每种衍生物由通式“IMAGE”表示，其中X表示选自下组的成员由具有1至5个碳原子的烷基，具有1至5个碳原子的烷氧基，卤素原子，具有7至10个总碳原子的芳基取代的烷氧基，具有2至6个总碳原子的烷氧基羰基组成的芳基和具有 6至10个碳原子，n为整数1至4中的任一个，X为相同基团或在n为至少2的情况下为不同基团。

29. 发明授权

US07050099B2 Solid-state image pickup apparatus 有权
公开(公告)号：US07050099B2
公开(公告)日：2006-05-23
申请号：US10125082
申请日：2002-04-18
申请人： Kentaro Takakura , Toshiya Fujii , Hiroyoshi Komobuchi , Yasuhiro Morinaka , Kazuyuki Inokuma
发明人： Kentaro Takakura , Toshiya Fujii , Hiroyoshi Komobuchi , Yasuhiro Morinaka , Kazuyuki Inokuma
IPC分类号： H04N5/202
CPC分类号： H04N5/2176 , H04N5/3653 , H04N5/3728
摘要： Gray level data of boundary pixels that are adjacent to a block boundary in a photoelectric conversion section is stored. Then, a cumulative histogram regarding the number of pixels for different gray levels is produced based on the stored gray level data separately for each block, and a data table representing the correspondence between each gray level before correction and that after correction for the block to be corrected is produced so as to reduce the difference between the cumulative histograms. The data table is stored in a correction data RAM. By using the data table, the outputs of the block to be corrected are non-linearly corrected for different gray levels.

30. 发明授权

US5304661A Substituted-acyclic terpene compound 失效
标题翻译：取代的非环萜烯化合物
公开(公告)号：US5304661A
公开(公告)日：1994-04-19
申请号：US44602
申请日：1993-04-09
申请人： Hisao Takayanagi , Yasunori Kitano , Yasuhiro Morinaka
发明人： Hisao Takayanagi , Yasunori Kitano , Yasuhiro Morinaka
IPC分类号： C07C33/02 , C07C43/178 , C07C43/315 , C07C45/44 , C07C45/51 , C07C45/63 , C07C45/67 , C07C47/21 , C07C47/24 , C07C47/263 , C07C47/277 , C07C49/203 , C07C49/227 , C07C49/24 , C07C49/255 , C07C49/587 , C07C69/007 , C07C69/738 , C07C255/07 , C07C255/10 , C07C255/15 , C07C255/46 , C07C309/65 , C07D309/06 , C07D309/12 , C07F7/18 , C07D315/00
CPC分类号： C07F7/1856 , C07C255/07 , C07C255/10 , C07C255/15 , C07C255/46 , C07C309/65 , C07C33/02 , C07C43/178 , C07C43/315 , C07C45/44 , C07C45/512 , C07C45/516 , C07C45/63 , C07C45/673 , C07C45/676 , C07C47/21 , C07C47/24 , C07C47/263 , C07C47/277 , C07C49/203 , C07C49/227 , C07C49/24 , C07C49/255 , C07C49/587 , C07C69/007 , C07C69/738 , C07D309/06 , C07D309/12 , C07F7/1852 , C07C2101/18
摘要： Acyclic terpene compounds useful as intermediates for producing sarcophytol A which have an anti-carcinogenic promotor activity and anti-tumor activity, which compounds are shown by the general formula (I): ##STR1##
摘要翻译：用于制备具有抗致癌促进剂活性和抗肿瘤活性的唾液酸A的中间体的无环萜烯化合物，该化合物由通式（I）表示：（*化学结构*）（I）

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