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21. 发明授权

US5201932A Carboxamides 失效
公开(公告)号：US5201932A
公开(公告)日：1993-04-13
申请号：US877365
申请日：1992-05-04
申请人： Volker Maywald , Wolfgang Freund , Gerhard Hamprecht , Thomas Kuekenhoehner , Peter Plath , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Volker Maywald , Wolfgang Freund , Gerhard Hamprecht , Thomas Kuekenhoehner , Peter Plath , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/80 , C07D261/18 , C07D275/02 , C07D275/03
CPC分类号： C07D275/03 , A01N43/80 , C07D261/18
摘要： Carboxamides Ia, Ib, Ic and Id ##STR1## (X=O, S; R.sup.1 =H, halogen, substituted or unsubstituted alkyl, substituted or unsubstituted benzyl, alkoxy, alkylthio, haloalkoxy, haloalkylthio, substituted or unsubstituted phenyl, substituted or unsubstituted phenoxy or phenylthio, a substituted or unsubstituted 5- or 6-membered heterocyclic radical containing one or two heteroatoms, cycloalkyl-substituted alkyl, substituted or unsubstituted alkenyl which may be epoxidized, substituted or unsubstituted alkynyl, substituted or unsubstituted cycloalkyl or cycloalkenyl; R.sup.1 '=cycloalkyl-substituted alkyl, substituted or unsubstituted alkenyl which may be epoxidized, substituted or unsubstituted cycloalkenyl; R.sup.2 =CHO, 4,5-dihydrooxazol-2-yl, COYR.sup.5, CONR.sup.6 R.sup.7 ; Y=O, S; R.sup.5 =H, substituted or unsubstituted alkyl, cycloalkyl, substituted or unsubstituted alkenyl, substituted or unsubstituted cycloalkenyl, substituted or unsubstituted alkynyl, substituted or unsubstituted phenyl, a 5- or 6-membered heterocyclic radical containing up to 3 heteroatoms, benzotriazole, N-phthalimido, tetrahydrophthalimido, succinimido, maleiimido, 2,2-dimethyl-1,3-dioxolan-4-ylmethyl, 1,3-dioxolan-2-on-4-ylmethyl, and when Y.dbd.O: one equivalent of a cation from the group of the alkali or alkaline earth metals, Mn, Cu, Fe ammonium and substituted ammonium, a radical --N.dbd.CR.sup.8 R.sup.9 or --W--Z; R.sup.8, R.sup.9 .dbd.H, substituted or unsubstituted alkyl, substituted or unsubstituted haloalkyl, cycloalkyl, alkoxy, furanyl, substituted or unsubstituted phenyl; R.sup.8 +R.sup.9 =4-7-membered methylene chain; W=alkylene chain, ethoxyethylene chain, butylene, butynylene chain; Z=a molecular moiety bonded to W in the .omega.-position and is the same as that linked to W in the .alpha.-position of W; R.sup.6 .dbd.H, alkyl, cycloalkyl; R.sup.7 .dbd.H; alkyl; --C(O-alkyl).dbd.N--H or --(O--alkyl).dbd.N--alkyl; R.sup.6 +R.sup.7 =4-5-membered methylene chain; R.sup.3 .dbd.H, substituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl; R.sup.4 .dbd.H, OH, alkoxy, subsituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted alkenyl, substituted or unsubstituted alkynyl, di-(C.sub.1 -C.sub.4)-alkylamino, a substituted or unsubstituted 5- or 6-membered heterocyclic radical containing one or two heteroatoms, substituted or unsubstituted phenyl, substituted or unsubstituted naphthyl; R.sub.3 +R.sub.4 =4-7-membered methylene chain which may be interrupted by O, S or N--CH.sub.3, or --(CH.sub.2).sub.3 --CO--)and their environmentally tolerated salts.The compounds Ia to Id are suitable as herbicides.

22. 发明授权

US5069708A Pyrimido(5,4-e)-as-triazine-5,7(6H,8H)-diones 失效
标题翻译：嘧啶并（5,4-e）-as-三嗪-5,7（6H，8H） - 二酮
公开(公告)号：US5069708A
公开(公告)日：1991-12-03
申请号：US547160
申请日：1990-07-03
申请人： Norbert Meyer , Ulrich Shirmer , Peter Plath , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Norbert Meyer , Ulrich Shirmer , Peter Plath , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/90 , C07D487/04
CPC分类号： A01N43/90
摘要： Herbicidal agents containing a pyrimido[5,4-e]-as-triazine-5,7-(6H,8H)-dione Ia ##STR1## (R.sup.1, R.sup.2 .dbd.H, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.2 -C.sub.8 -alkenyl, phenyl or benzyl, R.sup.3 .dbd.H, halogen, nitro, C.sub.1 -C.sub.8 -alkyl which may carry up to three further substituents, C.sub.2 -C.sub.6 -alkenyl, phenyl-C.sub.2 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -cycloalkyl which may carry up to 3 C.sub.1 -C.sub.4 -alkyl substituents, a 5- or 6-membered heterocyclic structure where up to 2 of the ring members are O, S or NR.sup.4 ; --CO--R.sup.4 or --CO--O--R.sup.4 ; phenyl or hetaryl, which may carry up to 3 further substituents; or ZR.sup.6 ; R.sup.4 .dbd.H, C.sub.1 -C.sub.6 -alkyl; Z.dbd.O, S or --N(R.sup.7)--; R.sup.6 .dbd.H, C.sub.1 -C.sub.6 -alkyl, phenyl or benzyl, which may carry up to 3 further substituents; R.sup.7 .dbd.H, C.sub.1 -C.sub.6 -alkyl or R.sup.6 and R.sup.7 together with nitrogen form a 5- or 6-membered ring which may contain O; n=0 or 1) or a salt of Ia with a mineral acid.
摘要翻译：含有嘧啶并[5,4-e] -as-三嗪-5,7-（6H，8H） - 二酮Ia（Ia）（R1，R2 = H，C1-C6-烷基，C3- C 2 -C 6环烷基，C 2 -C 8 - 烯基，苯基或苄基，R 3 = H，卤素，硝基，可带有至多三个其它取代基的C 1 -C 8烷基，C 2 -C 6 - 链烯基，苯基-C 2 -C 6 - 烯基，可含有3个C 1 -C 4烷基取代基的C 3 -C 6环烷基，其中至多2个环成员为O，S或NR 4的5或6元杂环结构; -CO-R 4或-CO- R 4 = H，C 1 -C 6 - 烷基; Z = O，S或-N（R 7） - ; R 6 = H，C 1 -C 6烷基; - 烷基，苯基或苄基，其可以带有多达3个其它取代基; R 7 = H，C 1 -C 6 - 烷基或者R 6和R 7与氮一起形成5-或6-元环，其可以含有O; n = 0或 1）或Ia与无机酸的盐。

23. 发明授权

US5076831A 1,8-napthalenedicarboximides as antidotes 失效
标题翻译：作为抗体的1,8-壬基二氧嘧啶
公开(公告)号：US5076831A
公开(公告)日：1991-12-31
申请号：US615865
申请日：1990-11-20
申请人： Thomas Saupe , Norbert Meyer , Peter Plath , Ulrich Schirmer , Bruno Wuerzer , Karl-Otto Westphalen , Manfred Patsch , Juergen Pfister
发明人： Thomas Saupe , Norbert Meyer , Peter Plath , Ulrich Schirmer , Bruno Wuerzer , Karl-Otto Westphalen , Manfred Patsch , Juergen Pfister
IPC分类号： A01N25/32 , A01N39/02 , A01N39/04 , A01N43/42 , C07D221/14 , C07D401/12 , C07D405/12 , C07D409/12 , C07D471/06
CPC分类号： C07D221/14 , A01N25/32 , C07D401/12 , C07D405/12 , C07D409/12 , C07D471/06
摘要： Substituted 1,8-naphthalenedicarboximides of the formula: ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, X, Y, and Z have the meanings recited in the disclosure are disclosed as new compounds suitable for use as antidotes in herbicidal compositions.
摘要翻译：其中R 1，R 2，R 3，R 4，R 5，R 6，X，Y和Z具有本公开中所述的含义的取代的1,8-萘二甲酰亚胺如下所示：其中R1，R2，R3，R4，R5，R6，X，Y和Z具有适合用作解毒剂的新化合物除草组合物。

24. 发明授权

US5217523A Pyrazole-3-carboxamides, herbicidal compositions and use 失效
标题翻译：吡唑-3-甲酰胺，除草组合物和用途
公开(公告)号：US5217523A
公开(公告)日：1993-06-08
申请号：US877366
申请日：1992-05-04
申请人： Klaus Ditrich , Gerhard Hamprecht , Peter Plath , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Klaus Ditrich , Gerhard Hamprecht , Peter Plath , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： C07D231/14 , C07D401/04 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/04 , C07D405/12 , C07D405/14 , C07D409/04 , C07D409/12 , C07D409/14 , C07D413/04 , C07D417/14
CPC分类号： C07D401/04 , C07D231/14 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/04 , C07D405/12 , C07D405/14 , C07D409/04 , C07D409/12 , C07D409/14 , C07D413/04 , C07D417/14
摘要： Pyrazole-3-carboxamides of the general formula I ##STR1## where the substituents have the following meaning: R.sup.1 hydrogen;substituted or unsubstituted C.sub.3 -C.sub.8 -cycloalkyl or C.sub.1 C.sub.6 -alkyl;R.sup.2 hydroxy; amino; C.sub.1 -C.sub.4 -alkylamino; di-C.sub.1 -C.sub.4 -alkylamino, aminocarbonyl-C.sub.1 -C.sub.6 -alkyl; substituted or unsubstituted C.sub.1 -C.sub.4 -alkoxy, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, phenyl or naphthyl,a substituted or unsubstituted 5- to 6-membered heterocyclic ring;one of the groups mentioned for R.sup.1 orR.sup.1 and R.sup.2 together denote a 4- to 7-membered chain which may contain, in addition to methylene groups one of the following groups as ring member: oxygen, sulfur N-methyl or carbonyl;R.sup.3 a substituted or unsubstituted 5- to 6-membered heterocyclic ring.substituted or unsubstituted C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 alkynyl, 5,6,7,8-tetrahydronaphthyl or phenyl orone of the groups mentioned for R.sup.1 ;R.sup.4 nitro; cyano; carboxyl; halogen; substituted or unsubstituted C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.4 -alkylthio, orone of the groups mentioned for R.sup.3 ;R.sup.5 4,5-dihydroxazol-2-yl or a group COYR.sup.6 ;Y hydrogen;R.sup.6 C.sub.3 -C.sub.8 -cycloalkyl, substituted or unsubstituted C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, C.sub.5 -C.sub.7 -cycloalkenyl or phenyl,a substituted or unsubstituted 5- or 6-membered heterocyclic ring; phthalimido; tetrahydrophthalimido; succinimido; maleiimido; benzotriazolyl ora group --N.dbd.CR.sup.7 R.sup.8, whereR.sup.7 is hydrogen or C.sub.1 -C.sub.6 -alkyl andR.sup.8 is C.sub.3 -C.sub.6 -cycloalkyl, phenyl, furyl or a radical R.sup.7 orR.sup.7, R.sup.8 together denote a 4- to 7-membered alkylene chain,and their agriculturally useful salts, Y not denoting oxygen and R.sup.1 not denoting hydrogen when R.sup.3 is hydrogen and R.sup.4 is nitro, trifluoromethyl, halogen or C.sub.1 -C.sub.4 -alkoxy and --YR.sup.6 not denoting ethoxy when R.sup.1 is hydrogen, R.sup.4 is methyl and R.sup.2 is phenyl or substituted phenyl.
摘要翻译：吡唑-3-甲酰胺，其通式为Ⅰ，其中取代基具有下列含义：R 1氢; 取代或未取代的C 3 -C 8 - 环烷基或C 1 -C 6烷基; R2羟基; 氨基; C 1 -C 4烷基氨基; 二-C 1 -C 4烷基氨基，氨基羰基-C 1 -C 6 - 烷基; 取代或未取代的C 1 -C 4 - 烷氧基，C 3 -C 6 - 烯基，C 3 -C 6 - 炔基，苯基或萘基，取代或未取代的5至6元杂环; 对于R1或R1和R2提及的基团之一一起表示4至7元链，除了亚甲基之外，还可以含有以下基团之一作为环成员：氧，硫，N-甲基或羰基; R3是取代或未取代的5至6元杂环。取代或未取代的C 3 -C 6 - 烯基，C 3 -C 6炔基，5,6,7,8-四氢萘基或苯基或提及的R 1的一个基团; R4硝基; 氰基; 羧基; 卤素; 取代或未取代的C 1 -C 4 - 烷氧基或C 1 -C 4 - 烷硫基，或提及的基团之一; R5 4,5-二羟基恶唑-2-基或COYR 6基; Y氢; R 6 C 3 -C 8 - 环烷基，取代或未取代的C 1 -C 6 - 烷基，C 3 -C 6 - 烯基，C 3 -C 6 - 炔基，C 5 -C 7 - 环烯基或苯基，取代或未取代的5元或6元杂环; 邻苯二甲酰亚氨基; 四氢邻苯二甲酰亚胺琥珀酰亚胺马来西亚苯并三唑基或基团-N = CR 7 R 8，其中R 7是氢或C 1 -C 6烷基，R 8是C 3 -C 6环烷基，苯基，呋喃基或基团R 7或R 7，R 8一起表示4至7元亚烷基链和其农业上有用的盐，Y不表示氧，当R 3为氢时，R 1不表示氢，R 4为硝基，三氟甲基，卤素或C 1 -C 4 - 烷氧基，而R 1为氢时未表示乙氧基，R 4为甲基，R 2为R 2 是苯基或取代的苯基。

25. 发明授权

US5356860A Styrene derivatives useful as herbicides and defoliants 失效
标题翻译：苯乙烯衍生物可用作除草剂和脱叶剂
公开(公告)号：US5356860A
公开(公告)日：1994-10-18
申请号：US61535
申请日：1993-05-14
申请人： Bernd Schaefer , Lothar Rueb , Peter Schaefer , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
发明人： Bernd Schaefer , Lothar Rueb , Peter Schaefer , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
IPC分类号： A01N37/32 , A01N37/46 , A01N43/36 , A01N43/38 , A01N43/56 , A01N43/90 , C07D207/44 , C07D207/452 , C07D209/48 , C07D231/56 , C07D513/04 , C07D207/24 , C07D237/26 , C07D513/14
CPC分类号： C07D207/452 , A01N37/32 , A01N37/46 , A01N43/56 , A01N43/90 , C07D209/48 , C07D231/56 , C07D513/04
摘要： Abstract of the Disclosure: Styrene derivatives I ##STR1## where R.sup.1 is H or halogen, R.sup.2 is halogen, R.sup.3 is H, halogen or C.sub.1 -C.sub.4 -alkyl, R.sup.4 is CN or C.sub.1 -C.sub.6 -alkylcarbonyl and A is a heterocyclic radical A.sub.1 to A.sub.5 : ##STR2## where R.sup.5 and R.sup.6 are H, CH.sub.3 or C.sub.2 H.sub.5, n is 0 or 1 and X is oxygen or sulfur, with the proviso that R.sup.4 is alkylcarbonyl when R.sup.1 is H and at the same time A is A.sub.2 where n is 0, and agriculturally useful salts thereof, processes for the preparation of the styrene derivatives I and herbicides containing them.
摘要翻译：公开内容摘要：苯乙烯衍生物I其中R 1是H或卤素，R 2是卤素，R 3是H，卤素或C 1 -C 4烷基，R 4是CN或C 1 -C 6烷基羰基，A是杂环基 A1至A5： A1 A2 A3 A4 A5其中R5和R6为H，CH3或C2H5，n为0或1，X为氧或硫，当R 1是H时，R 4是烷基羰基，同时A是其中n是0的A2，其农业上有用的盐，制备苯乙烯衍生物I的方法和含有它们的除草剂。

26. 发明授权

US5284821A Oxazole- and thiazolecarboxamides 失效
标题翻译：恶唑和噻唑甲酰胺
公开(公告)号：US5284821A
公开(公告)日：1994-02-08
申请号：US919457
申请日：1992-07-27
申请人： Klaus Ditrich , Volker Maywald , Gerhard Hamprecht , Albrecht Harreus , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Klaus Ditrich , Volker Maywald , Gerhard Hamprecht , Albrecht Harreus , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/74 , C07D263/34 , C07D277/56 , C07D417/04 , A01N43/76
CPC分类号： C07D263/34 , A01N43/74 , C07D277/56 , C07D417/04
摘要： Oxazole- and thiazolecarboxamides of the formulae Ia and Ib ##STR1## where the substituents have the following meanings: X oxygen or sulfur;R.sup.1 hydrogen; halogen; substituted or unsubstituted C.sub.1 -C.sub.6 -alkyl, benzyl, cycloalkyl, alkenyl, alkynyl, phenyl, phenoxy or phenylthio; alkoxy; alkylthio; haloalkoxy; haloalkylthio; or a substituted or unsubstituted 5- or 6-membered heterocyclic radical;R.sup.2 formyl, 4,5-dihydrooxazol-2-yl or --COYR.sup.5 ;Y oxygen or sulfur;R.sup.5 hydrogen; cycloalkyl; substituted or unsubstituted alkyl, phenyl, benzyl, alkenyl, cycloalkenyl or alkynyl; a substituted or unsubstituted 5- or 6-membered heterocyclic radical; phthalimido; tetrahydrophthalimido; succinimido; maleiimido; one equivalent of a cation; or--N.dbd.CR.sup.6 R.sup.7 ; R.sup.6, R.sup.7 hydrogen; alkyl; cycloalkyl; phenyl; furyl or together a methylene chain of 4 to 7 members;R.sup.3 hydrogen or substituted or unsubstituted alkyl or cycloalkyl;R.sup.4 hydroxy; alkoxy; substituted or unsubstituted alkyl, cycloalkyl, alkenyl, alkynyl, phenyl or naphthyl; a substituted or unsubstituted 5- or 6-membered heterocyclic radical; or R.sup.3 and R.sup.4 together are --(CH.sub.2).sub.n --Y.sub.p --(CH.sub.2).sub.q --, where n and q are 1, 2 or 3, p is 0 or 1 and Y is oxygen, sulfur or N-methyl, or form a radical of the formula --(CH.sub.2).sub.3 --CO--, and their environmentally tolerated salts,X in formula Ib not being sulfur when R.sup.1 is 3-pyridyl, R.sup.2 is CO.sub.2 CH.sub.2 CH.sub.3 or R.sup.3 is hydrogen, and X in formula Ia X not being sulfur and R.sup.1 not being thien-2-yl when YR.sup.5 is OH, R.sup.3 is hydrogen and R.sup.4 is methyl, processes for manufacturing such compounds and herbicidal agents containing compounds of the formulae Ia or Ib as active ingredients.
摘要翻译：式Ia和Ib的恶唑和噻唑甲酰胺其中取代基具有以下含义：X氧或硫; R1氢; 卤素; 取代或未取代的C 1 -C 6烷基，苄基，环烷基，烯基，炔基，苯基，苯氧基或苯硫基; 烷氧基烷硫基卤代烷氧基卤代烷硫基; 或取代或未取代的五元或六元杂环基; R2甲酰基，4,5-二氢恶唑-2-基或-COYR 5; Y氧或硫; R5氢; 环烷基取代或未取代的烷基，苯基，苄基，烯基，环烯基或炔基; 取代或未取代的5或6元杂环基; 邻苯二甲酰亚氨基四氢邻苯二甲酰亚胺琥珀酰亚胺马来西亚一个阳离子; 或-N = CR 6 R 7; R6，R7氢; 烷基; 环烷基苯基; 呋喃基或一起形成4至7个成员的亚甲基链; R3氢或取代或未取代的烷基或环烷基; R4羟基烷氧基取代或未取代的烷基，环烷基，烯基，炔基，苯基或萘基; 取代或未取代的5或6元杂环基; 或者R 3和R 4一起是 - （CH 2）n -Yp-（CH 2）q - ，其中n和q是1,2或3，p是0或1，Y是氧，硫或N-甲基，或形成式（（CH2）3-CO-）及其环境耐受盐的基团，当R1为3-吡啶基时，式Ib中的X不为硫，R2为CO2CH2CH3或R3为氢，式Ia中的X为硫，并且当YR 5是OH时，R 1不是噻吩-2-基，R 3是氢，R 4是甲基，制备这种化合物的方法和含有式Ia或Ib化合物的除草剂作为活性成分。

27. 发明授权

US5262387A Pyridine derivatives and their use for controlling undesirable plant growth 失效
标题翻译：吡啶衍生物及其用于控制不希望的植物生长的用途
公开(公告)号：US5262387A
公开(公告)日：1993-11-16
申请号：US783310
申请日：1991-11-20
申请人： Gerhard Hamprecht , Norbert Goetz , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Gerhard Hamprecht , Norbert Goetz , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/40 , A01N43/90 , C07D213/81 , C07D213/82 , C07D471/04
CPC分类号： C07D213/81 , A01N43/40 , A01N43/90 , C07D213/82 , C07D471/04
摘要： Pyridine derivatives of the formulae ##STR1## wherein W, X, Y and Z are each C--R.sup.4, N or N.fwdarw.O, with the proviso that the ring contains only one heteroatom, and the substituents R.sup.1, R.sup.2 and R.sup.3 have the following meanings:R.sup.1 is alkoxy, substituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted alkenyl, or substituted or unsubstituted alkynyl,R.sup.2 is hydrogen,R.sup.3 is formyl, 4,5-dihydrooxazol-2-yl or --CO--A--R.sup.5 or --CO--NR.sup.6.sup.R.sup.7, whereR.sup.4 is halogen, nitro, cyano, substituted or unsubstituted alkyl, substituted or unsubstituted benzyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted alkenyl, substituted or unsubstituted alkynyl, alkoxy, alkylthio, haloalkoxy, haloalkylthio, alkenyloxy, alkynyloxy, alkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, substituted or unsubstituted phenoxy or phenylthio, a substituted or unsubstituted 5- or 6-membered heterocyclic radical having one or two heteroatoms selected from the group consisting of oxygen, sulfur and nitrogen, or is substituted or unsubstituted phenyl,A is oxygen or sulfur,R.sup.5 is hydrogen, substituted or unsubstituted alkyl, substituted or unsubstituted benzyl, cycloalkyl, substituted or unsubstituted phenyl,one equivalent of a cation or the radical --N.dbd.CR.sup.8 R.sup.9 andR.sup.6 and R.sup.7 are hydrogen or alkyl or together denote a methylene chain having 4 or 5 members,their agriculturally utilizable salts, and their use for controlling unwanted plant growth.
摘要翻译：其中W，X，Y和Z各自为C-R 4，N或N-> O的吡啶衍生物，条件是环仅含有一个杂原子，并且取代基R 1，R 2和 R3具有以下含义：R 1是烷氧基，取代或未取代的烷基，取代或未取代的环烷基，取代或未取代的烯基，或取代或未取代的炔基，R 2是氢，R 3是甲酰基，4,5-二氢恶唑-2-基或 - CO-A-R5或-CO-NR6R7，其中R4是卤素，硝基，氰基，取代或未取代的烷基，取代或未取代的苄基，取代或未取代的环烷基，取代或未取代的烯基，取代或未取代的炔基，烷氧基，烷硫基，卤代烷氧基卤代烷硫基，烯氧基，炔氧基，烷基亚磺酰基，烷基磺酰基，卤代烷基磺酰基，取代或未取代的苯氧基或苯硫基，取代或未取代的具有一个或两个选自基团的杂原子的5-或6-元杂环基氧，硫和氮的取代基，或者是取代或未取代的苯基，A是氧或硫，R5是氢，取代或未取代的烷基，取代或未取代的苄基，环烷基，取代或未取代的苯基，1当量的阳离子或基团 -N = CR8R9，R6和R7是氢或烷基或一起表示具有4或5个成员的亚甲基链，它们的农业上可利用的盐，以及它们用于控制不想要的植物生长的用途。

28. 发明授权

US5258356A Substituted 1,8-naphthyridines, their preparation and their use as antidotes 失效
标题翻译：取代的1,8-萘啶，其制备及其用作解毒剂
公开(公告)号：US5258356A
公开(公告)日：1993-11-02
申请号：US13202
申请日：1993-02-01
申请人： Thomas Saupe , Peter Schaefer , Norbert Meyer , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Thomas Saupe , Peter Schaefer , Norbert Meyer , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N25/32 , C07D471/04
CPC分类号： C07D471/04 , A01N25/32
摘要： A combination of a variety of herbicides with safening agents which are substituted 1,8-naphthyridines of the formula ##STR1## where R.sup.1 is mercapto, hydroxyl, halogen, benzylthio, amino or NR.sup.2 R.sup.3, whereR.sup.2 is a group ##STR2## where A is C.sub.1 -C.sub.8 -alkyl, R.sup.3 is hydrogen, XR.sup.4, where X is oxygen or sulfur and R.sup.4 is C.sub.1 -C.sub.12 -alkyl,R.sup.5 and R.sup.7 are each hydrogen, C.sub.1 -C.sub.12 -alkyl, hydroxyl, halogen, mercapto, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, dialkylamino where each alkyl is of 1 to 6 carbon atoms, phenoxy or phenylthio, halo-(C.sub.1 -C.sub.3)-alkyl, C.sub.1 -C.sub.4 -alkoxy-(C.sub.1 -C.sub.3)-alkyl, andR.sup.6 is hydrogen, C.sub.1 -C.sub.12 -alkyl, carboxyl or C.sub.1 -C.sub.4 -alkoxycarbonyl or the plant-tolerated salts thereof.
摘要翻译：各种除草剂与安全剂的组合，其为R1为巯基，羟基，卤素，苄硫基，氨基或NR2R3的式VIII取代的1,8-萘啶，其中R2为基团，其中A 是C 1 -C 8 - 烷基，R 3是氢，XR 4，其中X是氧或硫，R 4是C 1 -C 12烷基，R 5和R 7各自是氢，C 1 -C 12烷基，羟基，卤素，巯基，C 1 -C 4 - 烷氧基，C 1 -C 4烷氧基 - （C 1 -C 3） - 烷基，和C 1 -C 4 - 烷氧基 - （C 1 -C 3） - 烷基， R6是氢，C1-C12-烷基，羧基或C1-C4-烷氧基羰基或其植物耐受的盐。

29. 发明授权

US5201934A Carboxamides and their use as herbicides 失效
标题翻译：羧甲酰胺及其作为除草剂的用途
公开(公告)号：US5201934A
公开(公告)日：1993-04-13
申请号：US592287
申请日：1990-10-03
申请人： Peter Muenster , Gerd Steiner , Wolfgang Freund , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Peter Muenster , Gerd Steiner , Wolfgang Freund , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/08 , A01N43/10 , A01N43/28 , A01N43/78 , C07D307/68 , C07D333/38 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D409/14 , C07D413/04 , C07D417/12 , C07D417/14 , C07D495/04
CPC分类号： C07D407/12 , A01N43/08 , A01N43/10 , A01N43/28 , C07D307/68 , C07D333/38 , C07D409/12 , C07D417/12
摘要： Carboxamides of the formulae Ia to Ic ##STR1## where X is oxygen or sulfur;R.sup.1 is hydrogen or substituted or unsubstituted cycloalkyl or alkyl;R.sup.2 is hydroxy, alkoxy, cyanoalkyl, substituted or unsubstituted alkenyl, alkynyl, phenyl or naphthyl, or one of the groups stated for R.sup.1 ;R.sup.3 and R.sup.4 are nitro, cyano, halogen, substituted or unsubstituted amino, alkoxy, alkylthio, substituted or unsubstituted alkenyl, alkynyl, phenyl, phenoxy or phenylthio, or one of the groups stated for R.sup.1 ;R.sup.5 is formyl, 4,5-dihydrooxazol-2-yl or COYR.sup.6 (Y.dbd.O,S);R.sup.6 is hydrogen, cycloalkyl, substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkenyl or phenyl,phthalimido, tetrahydrophthalimido, succinimido, maleimido, benzotriazolyl ora group --N.dbd.CR.sup.7 R.sup.8, whereR.sup.7 and R.sup.8 are hydrogen or alkyl, and R.sup.8 may also be cycloalkyl, phenyl, or R.sup.7 and R.sup.8 together form a 4- to 7-membered alkylene chain;and if R.sup.5 is carboxyl, methoxycarbonyl or ethoxycarbonyl and R.sup.2 is hydrogen, R.sup.3 is not hydrogen and R.sup.4 is not hydrogen or methyl, and if R.sup.5 is carboxyl, methoxycarbonyl or ethoxycarbonyl and R.sup.4 is hydrogen, R.sup.3 is not hydrogen or R.sup.2 is not one of the following groups: hydrogen, C.sub.1 -C.sub.4 -alkyl, phenyl, 2-(3,4-dimethoxyphenyl)ethyl or 2,5-dichlorothien-3-yl;processes for the manufacture of compounds I and herbicidal agents containing them.
摘要翻译：式Ia至Ic的酰胺酰胺其中X是氧或硫; R1是氢或取代或未取代的环烷基或烷基; R2是羟基，烷氧基，氰基烷基，取代或未取代的链烯基，炔基，苯基或萘基，或为R1所述的一个基团; R3和R4是硝基，氰基，卤素，取代或未取代的氨基，烷氧基，烷硫基，取代或未取代的烯基，炔基，苯基，苯氧基或苯硫基，或为R1表示的基团之一; R5是甲酰基，4,5-二氢恶唑-2-基或COYR 6（Y = O，S）; R 6是氢，环烷基，取代或未取代的烷基，烯基，炔基，环烯基或苯基，邻苯二甲酰亚氨基，四氢邻苯二甲酰亚胺基，琥珀酰亚胺基，马来酰亚胺基，苯并三唑基或基团-N = CR 7 R 8，其中R 7和R 8是氢或烷基，环烷基，苯基或R7和R8一起形成4-至7-元亚烷基链; 如果R5是羧基，甲氧基羰基或乙氧基羰基，R2是氢，R3不是氢，R4不是氢或甲基，如果R5是羧基，甲氧基羰基或乙氧基羰基，R4是氢，R3不是氢或R2不是以下基团：氢，C 1 -C 4 - 烷基，苯基，2-（3,4-二甲氧基苯基）乙基或2,5-二氯噻吩-3-基; 制备化合物I和含有它们的除草剂的方法。

30. 发明授权

US5171353A Sulfonamides 失效
标题翻译：磺胺
公开(公告)号：US5171353A
公开(公告)日：1992-12-15
申请号：US521032
申请日：1990-05-09
申请人： Klaus Fischer , Horst Mayer , Klaus Ditrich , Gerhard Hamprecht , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Klaus Fischer , Horst Mayer , Klaus Ditrich , Gerhard Hamprecht , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/90 , C07D471/04 , C07D473/06 , C07D473/40
CPC分类号： C07D471/04 , A01N43/90 , C07D473/06 , C07D473/40
摘要： Sulfonamides of the general formula I ##STR1## where R.sup.1 is hydrogen of C.sub.1 -C.sub.4 -alkyl,R.sup.2 is hydrogen or substituted or unsubstituted C.sub.1 -C.sub.6 -alkyl; C.sub.3 -C.sub.4 -alkenyl; C.sub.3 -C.sub.4 -alkynyl or substituted or unsubstituted saturated or singly unsaturated 5- to 7- membered heteroaryl;R.sup.3 and R.sup.4 are halogen; substituted or unsubstituted C.sub.1 -C.sub.4 -alkoxy C.sub.1 -C.sub.4 -alkylthio, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -alkenyloxy, C.sub.2 -C.sub.6 -alkenylthio, C.sub.2 -C.sub.6 -alkynyl, C.sub.2 -C.sub.6 -alkynyloxy, C.sub.2 -C.sub.6 -alkynylthio, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -cycloalkylthio, C.sub.5 -C.sub.6 -cycloalkenyl, C.sub.3 -C.sub.6 -cycloalkoxy, C.sub.5 -C.sub.6 -cycloalkenyloxy, C.sub.5 -C.sub.6 -cycloalkenylthio, phenyl, phenoxy, phenylthio, benzyl, benzyloxy or benzylthio;the group given for R.sup.2, or NR.sup.7 R.sup.8, where R.sup.7 and R.sup.8 are hydrogen, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.5 -C.sub.6 -cycloalkenyl, substituted or unsubstituted phenyl and/or benzyl bedeuten, or issubstituted or unsubstituted C.sub.4 -C.sub.6 -alkylene which may be interrupted or oxygen, sulfur or nitrogen;X is nitrogen or .dbd.CR.sup.5 14 ,where R.sup.5 is one of the radicals R.sup.3,n is 0 or 1 andA is substituted or unsubstituted mono- or dinuclear aryl containing one or two nitrogen, oxygen and/or sulfur atoms,and their agriculturally useful salts, and herbicidal and growth-regulating agents containing them.
摘要翻译：其中R 1是C 1 -C 4 - 烷基的氢，R 2是氢或被取代或未被取代的C 1 -C 6 - 烷基的磺酰胺， C3-C4-烯基; C3-C4-炔基或取代或未取代的饱和或单不饱和5-至7-元杂芳基; R3和R4是卤素; 取代或未取代的C 1 -C 4 - 烷氧基C 1 -C 4 - 烷硫基，C 2 -C 6 - 链烯基，C 2 -C 6 - 烯氧基，C 2 -C 6 - 烯硫基，C 2 -C 6炔基，C 2 -C 6 - 炔氧基，C 2 -C 6 - 炔硫基， C 3 -C 6环烷基，C 3 -C 6环烷硫基，C 5 -C 6环环烯基，C 3 -C 6环烷氧基，C 5 -C 6环环烯氧基，C 5 -C 6环环硫基，苯基，苯氧基，苯硫基，苄基，苄氧基或苄硫基; R2或NR7R8的基团，其中R7和R8是氢，C1-C6-烷基，C3-C6-烯基，C3-C6-炔基，C3-C6-环烷基，C5-C6-环烯基，取代或未取代的苯基或/或苄基叔丁基醚，或者是可被中断的取代或未取代的C 4 -C 6亚烷基或氧，硫或氮; X是氮或= CR514，其中R5是基团R3之一，n是0或1，A是含有一个或两个氮，氧和/或硫原子的取代或未取代的单核或二核芳基及其农业上有用的盐，和含有它们的除草和生长调节剂。

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