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11. 发明授权

US5135927A Microbicidal composition 失效
标题翻译：杀菌组合物
公开(公告)号：US5135927A
公开(公告)日：1992-08-04
申请号：US617702
申请日：1990-11-26
申请人： Werner Topfl , Robert Nyfeler , Werner Fory
发明人： Werner Topfl , Robert Nyfeler , Werner Fory
IPC分类号： A01N43/78 , C07D277/56 , C07D277/60 , C07D417/06 , C07D417/12 , C07D493/04 , C07F9/6539
CPC分类号： C07D277/60 , A01N43/78 , C07D277/56 , C07D417/06 , C07D417/12 , C07D493/04 , C07F9/6539
摘要： A microbicidal composition contains as active ingredient 2-chloro-4-trifluoromethylthiazol-5-carboxylic acid derivatives of the formula I ##STR1## R is an organic radical with up to 40 carbon atoms, which optionally contains nitrogen, oxygen or sulfur atoms and which can be transformed by hydrolosis or oxydation into the directly to the thiazol ring bound carboxyl rest.These compounds have good microbicidal activity and are used for the control and prevention of infestation of plants by phytophathogenic microorganismes.
摘要翻译：杀微生物组合物含有作为活性成分的式I的2-氯-4-三氟甲基噻唑-5-羧酸衍生物（I）R是具有至多40个碳原子的有机基团，其任选地含有氮，氧或硫原子，其可以通过水痘病毒或氧化反应直接转化成噻唑环结合的羧基。这些化合物具有良好的杀微生物活性，用于通过植物致病性微生物控制和预防植物侵染。

12. 发明授权

US5342823A Sulfonylureas 失效
标题翻译：磺脲类
公开(公告)号：US5342823A
公开(公告)日：1994-08-30
申请号：US18603
申请日：1993-02-17
申请人： Rainer Kuhlmeyer , Werner Topfl , Werner Fory
发明人： Rainer Kuhlmeyer , Werner Topfl , Werner Fory
IPC分类号： A01N47/36 , C07D213/80 , C07D231/18 , C07D405/12 , C07D405/14 , C07D409/12 , C07D409/14 , C07D521/00 , F16N11/04 , F16N11/08 , C07D407/14 , A01N43/54
CPC分类号： C07D521/00 , A01N47/36 , C07D405/12 , C07D409/12 , F16N11/04 , F16N11/08 , F16N2230/10
摘要： N-Arylsulfonyl-N'-pyrimidinyl-and N'-triazinylureas of formula I ##STR1## wherein Q is ##STR2## R is hydrogen or methyl; R.sub.1 is hydrogen, fluoro, chloro, C.sub.1 -C.sub.4 alkyl or methoxy;R.sub.2 is hydrogen, fluoro or chloro;R.sub.3, R.sub.4, R.sub.5, R.sub.6 and R.sub.7 are each independently of one another hydrogen or C.sub.1-C.sub.4 alkyl;R.sub.8, R.sub.9, R.sub.10, R.sub.11 and R.sub.12 are each independently of one another hydrogen or C.sub.1 -C.sub.4 alkyl;R.sub.13, R.sub.14, R.sub.15, R.sub.16 and R.sub.17 are each independently of one another hydrogen or C.sub.1 -C.sub.4 alkyl;Z is methyl or 2-pyridyl;E is methine or nitrogen;X is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 haloalkylthio, C.sub.1 -C.sub.4 alkylthio,C.sub.2 -C.sub.5 alkoxyalkyl, C.sub.2 -C.sub.5 alkoxyalkoxy, C.sub.2 -C.sub.5 alkylthioalkyl or cyclopropyl;Y is C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 haloalkylthio,C.sub.1 -C.sub.4 alkylthio, halogen, C.sub.2 -C.sub.5 alkoxyalkyl, C.sub.2 -C.sub.5 alkoxyalkoxy, amino, C.sub.1 -C.sub.3 alkylamino or di-(C.sub.1 -C.sub.3 alkyl)amino;and the salts of these compounds with amines, alkali metal or alkaline earth metal bases or with quaternary ammonium bases, have good pre-and postemergence selective herbicidal and growth regulating properties.
摘要翻译：（Q）（Q 3）（Q 3）（Q 3）R 3是氢或甲基; R 3是氢或甲基; R 3是氢或甲基。 R 1是氢，氟，氯，C 1 -C 4烷基或甲氧基; R2是氢，氟或氯; R3，R4，R5，R6和R7各自独立地为氢或C1-C4烷基; R8，R9，R10，R11和R12各自独立地为氢或C1-C4烷基; R 13，R 14，R 15，R 16和R 17各自独立地为氢或C 1 -C 4烷基; Z是甲基或2-吡啶基; E是次甲基或氮; X是C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基，C 1 -C 4卤代烷硫基，C 1 -C 4烷硫基，C 2 -C 5烷氧基烷基，C 2 -C 5烷氧基烷氧基，C 2 -C 5烷硫基烷基或环丙基; Y是C1-C4烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4卤代烷基，C1-C4卤代烷硫基，C1-C4烷硫基，卤素，C2-C5烷氧基烷基，C2-C5烷氧基烷氧基，氨基，C1-C3烷基氨基或二 - （C1-C3烷基）氨基 ; 并且这些化合物与胺，碱金属或碱土金属碱或季铵碱的盐具有良好的芽前和芽后选择性除草和生长调节性质。

13. 发明授权

US4992434A Microbicidal composition 失效
标题翻译：杀菌组合物
公开(公告)号：US4992434A
公开(公告)日：1991-02-12
申请号：US336166
申请日：1989-04-11
申请人： Werner Topfl , Robert Nyfeler , Werner Fory
发明人： Werner Topfl , Robert Nyfeler , Werner Fory
IPC分类号： A01N43/78 , C07D277/56 , C07D277/60 , C07D417/06 , C07D417/12 , C07D493/04 , C07F9/6539
CPC分类号： C07D277/60 , A01N43/78 , C07D277/56 , C07D417/06 , C07D417/12 , C07D493/04 , C07F9/6539
摘要： A microbicidal compostion contains as active ingredient 2-chloro-4-trifluoromethylthiazol-5-carbonic acid derivatives of the formula I ##STR1## R is organic radical with up to 40 carbon atoms, which optionally contains nitrogen, oxygen or sulfur atoms and which can be transformed by hydrolosis or oxydation into the directly to the thiazol ring bound carboxyl rest. These compounds have good microbicidal activity and are used for the control and prevention of infestation of plants by phytophathogenic microorganisms.
摘要翻译：杀微生物组合物含有作为活性成分的式I的2-氯-4-三氟甲基噻唑-5-碳酸衍生物（I）R是具有多达40个碳原子的有机基团，其任选地含有氮，氧或硫原子并且其可以通过水痘病毒或氧化反应直接转化成噻唑环结合的羧基。这些化合物具有良好的杀菌活性，用于通过植物致病微生物控制和预防植物侵染。

14. 发明授权

US4664695A N-phenylsulfonyl-N'-pyrimidinylureas as herbicides and plant growth regulants 失效
标题翻译： N-苯基磺酰基-N'-嘧啶基脲作为除草剂和植物生长调节剂
公开(公告)号：US4664695A
公开(公告)日：1987-05-12
申请号：US717637
申请日：1985-03-29
申请人： Rolf Schurter , Rudolph C. Thummel , Werner Topfl , Willy Meyer , Dieter Durr
发明人： Rolf Schurter , Rudolph C. Thummel , Werner Topfl , Willy Meyer , Dieter Durr
IPC分类号： C07D249/16 , A01N47/36 , C07C67/00 , C07C301/00 , C07C311/39 , C07D207/38 , C07D207/40 , C07D207/404 , C07D239/42 , C07D239/46 , C07D239/47 , C07D251/16 , C07D251/18 , C07D251/22 , C07D251/46 , C07D251/52 , C07D275/02 , C07D521/00 , C07D239/69 , A01N43/54 , C07D401/12 , C07D417/12
CPC分类号： C07D207/404 , A01N47/36 , C07D207/38 , C07D239/42 , C07D239/47 , C07D251/16 , C07D275/02 , C07D521/00
摘要： N-Phenylsulfonyl-N'-pyrimidinylureas of the general formula I ##STR1## and the salts of these compounds with amines, alkali metal bases or alkaline earth metal bases or with quaternary ammonium bases, have good selective herbicidal and growth regulating properties when applied pre- and postemergence.The symbols in formula I have the following meanings:R.sub.1 is hydrogen, halogen, nitro, cyano, or an alkyl, alkoxy, alkylthio, alkylsulfonyl, alkylcarbonyl, alkylcarbamoyl or alkoxycarbonyl group, each unsubstituted or substituted by halogen or alkoxy,R.sub.2 is hydrogen, halogen, alkyl, or an alkyl, alkoxy or alkylthio group, each unsubstituted or substituted by halogen or alkoxy,R.sub.3 is alkyl, haloalkyl, alkoxy or haloalkoxy,R.sub.4 is hydrogen, halogen, R.sub.3, alkylamino or dialkylamino,R.sub.5 is hydrogen, alkyl or alkoxy, andX is an alkenylamino, cycloalkylamino or cycloalkenylamino group which may be further substituted, or is a carbamoylamido or sulfonylamino group as defined in the description, or is a 5- or 6-membered saturated heterocyclic ring system which is bonded through the nitrogen atom and which may contain a further oxygen, sulfur or nitrogen atom in the ring and must contain at least one oxo group.
摘要翻译：具有通式I（I）的N-苯基磺酰基-N'-嘧啶基和这些化合物与胺，碱金属碱或碱土金属碱或季铵碱的盐具有良好的选择性除草和生长调节性质应用于芽前和芽后。式I中的符号具有以下含义：R 1是氢，卤素，硝基，氰基或烷基，烷氧基，烷硫基，烷基磺酰基，烷基羰基，烷基氨基甲酰基或烷氧基羰基，各自未被取代或被卤素或烷氧基取代，卤素，烷基或烷基，烷氧基或烷硫基，各自未被取代或被卤素或烷氧基取代，R3是烷基，卤代烷基，烷氧基或卤代烷氧基，R4是氢，卤素，R3，烷基氨基或二烷基氨基，R5是氢，烷基或烷氧基，X是可以被进一步取代的链烯基氨基，环烷基氨基或环烯基氨基，或者是说明书中定义的氨基甲酰氨基或磺酰氨基，或是通过氮键合的5或6元饱和杂环体系原子，并且其可以在环中含有另外的氧，硫或氮原子，并且必须含有至少一个氧代基团。

15. 发明授权

US4632695A N-phenylsulfonyl-N'-triazinylureas as herbicides and plant growth regulants 失效
标题翻译： N-苯基磺酰基-N'-三嗪基脲作为除草剂和植物生长调节剂
公开(公告)号：US4632695A
公开(公告)日：1986-12-30
申请号：US806168
申请日：1985-12-06
申请人： Rolf Schurter , Rudolph C. Thummel , Werner Topfl , Willy Meyer , Dieter Durr
发明人： Rolf Schurter , Rudolph C. Thummel , Werner Topfl , Willy Meyer , Dieter Durr
IPC分类号： C07D249/16 , A01N47/36 , C07C67/00 , C07C301/00 , C07C311/39 , C07D207/38 , C07D207/40 , C07D207/404 , C07D239/42 , C07D239/46 , C07D239/47 , C07D251/16 , C07D251/18 , C07D251/22 , C07D251/46 , C07D251/52 , C07D275/02 , C07D521/00 , A01N43/66 , A01N43/70
CPC分类号： C07D207/404 , A01N47/36 , C07D207/38 , C07D239/42 , C07D239/47 , C07D251/16 , C07D275/02 , C07D521/00
摘要： N-Phenylsulfonyl-N'-triazinylureas of the general formula I ##STR1## and the salts of these compounds with amines, alkali metal bases or alkaline earth metal bases or with quaternary ammonium bases, have good selective herbicidal and growth regulating properties when applied pre- and postemergence. The symbols in formula I have the following meanings:R.sub.1 is hydrogen, halogen, nitro, cyano, or an alkyl, alkoxy, alkylthio, alkylsulfonyl, alkylcarbonyl, alkylcarbamoyl or alkoxycarbonyl group, each unsubstituted or substituted by halogen or alkoxy,R.sub.2 is hydrogen, halogen, alkyl, or an alkyl, alkoxy or alkylthio group, each unsubstituted or substituted by halogen or alkoxy,R.sub.3 is alkyl, haloalkyl, alkoxy or haloalkoxy,R.sub.4 is hydrogen, halogen, R.sub.3, alkylamino or dialkylamino,R.sub.5 is hydrogen, alkyl or alkoxy, andX is an alkenylamino, cycloalkylamino or cycloalkenylamino group which may be further substituted, or is a carbamoylamido or sulfonylamino group as defined in the description, or is a 5- or 6-membered saturated heterocyclic ring system which is bonded through the nitrogen atom and which may contain a further oxygen, sulfur or nitrogen atom in the ring and must contain at least one oxo group.
摘要翻译：具有通式I（I）的N-苯基磺酰基-N'-三嗪基和这些化合物与胺，碱金属碱或碱土金属碱或季铵碱的盐具有良好的选择性除草和生长调节性质应用于芽前和芽后。式I中的符号具有以下含义：R 1是氢，卤素，硝基，氰基或烷基，烷氧基，烷硫基，烷基磺酰基，烷基羰基，烷基氨基甲酰基或烷氧基羰基，各自未被取代或被卤素或烷氧基取代，卤素，烷基或烷基，烷氧基或烷硫基，各自未被取代或被卤素或烷氧基取代，R3是烷基，卤代烷基，烷氧基或卤代烷氧基，R4是氢，卤素，R3，烷基氨基或二烷基氨基，R5是氢，烷基或烷氧基，X是可以被进一步取代的链烯基氨基，环烷基氨基或环烯基氨基，或者是说明书中定义的氨基甲酰氨基或磺酰氨基，或是通过氮键合的5或6元饱和杂环体系原子，并且其可以在环中含有另外的氧，硫或氮原子，并且必须含有至少一个氧代基团。

16. 发明授权

US4685961A Herbicidal sulfonylureas 失效
标题翻译：除草磺酰脲类
公开(公告)号：US4685961A
公开(公告)日：1987-08-11
申请号：US699388
申请日：1985-02-07
申请人： Werner Topfl , Willy Meyer , Hans-Dieter Schneider
发明人： Werner Topfl , Willy Meyer , Hans-Dieter Schneider
IPC分类号： A01N47/36 , C07D239/42 , C07D239/46 , C07D239/48 , C07D239/52 , C07D249/08 , C07D251/52 , C07D403/12 , C07D521/00 , C07D239/69 , A01N43/54 , A01N43/707
CPC分类号： C07D239/42 , A01N47/36 , C07D231/12 , C07D233/56 , C07D239/47 , C07D239/48 , C07D239/52 , C07D249/08 , C07D251/52 , C07D403/12 , C07D521/00
摘要： Novel substituted N-sulfonyl-N'-pyrimidinylureas or N-sulfonyl-N'-triazinylureas of the formula I ##STR1## have good pre- and postemergence selective herbicidal and growth regulating properties.In this formula E is nitrogen or --CH.dbd., the group ##STR2## is a phenyl, naphthyl, furyl, thiophenyl, pyrrole or pyridinyl radical which is substituted in accordance with the definitions ofR.sup.1 and R.sup.2,R.sup.3 and R.sup.4 are hydrogen, lower alkyl or lower alkoxy, or one of R.sup.3 and R.sup.4 may also be halogen, lower alkenyl, lower haloalkenyl, lower haloalkoxy, amino, lower alkylamino, --CH(OCH.sub.3).sub.2, a cyclised ketal group or a saturated 5- to 7-membered heterocycle which is bound through the nitrogen atom,R.sup.5 is hydrogen, lower alkyl, lower haloalkyl, or an unsubstituted or substituted phenyl, benzyl or naphthyl radical, andR.sup.6 is an alkyl, acyl or acylamido radical which is bound through sulfur or a sulfinyl or sulfonyl group and is as defined in the description, or is a 5- to 7-membered heterocyclic amino radical which is bound through the nitrogen atom.These compounds are particularly suitable for selectively controlling weeds in crops of cereals.
摘要翻译：式I（I）的新型取代的N-磺酰基-N'-嘧啶基或N-磺酰基-N'-三嗪基脲具有良好的芽前和芽后选择性除草和生长调节性质。在该式中，E是氮或-CH =，根据R1和R2的定义被取代的苯基，萘基，呋喃基，噻吩基，吡咯基或吡啶基，R3和R4是氢，低级烷基或低级烷氧基，或者R 3和R 4中的一个也可以是卤素，低级链烯基，低级卤代烯基，低级卤代烷氧基，氨基，低级烷基氨基，-CH（OCH 3）2，环化的缩酮基或饱和的5-至7-元通过氮原子结合的杂环，R5是氢，低级烷基，低级卤代烷基或未取代或取代的苯基，苄基或萘基，R6是通过硫或亚磺酰基结合的烷基，酰基或酰基酰氨基，磺酰基，如描述中所定义，或是通过氮原子结合的5-至7-元杂环氨基。这些化合物特别适用于选择性地控制谷物作物中的杂草。

17. 发明授权

US4559078A Herbicidal and growth regulator phosphorus-containing N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N'-triazinylureas 失效
标题翻译：除草生长调节剂含磷的N-苯基磺酰基-N'-嘧啶基脲和N-苯基磺酰基-N'-三嗪基脲
公开(公告)号：US4559078A
公开(公告)日：1985-12-17
申请号：US562659
申请日：1983-12-19
申请人： Ludwig Maier , Willy Meyer , Konrad Oertle , Achim Roloff , Werner Topfl
发明人： Ludwig Maier , Willy Meyer , Konrad Oertle , Achim Roloff , Werner Topfl
IPC分类号： A01N57/16 , A01N57/08 , A01N57/24 , C07D521/00 , C07F9/30 , C07F9/32 , C07F9/38 , C07F9/40 , C07F9/53 , C07F9/6512 , C07F9/6521 , C07F9/65
CPC分类号： C07D521/00 , A01N57/08 , C07F9/304 , C07F9/3229 , C07F9/3808 , C07F9/3834 , C07F9/4006 , C07F9/4015 , C07F9/4021 , C07F9/4056 , C07F9/5325 , C07F9/65127 , C07F9/65217
摘要： Phosphorus-containing N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N'-triazinylureas of the formula ##STR1## and the salts of these compounds with amines, alkali or alkaline earth metal bases or quaternary ammonium bases have good pre-emergence and post-emergence selective herbicidal and growth-regulating properties.In this formula, X is a group ##STR2## Y is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, trifluoromethyl, C.sub.2 -C.sub.5, alkenyl, C.sub.2 -C.sub.5 -alkynyl, nitro, --COOR.sup.6 or --Q--R.sup.6, Z is nitrogen or the methine group, E is oxygen or sulfur, R.sup.1 is hydrogen or C.sub.1 -C.sub.5 -alkyl and R.sup.2 and R.sup.3 independently of one another are C.sub.1 -C.sub.3 -alkyl, C.sub.1 -C.sub.3 -alkoxy, C.sub.1 -C.sub.3 -halogenoalkyl, C.sub.1 -C.sub.3 -halogenoalkoxy, cyclopropyl, amino, methylamino or dimethylamino, and A is oxygen, sulfur, C.sub.1 -C.sub.5 -alkylene, C.sub.2 -C.sub.5 -alkenylene, C.sub.1 -C.sub.5 -halogenoalkylene or --NR.sup.7 --(CH.sub.2).sub.m --; --CH.sub.2 --NH--(CH.sub.2).sub.m --; --(CH.sub.2).sub.m --NR.sup.7 -- or --O--(CH.sub.2).sub.p --, --S--(CH.sub.2).sub.p --, --(CH.sub.2).sub.p --O-- or --(CH.sub.2).sub.p --S--, n is zero or one, G is oxygen or sulfur, R.sup.4 is C.sub.1 -C.sub.5 -alkoxy, C.sub.1 -C.sub.5 -halogenoalkoxy, C.sub.1 -C.sub.5 -alkylthio, C.sub.1 -C.sub.5 -alkyl, C.sub.1 -C.sub.5 -halogenoalkyl, phenyl or hydroxyl, R.sup.5 is hydrogen, C.sub.1 -C.sub.5 -alkoxy, C.sub.1 -C.sub.5 -halogenoalkoxy, C.sub.1 -C.sub.5 -alkylthio, C.sub.1 -C.sub.5 -alkyl or hydroxyl, R.sup.6 is C.sub.1 -C.sub.5 -alkyl, C.sub.1 -C.sub.5 -halogenoalkyl or C.sub.2 -C.sub.6 -alkoxyalkyl, Q is oxygen, sulfur, --SO-- or --SO.sub.2 --, R.sup.7 is hydrogen, C.sub.1 -C.sub.5 -alkyl, phenyl, benzyl or phenyl which is substituted by C.sub.1 -C.sub.5 -alkyl, halogen or nitro, m is a number from zero to three, p is a number from zero to two and r is one or two.
摘要翻译：具有式“IMAGE”的含磷N-苯基磺酰基-N'-嘧啶基脲和N-苯基磺酰基-N'-三嗪基脲和这些化合物与胺，碱金属或碱土金属碱或季铵碱的盐具有良好的出苗前和出苗后选择性除草和生长调节性质。在该式中，X是基团Y是氢，卤素，C 1 -C 5 - 烷基，三氟甲基，C 2 -C 5，烯基，C 2 -C 5炔基，硝基，-COOR 6或-Q-R 6，Z是氮或次甲基，E是氧或硫，R1是氢或C1-C5-烷基，R2和R3彼此独立地是C1-C3-烷基，C1-C3-烷氧基，C1-C3-卤代烷基，C1-C3 - 卤代烷氧基，环丙基，氨基，甲基氨基或二甲基氨基，A是氧，硫，C1-C5-亚烷基，C2-C5-亚烯基，C1-C5-卤代亚烷基或-NR7-（CH2）m- -CH 2 -NH-（CH 2）m - ; - （CH 2）m -NR 7 - 或-O-（CH 2）p - ， - S-（CH 2）p - ， - （CH 2）p O-或 - （CH 2）p -S-，n为0或1，G为氧或硫，R4是C1-C5-烷氧基，C1-C5-卤代烷氧基，C1-C5-烷硫基，C1-C5-烷基，C1-C5-卤代烷基，苯基或羟基，R5是氢，C1-C5-烷氧基，C1 -C 5 - 卤代烷氧基，C 1 -C 5 - 烷硫基，C 1 -C 5 - 烷基或羟基，R 6是C 1 -C 5 - 烷基，C 1 -C 5 - 卤代烷基或C 2 -C 6 - 烷氧基烷基，Q是氧，硫，-SO-或 - SO 2 - ，R 7为氢，C 1 -C 5 - 烷基，苯基，苄基或被C 1 -C 5 - 烷基，卤素或硝基取代的苯基，m为0至3的数，p为0至2的数， r是一两个。

18. 发明授权

US4940792A Herbicidal sulfonylureas 失效
标题翻译：除草磺酰脲类
公开(公告)号：US4940792A
公开(公告)日：1990-07-10
申请号：US128761
申请日：1987-12-04
申请人： Werner Topfl , Willy Meyer , Hans-Dieter Schneider
发明人： Werner Topfl , Willy Meyer , Hans-Dieter Schneider
IPC分类号： A01N47/36 , C07D239/42 , C07D239/46 , C07D239/48 , C07D239/52 , C07D249/08 , C07D251/52 , C07D403/12 , C07D521/00
CPC分类号： C07D239/42 , A01N47/36 , C07D231/12 , C07D233/56 , C07D239/47 , C07D239/48 , C07D239/52 , C07D249/08 , C07D251/52 , C07D403/12 , C07D521/00
摘要： Novel substituted N-sulfonyl-N'-pyrimidinylureas or N-sulfonyl-N'-triazinylureas of the formula I ##STR1## have good pre- and postemergence selective herbicidal and growth regulating properties.In this formulaE is nitrogen or --CH.dbd.,the group ##STR2## is a phenyl, naphthyl, furyl, thiophenyl, pyrrole or pyridinyl radical which is substituted in accordance with the definitions ofR.sup.1 and R.sup.2,R.sup.3 and R.sup.4 are hydrogen, lower alkyl or lower alkoxy, or one of R.sup.3 and R.sup.4 may also be halogen, lower alkenyl, lower haloalkenyl, lower haloalkoxy, amino, lower alkylamino, --CH(OCH.sub.3).sub.2, a cyclized ketal group or a saturated 5- or 7-membered heterocycle which is bound through the nitrogen atom,R.sup.5 is hydrogen, lower alkyl, lower haloalkyl, or an unsubstituted or substituted phenyl, benzyl or naphthyl radical, andR.sup.6 is an alkyl, acyl or acylamido radical which is bound through sulfur or a sulfinyl or sulfonyl group and is as defined in the description, or is a 5- to 7-membered heterocyclic amino radical which is bound through the nitrogen atom.These compounds are particularly suitable for selectively controlling weeds in crops of cereals.

19. 发明授权

US4764203A Herbicidal sulfonylureas 失效
标题翻译：除草磺酰脲类
公开(公告)号：US4764203A
公开(公告)日：1988-08-16
申请号：US53912
申请日：1987-05-26
申请人： Werner Topfl , Willy Meyer , Hans-Dieter Schneider
发明人： Werner Topfl , Willy Meyer , Hans-Dieter Schneider
IPC分类号： A01N47/36 , C07D239/42 , C07D239/46 , C07D239/48 , C07D239/52 , C07D249/08 , C07D251/52 , C07D403/12 , C07D521/00 , A01N43/66 , C07D251/18 , C07D251/46 , C07D251/70
CPC分类号： C07D239/42 , A01N47/36 , C07D231/12 , C07D233/56 , C07D239/47 , C07D239/48 , C07D239/52 , C07D249/08 , C07D251/52 , C07D403/12 , C07D521/00
摘要： Novel substituted N-sulfonyl-N'-pyrimidinylureas or N-sulfonyl-N'-triazinylureas of the formula I ##STR1## have good pre- and postemergence selective herbicidal and growth regulating properties.In this formulaE is nitrogen or --CH.dbd.,the group ##STR2## is a phenyl, naphthyl, furyl, thiophenyl, pyrrole or pyridinyl radical which is substituted in accordance with the definitions of R.sup.1 and R.sup.2,R.sup.3 and R.sup.4 are hydrogen, lower alkyl or lower alkoxy, or one of R.sup.3 and R.sup.4 may also be halogen, lower alkenyl, lower haloalkenyl, lower haloalkoxy, amino, lower alkylamino, --CH(OCH.sub.3).sub.2, a cyclized ketal group or a saturated 5- to 7-membered heterocycle which is bound through the nitrogen atom,R.sup.5 is hydrogen, lower alkyl, lower haloalkyl, or an unsubstituted or substituted phenyl, benzyl or naphthyl radical, andR.sup.6 is an alkyl, acyl or acylamido radical which is bound through sulfur or a sulfinyl or sulfonyl group and is as defined in the description, or is a 5- to 7-membered heterocyclic amino radical which is bound through the nitrogen atom.These compounds are particularly suitable for selectively controlling weeds in crops of cereals.
摘要翻译：式I（I）的新型取代的N-磺酰基-N'-嘧啶基或N-磺酰基-N'-三嗪基脲具有良好的芽前和芽后选择性除草和生长调节性质。在该式中，E是氮或-CH =，根据R1和R2的定义被取代的苯基，萘基，呋喃基，噻吩基，吡咯基或吡啶基，R3和R4是氢，低级烷基或低级烷氧基，或者R 3和R 4中的一个也可以是卤素，低级烯基，低级卤代烯基，低级卤代烷氧基，氨基，低级烷基氨基，-CH（OCH 3）2，环状缩酮基或饱和的5-至7-元通过氮原子结合的杂环，R5是氢，低级烷基，低级卤代烷基或未取代或取代的苯基，苄基或萘基，R6是通过硫或亚磺酰基结合的烷基，酰基或酰基酰氨基，磺酰基，如描述中所定义，或是通过氮原子结合的5-至7-元杂环氨基。这些化合物特别适用于选择性地控制谷物作物中的杂草。

20. 发明授权

US4551531A 4-Difluoromethoxy-2-amino-pyrimidines 失效
标题翻译： 4-二氟甲氧基-2-氨基 - 嘧啶
公开(公告)号：US4551531A
公开(公告)日：1985-11-05
申请号：US641140
申请日：1984-07-26
申请人： Willy Meyer , Karl Gass , Werner Topfl , Rolf Schurter , Georg Pissiotas
发明人： Willy Meyer , Karl Gass , Werner Topfl , Rolf Schurter , Georg Pissiotas
IPC分类号： C07D239/47 , A01N47/36 , A01P13/00 , C07D239/42 , C07D239/46 , C07D239/48 , C07D239/52 , C07D239/54 , C07D239/545 , C07D239/56 , C07D251/46 , C07D521/00
CPC分类号： C07D239/47 , A01N47/36 , C07D239/48 , C07D239/52 , C07D239/545 , C07D239/56 , C07D251/46 , C07D521/00
摘要： The invention relates to N-arylsulfonyl-N'-pyrimidinyl ureas of the general formula ##STR1## and to the salts thereof with amines, alkali metal hydroxides or alkaline earth metal hydroxides or with quaternary ammonium bases. These compounds have good pre- and postemergence selective herbicidal and growth regulating properties.In the formula, R.sub.18 is hydrogen, alkyl or alkoxy, X is an unsubstituted or substituted phenyl radical or an unsubstituted or substituted naphthyl radical, Y is C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkoxy, C.sub.1 -C.sub.3 alkylthio, C.sub.2 -C.sub.3 alkoxyalkyl, halogen or an unsubstituted amino group and Z is oxygen or sulfur.
摘要翻译：本发明涉及通式为（I）的N-芳基磺酰基-N'-嘧啶基脲，以及其与胺，碱金属氢氧化物或碱土金属氢氧化物或季铵碱的盐。这些化合物具有良好的芽前和芽后选择性除草和生长调节性质。式中，R 18为氢，烷基或烷氧基，X为未取代或取代的苯基或未取代或取代的萘基，Y为C1-C3烷基，C1-C3卤代烷基，C1-C3烷氧基，C1-C3卤代烷氧基，C1-C3烷硫基， C 2 -C 3烷氧基烷基，卤素或未取代的氨基，Z是氧或硫。

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