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141. 发明授权

US4522838A 2-Acetyl-1-pyrroline and its use for flavoring foods 失效
标题翻译： 2-乙酰基-1-吡咯啉及其用于调味食品的用途
公开(公告)号：US4522838A
公开(公告)日：1985-06-11
申请号：US500049
申请日：1983-06-01
申请人： Ronald G. Buttery , Louisa C. Ling , Bienvenido O. Juliano
发明人： Ronald G. Buttery , Louisa C. Ling , Bienvenido O. Juliano
IPC分类号： A23L27/20 , C07D207/20 , C11B9/00 , C07D207/00 , A23L1/226
CPC分类号： C07D207/20 , A23L27/2054 , C11B9/0092
摘要： The compound, 2-acetyl-1-pyrroline and its use in flavoring foods, particularly in imparting a "scented" rice flavor to foods, are disclosed.
摘要翻译：该化合物2-乙酰基-1-吡咯啉及其在调味食品中的用途，特别是赋予食品“香味”米味的用途。

142. 发明授权

US4430456A Polyurethane-forming process using amino and amido dialkyl tin carboxylates 失效
标题翻译：使用氨基和酰氨基二烷基锡羧酸盐的聚氨酯形成方法
公开(公告)号：US4430456A
公开(公告)日：1984-02-07
申请号：US418519
申请日：1982-09-16
申请人： Ibrahim S. Bechara , Rocco L. Mascioli
发明人： Ibrahim S. Bechara , Rocco L. Mascioli
IPC分类号： C07F7/22 , C08G18/24 , C08G18/14 , C07D207/00
CPC分类号： C07F7/2244 , C08G18/246
摘要： Amino and amido dialkyltin dicarboxylates and stannoxy carboxylates are prepared by first reacting an amine or amino alcohol with a dicarboxylic acid anhydride, followed by reaction of the resulting product with a dialkyltin oxide. The obtained compounds are useful as catalysts for promoting reaction of organic isocyanates with organic compounds having one or more active hydrogen-containing groups.
摘要翻译：通过首先使胺或氨基醇与二羧酸酐反应，然后将所得产物与二烷基氧化锡反应来制备二羧酸氨基和酰氨基二烷基锡二羧酸酯和烷氧基羧酸盐。所得化合物可用作促进有机异氰酸酯与具有一个或多个含活性氢基团的有机化合物的反应的催化剂。

143. 发明授权

US4343740A Hydroxylalkyl hydroxy-aromatic condensation products as fuel and lubricant additives 失效
标题翻译：羟基烷基羟基 - 芳族缩合产物作为燃料和润滑剂添加剂
公开(公告)号：US4343740A
公开(公告)日：1982-08-10
申请号：US279399
申请日：1981-07-01
申请人： Charles P. Bryant
发明人： Charles P. Bryant
IPC分类号： C08F8/00 , C10L1/18 , C10L1/22 , C10M159/12 , C07D207/00
CPC分类号： C10M159/12 , C08F8/00 , C10L1/1817 , C10L1/221
摘要： Condensation products made by reacting an .alpha.-hydroxyalkyl hydroxy-aromatic compound also having at least one non-fused hydrocarbyl substituent with at least one olefinic nitrile, carboxylic acid or carboxylic acid derivative are useful as additives for fuels and lubricants. The total number of carbon atoms in the non-fused hydrocarbyl substituents is at least about 7 while the .alpha.-hydroxyalkyl group contains from 1 to about 36 carbons and the olefinic acid or nitrile reactant usually contains 2 to about 40 carbon atoms. Products made from hydroxymethyl alkyl-substituted phenols and .alpha.,.beta.-olefinic acid derivatives such as maleic anhydride are particularly useful. Similarly useful post-treated products can be made from these condensation products by further reaction with alcohols, amines, metal salts or metals.
摘要翻译：通过使具有至少一个非稠合烃基取代基的α-羟基烷基羟基 - 芳族化合物与至少一种烯属腈，羧酸或羧酸衍生物反应制得的缩合产物可用作燃料和润滑剂的添加剂。非稠合烃基取代基中的碳原子总数为至少约7，而α-羟基烷基含有1至约36个碳，并且烯属酸或腈反应物通常含有2至约40个碳原子。由羟甲基烷基取代的酚和α，β-烯烃酸衍生物如马来酸酐制成的产品是特别有用的。类似地，有用的后处理产物可以通过与醇，胺，金属盐或金属的进一步反应从这些缩合产物制备。

144. 发明授权

US4336194A Benzyl pyrrolyl methyl carboxylate insecticides and acaricides 失效
标题翻译：苄基吡咯甲酸甲酯杀虫剂和杀螨剂
公开(公告)号：US4336194A
公开(公告)日：1982-06-22
申请号：US57282
申请日：1979-07-13
申请人： Tadashi Ohsumi , Nobushige Itaya , Masachika Hirano
发明人： Tadashi Ohsumi , Nobushige Itaya , Masachika Hirano
IPC分类号： A01N43/36 , A01N53/04 , C07D207/00 , C07D207/32 , C07D207/323 , C07D207/325 , C07D207/452
CPC分类号： C07D207/323 , C07D207/325
摘要： Carboxylic acid esters of the formula (I), ##STR1## wherein X is a hydrogen atom, or a C.sub.1 -C.sub.3 alkyl or a C.sub.1 -C.sub.3 alkoxyl group or a halogen atom linked to the meta or para position and R.sub.1 is a group of the formula (II) or (III), ##STR2## wherein R.sub.2 is a hydrogen atom or a methyl group, and when R.sub.2 is a methyl group R.sub.3 is also a methyl group, and when R.sub.2 is a hydrogen atom R.sub.3 is a group of the formula, ##STR3## (wherein R.sub.5 is a halogen atom or a C.sub.1 -C.sub.3 alkyl, vinyl or a C.sub.1 -C.sub.3 alkoxymethyl group, R.sub.6 is a hydrogen or halogen atom or a methyl group, or, taken together, R.sub.5 and R.sub.6 may form a tetramethylene group by connecting together at ends thereof), R.sub.4 is a halogen atom or a C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxyl or 3,4-methylenedioxy group, n is 1 or 2 and Y is a isopropyl or cyclopropyl group. These carboxylic acid esters are produced by reacting the reactive derivatives of a carboxylic acid represented by the formula, ##STR4## wherein R.sub.1 is a group of the formula (II) or (III), ##STR5## wherein R.sub.2, R.sub.3, R.sub.4, n and Y are as defined above, and Z is a halogen atom, with an alcohol of the formula (IV), ##STR6## wherein X is as defined above, in the presence of an acid-binding agent. These carboxylic acid esters are useful as insecticides and acaricides.
摘要翻译：式（I）的羧酸酯，其中X为氢原子，或C1-C3烷基或C1-C3烷氧基或与间位或对位连接的卤素原子，R1为式（II）或（III）的基团，其中R2是氢原子或甲基，当R2是甲基时，R3也是甲基，当R2是氢原子时R3是式中的一组基团（其中R 5为卤素原子或C 1 -C 3烷基，乙烯基或C 1 -C 3烷氧基甲基，R 6为氢或卤素原子或甲基，或一起为R 5 R 6是卤原子或C 1 -C 3烷基，C 1 -C 3烷氧基或3,4-亚甲二氧基，n是1或2，Y是异丙基或环丙基。这些羧酸酯通过使下式表示的羧酸的反应性衍生物，其中R 1是式（II）或（III）的基团，其中R 2，R 3，R 4，n 和Y如上定义，并且Z是卤素原子，与式（IV）的醇，其中X如上定义，在酸结合剂存在下，其中X如上定义。这些羧酸酯可用作杀虫剂和杀螨剂。

145. 发明授权

US4211776A N-Substituted 2-methoxybenzenesulphonamides, process for preparing them and medicaments containing them 失效
标题翻译： N-取代的2-甲氧基苯磺酰胺，其制备方法和含有它们的药物
公开(公告)号：US4211776A
公开(公告)日：1980-07-08
申请号：US947623
申请日：1978-10-02
申请人： Robert C. Moreau , Jean-Paul Fournier
发明人： Robert C. Moreau , Jean-Paul Fournier
IPC分类号： C07C205/26 , C07D295/12 , C07D295/13 , A61K31/32 , A61K31/40 , C07D207/00 , C07D209/00
CPC分类号： C07D295/13 , C07C205/26 , C07C309/00
摘要： The invention relates to new N-substituted benzenesulphonamides of general formula ##STR1## in which n is 2 or 3,R.sub.1 and R.sub.2 are hydrogen atoms, methyl, ethyl groups, or jointly form with the nitrogen a nitrogenized heterocyclic ring having 5 or 6 members, in particular a piperidino, pyrrolidino or morpholino group.R.sub.3 is a hydrogen atom, an NO.sub.2 group, an NH.sub.2 group, or a halogen,R.sub.4 is a hydrogen, a halogen, NH.sub.2 group or a sulphonamide group.These compounds are useful as active substances of medicaments, in particular as antiemetic.
摘要翻译：本发明涉及通式为“IMAGE”的新的N-取代苯磺酰胺，其中n为2或3，R 1和R 2为氢原子，甲基，乙基或与氮一起形成具有5或6个成员的氮杂环，特别是哌啶子基，吡咯烷子基或吗啉代基团。 R3是氢原子，NO2基，NH2基或卤素，R4是氢，卤素，NH2基或磺酰胺基。这些化合物可用作药物的活性物质，特别是作为止吐剂。

146. 发明授权

US4145264A Preparation of metal-free phthalocyanines 失效
标题翻译：无金属酞菁的制备
公开(公告)号：US4145264A
公开(公告)日：1979-03-20
申请号：US884892
申请日：1978-03-09
申请人： Peter Thoma , Wolfgang Habermann , Joachim Kranz
发明人： Peter Thoma , Wolfgang Habermann , Joachim Kranz
IPC分类号： C09B47/30 , C09B47/067 , C25B3/04 , C07D207/00 , C09B47/04
CPC分类号： C09B47/067
摘要： Metal-free phthalocyanines (PC) are prepared by electrolysis, at inert electrodes, of aromatic o-dinitriles in organic liquids which contain small amounts of dissolved electrolytically conductive compounds, in the presence of hydrogen or of a compound which eliminates hydrogen under the reaction conditions and in the presence of alkaline compounds (as activators). The PC formed may be isolated in the pure form by filtration. The product contains from 90 to 99% of PC. It is used for the preparation of PC-based pigments.

147. 发明授权

US4118417A Process for resolving cis-1-substituted phenyl-1,2-cyclopropanedicarboxylic acids 失效
标题翻译：拆分顺式-1-取代苯基-1,2-环丙烷二羧酸的方法
公开(公告)号：US4118417A
公开(公告)日：1978-10-03
申请号：US809340
申请日：1977-06-23
申请人： Joseph William Epstein
发明人： Joseph William Epstein
IPC分类号： C07C33/36 , C07D209/52 , C07C63/00 , C07D207/00
CPC分类号： C07C33/36 , C07D209/52
摘要： A method for resolving racemic substituted cyclopropanedicarboxylic acids which are useful as intermediates for the preparation of substituted phenyl azabicyclohexanes which possess anxyolitic and analgesic activity.
摘要翻译：用于拆分外消旋取代的环丙烷二羧酸的方法，其可用作制备具有羟基和镇痛活性的取代的苯基氮杂双环己烷的中间体。

148. 发明授权

US11524940B1 Inhibitors of cysteine proteases and methods of use thereof 有权
公开(公告)号：US11524940B1
公开(公告)日：2022-12-13
申请号：US17525514
申请日：2021-11-12
申请人： Pardes Biosciences, Inc.
发明人： Lee D. Arnold , Andy Jennings , Walter Keung
IPC分类号： C07D207/00 , A61K31/40 , A61P31/14 , C07D213/90 , A61K45/06
摘要： The disclosure provides compounds with warheads and their use in treating medical diseases or disorders, such as viral infections. Pharmaceutical compositions and methods of making various compounds with warheads are provided. The compounds are contemplated to inhibit proteases, such as the 3C, CL- or 3CL-like protease.

149. 发明授权

US11524934B2 Phenylamine compounds 有权
公开(公告)号：US11524934B2
公开(公告)日：2022-12-13
申请号：US16605847
申请日：2018-04-18
申请人： PI INDUSTRIES LTD.
发明人： Maruti Naik , Vishal A. Mahajan , Gulab E. Walunj , Dipak D. Nivdunge , Sulur G. Manjunatha , Ruchi Garg , Santosh Shridhar Autkar , Nitin Ramesh Tembhare , Hagalavadi M. Venkatesha , Konstantin Poscharny , Alexander G. M. Klausener
IPC分类号： C07C257/12 , C07D207/00 , A01N37/00 , A01N39/00 , A01N43/00 , A01N37/52 , A01N43/36 , A01N43/38 , A01N43/40 , A01N43/50 , A01N43/52 , A01N43/56 , A01N43/653 , A01N43/78 , A01N43/84 , A01N43/90 , C07C323/45 , C07D207/36 , C07D209/12 , C07D213/81 , C07D231/44 , C07D231/56 , C07D235/04 , C07D239/26 , C07D249/08 , C07D277/68 , C07D295/16 , C07D471/04
摘要： The present invention relates to 4-substituted phenylamidine derivatives of the general formula (I), wherein R5-R6, ArA4, D, G, B, Q and an integer m have the meanings as defined in the description. The invention further relates to methods for their preparation and use of said compounds for controlling undesired phytopathogenic microorganisms, and agents for said purpose, comprising said phenylamine derivatives. This invention further relates to a method for controlling undesired phytopathogenic microorganisms by application of said 4-substituted phenylamidine derivatives of general formula (I) to such undesired microorganisms and/or to their habitat, according to the invention.

150. 发明授权

US11174231B1 Inhibitors of cysteine proteases and methods of use thereof 有权
公开(公告)号：US11174231B1
公开(公告)日：2021-11-16
申请号：US17322221
申请日：2021-05-17
申请人： Pardes Biosciences, Inc.
发明人： Lee D. Arnold , Andy Jennings , Walter Keung
IPC分类号： C07D207/00 , A61K31/40 , A61P31/14 , C07D213/90 , A61K45/06
摘要： The disclosure provides compounds with warheads and their use in treating medical diseases or disorders, such as viral infections. Pharmaceutical compositions and methods of making various compounds with warheads are provided. The compounds are contemplated to inhibit proteases, such as the 3C, CL- or 3CL-like protease.

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