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1. 发明申请

US20110319622A1 PROCESS OF PRODUCING BLEACH BOOSTERS 有权
标题翻译：生产漂白剂的方法
公开(公告)号：US20110319622A1
公开(公告)日：2011-12-29
申请号：US13224621
申请日：2011-09-02
申请人： Ludwig Völkel , Christian Bittner , Ingo Münster , Frank Dietsche , Wolfgang Schrof
发明人： Ludwig Völkel , Christian Bittner , Ingo Münster , Frank Dietsche , Wolfgang Schrof
IPC分类号： C07D217/10
CPC分类号： C07D217/10 , C07D217/04 , C07D498/04
摘要： This invention relates to a process of producing compounds, which are useful as bleach boosters, as well as to the compounds, which are obtainable using said process, and to their use.
摘要翻译：本发明涉及生产可用作漂白助剂的化合物的方法，以及可使用所述方法获得的化合物及其用途。

2. 发明申请

US20050261334A1 Bis-pyridino containing compounds for the use in the treatment of CNS pathologies 审中-公开
标题翻译：用于治疗中枢神经系统病变的含双吡啶的化合物
公开(公告)号：US20050261334A1
公开(公告)日：2005-11-24
申请号：US11027675
申请日：2005-01-03
申请人： Peter Crooks , Linda Dwoskin , Joshua Ayers , Vladimir Grinevich , Sangeetha Sumithran
发明人： Peter Crooks , Linda Dwoskin , Joshua Ayers , Vladimir Grinevich , Sangeetha Sumithran
IPC分类号： A61K31/444 , A61K31/4709 , C07D213/16 , C07D213/22 , C07D215/10 , C07D217/10 , C07D401/04 , C07D401/14 , C07D41/02
CPC分类号： C07D215/10 , C07D213/06 , C07D213/22 , C07D217/10 , C07D401/14
摘要： N-n-Alkylation of nicotine converts nicotine from an agonist into an antagonist specifically for neuronal nicotinic acetylcholine receptor subtypes mediating nicotine-evoked dopamine release. Conformationally restricted analogs exhibit both high affinity and selectivity at this site, and are able to access the brain due to their ability to act as substrates for the blood-brain barrier choline transporter.
摘要翻译：尼古丁的N-n-烷基化将尼古丁从激动剂转化成特异性用于神经元烟碱乙酰胆碱受体亚型的拮抗剂，其介导尼古丁诱发的多巴胺释放。构象限制的类似物在该位点表现出高亲和力和选择性，并且由于其作为血脑屏障胆碱转运蛋白底物的能力，能够进入大脑。

3. 发明授权

US06958205B2 Image forming material and ammonium compound 有权
标题翻译：成像材料和铵化合物
公开(公告)号：US06958205B2
公开(公告)日：2005-10-25
申请号：US10201557
申请日：2002-07-24
申请人： Kaoru Iwato , Tadahiro Sorori
发明人： Kaoru Iwato , Tadahiro Sorori
IPC分类号： G03F7/004 , B41C1/10 , B41M5/36 , B41N1/14 , C07D211/42 , C07D211/46 , C07D217/10 , C07D295/02 , C07D295/037 , C07D295/06 , C07D295/073 , C07D295/08 , C07D295/096 , C07D295/10 , C07D295/108 , C07D295/12 , C07D295/14 , C07D295/155 , C07D295/16 , C07D295/192 , C07D471/06 , C07D471/10 , C07D487/10 , G03F7/00
CPC分类号： C07D217/10 , B41C1/1008 , B41C1/1016 , B41C2201/04 , B41C2201/14 , B41C2210/02 , B41C2210/06 , B41C2210/22 , B41C2210/24 , B41C2210/262 , C07D211/42 , C07D211/46 , C07D295/037 , C07D295/073 , C07D295/096 , C07D295/108 , C07D295/155 , C07D295/192 , C07D471/06 , C07D471/10 , C07D487/10 , Y10S430/165
摘要： An image forming material includes an image forming layer containing a water-insoluble and alkali-soluble resin, a light-heat converting agent and a compound represented by the following general formula (1). In general formula (1), R1 to R3 independently represent an organic group, where R1 represents a residue forming a ring containing a N1 atom, R2 and R3 may bond to each other to form a ring or at least one of R2 and R3 may bond to R1 to form a ring and X− represents a conjugate base of an organic acid or inorganic acid. The ring containing the N1 atom is preferably a piperidine ring.
摘要翻译：成像材料包括含有水不溶性和碱溶性树脂的图像形成层，光热转换剂和由以下通式（1）表示的化合物。在通式（1）中，R 1至R 3独立地表示有机基团，其中R 1表示形成含有氮原子，R 2和R 3可以彼此键合以形成环或至少一个R 2， R 1和R 3可以键合到R 1以形成环，X - 表示有机酸或无机酸的共轭碱。含有N 1〜O原子的环优选为哌啶环。

4. 发明授权

US5767129A Substituted quinolines and isoquinolines as calcium channel blockers, their preparation and the use thereof 失效
公开(公告)号：US5767129A
公开(公告)日：1998-06-16
申请号：US698010
申请日：1996-08-13
申请人： Po-Wai Yuen
发明人： Po-Wai Yuen
IPC分类号： C07D217/04 , C07D217/10 , A61K31/47 , C07D215/02 , C07D215/16 , C07D217/22
CPC分类号： C07D217/04 , C07D217/10
摘要： The present invention relates to novel substituted quinolines and isoquinolines and derivatives thereof useful in the treatment of neurological disorders. Methods of preparing the compounds, intermediates useful in the preparation and pharmaceutical compositions containing the compounds are also included. The compounds are useful in treating pain, cerebral ischemia, and other cerebrovascular disorders.

5. 发明授权

US5710116A Color-safe bleach boosters, compositions and laundry methods employing same 失效
公开(公告)号：US5710116A
公开(公告)日：1998-01-20
申请号：US697748
申请日：1996-08-29
申请人： Gregory Scot Miracle , Michael Eugene Burns , Patti Jean Kellett , James Charles Theophile Roger Burckett-St. Laurent
发明人： Gregory Scot Miracle , Michael Eugene Burns , Patti Jean Kellett , James Charles Theophile Roger Burckett-St. Laurent
IPC分类号： C07D217/10 , C07D498/04 , C11D3/28 , C11D3/34 , C11D3/39 , C11D3/395 , D06L3/02
CPC分类号： D06L3/021 , C07D217/10 , C11D3/349 , C11D3/392
摘要： Bleach boosters comprising zwitterionic imines and anionic imine polyions having a net negative charge are disclosed. The bleach boosters increase bleaching effectiveness in lower temperature solutions and demonstrate superior color safety profiles. The bleach boosters are ideally suited for inclusion into bleaching compositions including those with detersive surfactants and enzymes. Also provided is a laundry additive product including zwitterionic imines and anionic imine polyions with a net negative charge as bleach boosters. A method for laundering a fabric employing the bleach boosters of the present invention is also disclosed.

6. 发明授权

US5438140A Production of nickelized shaped articles 失效
标题翻译：镍化物品的生产
公开(公告)号：US5438140A
公开(公告)日：1995-08-01
申请号：US211726
申请日：1994-04-28
申请人： Alfred Oftring , Bernd Burkhart , Volker Schwendemann , Klaus Glaser
发明人： Alfred Oftring , Bernd Burkhart , Volker Schwendemann , Klaus Glaser
IPC分类号： C07D215/10 , C07D213/20 , C07D217/10 , C25D3/18 , C07D217/00
CPC分类号： C25D3/18
摘要： Nickelized shaped articles are produced by electrodeposition of nickel from aqueous acidic baths containing as essential constituents one or more nickel salts, one or more inorganic acids and one or more brighteners, the brighteners used being cyclic ammonium compounds I ##STR1## where the nitrogen atom is part of a pyridine, quinoline or isoquinoline ring system which can additionally carry one or two C.sub.1 -C.sub.4 -alkyl substituents,R.sup.1 and R.sup.2 are each hydrogen or C.sub.1 -C.sub.4 alkyl,A is a group of the formula --CO--O--R.sup.3, --CO--CH.sub.2 --CO--O--R.sup.3, --O--CO--R.sup.3 or --O--R.sup.3,whereR.sup.3 is C.sub.1 -C.sub.12 -alkyl, C.sub.5 -C.sub.8 -cycloalkyl, C.sub.7 -C.sub.12 -phenylalkyl or phenyl which can be substituted by one or two C.sub.1 -C.sub.4 -alkyl radicals, C.sub.1 -C.sub.4 -alkoxy radicals, halogen atoms, hydroxyl groups, phenyl radicals or C.sub.1 -C.sub.4 alkoxycarbonyl groups, m is from 0 to 10, n is from 1 to 4, p is 0 or 1, and X.sup..crclbar. is an n-valent inorganic or organic anion which promotes water solubility,with the proviso that for p=0 and A=--CO--O--C.sub.1 -C.sub.12 -alkyl m must not be 1, 2 or 3 and under the same conditions R.sup.1 must not be hydrogen when m is 0.
摘要翻译： PCT No.PCT / EP92 / 02180第 371日期1994年04月28日 102（e）日期1994年4月28日PCT提交1992年9月21日PCT公布。公开号WO93 / 09275 日期：1993年5月13日。镍铁成型制品是通过从含有酸性浴的电解沉积镍制成的，该酸性浴包含作为必需组分的一种或多种镍盐，一种或多种无机酸和一种或多种增白剂，所用的增白剂是环状铵化合物I IMAGE （I）其中氮原子是可另外携带一个或两个C 1 -C 4烷基取代基的吡啶，喹啉或异喹啉环体系的一部分，R 1和R 2各自为氢或C 1 -C 4烷基，A为式-CO-O-R3，-CO-CH2-CO-O-R3，-O-CO-R3或-O-R3，其中R3是C1-C12-烷基，C5-C8-环烷基，C7-C12- 可以被一个或两个C 1 -C 4烷基，C 1 -C 4烷氧基，卤原子，羟基，苯基或C 1 -C 4烷氧基羰基取代的苯基烷基或苯基，m为0至10，n为1 至4，p为0或1，并且X（ - ）是促进水溶性的n价无机或有机阴离子，条件是对于p = 0且A = -CO-O-C 1 -C 12烷基m 麝香 t不为1,2或3，在相同条件下，当m为0时，R1不能为氢。

7. 发明授权

US5216150A Derivatives of isoquinoline (and naphthalene) sulfonamides 失效
标题翻译：异喹啉（和萘）磺酰胺的衍生物
公开(公告)号：US5216150A
公开(公告)日：1993-06-01
申请号：US758808
申请日：1991-09-12
申请人： Hiroyoshi Hidaka , Tomohiko Ishikawa , Masatoshi Hagiwara , Tsutomu Inoue , Kenji Naitoh , Osamu Sakuma , Masayuki Yuasa , Tadashi Morita , Tadashi Toshioka , Isao Umezawa , Takashi Inaba
发明人： Hiroyoshi Hidaka , Tomohiko Ishikawa , Masatoshi Hagiwara , Tsutomu Inoue , Kenji Naitoh , Osamu Sakuma , Masayuki Yuasa , Tadashi Morita , Tadashi Toshioka , Isao Umezawa , Takashi Inaba
IPC分类号： C07C311/16 , C07D217/02 , C07D217/10 , C07D401/12 , C07D401/14 , C07D405/12 , C07D409/12 , C07D491/10
CPC分类号： C07D401/12 , C07C311/16 , C07D217/02 , C07D217/10 , C07D401/14 , C07D405/12 , C07D409/12 , C07D491/10
摘要： Novel quinoline sulfonamino derivatives having a vessel smooth muscle relaxation activity as well as a platelet agglutination inhibitory activity and inhibitory activity to protein kinase A, myosin light chain kinase, proteinkinase C, and calmodulindependent proteinkinase II, but having little action or cardio function; a process for the production of the derivatives, and a pharmaceutical composition containing the derivative.
摘要翻译：具有血管平滑肌松弛活性的新型喹啉磺氨基衍生物以及血小板凝集抑制活性和对蛋白激酶A，肌球蛋白轻链激酶，蛋白激酶C和钙调蛋白依赖性蛋白激酶II的抑制活性，但几乎没有作用或心脏功能; 制备衍生物的方法和含有该衍生物的药物组合物。

8. 发明授权

US5059608A Bicyclic amine compound and a process for the preparation thereof 失效
标题翻译：双环胺化合物及其制备方法
公开(公告)号：US5059608A
公开(公告)日：1991-10-22
申请号：US327813
申请日：1989-03-23
申请人： Hisashi Takasugi , Atsushi Kuno , Mitsuru Ohkubo
发明人： Hisashi Takasugi , Atsushi Kuno , Mitsuru Ohkubo
IPC分类号： A61K31/47 , A61K31/472 , A61K31/55 , A61P25/00 , A61P25/08 , C07D217/02 , C07D217/04 , C07D217/06 , C07D217/10 , C07D217/14 , C07D217/16 , C07D223/16 , C07D401/06 , C07D405/04 , C07D409/04
CPC分类号： C07D223/16 , C07D217/02 , C07D217/04 , C07D217/06 , C07D217/14 , C07D217/16 , C07D405/04 , C07D409/04 , Y02P20/55
摘要： The invention relates to a compound useful as an anticonvulsant, and for treatment of delayed neuronal death, the compound being a bicyclic amine of the formula: ##STR1## wherein R.sup.1 is lower alkyl,R.sup.2 is aryl which may have one or more suitable substituent(s), cyclo(lower)alkyl or heterocyclic group,R.sup.3 is hydrogen, lower alkyl which may have one or more suitable substituent(s), lower alkenyl, or acyl which may have one or more suitable substituent(s),R.sup.4 is hydrogen, lower alkyl, or hydroxy(lower)alkyl,R.sup.5 is hydrogen, lower alkyl, halogen, or protected amino, andn is an integer of 1 or 2, with the proviso that when R.sup.3 is lower alkyl which may have one or more suitable substituent(s), R.sup.2 is cyclo(lower)alkyl or heterocyclic group,or a pharmaceutically acceptable salt thereof.
摘要翻译：本发明涉及可用作抗惊厥药并用于治疗延迟性神经元死亡的化合物，该化合物为下式的双环胺：其中R 1为低级烷基，R 2为可具有一个或多个合适取代基的芳基（ s），环（低级）烷基或杂环基，R 3是氢，可具有一个或多个合适取代基的低级烷基，可具有一个或多个合适取代基的低级烯基或酰基，R 4是氢，低级烷基或羟基（低级）烷基，R 5为氢，低级烷基，卤素或被保护的氨基，n为1或2的整数，条件是当R 3为低级烷基时，其可具有一个或多个合适的取代基，R2是环（低级）烷基或杂环基，或其药学上可接受的盐。

9. 发明授权

US4982312A Charge transfer complex and solid electrolytic capacitor employing the same 失效
标题翻译：电荷转移复合物和采用其的固体电解电容器
公开(公告)号：US4982312A
公开(公告)日：1991-01-01
申请号：US428231
申请日：1989-10-27
申请人： Shuko Shindo , Tsuyoshi Aoyama , Yoji Yamaguchi , Isao Isa , Makoto Ebisawa
发明人： Shuko Shindo , Tsuyoshi Aoyama , Yoji Yamaguchi , Isao Isa , Makoto Ebisawa
IPC分类号： C07C255/31 , C07D213/22 , C07D215/10 , C07D217/10 , H01G9/02 , H01G9/028
CPC分类号： H01G9/028 , C07C255/31 , C07D213/22 , C07D215/10 , C07D217/10
摘要： A charge transfer complex comprising N,N'-alkylene-di-3,5-lutidine as a donor and 7,7,8,8-tetracyanoquinodimethane as an acceptor, the molar ratio of the acceptor to the donor of the charge transfer complex being between 3.0 and 5.0 has a high melting point and excellent electrical conductivity as an electrolyte for a capacitor. A solid electrolytic capacitor employing said charge transfer complex has reduced current leakage and high temperature load characteristics. A chip-type solid electrolytic capacitor employing said charge transfer complex has reduced current leakage, high temperature load characteristics and excellent thermal stability and life characteristics.

10. 发明授权

US4945098A Novel propane-1,3-diol derivatives and use 失效
标题翻译：新型丙-1,3-二醇衍生物和用途
公开(公告)号：US4945098A
公开(公告)日：1990-07-31
申请号：US78525
申请日：1987-07-10
申请人： Gunnar Grue-Sorensen , Christian K. Nielsen
发明人： Gunnar Grue-Sorensen , Christian K. Nielsen
IPC分类号： C07C271/08 , C07C67/00 , C07C213/00 , C07C227/00 , C07C227/08 , C07C229/12 , C07C239/00 , C07C271/06 , C07C325/00 , C07C333/02 , C07D213/00 , C07D217/10 , C07D277/10 , C07D277/22 , C07D277/24 , C07D453/00
CPC分类号： C07D277/24 , C07C271/06 , C07C333/02
摘要： A derivative of 2-methylenepropane-1,3-diol of the general formula I ##STR1## where O--A.sup.1 and O--A.sup.2, which can be the same or different, each represents O, O--C(O), O--C(O)NH, O--C(S)NH or O--C(O)O, R.sup.1 represents an alkyl or alkenyl group of 10-22 carbon atoms, n is an integer from 1 to 11, B.sup.+ represents a quaternary ammonium group, either N.sup.+ R.sup.4 R.sup.5 R.sup.6, or N.sup.+ (Het), where R.sup.4, R.sup.5 and R.sup.6 are similar or different alkyl groups of 1-4 carbon atoms, or two or all of R.sup.4, R.sup.5 and R.sup.6 may be incorporated into a cyclic or bicyclic structure, which may contain additional hetero atoms; X.sup.- means the anion of a pharmceutically acceptable inorganic or organic acid; and R.sup.2 and R.sup.3 are the same or different, and represent hydrogen or alkl groups of 1-4 carbon atoms.The present compounds have been shown to possess a PAF antagonistic effect and an inhibitory effect on the growth of tumor cells, and are thus valuable in the human and veterinary practice as platelet aggregation inhibitors, anti-thrombotic agents, anti-asthmatic agents, anti-allergic agents, anti-inflammatory agents, anti-hypotensive agents, anti-ulcer agents, anti-psoriatic agents, anti-graft rejection agents, anti-conception agents and anti-tumor agents.
摘要翻译： PCT No.PCT / DK86 / 00128 Sec。 371日期1987年7月10日第 102（e）日期1987年7月10日PCT提交1986年11月20日PCT公布。公开号WO87 / 03281 日本6月4日，1987.通式I的2-亚甲基丙烷-1,3-二醇的衍生物，其中O-A1和O-A2可以相同或不同，各自表示O，OC （O），OC（O）NH，OC（S）NH或OC（O）O，R 1表示10-22个碳原子的烷基或链烯基，n为1至11的整数，B +表示季铵基团，N + R4R5R6或N +（Het），其中R4，R5和R6是1-4个碳原子的相似或不同的烷基，或者R4，R5和R6中的两个或全部可以并入环状或双环结构，其可以含有额外的杂原子; X-表示药物可接受的无机或有机酸的阴离子; R2和R3相同或不同，表示1-4个碳原子的氢或烷基。本发明化合物已显示具有PAF拮抗作用和对肿瘤细胞生长的抑制作用，因此在人和兽医学实践中作为血小板聚集抑制剂，抗血栓形成剂，抗哮喘药，抗 - 过敏剂，抗炎剂，抗低血压剂，抗溃疡剂，抗牛皮癣剂，抗移植物排斥剂，抗受孕剂和抗肿瘤剂。

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