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1. 发明专利

JP2013028573A Amino acid derivative and manufacturing method for the same 审中-公开
标题翻译：氨基酸衍生物及其制备方法
公开(公告)号：JP2013028573A
公开(公告)日：2013-02-07
申请号：JP2011167310
申请日：2011-07-29
申请人： Kyoto Univ , 国立大学法人京都大学
发明人： KAWABATA TAKEO , YOSHIMURA TOMOYUKI
IPC分类号： C07C271/22 , C07C269/06 , C07D239/04
摘要： PROBLEM TO BE SOLVED: To provide an amino acid derivative that can be manufactured in a high yield and at a high optical purity and a manufacturing method for the same, and a production intermediate of the amino acid derivative and a manufacturing method for the same.SOLUTION: The amino acid derivative is represented by formula (VI) (wherein Rand Rare each an optionally substituted 1-4C aliphatic hydrocarbon group or an optionally substituted 6-12C aryl group; R's are each independently a hydrogen atom or an alkoxycarbonyl group represented by formula (II) (wherein Ris a 1-4C aliphatic hydrocarbon group or a 6-12C aryl group); and Ris a 1-4C alkylene group). There are also provided a manufacturing method for the amino acid derivative, a production intermediate of the amino acid derivative and a manufacturing method for the same.
摘要翻译：待解决的问题：为了提供可以以高产率和高光学纯度制造的氨基酸衍生物及其制备方法，以及氨基酸衍生物的制备方法和制备方法一样。解决方案：氨基酸衍生物由式（VI）表示（其中R 1 和R 2 分别为任选取代的1-4C脂族烃基或任选取代的6-12C芳基; R 6各自独立地为氢原子或由式（II）表示的烷氧基羰基，（其中R 5 是1-4C脂肪族烃基或6-12C芳基）; R 8 1-4C亚烷基）。还提供了氨基酸衍生物的制造方法，氨基酸衍生物的制造中间体及其制造方法。版权所有（C）2013，JPO＆INPIT

2. 发明专利

JPWO2004058676A1 パーフルオロアリルオキシ化合物及び該化合物を含有した液晶組成物有权
公开(公告)号：JPWO2004058676A1
公开(公告)日：2006-04-27
申请号：JP2005509739
申请日：2003-12-04
申请人：旭電化工業株式会社
发明人：裕克科野 , 裕克科野 , 孝洋大塚 , 孝洋大塚 , 入沢　正福 , 正福入沢
IPC分类号： C07C43/225 , C07C69/773 , C07D239/04 , C09K19/04 , C09K19/12 , C09K19/16 , C09K19/18 , C09K19/20 , C09K19/30 , C09K19/32 , C09K19/34 , C09K19/42 , G02F1/13
CPC分类号： C09K19/2007 , C07D239/04 , C09K19/0403 , C09K19/12 , C09K19/16 , C09K19/18 , C09K19/3003 , C09K19/3028 , C09K19/3059 , C09K19/3066 , C09K19/3068 , C09K19/322 , C09K19/3402 , C09K19/3444 , C09K19/3458 , C09K19/3469 , C09K19/3491 , C09K19/42 , C09K2019/0444 , C09K2019/0466 , C09K2019/3422 , Y10T428/10
摘要：本発明は、下記一般式(I)で表される新規なパーフルオロアリルオキシ化合物及び該化合物を含有してなる液晶組成物に関するものであり、本発明のパーフルオロアリルオキシ化合物は液晶材料として有用なものである。

3. 发明专利

JP2005510471A Cisplatin formulation of reduced toxicity and how to use it 审中-公开
公开(公告)号：JP2005510471A
公开(公告)日：2005-04-21
申请号：JP2003530209
申请日：2002-09-20
申请人：トスクインコーポレーティッド
发明人：パトリックフォガーティ
IPC分类号： C07D239/04 , A61K31/16 , A61K31/167 , A61K31/439 , A61K31/4462 , A61K31/505 , A61K31/513 , A61K31/535 , A61K33/24 , A61K45/00 , A61K45/06 , A61K47/22 , A61P35/00 , A61P43/00
CPC分类号： A61K45/06 , A61K31/16 , A61K31/167 , A61K31/439 , A61K31/4462 , A61K31/505 , A61K31/513 , A61K31/535 , A61K33/24 , A61K47/22 , A61K2300/00
摘要：減少した宿主の毒性が観察されるシスプラチン活性剤を用いる方法が提供される。本方法において、有効量のシスプラチン活性剤が、本発明のシスプラチン毒性減少剤の投与と共に宿主に投与される。また、本方法の実施に用いられる組成物、即ち、減少した毒性を有する薬学的組成物が提供され、これは、シスプラチン活性剤が、有効なシスプラチンの抗増殖活性を維持するが、望ましくないシスプラチンの毒性のレベルを減少させるシスプラチン毒性減少剤と組み合わされている。さらに、様々な異なる疾患状態の治療における方法及び組成物を用いる方法も提供される。

5. 发明专利

JP2000516251A 失效
公开(公告)号：JP2000516251A
公开(公告)日：2000-12-05
申请号：JP51171098
申请日：1997-08-22
IPC分类号： A61K31/426 , A61K31/495 , A61K31/527 , A61K31/54 , A61K31/5517 , A61P1/02 , A61P1/12 , A61P11/06 , A61P17/02 , A61P27/02 , A61P29/00 , A61P35/00 , A61P43/00 , C07D233/02 , C07D233/38 , C07D239/04 , C07D239/06 , C07D239/10 , C07D243/04 , C07D265/06 , C07D265/14 , C07D277/06 , C07D279/06 , C07D409/14 , C07D413/14 , C07D487/04 , C07D495/10

6. 发明专利

JPH11246817A COATING COMPOSITION OR SEALING COMPOUND CURABLE BY EFFECT OF MOISTURE 失效
公开(公告)号：JPH11246817A
公开(公告)日：1999-09-14
申请号：JP33190398
申请日：1998-11-09
申请人： BAYER AG
发明人： WAMPRECHT CHRISTIAN , BLUM HARALD , PEDAIN JOSEF , HALPAAP REINHARD DR , KLEIN GERHARD , ARLT DIETER
IPC分类号： C07D233/02 , C07C269/02 , C07C271/20 , C07D239/04 , C07D263/04 , C07D265/06 , C07D413/00 , C08F20/34 , C08F20/36 , C08F220/36 , C08F246/00 , C08G18/32 , C08G18/67 , C08G18/72 , C08G18/75 , C08G18/81 , C09D133/04 , C09D133/10 , C09D133/14 , C09D175/00 , C09D175/14 , C09K3/10
摘要： PROBLEM TO BE SOLVED: To obtain a coating material or a sealing compound based on an olefinic unsaturated compound and curable by effects of moisture. SOLUTION: This coating composition or sealing compound contains a binary system of a polyisocyanate component and a blocked amino group-containing polyamine component as a binder. The polyisocyanate component is an isocyanate group-containing copolymer obtained from an olefinic unsaturated compound, having at least two average NCO functionality, containing 0.1-13 wt.% isocyanate groups bonded to tertiary carbon atom forming a part of an alicyclic ring and having 1,000-100,000 weight-average molecular weight measured by a gel permeation chromatography.

7. 发明专利

JP2945360B2 失效
公开(公告)号：JP2945360B2
公开(公告)日：1999-09-06
申请号：JP32952497
申请日：1997-11-13
申请人： UNIV FLORIDA
发明人： REIMONDO JEI BAAJERON
IPC分类号： A01N33/04 , A01N33/12 , A01N43/54 , A61K31/00 , A61K31/13 , A61K31/131 , A61K31/135 , A61K31/505 , A61K31/506 , A61K31/785 , A61P17/00 , A61P31/00 , A61P31/04 , A61P31/12 , A61P35/00 , C07C209/08 , C07C209/62 , C07C211/14 , C07C211/27 , C07C211/53 , C07D239/04
摘要： The present invention provides a compound having one of the formulae: Wherein: R1 and R6 may be the same or different and are H, alkyl or aralkyl having from 1 to 12 carbon atoms, provided that R1 and R6 are not H; R7 is H, alkyl, aryl or aralkyl having from 1 to 12 carbon atoms; m is an integer from 3 to 6, inclusive; and n is an integer from 3 to 6, inclusive, or (IV), a salt thereof especially for anti-neoplastic, anti-psoriasis, anti-viral or anti-retroviral therapy or for controlling the growth of insects.

8. 发明专利

JP2849851B2 失效
公开(公告)号：JP2849851B2
公开(公告)日：1999-01-27
申请号：JP7175490
申请日：1990-03-20
申请人： CHIBA SUPESHARUTEI CHEM HOORUDEINGU INC
发明人： RAMANASAN RAUICHANDORAN
IPC分类号： C07D239/04 , C07D211/46 , C07D211/58 , C07D211/66 , C07D211/94 , C07D241/08 , C08F4/04 , C08F8/30 , C08K5/3432 , C08K5/3435 , C08K5/3442 , C08K5/3462

9. 发明专利

JPH0794425B2 失效
公开(公告)号：JPH0794425B2
公开(公告)日：1995-10-11
申请号：JP24880891
申请日：1991-09-27
申请人： MERCK & CO INC
发明人： MERITSUSA ESU EGUBAATOSON , JOOJI DEE HAATOMAN , WASHIRU HARUCHENKO , UIRIAMU ERU RASUERU , MAAKU II DATSUGAN
IPC分类号： C07D211/30 , A61K31/185 , A61K31/195 , A61K31/215 , A61K31/255 , A61K31/265 , A61K31/40 , A61K31/4015 , A61K31/41 , A61K31/415 , A61K31/42 , A61K31/421 , A61K31/435 , A61K31/44 , A61K31/4409 , A61K31/4418 , A61K31/4427 , A61K31/4433 , A61K31/445 , A61K31/4465 , A61K31/451 , A61K31/452 , A61K31/495 , A61K31/496 , A61K31/505 , A61K31/55 , A61K31/66 , A61P7/02 , A61P43/00 , C07C311/02 , C07C311/06 , C07C311/13 , C07C311/19 , C07C313/06 , C07C313/20 , C07C323/59 , C07C327/12 , C07D207/08 , C07D207/09 , C07D207/10 , C07D207/12 , C07D207/26 , C07D207/273 , C07D209/12 , C07D209/30 , C07D211/18 , C07D211/22 , C07D211/32 , C07D211/46 , C07D213/75 , C07D223/08 , C07D233/02 , C07D233/64 , C07D237/08 , C07D239/04 , C07D239/26 , C07D241/04 , C07D241/12 , C07D249/04 , C07D249/08 , C07D263/46 , C07D267/10 , C07D401/12 , C07D401/14 , C07D403/10 , C07D403/12 , C07D403/14 , C07D409/12 , C07D413/12 , C07D413/14 , C07D453/02 , C07D453/06 , C07D471/08 , C07D487/08 , C07F9/38 , C07F9/40
摘要： Sulphonamido-phenylalkanoic acid derivs. of formula (I), and their salts, are new. In (I), R1 = Het1 opt. substd. NR6R7, R6R7NC- (=NR6)- R6R7NC(=NR6)NH-, R6C(=NR7)NR7- or a gp. (a) or (b); Het1 = a 4-8 member heterocyclic ring contg. 1-4 heteroatoms from N, O, S; R6, R7 = H, 0-10C alkyl or cycloalkyl, both opt. substd. Het2 = 1-4C alkanoylamino, 1-6C alkoxycarbonyl, 0-6C alkylamino; 1-10C alkylsulphonylamino, 4-10C aralkylsulphonylamino, 4-10C aralkyl, 1-10 1-10C alkaryl, 1-10C alkylthio 4-10C aralkylthio, 1-10C alkylsulphinyl, 4-10C aralkylsulphinyl, 1-10C alkylsulphonyl, 4-10C aralkylsulphonyl, aminosulphonyl, 1-10C alkylaminosulphonyl, 4-10C aralkylsulphonylamino, oxo, thio, or 1- or 2-ethenyl or 3- propenyl, all opt. substd.; "alkyl" = from alkane, alkene or alkyne; alkoxy = O-alkyl; aralkyl and alkaryl contain alkyl as defined above and aryl defined below; Het2 = a 5 or 6 membered satd. heterocyclic ring contg. 1-4 heteroatoms from N, O, S; aryl = a mono- or poly-cyclic ring system of 5- and 6-membered aromatic rings contg. 0-4 heteroatoms from N, O, S; R2, R3 = H, aryl, or 0-10C alkyl or cycloalkyl both opt. substd.; R4 = aryl, 1-10C alkyl or cycloalkyl, 4-1UC aralkyl, 1-10C alkoxyalkyl, 1-10C alkaryl, 1-10C alkylthioalkyl, 1-10C alkoxythioalkyl, 1-10C alkylamino, 4-10C aralkylamino, 1-10C alkanoylamino, 4-10C aralkanoylamino, 1-10C alkanoyl, 4-10C aralkanoyl, or 1-10C carboxyalkyl opt. substd. R5 = Het1, COR8, or CSR8; R8 = e.g. OH, 1-10C alkyloxy, 1-10C alkaryloxy, etc. X. Y, Z are opt. substits. and = NR6, O, S, SO, CO, CS CH(OH), SO2, CR6=CR7, CC, Het1, (opt. substd. at any atom with R6), aryl, CONR6, NR6CO, NR6SO2, or SO2NR6; m = 0-10; n = 0-10; and p = 0-3.

10. 发明专利

JPH07252193A ANTITUMORAL, ANTIVIRAL, ANTI-RETROVIRAL AND ANTIPARASITIC SPERMINE DERIVATIVE 失效
公开(公告)号：JPH07252193A
公开(公告)日：1995-10-03
申请号：JP24074494
申请日：1994-09-08
申请人： UNIV FLORIDA
发明人： BERGERON RAYMOND J
IPC分类号： A01N33/04 , A01N33/12 , A01N43/54 , A61K31/00 , A61K31/13 , A61K31/131 , A61K31/135 , A61K31/505 , A61K31/506 , A61K31/785 , A61P17/00 , A61P31/00 , A61P31/04 , A61P31/12 , A61P35/00 , C07C209/08 , C07C209/62 , C07C211/14 , C07C211/27 , C07C211/53 , C07D239/04
摘要： The present invention provides a compound having one of the formulae: Wherein: R1 and R6 may be the same or different and are H, alkyl or aralkyl having from 1 to 12 carbon atoms, provided that R1 and R6 are not H; R7 is H, alkyl, aryl or aralkyl having from 1 to 12 carbon atoms; m is an integer from 3 to 6, inclusive; and n is an integer from 3 to 6, inclusive, or (IV), a salt thereof especially for anti-neoplastic, anti-psoriasis, anti-viral or anti-retroviral therapy or for controlling the growth of insects.

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