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1. 发明专利

JPS6169751A Salicylamide derivative, its preparation and agent for controlling crubroot of cruficerous plant 失效
标题翻译：杀菌剂衍生物，其制备和控制CRUFICEROUS工厂CRUBROOT的代理
公开(公告)号：JPS6169751A
公开(公告)日：1986-04-10
申请号：JP19060584
申请日：1984-09-13
申请人： Nippon Tokushu Noyaku Seizo Kk
发明人： KURAHASHI YOSHIO , SHIOKAWA KOZO , GOSHIMA TOSHIO , TOSHIBE SHINZO , MATSUMOTO NOBORU , MORIIE KOUICHI
IPC分类号： A01N37/40 , C07C67/00 , C07C231/00 , C07C231/12 , C07C235/60
CPC分类号： A01N37/40
摘要： NEW MATERIAL:The compound of formula I (X is halogen).
EXAMPLE: N-[2,2,2-trichloro-1-(2,2,2-trichloroethoxy)ethyl]salicylamide.
USE: An agent for controlling crubroot of cruficerous plant. It exhibits excellent effect at a low dose, and no phytotoxicity to crops.
PREPARATION: The compound of formula I can be prepared by reacting the compound of formula II (Hal is halogen) with the compound of formula CX
3 CH
2 OH in an inert solvent other than water and alcohol (e.g. toluene), preferably in the presence of an acid acceptor (e.g. pyridine, alkali metal hydroxide, etc.) at 0W100°C.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新材料：式I化合物（X为卤素）。实施例：N- [2,2,2-三氯-1-（2,2,2-三氯乙氧基）乙基]水杨酰胺。用途：用于控制ous ous植物。。的药剂。它在低剂量下表现出优异的效果，对作物没有植物毒性。制备：式I化合物可以通过使式II化合物（Hal为卤素）与式CX3CH2OH化合物在除水和醇（如甲苯）以外的惰性溶剂中反应制备，优选在酸存在下受体（如吡啶，碱金属氢氧化物等）在0-100℃。

2. 发明专利

JPS6118751A N-benzyl-cyclopropanecarboxamide derivative, its preparation, its intermediate and agricultural and horticultural fungicide 失效
标题翻译： N-苄基 - 环丙烷氧羰基衍生物，其制备方法，其中间体和农业和农药生物
公开(公告)号：JPS6118751A
公开(公告)日：1986-01-27
申请号：JP13895584
申请日：1984-07-06
申请人： Nippon Tokushu Noyaku Seizo Kk
发明人： KURAHASHI YOSHIO , SHIOKAWA KOUZOU , TOSHIBE SHINZOU , SAKAWA SHINJI , MORIIE KOUICHI
IPC分类号： C07C231/02 , A01N53/00 , A01N53/12 , C07C67/00 , C07C231/00 , C07C233/59
摘要： NEW MATERIAL:A compound shown by the formula I (X is halogen; n is 1, or 2; R
1 is H, or halogen; R
2 s lower alkyl, halogen-substituted-lower alkyl; R
2 is halogen-substituted-lower alkyl when R
1 is halogen, and R
2 is lower alkyl when R
1 is halogen; R
3 is lower alkyl).
EXAMPLE: N-4-Chloro-α-methylbenzyl 1,2,2-trichloro-3,3-dimethylcyclopropanecarboxyamide.
USE: An agricultural and horticultural fungicide. Effective especially for blast of rice plant.
PREPARATION: A compound shown by the formula II is reacted with a compound shown by the formula III (A is OH, or halogen) in an inert solvent optionally in the presence of an acid binder (e.g., triethylamine) at 0W100°C to give a compound shown by the formula I.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新材料：由式I表示的化合物（X为卤素; n为1或2; R 1为H或卤素; R 2为低级烷基，卤素取代的低级烷基; R 2为 >当R 1为卤素时为卤素取代的低级烷基，当R 1为卤素时，R 2为低级烷基; R 3为低级烷基）。实施例：1,2,2-三氯-3,3-二甲基环丙烷甲酰胺的N-4-氯-α-甲基苄基。用途：农业和园艺杀菌剂。特别适用于水稻种植。制备：将式II化合物与式III化合物（A是OH或卤素）在惰性溶剂中反应，任选地在0-100℃的酸性粘合剂（如三乙胺）存在下反应。得到式I所示的化合物。

3. 发明专利

JPS6160682A Tetrahydroquinolin-1-ylcarbonylimidazole derivative, its intermediate, its production, herbicide, agricultural and horticultural fungicide 失效
标题翻译：四氢喹啉-1-酮亚胺咪唑衍生物，其中间体，其生产，除草剂，农业和农药杀真菌剂
公开(公告)号：JPS6160682A
公开(公告)日：1986-03-28
申请号：JP17939984
申请日：1984-08-30
申请人： Nippon Tokushu Noyaku Seizo Kk
发明人： KURAHASHI YOSHIO , SHIOKAWA KOZO , GOSHIMA TOSHIO , TOSHIBE SHINZO , KAJI SHUZO , MORIYA KOUICHI , HAYAKAWA HIDENORI
IPC分类号： C07D401/06 , A01N47/38 , C07D215/08 , C07D215/12 , C07D215/16 , C07D215/18 , C07D215/20 , C07D215/26 , C07D215/28 , C07D215/36 , C07D215/48 , C07D221/10 , C07D221/16 , C07D521/00
CPC分类号： C07D231/12 , A01N47/38 , C07D215/08 , C07D215/12 , C07D215/18 , C07D215/20 , C07D215/26 , C07D215/28 , C07D215/36 , C07D215/48 , C07D221/10 , C07D221/16 , C07D233/56 , C07D249/08
摘要： NEW MATERIAL:A compound shown by the formula I [X is halogen, lower alkyl, nitro, cyano, trifluoromethyl, (halogen-substituted)lower alkoxy, (halogen- substituted)lower alkylthio, lower alkylsulfonyl, phenyl, (halogen-substituted) phenylthio, or (substituted)phenoxy; n is 1W3, X is except Cl when n is 1, and all X are not Cl when n is 2 or 3; 2X and C at the 7- and the 8-positions of tetrahydroquinoline rig in the formula may be bonded to form 5W6 ring].
EXAMPLE: 1-[7,8-Dimethyl-1(H),2,3,4-tetrahydroquinolin-1-ylcarbonyl]imidazole.
USE: A herbicide, agricultural and horticultural fungicide. having low toxicity and improved selectivity.
PREPARATION: A compound shown by the formula III is reacted with imidazole shown by the formula IV.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新材料：由式I表示的化合物[X是卤素，低级烷基，硝基，氰基，三氟甲基，（卤素取代的）低级烷氧基，（卤素取代的）低级烷硫基，低级烷基磺酰基，苯基，（卤素取代的）苯硫基或（取代的）苯氧基; n为1-3，当n为1时，除了Cl之外，当n为2或3时，X不为Cl; 2X和C在7-和8位的四氢喹啉钻机的配方中可以键合形成5-6环]。实施例：1- [7,8-二甲基-1（H），2,3,4-四氢喹啉-1-基羰基]咪唑。用途：除草剂，农业和园艺杀菌剂。毒性低，选择性好。制备：式III化合物与式IV所示的咪唑反应。

4. 发明专利

JPS61130272A Beta-substituted amino-phenetylazole derivative, its intermediate, preparation thereof, and agricultural and horticultural fungicide 失效
标题翻译：取代的氨基 - 苯并噻唑衍生物，其中间体，其制备方法和农业和农业化学品
公开(公告)号：JPS61130272A
公开(公告)日：1986-06-18
申请号：JP25198184
申请日：1984-11-30
申请人： Nippon Tokushu Noyaku Seizo Kk
发明人： KURAHASHI YOSHIO , MORISHIMA NORIHISA , YAMAGUCHI NAOKO , MATSUMOTO NOBORU
IPC分类号： A01N43/50 , A01N43/653 , C07D233/61 , C07D249/08 , C07D521/00
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要： NEW MATERIAL:The β-substituted amino-phenetylazole derivative of formula I (X is N or CH; Y is O or S; R
1 is lower alkyl, halogen or lower alkoxy; R
2 is lower alkyl, halogen, lower alkoxy, trifluoromethyl, nitro, or methoxyiminomethyl; p is 0, 1 or 2; q is 0 or 1W3; l is 1W5; m is 0 or 1).
EXAMPLE: 1-[β-(3-Phenoxypropylamino)-2,4-dichlorophenetyl]- 1H-1,2,4-triazole.
USE: Useful as an agricultural and horticultural fungicide e.g. for gray mold of various vegetables, powdery mildew of cucumber, late blight of tomato, etc. It has low toxicity to warm-blooded animals.
PREPARATION: The compound of formula I can be prepared by reacting the compound of formula II with the compound of formula III, and reducing the resultant compound of formula IV.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新物质：式I的β-取代氨基 - 苯乙烯衍生物（X为N或CH; Y为O或S; R 1为低级烷基，卤素或低级烷氧基; R 2为低级烷基，卤素，低级烷氧基，三氟甲基，硝基或甲氧基亚氨基甲基; p为0,1或2; q为0或1-3; l为1-5; m为0或1）。实施例：1- [β-（3-苯氧基丙基氨基）-2,4-二氯苯乙基] -1H-1,2,4-三唑。用途：用作农业和园艺杀真菌剂，例如各种蔬菜灰霉病，黄瓜白粉病，番茄晚疫病等，对温血动物毒性低。制备：式I化合物可以通过使式II化合物与式III化合物反应，还原所得的式IV化合物来制备。

5. 发明专利

JPS6168470A Carbamoylimidazole derivative, its production and agricultural an horticultural fungicide 失效
标题翻译：卡巴胺咪唑衍生物，其生产和农业化学品
公开(公告)号：JPS6168470A
公开(公告)日：1986-04-08
申请号：JP18877884
申请日：1984-09-11
申请人： Nippon Tokushu Noyaku Seizo Kk
发明人： KUME TOYOHIKO , KURAHASHI YOSHIO , ISONO KUNIHIRO , SAKAWA SHINJI , MATSUMOTO NOBORU
IPC分类号： A01N47/38 , A01N20060101 , C07D20060101 , C07D233/56 , C07D233/60
摘要： NEW MATERIAL:A carbamoylimidazole derivative shown by the formula I (R
1 is lower alkyl, lower alkoxy-lower alkyl, or 3W8C cycloalkyl; R
2 is fluoro- substituted lower alkyl; X is O or S; Y is halogen, lower alkyl; m is 0, 1, or 2; n is 3W6).
EXAMPLE: 1{N-2-[2,6-Dichloro-4-(2,2,2-trifluoroethylthio)phenoxy]ethyl-N-propyl carbamoyl}imidazole.
USE: Useful as an agricultural and horticultural fungicide. Showing improved fungicidal effect on plant blights such as blast or rice plant, late blight of tomato, anthracnose of cucumber, bakanae disease of rice plant, etc., with a low concentration of agent, and exhibiting completely controlling effect.
PREPARATION: A compound shown by the formula II (Hal is halogen) is reacted with a compound shown by the formula III, and with N, N'-carbonyldimidazole to give a compound shown by the formula I.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新材料：式I所示的氨基甲酰咪唑衍生物（R 1是低级烷基，低级烷氧基 - 低级烷基或3-8C环烷基; R 2是氟取代的低级烷基; X是O或S; Y 是卤素，低级烷基; m是0,1或2; n是3-6）。实施例：1 {N-2- [2,6-二氯-4-（2,2,2-三氟乙硫基）苯氧基]乙基-N-丙基氨基甲酰基}咪唑。用途：用作农业和园艺杀菌剂。显示了对植物病害如爆破或水稻植物，西红柿晚疫病，黄瓜炭疽病，水稻植物等的杀虫效果改善，具有低浓度的药剂，具有完全控制作用。制备：将式II化合物（Hal为卤素）与式III化合物和N，N'-羰基二咪唑反应，得到式I所示的化合物。

6. 发明专利

JPS6115867A N-benzyl-cyclopropanecarboxamide derivative, its preparation and agricultural and horticultural fungicide 失效
标题翻译： N-苄基 - 环丙烷氧羰基衍生物，其制备和农业和农业生物
公开(公告)号：JPS6115867A
公开(公告)日：1986-01-23
申请号：JP13526884
申请日：1984-07-02
申请人： Nippon Tokushu Noyaku Seizo Kk
发明人： KURAHASHI YOSHIO , SHIOKAWA KOUZOU , TOSHIBE SHINZOU , SAKAWA SHINJI , SEIKE KOUICHI
IPC分类号： C07C231/00 , A01N53/00 , A01N53/12 , C07C67/00 , C07C231/02 , C07C233/59
摘要： NEW MATERIAL:The compound of formula I (X is halogen; n is 1 or 2; R
1 W R
3 are H or lower alkyl).
EXAMPLE: N-( 4-chloro-α-methylbenzyl )2,2-dichloro-1-methyl-(trans)-3-methylcyclopropanecarboxamide.
USE: An agricultural and horticultural insecticide. It exhibits excellent activity especially for the control of rice blast.
PREPARATION: The compound of formula I can be prepared by reacting the compound of formula II with the compound of formula III (A is OH or halogen) in a solvent at a temperature between -20°C and the boiling point of the reaction mixture, preferably at 0W100°C, optionally in the presence of an acid acceptor (e.g. alkali metal hydroxide, triethylamine, etc.).
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新材料：式I化合物（X为卤素; n为1或2; R 1 -R 3为H或低级烷基）。实施例：N-（4-氯-α-甲基苄基）2,2-二氯-1-甲基 - （反式）-3-甲基环丙烷甲酰胺。用途：农业和园艺杀虫剂。它表现出优异的活性，特别是用于控制稻瘟病。制备：式I化合物可以通过使式II化合物与式III化合物（A为OH或卤素）在溶剂中在-20℃和反应混合物的沸点之间，优选0-100℃，任选在酸受体（例如碱金属氢氧化物，三乙胺等）存在下进行。

7. 发明专利

JPS6160659A Substituted phenylsulfonylazole, its production, and agricultural and horticultural fungicide 失效
标题翻译：取代的苯并呋喃，其生产和农业和农业生物
公开(公告)号：JPS6160659A
公开(公告)日：1986-03-28
申请号：JP18257984
申请日：1984-09-03
申请人： Nippon Tokushu Noyaku Seizo Kk
发明人： SAITO JUNICHI , TAMURA TATSUO , KURAHASHI YOSHIO , UZAWA SHIGERU , MATSUMOTO NOBORU , YAMAGUCHI NAOKO
IPC分类号： A01N43/50 , A01N43/653 , C07D233/56 , C07D233/84 , C07D249/08 , C07D521/00
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要： NEW MATERIAL:A substituted phenylsulfonylazole shown by the formula I (X is N or CH: R is halogen, lower alkyl, lower alkoxy, trifluoromethyl, nitro, phenyl, or cycloalkyl; n is 1W3; R is not methyl when n is 1).
EXAMPLE: 1-(2,5-Xylylsulfonyl)imidazole.
USE: Useful as an agricultural and horticultural fungicide. Having improved controlling action and effect on plant blights in agriculture and horticulture. Showing improved effect especially on late blight of tomato, blast of rice plate, downy mildew of melon, downy mildew of grape, etc.
PREPARATION: A compound shown by the formula II (Hal is halogen is reacted with a compound shown by the formula III in a solvent such as preferably hexane, etc. or in a diluent in the presence of an acid binder such as pyridine, etc. at 0W100°C, to give a compound shown by the formula I.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新物质：由式I表示的取代的苯基磺酰基（X为N或CH：R为卤素，低级烷基，低级烷氧基，三氟甲基，硝基，苯基或环烷基; n为1-3;当n为 1）。实施例：1-（2,5-辛基磺酰基）咪唑。用途：用作农业和园艺杀菌剂。改善了对农业和园艺植物病害的控制作用和影响。显示改善效果，特别是对番茄晚疫病，稻瘟病，瓜类霜霉病，葡萄霜霉病等的制备：式Ⅱ化合物（Hal为卤素）与式Ⅲ化合物反应在溶剂如己烷等溶剂中，或在酸性粘合剂如吡啶等的存在下，在0-100℃下，在稀释剂中，得到式I所示的化合物。

8. 发明专利

JPS5724394A Phosphoric acid haloalkyl ester or haloalkenyl ester, preparation of said compound, and agricultural fungicide 失效
标题翻译：磷酸二甲酯或羟丙基酯，制备化合物和农药杀真菌剂
公开(公告)号：JPS5724394A
公开(公告)日：1982-02-08
申请号：JP9867180
申请日：1980-07-21
申请人： Nippon Tokushu Noyaku Seizo Kk
发明人： YAMADA YASUO , SAITOU JIYUNICHI , KURAHASHI YOSHIO , KUME TOYOHIKO , ISONO KUNIHIRO , SAKAWA SHINJI
IPC分类号： A01N57/10 , C07F9/09 , C07F9/165
摘要： NEW MATERIAL:The titled compound of formula I [R
1 is chlorine; R
2 is H; or R
1 and R
2 may together form a single bond; R
3 is 1W3C alkyl; R
4 is 1W4C alkyl or (substituted) phenyl; X is O or S; Y is O, S or NR
5 (R
5 is H or alkyl)].
EXAMPLE: 0-2,3,3-Trichloroallyl-0-2-cyanophenyl-0-methyl phosphate.
USE: Agriculatural and horticultural fungicide. It has excellent fungicidal activity, and effective to a wide variety of plant pathogenic fungi, especially to rice blast.
PROCESS: The compound of formula I is prepared by reacting the compound of formula II (Hal is halogen), e.g. 0-2,3,3,3-tetrachloropropyl-0-methyl phosphorochloride, with the compound of formula M
1 -Y-R
4 (M
1 is H or alkali metal atom), e.g. ethanol, phenol, etc., pref. in a solvent such as water, hexane, acetone, etc., in the presence of an acid acceptor (e.g. an alkali metal hydroxide).
COPYRIGHT: (C)1982,JPO&Japio
摘要翻译：新材料：式I的标题化合物[R 1]为氯; R 2是H; 或R 1和R 2可以一起形成单键; R 3是1-3C烷基; R 4是1-4C烷基或（取代的）苯基; X是O或S; Y是O，S或NR 5（R 5是H或烷基）]。实施例：0-2,3,3-三氯烯丙基-0-2-氰基苯基-O-甲基磷酸酯。用途：农业和园艺杀菌剂。具有优良的杀真菌活性，对各种植物致病真菌尤其是稻瘟病有效。方法：式I化合物通过使式II化合物（Hal为卤素）如 0-2,3,3,3-四氯丙基-O-甲基磷酰氯与式M 1 -Y-R 4的化合物（M 1是H或碱金属原子），例如乙醇，苯酚等。在溶剂如水，己烷，丙酮等中，在酸受体（例如碱金属氢氧化物）存在下进行。

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