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1. 发明授权

EP1201662B1 Preparation of thiazoles 失效
标题翻译：噻唑生产
公开(公告)号：EP1201662B1
公开(公告)日：2005-10-26
申请号：EP01129478.2
申请日：1997-12-17
申请人： Syngenta Participations AG
发明人： Pitterna, Thomas , Szcpepanski, Henry , Maienfisch, Peter , Hüter, Ottmar Franz , Rapold, Thomas , Senn, Marcel , Göbel, Thomas , O'Sullivan, Anthony Cornelius
IPC分类号： C07D277/32 , C07D277/16
CPC分类号： C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74

2. 发明公开

EP1577307A2 Preparation of thiazoles 失效
标题翻译：噻唑的制备
公开(公告)号：EP1577307A2
公开(公告)日：2005-09-21
申请号：EP05013434.5
申请日：1997-12-17
申请人： Syngenta Participations AG
发明人： Pitterna, Thomas , Szcpepanski, Henry , Maienfisch, Peter , Hueter, Ottmar Franz , Repold, Thomas , Senn, Marcel , Gobel, Thomas , O' Sullivan, Anthony Cornelius
IPC分类号： C07D277/36
CPC分类号： C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74
摘要： A process for the preparation of a compound of formula (I):
wherein R is C 1 -C 4 alkyl, hydroxy C 1 -C 4 alkyl, C 3 -C 4 alkenyl, chloro- C 3 -C 4 alkenyl, C 3 -C 4 alkynyl, an unsubstituted or chlorine-substituted phenyl or benzyl group, pyridyl, pyrimidinyl, thiazolyl, benzothilzolyl, cyclohexyl or -CH 2 -COO-C 1 -C 4 alkyl; and X is methylsulfonate, trufluoromethylsulfonate, p-toluenesulfonate or halogen, comprising reacting a compound of formula (IV)
wherein R is as defined for formula (I) and R 2 and R 3 are each independently H, C 1 -C 6 alkyl, C 3 -C 6 cycloalkyl, phenyl or together with the nitrogen atom to which they are bonded form a five- to seven-membered ring in which a -CH 2 - group has optionally been replaced by a hetero atom, selected from the group, consisting of O and S or by NR 9 and wherein the carbon chain of the five- to seven-membered ring is unsubstituted or is mono- or di-substituted by C 1 -C 4 alkyl, and R 9 is H, C 1 -C 6 alkyl, C 3 -C 6 cycloalkyl, phenyl or benzyl; with a compound of the formula halogen-C(=O)-O-C 1 -C 8 alkyl, halogen-C(=O)-O-phenyl or halogen-C(=O)-O-benzyl.
摘要翻译：制备式（I）化合物的方法：其中R为C 1 -C 4烷基，羟基C 1 -C 4烷基，C 3 -C 4烯基，氯-C 3 -C 4烯基，C 3 -C 4炔基，取代的苯基或苄基，吡啶基，嘧啶基，噻唑基，苯并噻唑基，环己基或-CH 2 -COO-C 1 -C 4烷基; X是甲磺酸根，三氟甲基磺酸根，对甲苯磺酸根或卤素，包括使其中R如对式（I）所定义且R 2和R 3各自独立地为H，C 1 -C 6烷基，C 3 -C 6环烷基，苯基或与它们所键合的氮原子一起形成五元至七元环，其中-CH 2 - 基团任选地被选自O和S的杂原子或被 NR9且其中五元至七元环的碳链未被取代或被C1-C4烷基单取代或二取代，且R9为H，C1-C6烷基，C3-C6环烷基，苯基或苄基; 与卤素-C（= O）-OC 1 -C 8烷基，卤素-C（= O）-O-苯基或卤素-C（= O）-O-苄基的化合物反应。

3. 发明公开

EP1577307A3 Preparation of thiazoles 失效
标题翻译：噻唑生产
公开(公告)号：EP1577307A3
公开(公告)日：2009-04-29
申请号：EP05013434.5
申请日：1997-12-17
申请人： Syngenta Participations AG
发明人： Pitterna, Thomas , Szcpepanski, Henry , Maienfisch, Peter , Hueter, Ottmar Franz , Repold, Thomas, Syngenta Crop Protection , Senn, Marcel, Syngenta Crop Protection , Gobel, Thomas , O' Sullivan, Anthony Cornelius
IPC分类号： C07D277/36
CPC分类号： C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74
摘要： A process for the preparation of a compound of formula (I):

wherein R is C 1 -C 4 alkyl, hydroxy C 1 -C 4 alkyl, C 3 -C 4 alkenyl, chloro- C 3 -C 4 alkenyl, C 3 -C 4 alkynyl, an unsubstituted or chlorine-substituted phenyl or benzyl group, pyridyl, pyrimidinyl, thiazolyl, benzothilzolyl, cyclohexyl or -CH 2 -COO-C 1 -C 4 alkyl; and X is methylsulfonate, trufluoromethylsulfonate, p-toluenesulfonate or halogen, comprising reacting a compound of formula (IV)

wherein R is as defined for formula (I) and R 2 and R 3 are each independently H, C 1 -C 6 alkyl, C 3 -C 6 cycloalkyl, phenyl or together with the nitrogen atom to which they are bonded form a five- to seven-membered ring in which a -CH 2 - group has optionally been replaced by a hetero atom, selected from the group, consisting of O and S or by NR 9 and wherein the carbon chain of the five- to seven-membered ring is unsubstituted or is mono- or di-substituted by C 1 -C 4 alkyl, and R 9 is H, C 1 -C 6 alkyl, C 3 -C 6 cycloalkyl, phenyl or benzyl; with a compound of the formula halogen-C(=O)-O-C 1 -C 8 alkyl, halogen-C(=O)-O-phenyl or halogen-C(=O)-O-benzyl.

4. 发明公开

EP1201662A1 Preparation of thiazoles 失效
标题翻译： Herstellung von Thiazolen
公开(公告)号：EP1201662A1
公开(公告)日：2002-05-02
申请号：EP01129478.2
申请日：1997-12-17
申请人： Syngenta Participations AG
发明人： Pitterna, Thomas , Szcpepanski, Henry , Maienfisch, Peter , Hüter, Ottmar Franz , Rapold, Thomas , Senn, Marcel , Göbel, Thomas , O'Sullivan, Anthony Cornelius
IPC分类号： C07D277/32 , C07D277/16
CPC分类号： C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74
摘要： There are described a process for the preparation of a compound of the formula
wherein

R is unsubstituted or substituted C 1 -C 12 alkyl, C 2 -C 4 alkenyl, C 2 -C 4 alkynyl, C 3 -C 6 cycloalkyl, aryl, heteroaryl or -SR 1 ;
R 1 is unsubstituted or substituted C 1 -C 12 alkyl, C 1 -C 4 alkenyl, C 2 -C 4 alkenyl, C 2 -C 4 alkynyl, cycloalkyl, aryl or heteroaryl; and X is a leaving group; which comprises

a) reacting a compound of the formula
wherein R is as defined above, with a water-removing agent; or
b) for the preparation of a compound (I) wherein X is halogen or a sulfonate, reacting a compound of the formula
wherein R is as defined for formula (I), with a halogenating agent or a sulfonylating agent; or
c) for the preparation of a compound (I) wherein X is halogen, reacting a compound
wherein R is as defined for formula (I); and

R 2 and R 3 are for example, H, C 1 -C 6 alkyl, C 3 -C 6 cycloalkyl, phenyl or benzyl;
with a compound of the formula halogen-C(=O)-O-C 1 -C 8 alkyl, halogen-C(=O)-O-aryl or halogen-C(=O)-O-benzyl;
intermediates for the preparation of the compounds (II) to (IV) and (VI) and a method for the preparation thereof.
摘要翻译：描述了制备式CHEM的化合物的方法，其中R是未取代的或取代的C 1 -C 12烷基，C 2 -C 4烯基，C 2 -C 4炔基，C 3 -C 6环烷基，芳基，杂芳基或-SR 1; R1是未取代的或取代的C1-C12烷基，C1-C4链烯基，C2-C4链烯基，C2-C4炔基，环烷基，芳基或杂芳基; X为离去群; 其包括a）使式（CHEM）化合物（其中R如上定义）与除水剂反应; 或b）用于制备其中X为卤素或磺酸盐的化合物（I），其中R为式（I）所定义的式CHEM的化合物与卤化剂或磺酰化剂反应; 或c）用于制备其中X为卤素的化合物（I），使化合物＆lt; CHEM＆gt;其中R如式（I）所定义; 和R 2和R 3是例如H，C 1 -C 6烷基，C 3 -C 6环烷基，苯基或苄基; 与卤素-C（= O）-O-C 1 -C 8烷基，卤素-C（= O）-O-芳基或卤素-C（= O）-O-苄基的化合物反应; 用于制备化合物（II）至（IV）和（VI）的中间体及其制备方法。

5. 发明公开

EP2500340A1 2-Cyanophenyl Sulfonamide Derivatives Useful as Pesticides 审中-公开
标题翻译： 2-氰基苯基磺酰胺衍生物
公开(公告)号：EP2500340A1
公开(公告)日：2012-09-19
申请号：EP12171459.6
申请日：2009-01-23
申请人： Syngenta Participations AG
发明人： Pitterna, Thomas , Renold, Peter , Hueter, Ottmar Franz , Zambach, Werner , Maienfisch, Peter
IPC分类号： C07D307/32 , C07D307/52 , C07D307/79 , C07D333/20 , C07D333/78 , C07D405/12 , C07D409/04 , C07D409/12 , A01N43/00 , A01P5/00 , A01P9/00 , C07D211/76 , C07D213/70 , C07D249/08 , C07C311/16 , C07C311/17 , C07C311/18 , C07C311/21 , C07D207/27
CPC分类号： C07D307/79 , A01N41/10 , A01N43/08 , A01N43/10 , A01N43/12 , A01N43/28 , A01N43/36 , A01N43/40 , A01N43/653 , C07C311/20 , C07C311/29 , C07C323/49 , C07C2601/08 , C07D207/27 , C07D249/08 , C07D307/32 , C07D307/52 , C07D333/20 , C07D333/78 , C07D405/12
摘要： A compound of the formula I

where, for example, W, X and Y are each CH;
R 1 and R 6 , independently of each other, are for example, selected from the group consisting of H, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C1-C6-alkoxy, C3-C8-cycloalkyl, R 7 C(=O), and a ring system;
provided that at least one of R 1 and R 6 is a
- partially or fully unsaturated ring system containing in at least one ring in the ring system at least one hetero atom selected from N, O and S, which ring system is bound (i.e. through the N bonded to R1 and R6 in formula I) either directly or via a a C1-C6-alkylene group to the remainder of the compound,
- a ring system having a 5- to 14-membered bicylic ring which may be unsubstituted or be substituted with 1, 2 or 3, independently of one another, radicals selected from halogen, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy and C1-C6-haloalkoxy, or

R 2 is, for example,H, halogen, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-haloalkoxy or C1-C6-alkoxy-C1-C6-alkoxy,
and/or salts thereof; and their use as as pesticidal agents.
摘要翻译：式I的化合物，其中例如W，X和Y各自为CH; R 1和R 6彼此独立地例如选自H，C 1 -C 6 - 烷基，C 2 -C 6 - 烯基，C 2 -C 6 - 炔基，C 1 -C 6 - 烷氧基，C 3 -C 8 环烷基，R 7 C（= O）和环系; 条件是R 1和R 6中的至少一个是在环系中至少一个环中含有至少一个选自N，O和S的杂原子的部分或完全不饱和的环系，该环系统被结合（即通过与式I中的R 1和R 6键合的N直接或经由C1-C6-亚烷基与化合物的其余部分键合， - 具有5至14元双环的环系，其可以是未取代的或为被1,2或3个彼此独立地取代为选自卤素，C 1 -C 6 - 烷基，C 1 -C 6 - 卤代烷基，C 1 -C 6 - 烷氧基和C 1 -C 6 - 卤代烷氧基的基团，或R 2是， H，卤素，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6 - 烷氧基，C 1 -C 6卤代烷氧基或C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，和/或其盐; 以及其作为杀虫剂的用途。

6. 发明公开

EP1581546A1 AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4''- OR 4'-POSITION 有权转让
标题翻译： AVERMECTIN-B1- UND AVERMECTIN-B1-MONOSACCHARID-DERIVATE MIT EINEM ALKOXYMETHYLSUBSTITUENTEN INDER 4'' - ODER 4'-STELLUNG
公开(公告)号：EP1581546A1
公开(公告)日：2005-10-05
申请号：EP03810843.7
申请日：2003-12-19
申请人： Syngenta Participations AG
发明人： Maienfisch, Peter , Murphy Kessabi, Fiona , Cassayre, Jérôme , Quaranta, Laura , Pitterna, Thomas , Hueter, Ottmar Franz , Jung, Pierre
IPC分类号： C07H17/08 , A61K31/70 , A61P33/00
CPC分类号： C07H17/08
摘要： Avermectin B1 and avermectin B1 monosaccharide derivative compounds having an alkoxymethyl substituent in the 4″- or 4′-position; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions are provided.
摘要翻译：在4“或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物化合物; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物的农药及其互变异构体; 并提供了这些化合物和组合物的制备方法。

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