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81. 发明授权

EP0592680B1 N-sulfonated carboxamide derivatives as fungicides for plants 失效
标题翻译：的N-磺化羧酰胺衍生物作为杀真菌剂对植物
公开(公告)号：EP0592680B1
公开(公告)日：2000-07-19
申请号：EP93905612.3
申请日：1993-03-03
申请人： KUMIAI CHEMICAL INDUSTRY CO., LTD. , IHARA CHEMICAL INDUSTRY CO., LTD.
发明人： URUSHIBATA, Ikumi, K.I Chem. Res. Inst. Co., Ltd , YOSHIMURA, Takumi, K.I Chem. Res. Inst. Co., Ltd , DEGUCHI, Takeshi, K.I Chem. Res. Inst. Co., Ltd , YONEKURA, Norihisa, K.I Chem. Res. Inst. Co., Ltd. , SAKAI, Junetsu , HAYASHI, Shigeru
IPC分类号： C07D239/52 , C07D251/14 , C07D239/28 , A01N43/54 , C07D239/47 , C07D239/42 , C07D239/34
CPC分类号： C07D239/28 , A01N43/54 , A01N43/66 , C07D239/30 , C07D239/34 , C07D239/42 , C07D239/47 , C07D239/52 , C07D251/20
摘要： An N-sulfonylated, six-membered nitrogenous aromatic carboxamide derivative represented by general formula (I), a process for producing the same, and a pest control agent containing the same as the active ingredient, wherein R1 represents alkyl, alkenyl, etc.; R2 represents hydrogen, alkyl, etc.; R?3 and R4¿ may be the same or different from each other and each represents alkyl, alkoxy, etc.; and X and Y may be the same or different from each other and each represents methine or nitrogen. The derivative exhibits an excellent efficacy even at a low concentration against various diseases caused by algal phytopathogenic bacteria, in particular, downy mildew, and also can control the growth of weeds in lowland and upland fields.

82. 发明公开

EP1003511A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS 失效
标题翻译： ALPHA 1A受体的拮抗剂
公开(公告)号：EP1003511A1
公开(公告)日：2000-05-31
申请号：EP98930349.0
申请日：1998-06-17
申请人： MERCK & CO., INC.
发明人： PATANE, Michael, A. , BOCK, Mark, G.
IPC分类号： A61K31/445 , A61K31/505 , C07D211/18 , C07D239/34 , C07D491/08 , C07D487/04 , C07D401/12 , C07D411/12 , C07D413/12
CPC分类号： C07D239/22 , C07D205/04 , C07D211/56 , C07D401/06 , C07D403/06 , C07D413/06 , C07D417/06 , C07D487/04 , C07D491/04
摘要： This invention relates to certain novel compounds and derivatives thereof, their synthesis, and their use as alpha la adrenergic receptor antagonists. One application of these compounds is in the treatment of benign prostatic hyperplasia. These compounds are selective in their ability to relax smooth muscle tissue enriched in the alpha 1a receptor subtype without at the same time inducing hypotension. One such tissue is found surrounding the urethral lining. Therefore, one utility of the instant compounds is to provide acute relief to males suffering from benign prostatic hyperplasia, by permitting less hindered urine flow. Another utility of the instant compounds is provided by combination with a human 5-alpha reductase inhibitory compound, such that both acute and chronic relief from the effects of benign prostatic hyperplasia are achieved.

83. 发明公开

EP0998285A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS 失效
标题翻译： ALPHA 1A受体ADRENERISCHEN的拮抗剂
公开(公告)号：EP0998285A1
公开(公告)日：2000-05-10
申请号：EP98930356.5
申请日：1998-06-17
申请人： MERCK & CO., INC.
发明人： PATANE, Michael, A. , BOCK, Mark, G. , SELNICK, Harold, G.
IPC分类号： A61K31/445 , A61K31/505 , C07D211/18 , C07D239/34 , C07D491/08 , C07D487/04 , C07D401/12 , C07D411/12 , C07D413/12
CPC分类号： C07D401/14 , C07D403/12 , C07D403/14 , C07D413/12 , C07D413/14 , C07D417/12
摘要： This invention relates to certain novel compounds and derivatives thereof, their synthesis, and their use as alpha 1a adrenoreceptor antagonists. The compounds of the present invention are useful for treating benign prostatic hyperplasia (BPH).

84. 发明公开

EP0945434A4 PROCESS FOR PRODUCING HALOGENATED HETEROARYL COMPOUNDS 失效
标题翻译：用于生产卤代杂芳
公开(公告)号：EP0945434A4
公开(公告)日：2000-02-23
申请号：EP97946159
申请日：1997-12-09
申请人： BANYU PHARMA CO LTD
发明人： OKADA SHIGEMITSU , USHIJIMA RYOSUKE , ISHIKAWA KIYOFUMI
IPC分类号： C07D213/61 , C07D213/79 , C07D213/85 , C07D215/48 , C07D241/44 , B01J27/16 , C07B39/00 , C07D239/34
CPC分类号： C07D213/79 , C07D213/61 , C07D213/85 , C07D215/48 , C07D241/44
摘要： A process for producing compounds represented by general formula (II), wherein X represents halogeno; A?1, A2, and A3¿ are the same or different and each represents carbon or nitrogen, provided that at least one of A?1, A2, and A3¿ is nitrogen; and R?1, R2, R3 and R4¿ are the same or different and each represents hydrogen, lower alkyl, cyano, carboxy, lower alkyloxycarbonyl, carbamoyl, halogeno, nitro, hydroxy, or lower aminoalkyl, provided that when R?1 and R2¿ are adjacent substituents, the two can be bonded to each other to form a five- or six-membered ring optionally having on the ring one substituent selected from the group consisting of lower alkyl, nitryl, carboxy, lower alkyloxycarbonyl, carbamoyl, halogeno, nitro, hydroxy, and lower aminoalkyl, characterized by reacting a compound represented by general formula (I), wherein A?1, A2, A3, R1, R2, R3, and R4¿ have the same meaning as the above, with a halogenated quaternary ammonium salt in the presence of phosphorus pentaoxide.

85. 发明公开

EP0973844A1 COMPOUNDS AND PROCESS FOR CONTROLLING CONE TILT ANGLE IN MIXTURES OF SMECTIC LIQUID CRYSTAL COMPOUNDS 失效
标题翻译：化合物和方法用于检查锥角蝶状结构连接的混合工
公开(公告)号：EP0973844A1
公开(公告)日：2000-01-26
申请号：EP98910468.2
申请日：1998-03-18
申请人： MINNESOTA MINING AND MANUFACTURING COMPANY
发明人： RADCLIFFE, Marc, D. , SAVU, Patricia, M. , SNUSTAD, Daniel, C. , SPAWN, Terence, D.
IPC分类号： C09K19/04 , C09K19/34 , C07D239/26 , C07D239/34
CPC分类号： C07D239/26 , C09K19/04 , C09K19/3469
摘要： A process for controlling the cone tilt angle of a tilted smectic liquid crystal composition comprises the step of combining (a) at least one liquid crystal composition comprising at least one smectic or latent smectic liquid crystal compound comprising (i) an aliphatic fluorocarbon terminal portion comprising a terminal fluoroalkyl or fluoroether group and an alkylene group having at least two carbon atoms and containing at least one catenary ether oxygen atom, (ii) an aliphatic hydrocarbon terminal portion, and (iii) a central core connecting the terminal portions, wherein the alkylene group of the aliphatic fluorocarbon terminal portion is directly linked to the central core by a moiety selected from the group consisting of a covalent bond, -CH=CH-, and -C C-; and (b) at least one liquid crystal composition comprising at least one smectic or latent smectic liquid crystal compound; with the provisos that at least one of the compositions (a) and (b) comprises at least one chiral liquid crystal compound and that the combining of compositions (a) and (b) provides an optically active, tilted chiral smectic liquid crystal composition. The process enables control of cone tilt angle and thereby control of the brightness characteristics of liquid crystal display devices.

86. 发明公开

EP0972770A1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof 有权
标题翻译：杀螨和杀虫活性，取代的嘧啶，以及它们的制备方法
公开(公告)号：EP0972770A1
公开(公告)日：2000-01-19
申请号：EP99305172.1
申请日：1999-06-30
申请人： American Cyanamid Company
发明人： Cuccia, Salvatore John , Wood, William Wakefield , Buckwalter, Brian Lee , Chiarello, John Francis , Fleming, Linda Barbara
IPC分类号： C07D239/42 , C07D239/26 , C07D239/46 , C07D239/34 , A01N43/54
CPC分类号： C07D239/26 , A01N43/54 , C07D239/34 , C07D239/42 , C07D239/47
摘要： The present invention provides compounds of Formula I
methods for their preparation and their use as acaricidal and insecticidal agents.
摘要翻译：本发明提供了式I化合物它们的制备方法和它们作为杀螨和杀虫剂的用途。

87. 发明公开

EP0885875A4 VINYLENE COMPOUNDS AND LIQUID-CRYSTAL COMPOSITION 失效
标题翻译：乙烯基化合物和液晶筹备工作
公开(公告)号：EP0885875A4
公开(公告)日：1999-10-13
申请号：EP97902613
申请日：1997-02-07
申请人： CHISSO CORP
发明人： KONDO TOMOYUKI , MATSUI SHUICHI , MIYAZAWA KAZUTOSHI , SEKIGUCHI YASUKO , NAKAGAWA ETSUO
IPC分类号： C07C69/75 , C07C69/753 , C07C69/76 , C07D213/79 , C07D213/80 , C07D239/28 , C07D239/34 , C07D319/06 , C09K19/04 , C09K19/30 , C07D213/24 , C07D239/24 , C09K19/20 , C09K19/34 , G02F1/13
CPC分类号： C07D213/79 , C07C69/75 , C07C69/753 , C07C69/76 , C07D213/80 , C07D239/28 , C07D239/34 , C07D319/06 , C09K19/04 , C09K19/3001 , C09K19/3068
摘要： Liquid-crystal compounds represented by the general formula (1): Ra-A1-Z1-A2-Z2-A3-(-Z3-A4-)-m-Rb and having a liquid-crystal phase over a wide temperature range, a low viscosity, and an improved threshold voltage; a liquid-crystal composition; and a liquid-crystal display element containing the liquid-crystal composition (1), wherein Ra represents C1-20 alkyl in which at least one -CH2- may be replaced with -O-, etc. and at least one hydrogen atom may be replaced with a halogen atom; Rb is the same as Ra or is halogeno or cyano; A1, A2, A3, and A4 each independently represents a divalent ring group; Z1, Z2, and Z3 each independently represents C2-C4 alkenylene, -COO-, a covalent bond, etc., provided that at least one of Z1, Z2, and Z3 represents C2-C4 alkenylene and at least one of them represents -COO- or -OCO-; and m is 0 or 1.

88. 发明公开

EP0945434A1 PROCESS FOR PRODUCING HALOGENATED HETEROARYL COMPOUNDS 失效
标题翻译： VERFAHREN ZUR HERSTELLUNG VON HALOGENIERTEN HETEROARYLVERBINDUNGEN
公开(公告)号：EP0945434A1
公开(公告)日：1999-09-29
申请号：EP97946159.7
申请日：1997-12-09
申请人： BANYU PHARMACEUTICAL CO., LTD.
发明人： OKADA, Shigemitsu, Banyu Pharm. Co. Ltd Okazaki st , USHIJIMA, Ryosuke, Banyu Pharm. Co. Ltd , ISHIKAWA, Kiyofumi, Banyu Pharm. Co Ltd R&D Lab
IPC分类号： C07D213/61 , C07D215/48 , C07D239/34 , B01J27/16
CPC分类号： C07D213/79 , C07D213/61 , C07D213/85 , C07D215/48 , C07D241/44
摘要： The present invention relates to a process for producing a compound represented by the following general formula [II]:
wherein X is a halogen atom, each of A 1 , A 2 and A 3 may be identical or different, is a carbon atom or a nitrogen atom, provided that at least one of A 1 , A 2 and A 3 is a nitrogen atom, and each of R 1 , R 2 , R 3 and R 4 may be identical or different, is a hydrogen atom, a lower alkyl group, a cyano group, a carboxyl group, a lower alkoxycarbonyl group, a carbamoyl group, a halogen atom, a nitro group, a hydroxyl group or an amino-(lower alkyl) group, provided that in cases where R 1 and R 2 are adjacent to each other, R 1 and R 2 may be combined with each other to form a 5- or 6-membered ring which may carry on the ring thereof one substituent selected from the group consisting of a lower alkyl group, a nitrile group, a carboxyl group, a lower alkoxycarbonyl group, a carbamoyl group, a halogen atom, a nitro group, a hydroxyl group and an amino-(lower alkyl) group; characterized by reacting a compound represented by the following general formula [I]:
wherein A 1 , A 2 , A 3 , R 1 , R 2 , R 3 and R 4 are as defined above, with a quaternary ammonium halide in the presence of phosphorus pentoxide.
摘要翻译：本发明涉及一种制备由以下通式表示的化合物的方法：其中X是卤素原子，A 1，A 2和A 3中的每一个可以相同或不同是碳原子或氮原子，条件是A 1，A 2和A 3中的至少一个为氮原子，R 1，R 2，R 3， 3>和R 4可以相同或不同，是氢原子，低级烷基，氰基，羧基，低级烷氧基羰基，氨基甲酰基，卤素原子，硝基，羟基基团或氨基 - （低级烷基）基团，条件是在R 1和R 2彼此相邻的情况下，R 1和R 2可以彼此结合形成5 - 或6元环，其可以带有一个选自低级烷基，腈基，羧基，低级烷氧基羰基，氨基甲酰基，卤素原子，硝基的取代基，羟基和氨基 - （低级烷基）基团; 其特征在于使由以下通式表示的化合物：其中A 1，A 2，A 3，R 1，R 2，R 3和R 4， >如上定义，在五氧化二磷的存在下与季铵卤化物反应。

89. 发明授权

EP0736001B1 ARYLESSIGSÄUREDERIVATE UND IHRE VERWENDUNG ALS FUNGIZIDE 失效
标题翻译：芳基乙酸衍生物和它们作为杀真菌剂使用
公开(公告)号：EP0736001B1
公开(公告)日：1999-06-09
申请号：EP95904446.2
申请日：1994-12-09
申请人： BAYER AG
发明人： KLEEFELD, Gerd , TIEMANN, Ralf , GERDES, Peter , HEINEMANN, Ulrich , DEHNE, Heinz-Wilhelm , DUTZMANN, Stefan , STENZEL, Klaus
IPC分类号： C07C251/52 , C07C235/34 , C07C255/64 , C07C251/60 , A01N37/50 , A01N37/36 , A01N43/00 , C07D417/04 , C07D213/54 , C07D333/24 , C07D213/53 , C07D239/34
CPC分类号： C07D213/53 , A01N37/50 , C07C251/52 , C07D213/63 , C07D239/52 , C07D285/08 , C07D333/32 , C07D417/04

90. 发明授权

EP0574418B1 ARYLSULFONYLHARNSTOFFE, VERFAHREN ZU IHRER HERSTELLUNG UND IHRE VERWENDUNG ALS HERBIZIDE UND WACHSTUMSREGULATOREN 有权转让
标题翻译： Arylsulfonylureas，其制造方法相同，它们作为除草剂和生长调节
公开(公告)号：EP0574418B1
公开(公告)日：1998-11-11
申请号：EP92904460.0
申请日：1992-02-12
申请人： Hoechst Schering AgrEvo GmbH
发明人： ORT, Oswald , BAUER, Klaus , BIERINGER, Hermann
IPC分类号： C07D239/42 , A01N47/36 , C07D239/47 , C07D239/52 , C07D239/34 , C07D251/46 , C07D251/14 , C07D251/42
CPC分类号： C07D521/00 , A01N47/36 , C07C311/16 , C07C311/65
摘要： The invention concerns new herbicidal and plant-growth regulation compounds of formula (I), in which Q, W, R?1, R2, R3¿, Y and Z as shown in formula (I) are as defined in claim 1, as well as salts of these compounds. They can be prepared by reacting new compounds of formula (II) with a heterocyclic carbamate of formula (III), in which R' is a substituted or unsubstituted alkyl or aryl group. Also possible is an analogue preparation by reacting a phenyl sulphonyl carbamate or sulphonyl isocyanate corresponding to formula (II) with a compound of formula (V). Such herbicides are particularly suited for the selective control of weeds.

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