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71. 发明授权

EP0002741B1 Perfluoroalkyl-iodo norbornane compounds and their use as surfactants 失效
标题翻译：全氟代碘代诺贝恩化合物及其作为表面活性剂的用途
公开(公告)号：EP0002741B1
公开(公告)日：1981-11-18
申请号：EP78101696.9
申请日：1978-12-15
申请人： CIBA-GEIGY AG
发明人： Brace, Neal O.
IPC分类号： C07C61/12 , C07C103/19 , C07C103/737 , C07D209/76 , C07B29/04 , C07C69/74 , C07D307/77 , B01F17/00
CPC分类号： C07C61/15 , C07D307/93

72. 发明公开

EP0002620A1 Cycloalkyl carboxylic esters, insecticidal compositions containing them, and methods for their preparation 失效
标题翻译： Cycloalkylcarboxylester，含有杀虫它们的制备方法和组合物。
公开(公告)号：EP0002620A1
公开(公告)日：1979-06-27
申请号：EP78300845.1
申请日：1978-12-18
申请人： COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION
发明人： Holan, George , O'Keefe, David Francis
IPC分类号： C07C61/40 , C07C62/32 , C07C69/74 , C07C121/75 , C07D307/40 , C07D317/60 , C07C149/30 , A01N37/08
CPC分类号： A01N37/48 , A01N37/08 , A01N37/10 , A01N37/34 , A01N37/38 , A01N43/08 , A01N43/30 , C07C61/15 , C07C61/40 , C07C62/12 , C07C62/34 , C07C69/753 , C07C69/757 , C07D317/60
摘要： New compounds are described that fall within the general formula I
wherein R' is hydrogen or a methoxy, ethoxy, propoxy, butoxy, tetrafluoroethoxy, methylthio, ethylthio, propylthio, fluoro, chloro, bromo, methyl, ethyl, or nitro group, and R 2 is hydrogen or a methyl group, or R' and R 2 together form a methylenedioxy group; and R 3 is hydrogen, or halogen or an esterifying group, as well as other derivatives of the acid. The I esterifying group may be a lower alkyl group, or one of the following groups (a) to (f):-

(a) 3-phenoxybenzyl
(b) 2-benzyl-4-furylmethyl
(c) a-cyano-3-phenoxybenzyl
(d) 3,4-methylenedioxybenzyl
(e) a-ethynyl-3-phenoxybenzyl
(f) α-cyano-3-(4'-chlorophenoxyl)-benzyl

and Y 1 , y 2 , Y 3 , Y 4 , Y 5 and Y 6 are the same or different groups and each is hydrogen or a fluoro, bromo or chloro group, with the proviso that when R' is fluoro, chloro, bromo or methyl and R 2 is hydrogen, then one of Y' to Y 6 is other than hydrogen. Processes of making the compounds are described. The compounds in which R 3 is one of groups (a) to (f) are insecticides and insecticidal methods and compositions containing them are described.
摘要翻译：新化合物被描述并落在通式I内... ... worin - [R <1>是氢或甲氧基，乙氧基，丙氧基，丁氧基，四氟乙氧基，甲硫基，乙硫基，丙，氟，氯，溴，甲基，乙基，或硝基，且R <2>是氢或甲基，或者R <1>和R <2>一起形成亚甲二氧基; 且R为氢<3>是，或卤素，或通过酯化基团，以及所述酸的其它衍生物。酯化基团可以是低级烷基，或下列基团的（a）至（f）中的一项： - ...（一）3-苯氧基...（B）2-苄基-4-呋喃基甲基...（c）中的α-氰基 -3-苯氧基苄基...（D）3,4-亚甲...（e）中的α- - 乙炔基-3-苯氧基苄...（F）α-氰基-3-（4分钟-chlorophenoxyl） - 苄基......和Y <1>，Y <2>，Y <3>，Y <4>ý<5>和Y <6>是相同的或不同的基团，各自为氢或氟，溴或氯基团，条件做当R <1 >是氟，氯，溴或甲基，R <2>是氢，则Y <1>中的一个为Y <6>不是氢。制备所述化合物的方法被描述。化合物，其中R <3>是基团（a）至（f）是杀虫剂和杀昆虫的方法和含有它们的组合物描述的一个。

73. 发明公开

EP2978456A1 RADIOLABELLING PROCESS 有权转让
标题翻译：放射性过程
公开(公告)号：EP2978456A1
公开(公告)日：2016-02-03
申请号：EP14713479.5
申请日：2014-03-28
申请人： GE Healthcare Limited
发明人： WICKSTROM, Torild
IPC分类号： A61K51/04 , C07B59/00
CPC分类号： A61K51/0402 , A61K51/0406 , A61K51/0497 , C07B59/001 , C07B2200/05 , C07C51/377 , C07C61/15 , C07C227/20 , C07C269/06 , C07C2601/04 , C07C271/24 , C07C229/48
摘要： The present invention relates to a novel composition comprising 1-amino-3[18F]-fluorocyclobutanecarboxylic acid ([18F]-FACBC) wherein said composition has certain superior properties in comparison with known compositions comprising [18F]-FACBC. Also provided by the invention is a method to obtain said composition.
摘要翻译：本发明涉及包含1-氨基-3- [18 F] - 氟环丁烷羧酸（[18 F] -FACBC）的新型组合物，其中所述组合物与包含[18 F] -FACBC的已知组合物相比具有某些优越性质。本发明还提供了获得所述组合物的方法。

74. 发明公开

EP2003113A4 PROCESS FOR PRODUCTION OF CARBOXYLIC ACID CHLORIDE COMPOUND 审中-公开
标题翻译：法生产碳酸氯化物的
公开(公告)号：EP2003113A4
公开(公告)日：2012-07-18
申请号：EP07740213
申请日：2007-03-29
申请人： AJINOMOTO KK
发明人： ISHIKAWA TATSUYA , KONDOU SHOUICHI , TAKAHASHI SATOJI
IPC分类号： C07C51/60 , C07B53/00 , C07B61/00 , C07C61/15 , C07C231/02 , C07C233/63
CPC分类号： C07C231/02 , C07B53/00 , C07C51/60 , C07C2601/14 , C07C61/15 , C07C233/63

75. 发明公开

EP2003113A1 PROCESS FOR PRODUCTION OF CARBOXYLIC ACID CHLORIDE COMPOUND 审中-公开
标题翻译： VERFAHREN ZUR PRODUKTION EINERCARBONSÄURECHLORIDVERBINDUNG
公开(公告)号：EP2003113A1
公开(公告)日：2008-12-17
申请号：EP07740213.9
申请日：2007-03-29
申请人： Ajinomoto Co., Inc.
发明人： ISHIKAWA, Tatsuya , KONDOU, Shouichi , TAKAHASHI, Satoji
IPC分类号： C07C51/60 , C07C61/15 , C07C231/02 , C07C233/63 , C07B53/00 , C07B61/00
CPC分类号： C07C231/02 , C07B53/00 , C07C51/60 , C07C2601/14 , C07C61/15 , C07C233/63
摘要： The present invention discloses methods for producing a carboxylic acid chloride compound which comprises the step of reacting an alkyl-substituted cyclohexyl carboxylic acid with a chlorinating agent in the presence of a specific urea compound. According to this invention, it is possible to produce a carboxylic acid chloride compound which has high reaction speed, and whose product has high purity or high yield. Thus produced carboxylic acid chloride compound is useful as an intermediate for producing D-phenylalanine derivatives which are used as agents for treating diabetes.
摘要翻译：本发明公开了制备羧酰氯化合物的方法，其包括在特定脲化合物存在下使烷基取代的环己基羧酸与氯化剂反应的步骤。根据本发明，可以制备反应速度快，产物纯度高，产率高的羧酸酰氯化合物。这样制得的羧酰氯化合物可用作生产D-苯丙氨酸衍生物的中间体，其用作治疗糖尿病的药物。

76. 发明公开

EP1303474A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY PURE PYRETHROID INSECTICIDES 有权
标题翻译：用于生产对映纯的拟除虫菊酯杀虫剂
公开(公告)号：EP1303474A1
公开(公告)日：2003-04-23
申请号：EP01949710.6
申请日：2001-07-16
申请人： Syngenta Limited
发明人： BROWN, Stephen, Martin , GOTT, Brian, David
IPC分类号： C07C51/41 , C07C51/43 , C07C51/60 , C07C69/34 , C07C69/62 , C07C53/23 , C07C51/09 , A01N53/00
CPC分类号： C07C51/60 , C07B2200/07 , C07C51/09 , C07C51/412 , C07C61/15 , C07C67/14 , C07C61/40 , C07C53/21 , C07C53/50 , C07C69/743
摘要： A process for producing compounds of formula (VIIa) and (VIIb) wherein X is a leaving group; Y and Y1 are idependently Cl or Br; and Z is Cl, Br or a haloalkyl group which process comprises a) reacting a compound of formula (VII) wherein X, Y, Y1 and Z are as defined for compounds (VIIa) and (VIIb) with a substantially optically pure chiral amine in a solvent to form a diastereoisomeric salt; b) separating the diastereomeric salt of each enantiomer; c) converting the diastereomeric salt of each anantiomer separately to compounds of formulae (VIIa) and (VIIb) respectively by acid or base hydrolysis, the use of the compounds in making pyrethroid insecticides and novel intermediates.

77. 发明授权

EP0726244B1 Process for producing 2-fluorocyclopropanecarboxylic acid 失效
标题翻译：一种用于2-氟环丙烷羧酸的制备方法
公开(公告)号：EP0726244B1
公开(公告)日：1998-08-12
申请号：EP96300680.4
申请日：1996-01-31
申请人： SUMITOMO CHEMICAL COMPANY LIMITED , Daiichi Pharmaceutical Co., Ltd.
发明人： Itaya, Nobushige , Wakita, Ryuhei , Kubo, Asako , Sasaki, Mikio , Namba, Takashi , Yukimoto, Yusuke
IPC分类号： C07C51/347 , C07C61/15
CPC分类号： C07C61/15 , C07C51/377

78. 发明公开

EP0712831A4 SELECTIVE DEHALOGENATION METHOD 失效
标题翻译：选择性脱卤
公开(公告)号：EP0712831A4
公开(公告)日：1996-09-25
申请号：EP94923063
申请日：1994-08-03
申请人： DAIICHI SEIYAKU CO
发明人： AKIBA TOSHIFUMI , IKEYA TAKANOBU , KAWANISHI HIROFUMI , YUKIMOTO YUSUKE , KAMIHARA SHINJI , EBATA TSUTOMU
IPC分类号： C07C51/377 , C07C67/317 , C07C61/15 , C07C51/347 , C07C69/74
CPC分类号： C07C51/377 , C07C67/317 , C07C61/15 , C07C69/74
摘要： A convenient process for producing a compound represented by general formula (2) by the catalytic hydrogenolysis of a compound represented by general formula (1) or (3) in the presence of a base, wherein R represents hydrogen or C1-C4 alkyl; and X represents chlorine or bromine. The obtained compound can be used as an intermediate for producing medicines.

79. 发明公开

EP0712831A1 SELECTIVE DEHALOGENATION METHOD 失效
标题翻译：选择性脱卤方法
公开(公告)号：EP0712831A1
公开(公告)日：1996-05-22
申请号：EP94923063.5
申请日：1994-08-03
申请人： DAIICHI PHARMACEUTICAL CO., LTD.
发明人： AKIBA, Toshifumi, Daiichi Pharmaceutical Co. Ltd. , IKEYA, Takanobu, Daiichi Pharmaceutical Co., Ltd. , KAWANISHI, Hirofumi, Daiichi Pharmaceutical Co. L , YUKIMOTO, Yusuke Daiichi Pharmaceutical Co., Ltd. , KAMIHARA, Shinji Daiichi Pharmaceutical Co., Ltd. , EBATA, Tsutomu Daiichi Pharmaceutical Co., Ltd.
IPC分类号： C07C61/15 , C07C51/347 , C07C69/74 , C07C67/317
CPC分类号： C07C51/377 , C07C67/317 , C07C61/15 , C07C69/74
摘要： A convenient process for producing a compound represented by general formula (2) by the catalytic hydrogenolysis of a compound represented by general formula (1) or (3) in the presence of a base, wherein R represents hydrogen or C₁-C₄ alkyl; and X represents chlorine or bromine. The obtained compound can be used as an intermediate for producing medicines.
摘要翻译：通过通式（1）或（3）代表的化合物在碱存在下的催化氢解生产通式（2）代表的化合物的简便方法，其中R代表氢或C 1 -C 4烷基; X代表氯或溴。所获得的化合物可以用作生产药物的中间体。

80. 发明授权

EP0341475B1 Stereoisomere von N-(R)-1-Aryl-ethyl)-1-alkyl-2,2-dichlo-cyclopropancarbonsäureamiden 失效
标题翻译： N-（R）-1-芳基 - 乙基）-1-烷基-2,2-二氯甲基碳酰胺的立体异构体
公开(公告)号：EP0341475B1
公开(公告)日：1993-09-29
申请号：EP89107326.4
申请日：1989-04-24
申请人： BAYER AG
发明人： Kraatz, Udo, Dr. , Hänssler, Gerd, Dr.
IPC分类号： C07C233/57 , C07C231/02 , C07C61/15 , C07C69/635 , A01N53/00
CPC分类号： A01N53/00 , C07C61/15 , C07C233/58 , C07C2601/02

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