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1. 发明授权

US5986135A Fungicidal trifluoromethylalkylamino-triazolopyrimidines 失效
标题翻译：杀真菌三氟甲基烷基氨基 - 三唑并嘧啶
公开(公告)号：US5986135A
公开(公告)日：1999-11-16
申请号：US160894
申请日：1998-09-25
申请人： Waldemar Pfrengle , Klaus-Juergen Pees , Guido Albert , Paul Carter , Annerose Rehnig , Henry Van Tuyl Cotter
发明人： Waldemar Pfrengle , Klaus-Juergen Pees , Guido Albert , Paul Carter , Annerose Rehnig , Henry Van Tuyl Cotter
IPC分类号： C07D487/04 , A01N43/90 , C07C209/88 , C07C211/15
CPC分类号： C07D487/04 , C07C209/88 , C07B2200/07
摘要： An improved process for the preparation of (S)-1,1,1-trifluoroalkyl-2-amines of formula IIIA, ##STR1## where R.sup.1 is a C.sub.1-6 alkyl group, from the corresponding racemic mixture, which process includes treating 1 part by mole of the racemic mixture with approximately 0.3 to 0.7 part by mole of D-(-)-tartaric acid in the presence of an inert solvent.
摘要翻译：从相应的外消旋混合物制备式IIIA（其中R 1为C 1-6烷基）的（S）-1,1,1-三氟烷基-2-胺的改进方法，该方法包括处理1摩尔的外消旋混合物，在惰性溶剂的存在下，约0.3〜0.7份摩尔的D - （ - ） - 酒石酸。

2. 发明授权

US06204269B1 Fungicidal trifluoromethylalkylamino-triazolopyrimidines 失效
标题翻译：杀真菌三氟甲基烷基氨基 - 三唑并嘧啶
公开(公告)号：US06204269B1
公开(公告)日：2001-03-20
申请号：US09406574
申请日：1999-09-24
申请人： Waldemar Pfrengle , Klaus-Juergen Pees , Guido Albert , Paul Carter , Annerose Rehnig , Henry Van Tuyl Cotter
发明人： Waldemar Pfrengle , Klaus-Juergen Pees , Guido Albert , Paul Carter , Annerose Rehnig , Henry Van Tuyl Cotter
IPC分类号： A01N4390
CPC分类号： C07D487/04 , C07B2200/07 , C07C209/88 , C07C211/15
摘要： The novel optically active compounds of formula I: (R1, Hal and L1 through L5 are defined in the specification) wherein the enantiomeric excess of the (S)-enantiomer is at least 70%., show enhanced selective fungicidal activity. The new compounds are processed with carriers, and optionally with adjuvants, to form fungicidal compositions.
摘要翻译：式（I）的新型光学活性化合物：（R 1，Hal和L 1至L 5在本说明书中定义），其中（S） - 对映异构体的对映异构体过量至少为70％，表现出增强的选择性杀真菌活性。新的化合物用载体和任选地与佐剂一起加工以形成杀真菌组合物。

3. 发明授权

US07084146B2 Fungicidal trifluoromethylalkylamino-triazolopyrimidines 失效
标题翻译：杀真菌三氟甲基烷基氨基 - 三唑并嘧啶
公开(公告)号：US07084146B2
公开(公告)日：2006-08-01
申请号：US09840488
申请日：2001-04-23
申请人： Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
发明人： Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
IPC分类号： C07D487/04 , A01N43/90
CPC分类号： C07D487/04 , A01N43/90
摘要： The novel compounds of formula I: wherein R1 is hydrogen or methyl; R2 is hydrogen, or an optionally substituted alkyl, alkenyl, alkynyl, alkadienyl or phenyl group; Hal is halogen; and L1 through L5 are each hydrogen, halogen, alkyl, alkoxy or nitro, provided that at least one of L1 through L5 represents nitro or alkoxy; show selective fungicidal activity. The new compounds are processed with carriers and adjuvants to fungicidal compositions.
摘要翻译：式I的新化合物：其中R 1是氢或甲基; R 2是氢或任选取代的烷基，烯基，炔基，链二烯基或苯基; 卤素是卤素; 和L 1至L 5各自为氢，卤素，烷基，烷氧基或硝基，条件是L 1至L 2中的至少一个， SUP> 5表示硝基或烷氧基; 显示选择性杀真菌活性。新的化合物用载体和佐剂加工成杀真菌剂。

4. 再颁专利

USRE40332E1 Fungicidal trifluoromethylalkylamino-triazolopyrimidines 失效
标题翻译：杀真菌三氟甲基烷基氨基 - 三唑并嘧啶
公开(公告)号：USRE40332E1
公开(公告)日：2008-05-20
申请号：US10643707
申请日：2003-08-20
申请人： Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
发明人： Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
IPC分类号： C07D239/00 , C07D487/00 , C07D487/04 , A61K31/505 , A61K43/54
CPC分类号： C07D487/04 , A01N43/90
摘要： The novel compounds of formula I: wherein (R1, R2, Hal and L1 through L5 are defined in the specification) show selective fungicidal activity. The new compounds may be processed with carriers and adjuvants to produce fungicidal compositions.
摘要翻译：式I的新化合物：其中（R 1，R 2，R 2，Hal和L 1至L 5）在规范中定义）显示选择性杀真菌活性。可以用载体和佐剂处理新的化合物以产生杀真菌组合物。

5. 发明授权

US5948783A Fungicidal trifluoromethylalkylamino-triazolopyrimidines 失效
标题翻译：杀真菌三氟甲基烷基氨基 - 三唑并嘧啶
公开(公告)号：US5948783A
公开(公告)日：1999-09-07
申请号：US54580
申请日：1998-04-03
申请人： Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
发明人： Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
IPC分类号： A01N43/90 , C07D487/04 , A01N43/54
CPC分类号： C07D487/04 , A01N43/90
摘要： The novel compounds of formula I: ##STR1## wherein R.sup.1, R.sup.2, Hal and L.sup.1 through L.sup.5, are defined in the specification show selective fungicidal activity.
摘要翻译：式I的新化合物：其中R1，R2，Hal和L1至L5在本说明书中定义为选择性杀真菌活性。

6. 发明授权

US06255309B1 Fungicidal trifluoromethylalkylamino-triazolopyrimidines 有权
标题翻译：杀真菌三氟甲基烷基氨基 - 三唑并嘧啶
公开(公告)号：US06255309B1
公开(公告)日：2001-07-03
申请号：US09272916
申请日：1999-03-19
申请人： Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
发明人： Klaus-Juergen Pees , Guenter Krummel , Henry Van Tuyl Cotter , Guido Albert , Annerose Rehnig , Leslie May , Waldemar Pfrengle
IPC分类号： A61K31505
CPC分类号： C07D487/04 , A01N43/90
摘要： The novel compounds of formula I: wherein (R1, R2, Hal and L1 through L5 are defined in the specification) show selective fungicidal activity. The new compounds may be processed with carriers and adjuvants to produce fungicidal compositions.
摘要翻译：式I的新化合物：其中（R1，R2，Hal和L1至L5在说明书中定义）表示选择性杀真菌活性。可以用载体和佐剂处理新的化合物以产生杀真菌组合物。

7. 发明授权

US06380202B1 Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines 失效
标题翻译：杀真菌氟取代的7-杂环基 - 三唑并嘧啶
公开(公告)号：US06380202B1
公开(公告)日：2002-04-30
申请号：US09405658
申请日：1999-09-24
申请人： Klaus-Juergen Pees , Annerose Rehnig , Guido Albert
发明人： Klaus-Juergen Pees , Annerose Rehnig , Guido Albert
IPC分类号： A61K31519
CPC分类号： C07D487/04 , A01N43/90 , A61K31/519
摘要： The novel compounds of formula I: wherein (R1, R2, Hal and L1 through L5 are defined in the specification) show selective fungicidal activity and high systemicity. The new compounds are processed with carriers and adjuvants to fungicidal compositions.
摘要翻译：式I的新化合物：其中（R1，R2，Hal和L1至L5在本说明书中定义）表示选择性杀真菌活性和高系统性。新的化合物用载体和佐剂加工成杀真菌剂。

8. 发明授权

US6020338A Fungicidal 7-alkyl-triazolopyrimidines 失效
标题翻译：杀真菌剂7-烷基 - 三唑并嘧啶
公开(公告)号：US6020338A
公开(公告)日：2000-02-01
申请号：US243851
申请日：1999-02-03
申请人： Waldemar Pfrengle , Klaus-Juergen Pees , Guido Albert
发明人： Waldemar Pfrengle , Klaus-Juergen Pees , Guido Albert
IPC分类号： A01N43/90 , C07D487/04 , A01N43/54
CPC分类号： C07D487/04 , A01N43/90
摘要： The novel compounds of formula I: whereinR.sup.1 represents an optionally substituted alkyl, alkenyl, alkynyl, alkadienyl, or aryl group, or an optionally substituted cycloalkyl or cycloalkenyl group, in which one CH.sub.2 group may also be replaced by O, S or NR.sup.2, in which R.sup.2 represents a hydrogen atom or an alkyl group;X represents a hydrogen or halogen atom, or an alkoxy, aryloxy, aralkyloxy, haloalkoxy, alkylthio, cyano, amino, alkylamino or dialkylamino group;L.sup.1, L.sup.2, L.sup.3, L.sup.4 and L.sup.5 each independently represent an hydrogen or halogen atom or an optionally substituted alkyl or alkoxy group or a nitro or cyano group show selective fungicidal activity. The new compounds are processed with carriers and, optionally, adjuvants, to afford fungicidal compositions, useful in agricultural applications.
摘要翻译：式I的新化合物：其中R 1表示任选取代的烷基，烯基，炔基，链二烯基或芳基，或任选取代的环烷基或环烯基，其中一个CH 2基团也可被O，S或NR 2取代，其中R2表示氢原子或烷基; X表示氢或卤素原子，或烷氧基，芳氧基，芳烷氧基，卤代烷氧基，烷硫基，氰基，氨基，烷基氨基或二烷基氨基; L1，L2，L3，L4和L5各自独立地表示氢或卤素原子或任选取代的烷基或烷氧基或硝基或氰基显示选择性杀真菌活性。用载体和任选的佐剂处理新的化合物，得到可用于农业应用的杀真菌组合物。

9. 发明申请

US20050282847A1 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines 失效
标题翻译：杀真菌剂5-苯基取代的2-（氰基氨基）嘧啶
公开(公告)号：US20050282847A1
公开(公告)日：2005-12-22
申请号：US11186087
申请日：2005-07-22
申请人： Klaus-Juergen Pees , Waldemar Pfrengle , Gavin Heffernan
发明人： Klaus-Juergen Pees , Waldemar Pfrengle , Gavin Heffernan
IPC分类号： C07D239/42 , A01N43/54 , A01N47/40 , A61K31/519 , C07D239/48 , C07D401/04 , C07D409/12 , C07D487/04
CPC分类号： C07D239/48 , A01N43/54 , A01N47/40 , C07D239/38 , C07D401/04 , C07D487/04
摘要： Pyrimidines of formula I in which R1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxy-carbonyl, wherein R1 groups are unsubstituted or substituted as defined in the specification; R2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR5 or a single bond, wherein R5 represents hydrogen or alkyl; or R1 and R5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.
摘要翻译：式I的嘧啶，其中R 1表示氢或烷基，卤代烷基，烯基，炔基，链烯基，烷氧基，环烷基，苯基或5-或6-元杂芳基或5-或6-元杂环基，含有一至四个氮原子或一至三个氮原子和一个硫或氧原子，或三烷基甲硅烷基，甲酰基或烷氧基 - 羰基，其中R 1是未被取代或如所定义的取代在规范中; R 2表示含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的未取代或取代的苯基，环烷基或5或6元杂芳基; R 3表示氢，卤素或烷基，烷氧基，烷硫基，烷基氨基或二烷基氨基; 其为未取代或取代的; R 4表示氢或烷基，烯基或炔基; 其为未取代或取代的; 并且X表示O，S，NR 5或单键，其中R 5表示氢或烷基; 或R 1和R 5连同中间的氮原子一起形成杂环; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制有害真菌的用途。

10. 发明授权

US06943252B2 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines 失效
标题翻译：杀真菌剂5-苯基取代的2-（氰基氨基）嘧啶
公开(公告)号：US06943252B2
公开(公告)日：2005-09-13
申请号：US10615352
申请日：2003-07-09
申请人： Klaus-Juergen Pees , Waldemar Pfrengle , Gavin Heffernan
发明人： Klaus-Juergen Pees , Waldemar Pfrengle , Gavin Heffernan
IPC分类号： C07D239/42 , A01N43/54 , A01N47/40 , A61K31/519 , C07D239/48 , C07D401/04 , C07D409/12 , C07D487/04 , C07D239/02
CPC分类号： C07D239/48 , A01N43/54 , A01N47/40 , C07D239/38 , C07D401/04 , C07D487/04
摘要： Pyrimidines of formula I in which R1 represents hydrogen or alkyl, haloalkyl, alkenyl, alkynyl, alkadienyl, alkoxy, cycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or tri-alkyl-silyl, formyl or alkoxycarbonyl, wherein R1 groups are unsubstituted or substituted as defined in the specification; R2 represents phenyl, cycloalkyl or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which are unsubstituted or substituted; R3 represents hydrogen, halogen or alkyl, alkoxy, alkylthio, alkylamino or dialkylamino; which are unsubstituted or substituted; R4 represents hydrogen or alkyl, alkenyl or alkynyl; which are unsubstituted or substituted; and X represents O, S, NR5 or a single bond, wherein R5 represents hydrogen or alkyl; or R1 and R5 together with the interjacent nitrogen atom form a heterocyclic ring; processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling harmful fungi.
摘要翻译：式I的嘧啶，其中R 1表示氢或烷基，卤代烷基，烯基，炔基，链烯基，烷氧基，环烷基，苯基或5-或6-元杂芳基或5-或6-元杂环基，其含有一至四个氮原子或一至三个氮原子和一个硫或氧原子，或三烷基甲硅烷基，甲酰基或烷氧基羰基，其中R 1'是未取代的或如规范; R 2表示含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的未取代或取代的苯基，环烷基或5或6元杂芳基; R 3表示氢，卤素或烷基，烷氧基，烷硫基，烷基氨基或二烷基氨基; 其为未取代或取代的; R 4表示氢或烷基，烯基或炔基; 其为未取代或取代的; 并且X表示O，S，NR 5或单键，其中R 5表示氢或烷基; 或R 1和R 5连同中间的氮原子一起形成杂环; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制有害真菌的用途。

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