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1. 发明授权

US5256666A 3-Isoxazolylphenyl compounds, their preparation and their use 失效
标题翻译： 3-异恶唑基苯基化合物，其制备及其应用
公开(公告)号：US5256666A
公开(公告)日：1993-10-26
申请号：US975733
申请日：1992-11-13
申请人： Stefan Mueller , Hans Theobald , Harald Rang , Volker Harries
发明人： Stefan Mueller , Hans Theobald , Harald Rang , Volker Harries
IPC分类号： A01N55/00 , A01N55/10 , C07F7/08 , C07F7/10 , A01N43/54 , A01N43/80 , C07D231/12 , C07D231/16
CPC分类号： A01N55/00 , C07F7/0812
摘要： 3-Isoxazolylphenyl compounds Ia and Ib ##STR1## where R is halogen; alkyl; haloalkyl; alkoxy; haloalkoxy; alkenyl; haloalkenyl; unsubstituted or substituted phenylethenyl; alkynyl; cycloalkyl; aryl; hetaryl; CO.sub.2 R.sup.6 or CONR.sup.7 R.sup.8,R.sup.6 is hydrogen, alkyl, cycloalkyl or benzyl;R.sup.7 and R.sup.8 are each hydrogen, alkyl, cycloalkyl or benzyl or, together with the nitrogen atom to which they are bonded, form a heterocyclic radical;n is 0, 1 or 2;R.sup.1 is halogen or alkyl;R.sup.2 is hydrogen; alkyl; alkenyl; alkynyl or cyano;R.sup.3 and R.sup.4 independently of one another are each unsubstituted or substituted alkyl, alkenyl, cycloalkyl, phenyl, naphthyl, pyridyl or pyrimidinyl; or R.sup.3 and R.sup.4 together form unsubstituted or substituted alkylene;R.sup.5 is hydrogen; unsubstituted or substituted alkyl or one of the groups stated for R.sup.3 ;X is CH.sub.2, O, S or NR.sup.9 andR.sup.9 is hydrogen, alkyl, cycloalkyl, alkenyl, alkynyl or unsubstituted or substituted benzyl, processes for their preparation, agents containing them and the use thereof.
摘要翻译： 3-异恶唑基苯基化合物Ia和Ib其中R是卤素; 烷基; 卤代烷基烷氧基卤代烷氧基烯基; 卤代烯基未取代或取代的苯乙烯基; 炔基; 环烷基芳基; 杂芳 CO 2 R 6或CONR 7 R 8，R 6是氢，烷基，环烷基或苄基; R 7和R 8各自为氢，烷基，环烷基或苄基，或与它们所键合的氮原子一起形成杂环基; n为0,1或2; R1是卤素或烷基; R2是氢; 烷基; 烯基; 炔基或氰基; 链烯基，环烷基，苯基，萘基，吡啶基或嘧啶基; R 3和R 4各自独立地为未取代或取代的烷基，烯基，环烷基，苯基，萘基，或者R 3和R 4一起形成未取代或取代的亚烷基; R5是氢; 未取代或取代的烷基或为R3表示的基团之一; X为CH 2，O，S或NR 9，R 9为氢，烷基，环烷基，烯基，炔基或未取代或取代的苄基，其制备方法，含有它们的试剂及其用途。

2. 发明授权

US5545664A Substituted phenoxymethylphenyl derivatives, their preparation and their use for controlling pests and fungi 失效
标题翻译：取代的苯氧基甲基苯基衍生物，其制备及其用于防治害虫和真菌的用途
公开(公告)号：US5545664A
公开(公告)日：1996-08-13
申请号：US409039
申请日：1995-03-23
申请人： Reinhard Kirstgen , Klaus Oberdorf , Hubert Sauter , Herbert Bayer , Wassilios Grammenos , Harald Rang , Volker Harries , Gisela Lorenz , Eberhard Ammermann
发明人： Reinhard Kirstgen , Klaus Oberdorf , Hubert Sauter , Herbert Bayer , Wassilios Grammenos , Harald Rang , Volker Harries , Gisela Lorenz , Eberhard Ammermann
IPC分类号： A01N37/38 , A01N37/50 , A01N37/52 , C07C251/48 , C07C251/50 , C07C255/62 , C07C255/64 , C07C259/02 , C07C259/10 , C07C259/18 , C07C323/47 , C07C327/58 , C07D317/18 , C07D333/28 , C07D521/00 , A01N37/34 , A61K31/275
CPC分类号： C07D231/12 , A01N37/50 , A01N37/52 , C07C251/48 , C07C255/64 , C07C259/02 , C07C259/10 , C07C259/18 , C07C327/58 , C07D233/56 , C07D249/08 , C07D317/18 , C07D333/28 , C07C2101/02 , C07C2101/08
摘要： Substituted phenoxymethylphenyl derivatives I ##STR1## X is .dbd.CH--OCH.sub.3, .dbd.C--CH.sub.3 or .dbd.N--OCH.sub.3 ; R.sup.1 is, inter alia,R.sup.2 and R.sup.3 are, inter alia,H, halogen, CN, NO.sub.2, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.2 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 --C.sub.2 -haloalkoxy;R.sup.4 is, inter alia,CN, Cl, Dr, C.sub.1 -C.sub.6 -alkoxy, C.sub.1 -C.sub.6 -alkylthio or C.sub.1 -C.sub.4 -haloalkoxy;R.sup.5 is, inter alia,NO.sub.2, CN, halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.4 -haloalkoxy;n is 0-4; Y is --O--, --NH--, --N(CH.sub.3)--; R.sup.6 is H, C.sub.1 -C.sub.4 -alkyl.The compounds are useful for controlling pests and fungi.
摘要翻译：取代的苯氧基甲基苯基衍生物I X为= CH-OCH 3，= C-CH 3或= N-OCH 3; R1尤其是R2和R3尤其是H，卤素，CN，NO2，C1-C4-烷基，C1-C2-卤代烷基，C1-C4-烷氧基或C1-C2-卤代烷氧基; R4尤其是CN，Cl，Dr，C 1 -C 6 - 烷氧基，C 1 -C 6 - 烷硫基或C 1 -C 4 - 卤代烷氧基; R5尤其是NO 2，CN，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4 - 烷氧基或C 1 -C 4 - 卤代烷氧基; n为0-4; Y是-O - ， - NH - ， - N（CH 3） - ; R6是H，C1-C4-烷基。这些化合物可用于防治害虫和真菌。

3. 发明授权

US5696161A Substituted phenoxymethylphenyl derivatives, their preparation and their use for controlling pests and fungi 失效
标题翻译：取代的苯氧基甲基苯基衍生物，其制备及其用于防治害虫和真菌的用途
公开(公告)号：US5696161A
公开(公告)日：1997-12-09
申请号：US645428
申请日：1996-05-13
申请人： Reinhard Kirstgen , Klaus Oberdorf , Hubert Sauter , Herbert Bayer , Wassilios Grammenos , Harald Rang , Volker Harries , Gisela Lorenz , Eberhard Ammermann
发明人： Reinhard Kirstgen , Klaus Oberdorf , Hubert Sauter , Herbert Bayer , Wassilios Grammenos , Harald Rang , Volker Harries , Gisela Lorenz , Eberhard Ammermann
IPC分类号： A01N37/38 , A01N37/50 , A01N37/52 , C07C251/48 , C07C251/50 , C07C255/62 , C07C255/64 , C07C259/02 , C07C259/10 , C07C259/18 , C07C323/47 , C07C327/58 , C07D317/18 , C07D333/28 , C07D521/00 , A61K31/19 , A61K31/215 , C07C255/07
CPC分类号： C07D231/12 , A01N37/50 , A01N37/52 , C07C251/48 , C07C255/64 , C07C259/02 , C07C259/10 , C07C259/18 , C07C327/58 , C07D233/56 , C07D249/08 , C07D317/18 , C07D333/28 , C07C2101/02 , C07C2101/08
摘要： Substituted phenoxymethylphenyl derivatives I ##STR1## X is .dbd.CH--OCH.sub.3, .dbd.CH--CH.sub.3 or .dbd.N--OCH.sub.3 ; R.sup.1 is, inter alia, R.sup.2 and R.sup.3 are, inter alia, H, halogen, CN, NO.sub.2, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.2 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.2 -haloalkoxy; R.sup.4 is, inter alia, CN, Cl, Br, C.sub.1 -C.sub.6 -alkoxy, C.sub.1 -C.sub.6 -alkylthio or C.sub.1 -C.sub.4 -haloalkoxy; R.sup.5 is, inter alia, NO.sub.2, CN, halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.4 -haloalkoxy; n is 0-4; Y is --O--, --NH--, --N(CH.sub.3)--; R.sup.6 is H, C.sub.1 -C.sub.4 -alkyl. The compounds are useful for controlling pests and fungi.
摘要翻译：取代的苯氧基甲基苯基衍生物I X为= CH-OCH 3，= CH-CH 3或= N-OCH 3; R1尤其是R2和R3尤其是H，卤素，CN，NO2，C1-C4-烷基，C1-C2-卤代烷基，C1-C4-烷氧基或C1-C2-卤代烷氧基; R4尤其是CN，Cl，Br，C1-C6-烷氧基，C1-C6-烷硫基或C1-C4-卤代烷氧基; R5尤其是NO 2，CN，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4 - 烷氧基或C 1 -C 4 - 卤代烷氧基; n为0-4; Y是-O - ， - NH - ， - N（CH 3） - ; R6是H，C1-C4-烷基。这些化合物可用于防治害虫和真菌。

4. 发明授权

US5403838A .alpha.-arylacrylic acid derivatives, their preparation and use for controlling pests and fungi 失效
标题翻译： α-芳基丙烯酸衍生物，它们的制备和用途，用于防治害虫和真菌
公开(公告)号：US5403838A
公开(公告)日：1995-04-04
申请号：US928038
申请日：1992-08-11
申请人： Reinhard Kirstgen , Hans Theobald , Hartmann Koenig , Albrecht Harreus , Klaus Oberdorf , Uwe Kardorff , Volker Harries , Gisela Lorenz , Eberhard Ammermann
发明人： Reinhard Kirstgen , Hans Theobald , Hartmann Koenig , Albrecht Harreus , Klaus Oberdorf , Uwe Kardorff , Volker Harries , Gisela Lorenz , Eberhard Ammermann
IPC分类号： A01N43/36 , A01N43/56 , A01N43/76 , A01N43/80 , C07D207/32 , C07D207/327 , C07D207/337 , C07D207/34 , C07D207/416 , C07D231/12 , C07D231/38 , C07D261/08 , C07D261/10 , C07D261/18 , C07D271/02 , C07D275/02 , C07D275/03 , C07D413/04 , C07D417/04 , C07F9/572 , C07F9/6503 , C07F9/653 , C07F9/6539 , C07D213/30 , C07D307/12 , C07D261/20
CPC分类号： C07D207/337 , A01N43/36 , A01N43/56 , A01N43/80 , C07D231/12 , C07D261/08 , C07D261/10 , C07D275/02 , C07D275/03 , C07D413/04 , C07F9/5722 , C07F9/65033 , C07F9/653 , C07F9/6539
摘要： .alpha.-Arylacrylic acid derivatives of the formula I ##STR1## where the substituents have the following meanings: X C, NY CR.sup.4, N, O, SZ CR.sup.5, N, O, Sn 0 to 4R.sup.1 hydrogen, nitro, cyano, halogen; alkyl, alkoxy, halogenated alkyl, halogenated alkoxy or alkylthio, or, when n is 2, 3 or 4, two adjacent substituents R.sup.1 may together denote a 1,3-butadien-1,4-diyl group which may be substituted;R.sup.2 alkyl; halogenated alkyl, halogen, cyano, nitro, alkoxycarbonyl, dimethylamino, R.sup.2 additionally denotes hydrogen;R.sup.3 hydrogen; substituted or unsubstituted alkyl; a substituted or unsubstituted cyclic structure, which may contain, in addition to carbon atoms, one to three heteroatoms; or a substituted or unsubstituted aromatic system, which may contain, in addition to carbon atoms, one to four nitrogen atoms and one to three heteroatoms;R.sup.4, R.sup.5 hydogen, alkyl; halogenated alKyl, halogen, cyano, nitro, dimethylamino, alkoxycarbonyland pesticides and fungicidal agents containing these compounds.
摘要翻译：式I的α-丙烯酰基丙酸衍生物（I）其中取代基具有以下含义：XC，NY CR4，N，O，SZ CR5，N，O，Sn 0至4 R1氢，硝基，氰基，卤素; 烷基，烷氧基，卤代烷基，卤代烷氧基或烷硫基，或当n为2,3或4时，两个相邻的取代基R1可以一起表示可被取代的1,3-丁二烯-1,4-二基; R2烷基; 卤代烷基，卤素，氰基，硝基，烷氧基羰基，二甲基氨基，R2另外表示氢; R3氢; 取代或未取代的烷基; 取代或未取代的环状结构，除了碳原子外，还可含有一至三个杂原子; 或取代或未取代的芳族体系，除了碳原子外，还可以含有一至四个氮原子和一至三个杂原子; R4，R5氢原子，烷基; 卤代烷基，卤素，氰基，硝基，二甲基氨基，烷氧基羰基，农药和含有这些化合物的杀真菌剂。

5. 发明授权

US5935965A 2-�(2-Alkoxy-6-trifluoromethylpyrimidin-4-yl)oxymethylene!phenylacetic acid derivatives, their preparation and intermediate therefor, and use thereof 失效
标题翻译： 2 - [（2-烷氧基-6-三氟甲基嘧啶-4-基）甲醛]苯乙酸衍生物及其制备方法及其中间体及其用途
公开(公告)号：US5935965A
公开(公告)日：1999-08-10
申请号：US836255
申请日：1997-05-06
申请人： Reinhard Kirstgen , Klaus Oberdorf , Franz Schutz , Hans Theobald , Volker Harries
发明人： Reinhard Kirstgen , Klaus Oberdorf , Franz Schutz , Hans Theobald , Volker Harries
IPC分类号： C07D239/54 , A01N43/54 , A01P7/02 , C07D239/52 , C07D239/56 , A61K31/505 , C07D239/34
CPC分类号： C07D239/56 , A01N43/54 , C07D239/52
摘要： 2-�(2-Alkoxy-6-trifluoromethylpyrimidin-4-yl)oxymethylene!-phenylacetic acid derivatives of the formula I ##STR1## where the index and the substituents have the following meanings: U is CH or N;V is O or NH;R is alkyl;R.sup.1 is cyano, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or phenyl;n is 0 or an integer from 1 to 4,processes and intermediates for their preparation, and their use are described.
摘要翻译： PCT No.PCT / EP95 / 04375。 371日期：1997年5月6日 102（e）日期1997年5月6日PCT提交1995年11月7日PCT公布。第WO96 / 16047号公报日期：19962年5月30日 - 指数和取代基具有以下含义的[（2-烷氧基-6-三氟甲基嘧啶-4-基）甲醛] - 苯基乙酸衍生物：U是CH或N; V是O或NH; R是烷基; R 1是氰基，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基或苯基; n为0或1〜4的整数，其制备方法和中间体及其用途进行了说明。

6. 发明授权

US5633268A Substituted ortho-ethenylphenylacetic acid derivatives 失效
标题翻译：取代邻乙烯基苯乙酸衍生物
公开(公告)号：US5633268A
公开(公告)日：1997-05-27
申请号：US433515
申请日：1995-05-12
申请人： Reinhard Kirstgen , Hans Theobald , Klaus Oberdorf , Reinhard Doetzer , Ralf Klintz , Bernd Schaefer , Volker Harries , Uwe Kardorff , Gisela Lorenz , Eberhard Ammermann
发明人： Reinhard Kirstgen , Hans Theobald , Klaus Oberdorf , Reinhard Doetzer , Ralf Klintz , Bernd Schaefer , Volker Harries , Uwe Kardorff , Gisela Lorenz , Eberhard Ammermann
IPC分类号： A01N37/06 , A01N37/10 , A01N37/30 , A01N37/34 , A01N37/36 , A01N37/50 , A01N43/40 , A01N43/72 , A01N43/80 , A01N43/824 , C07C69/65 , C07C69/734 , C07C69/738 , C07C205/42 , C07C205/53 , C07C205/56 , C07C235/34 , C07C235/36 , C07C235/38 , C07C235/72 , C07C239/20 , C07C239/22 , C07C243/32 , C07C243/38 , C07C251/40 , C07C251/48 , C07C251/52 , C07C251/64 , C07C251/66 , C07C255/14 , C07C255/38 , C07C255/41 , C07C255/62 , C07C255/64 , C07C255/66 , C07C259/06 , C07C271/60 , C07C291/02 , C07C323/10 , C07C323/62 , C07C327/20 , C07C327/38 , C07C331/02 , C07D295/32 , C07D285/08 , A61K31/41
CPC分类号： C07D295/32 , A01N37/36 , A01N37/50 , A01N43/80 , C07C205/42 , C07C205/53 , C07C205/56 , C07C235/34 , C07C235/36 , C07C235/38 , C07C239/22 , C07C243/32 , C07C243/38 , C07C251/40 , C07C251/48 , C07C251/52 , C07C251/66 , C07C255/14 , C07C255/38 , C07C255/41 , C07C255/62 , C07C255/64 , C07C255/66 , C07C259/06 , C07C271/60 , C07C69/65 , C07C69/734 , C07C2101/02 , C07C2101/08 , C07C2101/14 , C07C2103/74
摘要： Compounds of the formula I ##STR1## where the index and the substituents have the following meanings as defined in the specification.
摘要翻译： PCT No.PCT / EP93 / 03067 Sec。 371日期：1995年5月12日 102（e）日期1995年5月12日PCT提交1993年11月12日PCT公布。公开号WO94 / 11334 日期1994年5月26日化学式I 其中指数和取代基具有如说明书中定义的以下含义。

7. 发明授权

US5489605A Cyanooxime ethers, their preparation, agents containing them and their use 失效
标题翻译：氰基肟醚，它们的制备，含有它们的药剂及其用途
公开(公告)号：US5489605A
公开(公告)日：1996-02-06
申请号：US290938
申请日：1994-08-24
申请人： Klaus Oberdorf , Uwe Kardorff , Hans Theobald , Albrecht Harreus , Hartmann Koenig , Volker Harries
发明人： Klaus Oberdorf , Uwe Kardorff , Hans Theobald , Albrecht Harreus , Hartmann Koenig , Volker Harries
IPC分类号： C07D249/08 , A01N37/34 , A01N37/50 , A01N43/16 , A01N43/74 , A01N43/76 , A01N43/80 , A01N43/82 , A01N43/824 , C07C253/30 , C07C255/62 , C07C261/02 , C07C323/11 , C07C323/18 , C07C323/60 , C07C331/04 , C07D207/333 , C07D231/12 , C07D235/12 , C07D261/06 , C07D261/08 , C07D263/30 , C07D263/32 , C07D271/10 , C07D277/24 , C07D285/12 , C07D307/12 , C07D307/38 , C07D307/42 , C07D307/54 , C07D307/80 , C07D317/50 , C07D333/16 , C07D333/58 , C07D405/12 , C07D407/12 , C07D413/12 , C07D521/00 , C07C255/64
CPC分类号： C07C323/60 , A01N37/50 , A01N43/16 , A01N43/76 , A01N43/80 , C07D261/08 , C07D263/32
摘要： Cyanooxime ethers of the formula IR.sup.1 R.sup.2 CH--ON.dbd.C(CN)--R.sup.3 IwhereR.sup.1 is hydrogen or C.sub.1 -C.sub.4 -alkyl;R.sup.2 is an unsubstituted or substituted mononuclear to trinuclear aliphatic or aromatic ring system which, in addition to carbon atoms, may contain from one to four nitrogen atoms or from one to three hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen andR.sup.3 is unsubstituted or substituted alkyl or an unsubstituted or substituted aliphatic ring system which, in addition to carbon atoms, may contain one or two hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen,processes for their preparation, agents containing them and their use.
摘要翻译： PCT No.PCT / EP93 / 00371 Sec。 371日期：1994年8月24日 102（e）日期1994年8月24日PCT提交1993年2月17日PCT公布。公开号WO93 / 16985 PCT 日期：1993年9月2日。式I的R 1 R 2 CH-ON = C（CN）-R 3 I的芳氧基醚，其中R 1是氢或C 1 -C 4烷基; R2是未取代或取代的单核至三核脂族或芳环体系，其除了碳原子之外可以含有1-4个氮原子或1至3个选自氧，硫和氮的杂原子和R3和是未取代或取代的烷基或未取代或取代的脂族环系，其除碳原子外可含有一个或两个选自氧，硫和氮的杂原子，其制备方法，含有它们的试剂及其制备方法使用。

8. 发明授权

US07056941B1 2-[pyrazolyl and triazolyl-3′-oxymethylene]-phenyl-isoxazolones, triazolones and tetrazolones as pesticides and fungicides 失效
标题翻译： 2- [吡唑基和三唑基-3'-氧亚甲基] - 苯基 - 异恶唑酮，三唑酮和四唑酮作为农药和杀真菌剂
公开(公告)号：US07056941B1
公开(公告)日：2006-06-06
申请号：US09462647
申请日：1998-07-02
申请人： Bernd Müller , Hubert Sauter , Herbert Bayer , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Andreas Gypser , Arne Ptock , Reinhard Kirstgen , Norbert Götz , Roland Götz , Franz Röhl , Eberhard Ammermann , Volker Harries , Gisela Lorenz , Siegfried Strathmann
发明人： Bernd Müller , Hubert Sauter , Herbert Bayer , Markus Gewehr , Wassilios Grammenos , Thomas Grote , Andreas Gypser , Arne Ptock , Reinhard Kirstgen , Norbert Götz , Roland Götz , Franz Röhl , Eberhard Ammermann , Volker Harries , Gisela Lorenz , Siegfried Strathmann
IPC分类号： A01N43/653 , C07D249/12
CPC分类号： A01N43/80 , A01N43/653 , C07D249/12
摘要： 2-[Pyrazolyl- and triazolyl-3′-oxymethylene]phenylisoxazolones, -triazolones and -tetrazolones of formula I where: X is a group A, B or C, where # denotes the bond with the phenyl ring, Ra is hydrogen, halogen, alkyl or alkoxy, Rb is alkyl; Y is N or CRc, where Rc is hydrogen, halogen or alkyl; n is 0, 1, 2, 3 or 4, where the substituents R1 may be different if n is greater than 1; R1 is nitro, cyano, halogen, alkyl with or without substitution or alkoxy with or without substitution or is additionally, if n is 2, an optionally substituted 3 or 4 membered bridge which forms together with the ring to which it is attached a bicyclic partially unsaturated or aromatic radical; R2 is hydrogen, nitro, cyano, halogen, alkyl, haloalkyl, alkoxy, alkylthio or alkoxycarbonyl; R3 is optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aryl or optionally substituted hetaryl, their preparation and their use for controlling unwanted animal pests or harmful fungi.
摘要翻译： 2- [吡唑基 - 和三唑基-3'-甲醛]苯基异恶唑酮，式I的三唑酮和四唑酮其中：X是A，B或C基团，其中＃表示与苯环的键，R a 氢，卤素，烷基或烷氧基，R b是烷基; Y是N或CR，其中R c是氢，卤素或烷基; n为0,1,2,3或4，其中如果n大于1，则取代基R 1可以不同; R 1是硝基，氰基，卤素，具有或不具有取代的烷基或具有或不具有取代的烷氧基，或者另外，如果n是2，则与环一起形成的任选取代的3或4元桥其连接有双环部分不饱和或芳族基团; R 2是氢，硝基，氰基，卤素，烷基，卤代烷基，烷氧基，烷硫基或烷氧基羰基; R 3是任选取代的烷基，任选取代的环烷基，任选取代的芳基或任选取代的杂芳基，它们的制备及其用于防治有害动物害虫或有害真菌的用途。

9. 发明授权

US06537989B1 Azadioxacycloalkene derivatives, methods for the production thereof and their use as fungicides and pest control agents 失效
标题翻译： Azadioxacycalkalk衍生物，其生产方法及其作为杀真菌剂和害虫防治剂的用途
公开(公告)号：US06537989B1
公开(公告)日：2003-03-25
申请号：US09806608
申请日：2001-04-02
申请人： Markus Gewehr , Wassilios Grammenos , Hubert Sauter , Herbert Bayer , Andreas Gypser , Bernd Müller , Arne Ptock , Oliver Cullmann , Thomas Grote , Eberhard Ammermann , Gisela Lorenz , Siegfried Strathmann , Volker Harries
发明人： Markus Gewehr , Wassilios Grammenos , Hubert Sauter , Herbert Bayer , Andreas Gypser , Bernd Müller , Arne Ptock , Oliver Cullmann , Thomas Grote , Eberhard Ammermann , Gisela Lorenz , Siegfried Strathmann , Volker Harries
IPC分类号： A61K3155
CPC分类号： C07D273/00 , A01N43/88
摘要： The present invention relates to azadioxacycloalkenes of the formula I in which the substituents R1 to R5 and X, the index n and the bridge member W have the following meanings: R1 is C1-C4-alkyl, halogen, C1-C4-haloalkyl, C3-C6-cycloalkyl; R2 is C1-C4-alkyl, C1-C4-haloalkyl, C3-C4-alkenyl, C3-C4-haloalkenyl, C3-C4-alkynyl or C3-C4-haloalkynyl; R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl or unsubstituted or substituted phenyl; R4 is ═CRaRb, —CRd═CRaRb or ═N—ORc, where Ra, Rb, Rc and Rd are each as defined in claim 1; R5 is nitro, cyano, halogen, C1-C6-alkyl or, in the case that n is 2, additionally a bridge which is attached to two adjacent ring atoms; n is 0, 1, 2, 3 or 4, where the substituents R1 may be different if n is greater than 1; X is C1-C4-alkoxy-N═, C1-C4-alkoxy-CH═ or R6—CH═, where R6 is as defined in claim 1 W is unsubstituted or substituted C1-C3-alkylene.
摘要翻译：本发明涉及取代基R1至R5和X，指数n和桥连构件W具有以下含义的式Iin的二恶唑环烯烃：R1为C1-C4烷基，卤素，C1-C4卤代烷基，C3- C6-环烷基; R2是C1-C4-烷基，C1-C4卤代烷基，C3-C4-烯基，C3-C4-卤代烯基，C3-C4-炔基或C3-C4-卤代炔基; R3是氢，C1-C4- 烷基，C1-C4卤代烷基或未取代或取代的苯基; R4是= CRaRb，-CRd = CRaRb或= N-ORc，其中Ra，Rb，Rc和Rd分别如权利要求1中所定义; R5是硝基，氰基，卤素，C 1 -C 6 - 烷基，或在n为2的情况下，另外是连接到两个相邻环原子上的桥; n为0,1,2,3或4，其中如果n 大于1; X为C 1 -C 4 - 烷氧基-N =，C 1 -C 4 - 烷氧基-CH =或R 6 -CH =，其中R 6如权利要求1W中所定义，为未取代或取代的C 1 -C 3 - 亚烷基。

10. 发明授权

US06451790B1 Azadioxacycloalkenes and their use for combating harmful fungi and animal pests 失效
标题翻译： Azadioxacycalkalk烯及其用于防治有害真菌和动物害虫的用途
公开(公告)号：US06451790B1
公开(公告)日：2002-09-17
申请号：US09889164
申请日：2001-07-11
申请人： Markus Gewehr , Hubert Sauter , Bernd Müller , Wassilios Grammenos , Andreas Gypser , Arne Ptock , Oliver Cullmann , Jordi Tormo i Blasco , Eberhard Ammermann , Siegfried Strathmann , Gisela Lorenz , Volker Harries , Roland Götz , Thomas Grote
发明人： Markus Gewehr , Hubert Sauter , Bernd Müller , Wassilios Grammenos , Andreas Gypser , Arne Ptock , Oliver Cullmann , Jordi Tormo i Blasco , Eberhard Ammermann , Siegfried Strathmann , Gisela Lorenz , Volker Harries , Roland Götz , Thomas Grote
IPC分类号： C07D41312
CPC分类号： C07D413/12 , A01N43/82 , A01N43/88 , C07D231/20 , C07D249/12 , C07D413/14
摘要： Compounds of formula I wherein W is optionally substituted alkylene; Y is N or CRa; Ra is hydrogen, halogen or alkyl; R1n represents hydrogen or 1 to 4 substituents; R2 is hydrogen, nitro, cyano, halogen, alkyl, haloalkyl, alkoxy, alkylthio or alkoxycarbonyl; R3 is optionally substituted alkyl, cycloalkyl, aryl or hetaryl; A is N—OR4, CH—OR4, CH—SR4 or CHR5; R4 is alkyl or haloalkyl; R5 is halogen, alkyl or haloalkyl; methods and intermediates for their preparation. The compounds and compositions comprising them are useful for combating animal pests and harmful fungi.
摘要翻译：式I的化合物，其中W是任选取代的亚烷基; Y是N或CR a; R a是氢，卤素或烷基; R 11代表氢或1-4个取代基; R 2是氢，硝基，氰基，卤素，烷基，卤代烷基，烷氧基，烷硫基或烷氧基羰基; R3是任选取代的烷基，环烷基，芳基或杂芳基; A是N-OR4，CH-OR4，CH-SR4或CHR5; R4是烷基或卤代烷基; R5是卤素，烷基或卤代烷基;其制备方法和中间体。包含它们的化合物和组合物可用于对抗动物害虫和有害真菌。

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