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1. 发明授权

US06703347B2 Isothiazole derivatives and their use as pesticides 失效
标题翻译：异噻唑衍生物及其作为农药的用途
公开(公告)号：US06703347B2
公开(公告)日：2004-03-09
申请号：US10182425
申请日：2002-11-07
申请人： Sarah Armstrong , Nigel John Barnes , Susan Patricia Barnett , Eric Daniel Clarke , Patrick Jelf Crowley , Torquil Eoghan Macleod Fraser , David John Hughes , Christopher John Mathews , Roger Salmon , Stephen Christopher Smith , Russell Viner , William Guy Whittingham , John Williams , Alan John Whittle , William Roderick Mound , Christopher John Urch , Brian Leslie Pilkington
发明人： Sarah Armstrong , Nigel John Barnes , Susan Patricia Barnett , Eric Daniel Clarke , Patrick Jelf Crowley , Torquil Eoghan Macleod Fraser , David John Hughes , Christopher John Mathews , Roger Salmon , Stephen Christopher Smith , Russell Viner , William Guy Whittingham , John Williams , Alan John Whittle , William Roderick Mound , Christopher John Urch , Brian Leslie Pilkington
IPC分类号： C07D41712
CPC分类号： C07D417/12 , A01N43/80
摘要： A compound of formula (I), where A is optionally substituted alkylene, alkenylene, alkynylene, cycloalkylene, alkylenoxy, oxy(C1-6)alkylene, alkylenthio, thio(C1-6)alkylene, C1-6alkylenamino, amino(C1-6)alkylene, [C1-6alkyleneoxy(C1-6)alkylene], [C1-6alkylenethio(C1-6)alkylene], [1-6alkylenesulfinyl(C1-6)alkylene], [C1-6alkylenesulfonyl(C1-6)alkylene] or [C1-6alkyleneamino(C1-6)alkylene]; provided that A is not CH2 or CH2O; B is N,N-oxide or CR8; Y is O, S or NR9; Z is O, S or NR10; and R1, R2, R3, R4, R5, R6, R7, R8, R9, R10 are specified radicals; compositions containing them; process for making them; and their use as insecticides or fungicides.
摘要翻译：式（I）化合物，其中A为任选取代的亚烷基，亚烯基，亚炔基，亚环烷基，亚烷氧基，氧（C 1-6）亚烷基，烷基硫基，硫代（C 1-6）亚烷基，C 1-6亚烷基氨基，氨基（C 1-6））亚烷基，[C 1-6亚烷基氧基（C 1-6）亚烷基]，[C 1-6亚烷基硫醚（C 1-6）亚烷基]，[1-6亚烷基亚烷基（C 1-6）亚烷基] 或[C 1-6亚烷基氨基（C 1-6）亚烷基]; A不是CH2或CH2O; B是N，N-氧化物或CR 8; Y是O，S或NR 9; Z是O，S或NR 10; R 1，R 2，R 3，R 4，R 5，R 6，R 7，R 8，R 9，R 10，被指定为自由基; 含有它们的组合物; 制作过程; 并将其用作杀虫剂或杀真菌剂。

2. 发明授权

US06544989B2 Benzazoles: benzoxazole, benzthiazole and benzimidazole derivatives 失效
标题翻译：苯并唑：苯并恶唑，苯并噻唑和苯并咪唑衍生物
公开(公告)号：US06544989B2
公开(公告)日：2003-04-08
申请号：US09767880
申请日：2001-01-23
申请人： Christopher John Mathews , Russell Viner , Susan Patricia Barnett , Christopher John Urch , Stephen Christopher Smith , Patrick Jelf Crowley , William Guy Whittingham , Stephen Paul Heaney , John Williams , Torquil Eoghan Macleod Fraser , Eric Daniel Clarke , David John Hughes , Sarah Armstrong , Nigel John Barnes , Alan John Whittle , Brian Leslie Pilkington
发明人： Christopher John Mathews , Russell Viner , Susan Patricia Barnett , Christopher John Urch , Stephen Christopher Smith , Patrick Jelf Crowley , William Guy Whittingham , Stephen Paul Heaney , John Williams , Torquil Eoghan Macleod Fraser , Eric Daniel Clarke , David John Hughes , Sarah Armstrong , Nigel John Barnes , Alan John Whittle , Brian Leslie Pilkington
IPC分类号： C07D41712
CPC分类号： C07D417/12 , A01N43/80
摘要： The invention provides compounds of formula (I): where the substituents are as defined in the specification. The invention also provides processes for preparing the compounds, compositions comprising the compounds, methods of using the compounds and compositions to combat fungal diseases, and methods of using the compounds and compositions to combat or control insect, acarine, mollusc and nematode pests.
摘要翻译：本发明提供式（I）化合物：其中取代基如说明书中所定义。本发明还提供了制备化合物的方法，包含化合物的组合物，使用化合物和组合物来对抗真菌疾病的方法，以及使用化合物和组合物来对抗或控制昆虫，螨虫，软体动物和线虫的害虫的方法。

3. 发明授权

US5770741A Process for cylopropane derivatives 失效
标题翻译：环丙烷衍生物的方法
公开(公告)号：US5770741A
公开(公告)日：1998-06-23
申请号：US444663
申请日：1995-05-19
申请人： Patrick Jelf Crowley , Christopher John Urch , Paul Anthony Worthington
发明人： Patrick Jelf Crowley , Christopher John Urch , Paul Anthony Worthington
IPC分类号： C07C45/29 , C07C45/30 , C07C45/68 , C07C49/813 , C07D249/08 , C07D521/00
CPC分类号： C07D249/08 , C07C45/29 , C07C45/292 , C07C45/30 , C07C45/68 , C07C49/813 , C07D231/12 , C07D233/56
摘要： The invention provides a process for the preparation of a compound of the general formula (I): ##STR1## wherein X, Y and R.sup.1 to R.sup.7 are as defined. In the process, the olefinic analog of the compound of general formula (I) is treated with a halogen-bearing compound in the presence of metallic zinc.
摘要翻译：本发明提供了制备通式（I）的化合物的方法：其中X，Y和R 1至R 7如上所定义。在该方法中，通式（I）化合物的烯属类似物在金属锌存在下用含卤素化合物处理。

4. 发明授权

US5912254A Bicycle amine derivatives 失效
标题翻译：自行车胺衍生物
公开(公告)号：US5912254A
公开(公告)日：1999-06-15
申请号：US969635
申请日：1997-11-13
申请人： Nigel Douglas Bishop , Christopher John Urch , Terence Lewis , Raymond Leo Sunley , Roger Salmon , Christopher Richard Ayles Godfrey
发明人： Nigel Douglas Bishop , Christopher John Urch , Terence Lewis , Raymond Leo Sunley , Roger Salmon , Christopher Richard Ayles Godfrey
IPC分类号： C07D451/02 , A01N43/90 , A01N47/38 , C07D451/04 , C07D451/14 , C07D498/08 , C07D513/08 , C07D519/00 , A61K31/435 , C07D221/02
CPC分类号： C07D519/00 , A01N43/90 , A01N47/38
摘要： A compound of formula (I):P-R.sup.2 -Q (I)where each of P and Q is, independently, a group of formula (B): ##STR1## wherein J is a bidentate group of formula --CH.sub.2 --X--CH.sub.2 --(wherein X is methylene, sulfur or oxygen), X'C.dbd.CY or X'WC-CYZ (wherein X', W, Y and Z are independently hydrogen, hydroxy, acyloxy, alkoxy, alkylsilyloxy or halogen); R.sup.1 is an optionally substituted phenyl or 5-or 6-membered heterocyclic ring system containing from 1 to 3 heteroatoms individually selected from nitrogen, oxygen and sulfur atoms, and at least one unsaturation (double bond) between adjacent atoms in the ring, said heterocyclic ring being optionally fused to a benzene ring; or an acid addition salt, quaternary ammonium salt or N-oxide derived therefrom; an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor; a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.
摘要翻译：式（I）化合物：P-R 2 -Q（I）其中P和Q各自独立地是式（B）的基团：其中J是式-CH 2 -X-CH 2 - （其中X是亚甲基，硫或氧），X'C = CY或X'WC-CYZ（其中X'，W，Y和Z独立地是氢，羟基，酰氧基，烷氧基，烷基甲硅烷氧基或卤素）; R1是任选取代的苯基或5-或6-元杂环系，其含有1-3个分别选自氮，氧和硫原子的杂原子，以及环中相邻原子之间的至少一个不饱和键（双键），所述杂环环任选地与苯环稠合; 或由其衍生的酸加成盐，季铵盐或N-氧化物; 杀虫杀螨或杀线虫组合物，其包含式（I）化合物及其合适的载体或稀释剂; 一种防治昆虫，螨虫或线虫害虫的方法，包括用有效量的式（I）化合物或上述组合物处理害虫或害虫的场所。

5. 发明授权

US06573275B1 Bicyclic amines 失效
公开(公告)号：US06573275B1
公开(公告)日：2003-06-03
申请号：US10124696
申请日：2002-04-12
申请人： Christopher John Urch , Roger Salmon , Terence Lewis , Christopher Richard Ayles Godfrey , Martin Stephen Clough
发明人： Christopher John Urch , Roger Salmon , Terence Lewis , Christopher Richard Ayles Godfrey , Martin Stephen Clough
IPC分类号： C07D23924
CPC分类号： C07D451/02 , A01N43/90 , A01N47/16 , A01N47/22 , A01N47/38 , C07D401/04
摘要： A compound of formula (I): wherein R1 represents a group of formula (A) where each of W, X, Y and Z and Z represents either a group CR or the nitrogen atom, provided that not more than two of W, X, Y and Z represent the nitrogen atom and where each R present is independently selected from hydrogen and halogen atoms and cyano, amino, hydrazino, acylamino, hydroxy, alkyl, hydroxyalkyl, alkoxy, haloalkyl, haloalkoxy, alkenyl, alkenyloxy, alkoxyalkenyl, alkynyl, carboxylic acyl, alkoxycarbonyl, aryl and heterocyclyl groups, said groups comprising up to 6 carbon atoms, and wherein R2 represents hydrogen or cyano or a group selected from alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkanyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl or dithiocarboxyl groups, said groups comprising from 1 to 15 carbon atoms, said groups being optionally substituted with one or more substituents selected from, halogen, cyano, carboxyl, carboxylic acyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxy, nitro, haloalkyl, alkyl, amino, acylamino, imidate and phosphonato groups; and acid addition salts and quaternary ammonium salts and N-oxide derived therefrom. The compounds are useful as insecticides.

6. 发明授权

US06177442B1 Bicyclic amine derivatives 失效
标题翻译：双环胺衍生物
公开(公告)号：US06177442B1
公开(公告)日：2001-01-23
申请号：US09357750
申请日：1999-07-21
申请人： Christopher John Urch , Terence Lewis , Raymond Leo Sunley , Roger Salmon , Christopher Richard Ayles Godfrey , Christopher Ian Brightwell , Matthew Brian Hotson
发明人： Christopher John Urch , Terence Lewis , Raymond Leo Sunley , Roger Salmon , Christopher Richard Ayles Godfrey , Christopher Ian Brightwell , Matthew Brian Hotson
IPC分类号： A61K3146
CPC分类号： C07D451/02 , A01N43/90 , A01N47/16 , A01N47/18 , C07D451/04 , C07D451/06 , C07D451/14
摘要： The invention provides a compound of formula (I): wherein A represents a bidentate group of formula —CH2—X—CH2— (wherein X is methylene, sulfur or oxygen), X′C═CY or X′WC—CYZ (wherein X′, W, Y and Z are independently hydrogen, hydroxy, acyloxy, alkoxy, alkylsilyloxy, cyano or halogen, or X′ and W or Y and Z together with the carbon to which they are attached form a carbonyl group), provided that A is not CH2—CH2; Ar is an optionally substituted phenyl or 5- or 6-membered heterocyclic ring system containing from 1 to 3 heteroatoms individually selected from nitrogen, oxygen and sulfur atoms, and at least one unsaturation (double bond) between adjacent atoms in the ring, said heterocyclic ring being optionally fused to a benzene ring; aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkanyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl, dithiocarboxyl moieties of R, R3 and R4 comprise from 1 to 15 carbon atoms, and are optionally substituted with one or more substituents selected from, halogen, cyano, carboxyl, carboxylic acyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxy, nitro, haloalkyl, alkyl, amino, acylamino, imidate and phosphonato groups; or an acid addition salt, quaternary ammonium salt or N-oxide derived therefrom; an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor; a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.
摘要翻译：本发明提供式（I）化合物：其中A表示式-CH 2 -X-CH 2 - （其中X为亚甲基，硫或氧），X'C = CY或X'WC-CYZ（其中 X'，W，Y和Z独立地为氢，羟基，酰氧基，烷氧基，烷基甲硅烷氧基，氰基或卤素，或X'和W或Y和Z与它们所连接的碳一起形成羰基） A不是CH2-CH2; Ar是任选取代的苯基或5-或6-元杂环体系，其含有1-3个分别选自氮，氧和硫原子的杂原子，以及环中相邻原子之间的至少一个不饱和键（双键），所述杂环环任选地与苯环稠合; 芳基，杂芳基，芳烷基，杂芳基烷基，烯基，芳烯基，炔基，烷氧基羰基，链烷磺酰基，芳烃磺酰基，烷氧基羰基，芳烷氧基羰基，芳氧基羰基，杂环基烷基，氨基甲酰基，R，R3和R4的二硫代羧基部分包含1至15个碳原子，具有一个或多个选自卤素，氰基，羧基，羧基酰基，氨基甲酰基，烷氧基羰基，烷氧基，亚烷基二氧基，羟基，硝基，卤代烷基，烷基，氨基，酰氨基，亚胺基和膦酸基的取代基。或由其衍生的酸加成盐，季铵盐或N-氧化物; 杀虫杀螨或杀线虫组合物，其包含式（I）化合物及其合适的载体或稀释剂; 一种防治昆虫，螨虫或线虫害虫的方法，包括用有效量的式（I）化合物或上述组合物处理害虫或害虫的场所。

7. 发明授权

US06207676B1 Bicyclic amines 有权
标题翻译：双环胺
公开(公告)号：US06207676B1
公开(公告)日：2001-03-27
申请号：US09207195
申请日：1998-12-08
申请人： Christopher John Urch , Roger Salmon , Terence Lewis , Christopher Richard Ayles Godfrey , Martin Stephen Clough
发明人： Christopher John Urch , Roger Salmon , Terence Lewis , Christopher Richard Ayles Godfrey , Martin Stephen Clough
IPC分类号： A61K31439
CPC分类号： C07D451/02 , A01N43/90 , A01N47/16 , A01N47/22 , A01N47/38 , C07D401/04
摘要： A compound of formula (I): wherein R1 represents a group of formula (A) where each of W, X, Y and Z and Z represents either a group CR or the nitrogen atom, provided that not more than two of W, X, Y and Z represent the nitrogen atom and where each R present is independently selected from hydrogen and halogen atoms and cyano, amino, hydrazino, acylamino, hydroxy, alkyl, hydroxyalkyl, alkoxy, haloalkyl, haloalkoxy, alkenyl, alkenyloxy, alkoxyalkenyl, alkynyl, carboxylic acyl, alkoxycarbonyl, aryl and heterocyclyl groups, said groups comprising up to 6 carbon atoms, and wherein R2 represents hydrogen or cyano or a group selected from alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkanyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl or dithiocarboxyl groups, said groups comprising from 1 to 15 carbon atoms, said groups being optionally substituted with one or more substituents selected from, halogen, cyano, carboxyl, carboxylic acyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxy, nitro, haloalkyl, alkyl, amino, acylamino, imidate and phosphonato groups; and acid addition salts and quaternary ammonium salts and N-oxide derived therefrom. The compounds are useful as insecticides.
摘要翻译：式（I）的化合物：其中R 1表示式（A）的基团，其中W，X，Y和Z和Z各自表示基团CR或氮原子，条件是不大于2个W，X ，Y和Z代表氮原子，其中每个R独立地选自氢和卤素原子和氰基，氨基，肼基，酰氨基，羟基，烷基，羟基烷基，烷氧基，卤代烷基，卤代烷氧基，烯基，烯氧基，烷氧基烯基，炔基，羧基酰基，烷氧基羰基，芳基和杂环基，所述基团包含至多6个碳原子，并且其中R 2表示氢或氰基或选自烷基，芳基，杂芳基，芳烷基，杂芳基烷基，烯基，芳烯基，炔基，烷氧基羰基，链烷磺酰基，芳基磺酰基，烷氧基羰基，芳烷氧基羰基，芳氧基羰基，杂环基烷基，氨基甲酰基或二硫代羧基，所述基团包含1至15个碳原子，所述基团任选被一个或多个取代基se 由卤素，氰基，羧基，羧基酰基，氨基甲酰基，烷氧基羰基，烷氧基，亚烷基二氧基，羟基，硝基，卤代烷基，烷基，氨基，酰氨基，亚氨酸酯和膦酸酯基组成。和酸加成盐和季铵盐和由其衍生的N-氧化物。这些化合物可用作杀虫剂。

8. 发明授权

US06174894B1 Bicyclic amine derivatives 失效
标题翻译：双环胺衍生物
公开(公告)号：US06174894B1
公开(公告)日：2001-01-16
申请号：US09357749
申请日：1999-07-21
申请人： Christopher John Urch , Terence Lewis , Raymond Leo Sunley , Roger Salmon , Christopher Richard Ayles Godfrey , Christopher Ian Brightwell
发明人： Christopher John Urch , Terence Lewis , Raymond Leo Sunley , Roger Salmon , Christopher Richard Ayles Godfrey , Christopher Ian Brightwell
IPC分类号： A61K31435
CPC分类号： C07D451/02 , A01N43/90 , A01N47/16 , A01N47/18 , C07D451/04 , C07D451/06 , C07D451/14
摘要： The present invention provides a compound of Formula (I): wherein Ar is optionally substituted phenyl wherein the substutuents, if present, are selected from halogen atoms, cyano, alkyl, alkenyl, alkynyl, alkoxy, haloalkyl, haloalkenyl, alkylthio and alkyl amino groups; R represents hydrogen or cyano or a group selected from alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkenyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl, dithiocarboxyl or XR3 (where X represents oxygen or a group NR4); R3 and R4 are, independently, hydrogen, alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, heterocyclylalkyl, alkoxycarbonyl or carboxylic acyl each of which may be optionally substituted; R1 represents hydrogen, hydroxy, alkyl, alkoxy, amino, nitro, isocyanato, acylamino, hydroxyalkyl, optionally substituted heteroaryl, alkoxyalkyl, haloalkyl, halohydroxyalkyl, aralkyloxyalkyl, acyloxyalkyl, amidoximido, sulfonyloxyalkyl, aminoalkyl, alkoxycarbonylamino, acylaminoalkyl, cyanoalkyl, imino, formyl, acyl or carboxylic acid or an ester or amide thereof, or alkenyl or alkynyl either of which is optionally substituted; or an acid addition salt, quaternary ammonium salt or N-oxide derived therefrom; an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor; and a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.
摘要翻译：本发明提供式（I）的化合物：其中Ar是任选取代的苯基，其中如果存在这些取代基，则选自卤素原子，氰基，烷基，烯基，炔基，烷氧基，卤代烷基，卤代烯基，烷硫基和烷基氨基 ; R表示氢或氰基或选自烷基，芳基，杂芳基，芳烷基，杂芳基烷基，烯基，芳烯基，炔基，烷氧基羰基，链烷磺酰基，芳烃磺酰基，烯氧基羰基，芳烷氧基羰基，芳氧基羰基，杂环基烷基，氨基甲酰基，二硫代羧基或XR3（其中X表示氧或NR4组）; R 3和R 4独立地是氢，烷基，芳基，杂芳基，芳烷基，杂芳基烷基，烯基，芳烯基，炔基，杂环基烷基，烷氧基羰基或羧酰基，各自可以任选被取代; R 1表示氢，羟基，烷基，烷氧基，氨基，硝基，异氰酸酯基，酰氨基，羟基烷基，任选取代的杂芳基，烷氧基烷基，卤代烷基，卤代羟烷基，芳烷氧基烷基，酰氧基烷基，酰氨基亚氨基，磺酰氧基烷基，氨基烷基，烷氧基羰基氨基，酰氨基烷基，氰基烷基，亚氨基，甲酰基，酰基或羧酸或其酯或酰胺，或任选被取代的链烯基或炔基; 或由其衍生的酸加成盐，季铵盐或N-氧化物; 杀虫杀螨或杀线虫组合物，其包含式（I）化合物及其合适的载体或稀释剂; 以及一种防治昆虫，螨虫或线虫害虫的场所的方法，包括用有效量的式（I）化合物或上述组合物处理害虫或害虫的场所。

9. 发明授权

US6093726A Bicyclic amine derivatives 失效
标题翻译：双环胺衍生物
公开(公告)号：US6093726A
公开(公告)日：2000-07-25
申请号：US969639
申请日：1997-11-13
申请人： Christopher John Urch , Roger Salmon , Christopher Richard Ayles Godfrey
发明人： Christopher John Urch , Roger Salmon , Christopher Richard Ayles Godfrey
IPC分类号： A01N43/90 , A01N47/16 , A01N47/18 , C07D451/02 , C07D451/04 , C07D451/06 , C07D451/14 , C07D498/08 , A61K31/435 , C07D471/08
CPC分类号： C07D451/02 , A01N43/90 , A01N47/16 , A01N47/18 , C07D451/04 , C07D451/06 , C07D451/14
摘要： A compound of formula (I): ##STR1## wherein Ar is optionally substituted phenyl or optionally substituted 5-or 6-membered heterocyclic ring containing from 1 to 3 heteroatoms individually selected from nitrogen, oxygen and sulfur atoms, and at least one unsaturation (double bond) between adjacent atoms in the ring, said heterocyclic ring being optionally fused to a benzene ring; or an acid addition salt, quaternary ammonium salt or N-oxide derived therefrom, an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor, a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.
摘要翻译：式（I）的化合物：其中Ar是任选取代的苯基或含有1至3个选自氮，氧和硫原子的杂原子的任选取代的5或6元杂环，和至少一个不饱和键（双键）在环中的相邻原子之间，所述杂环任选地与苯环稠合; 或由其衍生的酸加成盐，季铵盐或N-氧化物，包含式（I）化合物及其合适的载体或稀释剂的杀虫，杀螨或杀线虫组合物，防治昆虫，螨虫或线虫的方法包括用有效量的式（I）化合物或上述组合物处理害虫或害虫的场所的场所的害虫。

10. 发明授权

US06391883B1 Bicyclic amines 有权
标题翻译：双环胺
公开(公告)号：US06391883B1
公开(公告)日：2002-05-21
申请号：US09602711
申请日：2000-06-26
申请人： Christopher John Urch , Roger Salmon , Terence Lewis , Christopher Richard Ayles Godfrey , Martin Stephen Clough
发明人： Christopher John Urch , Roger Salmon , Terence Lewis , Christopher Richard Ayles Godfrey , Martin Stephen Clough
IPC分类号： A61K31497
CPC分类号： C07D451/02 , A01N43/90 , A01N47/16 , A01N47/22 , A01N47/38 , C07D401/04
摘要： A compound of formula (I): wherein R1 represents a group of formula (A) where each of W, X, Y and Z and Z represents either a group CR or the nitrogen atom, provided that not more than two of W, X, Y and Z represent the nitrogen atom and where each R present is independently selected from hydrogen and halogen atoms and cyano, amino, hydrazino, acylamino, hydroxy, alkyl, hydroxyalkyl, alkoxy, haloalkyl, haloalkoxy, alkenyl, alkenyloxy, alkoxyalkenyl, alkynyl, carboxylic acyl, alkoxycarbonyl, aryl and heterocyclyl groups, said groups comprising up to 6 carbon atoms, and wherein R2 represents hydrogen or cyano or a group selected from alkyl, aryl, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, arenesulfonyl, alkanyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl or dithiocarboxyl groups, said groups comprising from 1 to 15 carbon atoms, said groups being optionally substituted with one or more substituents selected from, halogen, cyano, carboxyl, carboxylic acyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxy, nitro, haloalkyl, alkyl, amino, acylamino, imidate and phosphonato groups; and acid addition salts and quaternary ammonium salts and N-oxide derived therefrom. The compounds are useful as insecticides.
摘要翻译：式（I）的化合物：其中R 1表示式（A）的基团，其中W，X，Y和Z和Z各自表示基团CR或氮原子，条件是不大于2个W，X ，Y和Z代表氮原子，其中每个R独立地选自氢和卤素原子和氰基，氨基，肼基，酰氨基，羟基，烷基，羟基烷基，烷氧基，卤代烷基，卤代烷氧基，烯基，烯氧基，烷氧基烯基，炔基，羧基酰基，烷氧基羰基，芳基和杂环基，所述基团包含至多6个碳原子，并且其中R 2表示氢或氰基或选自烷基，芳基，杂芳基，芳烷基，杂芳基烷基，烯基，芳烯基，炔基，烷氧基羰基，链烷磺酰基，芳基磺酰基，烷氧基羰基，芳烷氧基羰基，芳氧基羰基，杂环基烷基，氨基甲酰基或二硫代羧基，所述基团包含1至15个碳原子，所述基团任选被一个或多个取代基se 由卤素，氰基，羧基，羧基酰基，氨基甲酰基，烷氧基羰基，烷氧基，亚烷基二氧基，羟基，硝基，卤代烷基，烷基，氨基，酰氨基，亚氨酸酯和膦酸酯基组成。和酸加成盐和季铵盐和由其衍生的N-氧化物。这些化合物可用作杀虫剂。

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