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1. 发明申请

WO2005123733A1 PYRIDOPYRAZINES FOR COMBATTING PHYTOPATHOGENIC FUNGI 审中-公开
标题翻译：用于混合致病性真菌的吡咯烷
公开(公告)号：WO2005123733A1
公开(公告)日：2005-12-29
申请号：PCT/EP2005/006706
申请日：2005-06-21
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , CROWLEY, Patrick, Jelf , MÜLLER, Urs , DOBLER, Markus , WILLIAMS, John
发明人： CROWLEY, Patrick, Jelf , MÜLLER, Urs , DOBLER, Markus , WILLIAMS, John
IPC分类号： C07D471/04
CPC分类号： C07D471/04
摘要： The compounds of the general formula (I) wherein R, R 1 , R 2 , R 8 , and R 9 are defined as set forth in the specification.
摘要翻译：其中R，R 1，R 2，R 8和R 9的通式（I）的化合物定义如说明书中所述。

2. 发明申请

WO2005123698A1 FUNGICIDES BASED ON NITROGEN-CONTAINING HETEROCYCLES 审中-公开
标题翻译：基于含氮杂质的杀真菌剂
公开(公告)号：WO2005123698A1
公开(公告)日：2005-12-29
申请号：PCT/EP2005/006687
申请日：2005-06-21
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , CROWLEY, Patrick, Jelf , MÜLLER, Urs , DOBLER, Markus , WILLIAMS, John
发明人： CROWLEY, Patrick, Jelf , MÜLLER, Urs , DOBLER, Markus , WILLIAMS, John
IPC分类号： C07D241/36
CPC分类号： C07D471/04 , A01N43/90
摘要： The compound of the general formula (I), wherein W, X, Y, Z, R, R 1 and R 2 are defined as set forth in the specification, useful as fungicide.
摘要翻译：通式（I）的化合物，其中W，X，Y，Z，R，R 1和R 2定义如说明书中所述，可用作杀真菌剂。

3. 发明申请

WO2004056829A1 FUNGICIDES BASED ON NITROGEN-CONTAINING HETEROCYCLES 审中-公开
标题翻译：基于含氮杂质的杀真菌剂
公开(公告)号：WO2004056829A1
公开(公告)日：2004-07-08
申请号：PCT/GB2003/005261
申请日：2003-12-03
申请人： SYNGENTA LIMITED , SYNGENTA PARTICIPATIONS AG , CROWLEY, Patrick, Jelf , DOBLER, Markus , MUELLER, Urs , WILLIAMS, John
发明人： CROWLEY, Patrick, Jelf , DOBLER, Markus , MUELLER, Urs , WILLIAMS, John
IPC分类号： C07D487/04
CPC分类号： C07D471/04
摘要： Fungicidal compounds having the general formula (1): formula (1) wherein W, Z and one of X and Y are N and the other one of X and Y is CR 8 ; R 8 is H, halo, C 1-4 alkyl, C 1-4 alkoxy, C 1-4 alkylthio or halo(C 1-4 )alkyl; R and R 2 are independently H, halo, C 1-8 alkyl, C 1-8 alkoxy, C 1-8 alkylthio, C 2-8 alkenyl, C 2-8 alkynyl, cyano or NR 3 R 4 , provided that at least one of R and R 2 is NR 3 R 4 ; R 1 is halo, C 1-8 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 3-8 cycloalkyl, C 3-8 cycloalkyl(C 1-6 )-alkyl, C 1-8 alkoxy, C 1-8 alkylthio, aryl, aryloxy, arylthio, heteroaryl, heteroaryloxy, heteroarylthio, aryl(C 1-4 )alkyl, aryl(C 1-4 )alkoxy, heteroaryl(C 1-4 )alkyl, heteroaryl(C 1-4 )alkoxy, aryl(C 1-4 )alkylthio, heteroaryl(C 1-4 )alkylthio, morpholino, piperidino or pyrrolidino; R 3 and R 4 are independently H, C 1-8 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, aryl, aryl(C 1-8 )- alkyl, C 3-8 cycloalkyl, C 3-8 cycloalkyl(C 1-6 )alkyl, heteroaryl, heteroaryl(C 1-8 )alkyl, NR 5 R 6 , provided that not both R 3 and R 4 are H or NR 5 R 6 , or R 3 and R 4 together form a C 3-7 alkylene or C 3-7 alkenylene chain optionally substituted with one or more C 1-4 alkyl or C 1-4 alkoxy groups, or, together with the nitrogen atom to which they are attached, R 3 and R 4 form a morpholine, thiomorpholine, thiomorpholine S-oxide or thiomorpholine S-dioxide ring or a piperazine or piperazine N -(C 1-4 )alkyl (especially N -methyl) ring; and R 5 and R 6 are independently H, C 1-8 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, aryl, aryl(C 1-8 )alkyl, C 3-8 cycloalkyl, C 3-8 cycloalkyl(C 1-6 )alkyl, heteroaryl or heteroaryl(C 1-8 )alkyl; any of the foregoing alkyl, alkenyl, alkynyl or cycloalkyl groups or moieties (other than for R 8 ) being optionally substituted with halogen, cyano, C 1-6 alkoxy, C 1-6 alkylcarbonyl, C 1-6 alkoxycarbonyl, C 1-6 haloalkoxy, C 1-6 alkylthio, tri(C 1-4 )alkylsilyl, C 1-6 alkylamino or C 1-6 dialkylamino, any of the foregoing morpholine, thiomorpholine, piperidine, piperazine and pyrrolidine rings being optionally substituted with C 1-4 alkyl (especially methyl), and any of the foregoing aryl or heteroaryl groups or moieties being optionally substituted with one or more substituents selected from halo, hydroxy, mercapto, C 1-6 alkyl, C 2-6 alkenyl, C 2-6 alkynyl, C 1-6 alkoxy, C 2-6 alkenyloxy, C 2-6 alkynyloxy, halo(C 1-6 )alkyl, halo(C 1-6 )alkoxy, C 1-6 alkylthio, halo(C 1-6 )alkylthio, hydroxy(C 1-6 )alkyl, C 1-4 alkoxy(C 1-6 )alkyl, C 3-6 cycloalkyl, C 3-6 cycloalkyl(C 1-4 )alkyl, phenoxy, benzyloxy, benzoyloxy, cyano, isocyano, thiocyanato, isothiocyanato, nitro, -NR"'R"", NHCOR"', -NHCONR"'R"", -CONR"'R"", -SO 2 R"', -OSO 2 R"', -COR"', -CR"'=NR"" or -N=CR "'R"", in which R"' and R"" are independently hydrogen, C 1-4 alkyl, halo-(C 1-4 )alkyl, C 1-4 alkoxy, halo(C 1-4 )alkoxy, C 1-4 alkylthio, C 3-6 cycloalkyl, C 3-6 cycloalkyl(C 1-4 )alkyl, phenyl or benzyl, the phenyl and benzyl groups being optionally substituted with halogen, C 1-4 alkyl or C 1-4 alkoxy.
摘要翻译：其中W，Z和X和Y之一是N，X和Y中的另一个是CR 8的通式（1）：式（1）的杀真菌化合物：式 R 8是H，卤素，C 1-4烷基，C 1-4烷氧基，C 1-4烷硫基或卤代（C 1-4）烷基; R和R 2独立地是H，卤素，C 1-8烷基，C 1-8烷氧基，C 1-8烷硫基，C 2-8烯基，C 2-8炔基，氰基或NR 3 R 4，条件是 R 3和R 2中的至少一个是NR 3 R 4; R 1是卤素，C 1-8烷基，C 2-8烯基，C 2-8炔基，C 3-8环烷基，C 3-8环烷基（C 1-6） - 烷基，C 1-8烷氧基，C 1-8烷硫基，芳基，芳氧基，芳硫基，杂芳基，杂芳氧基，杂芳硫基，芳基（C1-4）烷基，芳基（C1-4）烷氧基，杂芳基（C1-4）烷基，杂芳基（C1-4）烷氧基，芳基（C1-4），杂芳基（C 1-4）烷硫基，吗啉代，哌啶子基或吡咯烷子基; R 3和R 4独立地是H，C 1-8烷基，C 2-8烯基，C 2-8炔基，芳基，芳基（C 1-8） - 烷基，C 3-8环烷基，C 3-8环烷基 -6）烷基，杂芳基，杂芳基（C 1-8）烷基，NR 5 R 6，条件是不是R 3和R 4都不是H或NR 5 R 6，或 R 3和R 4一起形成任选被一个或多个C 1-4烷基或C 1-4烷氧基取代的C 3-7亚烷基或C 3-7亚烯基链，或者与它们所在的氮原子一起 R 3和R 4形成吗啉，硫代吗啉，硫代吗啉S-氧化物或硫代吗啉S-二氧化环或哌嗪或哌嗪N-（C 1-4）烷基（特别是N-甲基）环; R 5和R 6独立地为H，C 1-8烷基，C 2-8烯基，C 2-8炔基，芳基，芳基（C 1-8）烷基，C 3-8环烷基，C 3-8环烷基 -6）烷基，杂芳基或杂芳基（C 1-8）烷基; 氰基，C 1-6烷氧基，C 1-6烷基羰基，C 1-6烷氧基羰基，C 1-6卤代烷氧基，任选被烷基，烯基，炔基或环烷基中的任何一个（除R 8之外），C 1-6烷硫基，三（C 1-4）烷基甲硅烷基，C 1-6烷基氨基或C 1-6二烷基氨基，任何上述吗啉，硫代吗啉，哌啶，哌嗪和吡咯烷环任选被C 1-4烷基（特别是甲基）并且任何前述芳基或杂芳基基团或部分任选被一个或多个选自卤素，羟基，巯基，C 1-6烷基，C 2-6烯基，C 2-6炔基，C 1-6烷氧基， C 1-6烷氧基，C 1-6烷氧基，C 1-6烷氧基，C 1-6烷硫基，卤代（C 1-6）烷硫基，羟基（C 1-6）烷基， C 1-6）烷基，C 3-6环烷基，C 3-6环烷基

4. 发明申请

WO2004056826A1 FUNGICIDES 审中-公开
标题翻译：杀菌剂
公开(公告)号：WO2004056826A1
公开(公告)日：2004-07-08
申请号：PCT/GB2003/005273
申请日：2003-12-04
申请人： SYNGENTA LIMITED , SYNGENTA PARTICIPATIONS AG , CROWLEY, Patrick, Jelf , DOBLER, Markus , MUELLER, Urs , WILLIAMS, John
发明人： CROWLEY, Patrick, Jelf , DOBLER, Markus , MUELLER, Urs , WILLIAMS, John
IPC分类号： C07D471/04
CPC分类号： C07D239/42 , A01N43/90 , C07D471/04
摘要： Fungicidal compositions having the general formula (1): formula (1) wherein W and Y are both N and X and Z are both CR 8 or X and Z are both N and W and Y are both CR 8 , R 8 is H, halo, C 1-4 alkyl, C 1-4 alkoxy or halo(C 1-4 )alkyl; R and R 2 are independently H, halo, C 1-8 alkyl, C 1-8 alkoxy, C 1-8 alkylthio, C 2-8 alkenyl, C 2-8 alkynyl, cyano or NR 3 R 4 , provided that at least one of R and R 2 is NR 3 R 4 ; R 1 is halo, C 1-8 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 3-8 cycloalkyl, C 3-8 cycloalkyl(C 1-6 )-alkyl, C 1-8 alkoxy, C 1-8 alkylthio, aryl, aryloxy, arylthio, heteroaryl, heteroaryloxy, heteroarylthio, aryl(C 1-4 )alkyl, aryl(C 1-4 )alkoxy, heteroaryl(C 1-4 )alkyl, heteroaryl(C 1-4 )alkoxy, aryl(C 1-4 )alkylthio, heteroaryl(C 1-4 )alkylthio, morpholino, piperidino or pyrrolidino.
摘要翻译：具有通式（1）：式（1）的杀真菌组合物，其中W和Y都是N，X和Z都是CR 8或X和Z都是N和W，Y都是CR 8，R C 8是H，卤素，C 1-4烷基，C 1-4烷氧基或卤代（C 1-4）烷基; R和R 2独立地是H，卤素，C 1-8烷基，C 1-8烷氧基，C 1-8烷硫基，C 2-8烯基，C 2-8炔基，氰基或NR 3 R 4，条件是 R 3和R 2中的至少一个是NR 3 R 4; R 1是卤素，C 1-8烷基，C 2-8烯基，C 2-8炔基，C 3-8环烷基，C 3-8环烷基（C 1-6） - 烷基，C 1-8烷氧基，C 1-8烷硫基，芳基（C 1-4）烷基，芳基（C 1-4）烷氧基，杂芳基（C 1-4）烷基，杂芳基（C 1-4）烷氧基，芳基（C 1-4）烷硫基，杂芳基（C1-4）烷硫基，吗啉代，哌啶子基或吡咯烷子基。

5. 发明申请

WO2004056825A1 PYRIDODIAZINES AS PLANT FUNGICIDES 审中-公开
标题翻译： PYRIDODIAZINES作为植物杀真菌剂
公开(公告)号：WO2004056825A1
公开(公告)日：2004-07-08
申请号：PCT/GB2003/005250
申请日：2003-12-03
申请人： SYNGENTA LIMITED , SYNGENTA PARTICIPATIONS AG , CROWLEY, Patrick, Jelf , DOBLER, Markus , MUELLER, Urs , WILLIAMS, John
发明人： CROWLEY, Patrick, Jelf , DOBLER, Markus , MUELLER, Urs , WILLIAMS, John
IPC分类号： C07D471/04
CPC分类号： C07D471/04
摘要： Fungicidal compounds of general formula (1) wherein R, R 1 , R 2 , W, X, Y and Z are as defined in the specification.
摘要翻译：其中R，R 1，R 2，W，X，Y和Z的通式（1）的杀真菌化合物如说明书中所定义。

6. 发明申请

WO2004056824A2 FUNGICIDES 审中-公开
标题翻译：杀菌剂
公开(公告)号：WO2004056824A2
公开(公告)日：2004-07-08
申请号：PCT/GB2003/005248
申请日：2003-12-03
申请人： SYNGENTA LIMITED , SYNGENTA PARTICIPATIONS AG , CROWLEY, Patrick, Jelf , DOBLER, Markus , MUELLER, Urs , WILLIAMS, John
发明人： CROWLEY, Patrick, Jelf , DOBLER, Markus , MUELLER, Urs , WILLIAMS, John
IPC分类号： C07D471/04
CPC分类号： C07D471/04 , A01N43/90
摘要： Fungicidal compositions of the general formula (1): wherein one of W, X, Y and Z is N and the others are CR 8 ; R 8 is H, halo, C 1-4 alkyl, C 1-4 alkoxy or halo(C 1 - 4 )alkyl, provided that when X is CH, Z is N, R is NHNH 2 , R 1 is phenyl and R 2 is Cl, W and Y are not both CCH 3 ; one of R and R 2 is NR 3 R 4 and the other is halo, C 1-8 alkyl, C 1-8 alkoxy, C 1-8 alkylthio, C 2-8 alkenyl, C 2-8 alkynyl or cyano; R 1 is aryl, heteroaryl, morpholino, piperidino or pyrrolidino; R 3 and R 4 are independently H, C 1-8 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, aryl, aryl(C 1-8 )-alkyl, C 3-8 cycloalkyl, C3-8 cycloalkyl(C 1-6 )alkyl, heteroaryl, heteroaryl(C 1-8 )alkyl, NR 5 R 6 , provided that not both R 3 and R 4 are H or NR 5 R 6 , or R 3 and R 4 together form a C 3-7 alkylene or C 3-7 alkenylene chain optionally substituted with one or more C 1-4 alkyl or C 1-4 alkoxy groups, or, together with the nitrogen atom to which they are attached, R 3 and R 4 form a morpholine, thiomorpholine, thiomorpholine S-oxide or thiomorpholine S-dioxide ring or a piperazine or piperazine N -(C 1 - 4 )alkyl (especially N -methyl) ring; and R 5 and R 6 are independently H, C 1-8 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, aryl, aryl(C l-8 )-alkyl, C 3-8 cycloalkyl, C 3-8 cycloalkyl(C 1-6 )alkyl, heteroaryl or heteroaryl(C 1-8 )alkyl; any of the foregoing alkyl, alkenyl, alkynyl or cycloalkyl groups or moieties (other than for R 8 ) being optionally substituted with halogen, cyano, C 1-6 alkoxy , C 1-6 alkylcarbonyl, C 1-6 alkoxycarbonyl, C 1-6 haloalkoxy, C 1-6 alkylthio, tri(C 1-4 )alkylsilyl, C 1-6 alkylamino or C 1-6 ialkylamino, any of the foregoing morpholine, thiomorpholine, piperidine, piperazine and pyrrolidine rings being optionally substituted with C 1-4 alkyl (especially methyl), and any of the foregoing aryl or heteroaryl groups or moieties being optionally substituted with one or more substituents selected from halo, hydroxy, mercapto, C 1-6 alkyl, C 2-6 alkenyl, C 2-6 alkynyl, C 1-6 alkoxy, C 2-6 alkenyloxy, C 2-6 alkynyloxy, halo(C 1-6 )alkyl, halo(C 1-6 )alkoxy, C 1-6 alkylthio, halo(C 1-6 )alkylthio, hydroxy(C 1-6 )alkyl, C 1-4 alkoxy(C 1-6 )alkyl, C 1-6 cycloalkyl, C 3-6 cycloalkyl(C 1-4 )alkyl, phenoxy, benzyloxy, benzoyloxy, cyano, isocyano, thiocyanato, isothiocyanato, nitro, -NHCOR"', -NHCONR"'R"", -CONK"'R"", SO 2 R"', -OSO 2 R"', -COR"', -CR"'=NR" or -N=CR "'R"", in which R"' and R"" are independently hydrogen, C 1-4 alkyl, halo-(C 1-4 )alkyl, C 1-4 alkoxy, halo(C 1-4 )alkoxy, C 1-4 alkylthio, C 3-6 cycloalkyl, C 3-6 cycloalkyl(C 1-4 )alkyl, phenyl or benzyl groups beings optionally substituted with halogen, C 1-4 alkyl or C 1-4 alkoxy.
摘要翻译：通式（1）的杀真菌组合物：其中W，X，Y和Z中的一个为N，其余为CR 8; R 8为H，卤素，C 1-4烷基，C 1-4烷氧基或卤代（C 1-4）烷基，条件是当X为CH时，Z为N，R为NHNH 2，R 1为苯基且R <2>是Cl，W和Y不同时为CCH3; R 2和R 2之一是NR 3 R 4，另一个是卤素，C 1-8烷基，C 1-8烷氧基，C 1-8烷硫基，C 2-8烯基，C 2-8炔基或氰基; R 1是芳基，杂芳基，吗啉代，哌啶子基或吡咯烷子基; R 3和R 4独立地是H，C 1-8烷基，C 2-8烯基，C 2-8炔基，芳基，芳基（C 1-8） - 烷基，C 3-8环烷基，C 3-8环烷基 -6）烷基，杂芳基，杂芳基（C 1-8）烷基，NR 5 R 6，条件是不是R 3和R 4都不是H或NR 5 R 6，，或其中R 3和R 4一起形成任选被一个或多个C 1-4烷基或C 1-4烷氧基取代的C 3-7亚烷基或C 3-7亚烯基链，或与氮原子一起 R 3和R 4形成吗啉，硫代吗啉，硫代吗啉S-氧化物或硫代吗啉S-二氧化环或哌嗪或哌嗪N-（C 1-4）烷基（特别是N-甲基）环; R 5和R 6独立地为H，C 1-8烷基，C 2-8烯基，C 2-8炔基，芳基，芳基（C 1-8）烷基，C 3-8环烷基，C 3-8环烷基（ C 1-6）烷基，杂芳基或杂芳基（C 1-8）烷基; 氰基，C 1-6烷氧基，C 1-6烷基羰基，C 1-6烷氧基羰基，C 1 -C 6烷氧羰基，C 1-6烷氧基羰基， 6卤代烷氧基，C 1-6烷硫基，三（C 1-4）烷基甲硅烷基，C 1-6烷基氨基或C 1-6烷基氨基，任何上述吗啉，硫代吗啉，哌啶，哌嗪和吡咯烷环任选被C 1-4烷基取代甲基），并且任何前述芳基或杂芳基任选被一个或多个选自卤素，羟基，巯基，C 1-6烷基，C 2-6烯基，C 2-6炔基，C 1-6烷氧基， C 2-6烯氧基，C 2-6炔氧基，卤代（C 1-6）烷基，卤代（C 1-6）烷氧基，C 1-6烷硫基，卤代（C 1-6）烷硫基，羟基（C 1-6）烷基，烷氧基（C 1-6）烷基，C 1-6环烷基，C 3-6环烷基（C 1-4）烷基，苯氧基，苄氧基，苯甲酰氧基，氰基，异氰基，氰硫基，异硫氰酸根合，硝基，-NHCOR“ R“”，“ON”，“R”“，SO2R”'，-OSO R“'， - ”“，”NR“或-N = CR”'R“”，其中R“'和R”“独立地为氢，C 1-4烷基，卤代（C1- 4）烷基，C 1-4烷氧基，卤代（C 1〜

7. 发明申请

WO2006100038A1 TRIAZOLOPYRIMIDINE DERIVATIVES USEFUL AS FUNGICIDES 审中-公开
标题翻译：三唑并嘧啶衍生物有效用作杀真菌剂
公开(公告)号：WO2006100038A1
公开(公告)日：2006-09-28
申请号：PCT/EP2006/002591
申请日：2006-03-21
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , WENDEBORN, Sebastian , LAMBERTH, Clemens , NEBEL, Kurt , CROWLEY, Patrick, Jelf
发明人： WENDEBORN, Sebastian , LAMBERTH, Clemens , NEBEL, Kurt , CROWLEY, Patrick, Jelf
IPC分类号： C07D487/04 , C07D519/00 , A01N43/90 , A01P3/00
CPC分类号： A01N43/90 , C07D487/04
摘要： The present invention relates to novel triazolopyrimidine derivatives of formula I as active ingredients which have microbiocidal activity, in particular fungicidal activity wherein the substituents are as defined in claim 1.
摘要翻译：本发明涉及式I的新型三唑并嘧啶衍生物作为活性成分，其具有杀微生物活性，特别是杀真菌活性，其中取代基如权利要求1所定义。

8. 发明申请

WO2006100037A1 TRIAZOLOPYRIMIDINE DERIVATIVES USEFUL AS MICROBIOCIDES 审中-公开
标题翻译：三氮唑嘧啶衍生物作为微生物有用
公开(公告)号：WO2006100037A1
公开(公告)日：2006-09-28
申请号：PCT/EP2006/002590
申请日：2006-03-21
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , LAMBERTH, Clemens , WENDEBORN, Sebastian , NEBEL, Kurt , CROWLEY, Patrick, Jelf
发明人： LAMBERTH, Clemens , WENDEBORN, Sebastian , NEBEL, Kurt , CROWLEY, Patrick, Jelf
IPC分类号： C07D487/04 , C07D519/00 , A01N43/90
CPC分类号： C07D487/04 , A01N43/90
摘要： The present invention relates to novel triazolopyrimidine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein the substituents are as defined in Claim 1.
摘要翻译：本发明涉及具有杀微生物活性，特别是杀真菌活性的作为活性成分的式（I）的新型三唑并嘧啶衍生物，其中取代基如权利要求1所定义。

9. 发明申请

WO2008031566A2 NOVEL PYRIDOPYRAZINE DERIVATIVES 审中-公开
标题翻译：新型吡咯烷酮衍生物
公开(公告)号：WO2008031566A2
公开(公告)日：2008-03-20
申请号：PCT/EP2007/007912
申请日：2007-09-11
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , CROWLEY, Patrick, Jelf , LAMBERTH, Clemens , WENDEBORN, Sebastian, Volker , TRAH, Stephan
发明人： CROWLEY, Patrick, Jelf , LAMBERTH, Clemens , WENDEBORN, Sebastian, Volker , TRAH, Stephan
CPC分类号： C07D471/04 , A01N43/90
摘要： The present invention relates to novel N -oxide derivatives of pyridopyrazines of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity :wherein X is N + -O" and Y is N; or X is N and Y is N + -O"; or X and Y are both N + -O"; R is for example H, halo, cyano, C 1-6 alkyl or C 1-6 alkoxy; R 1 is optionally substituted aryl or heteroaryl; R 2 is for example halo, C 1-8 alkyl, C 3-8 CycloaIkyI, aryl, or heteroaryl; R 3 and R 4 independently of each other are for example H, C 1-8 alkyl, halo(d-8)alkyl, C 2-8 alkenyl, C 2-8 alkynyl or aryl; or R 3 and R 4 together with the nitrogen atom to which they are attached form a C 3-10 alkylene chain or C 3-7 alkenylene chain optionally substituted with halo, C 1-4 alkyl, C 1-4 haloalkyl, C1-4 alkoxy; or R 3 and R 4 together with the nitrogen atom to which they are attached form for example a morpholine, thiomorpholine or thiomorpholine S-oxide ring; or R 3 and R 4 together with the nitrogen atom to which they are attached form a bicyclic annelated or fused ring; and R 7 and R 8 independently of each other are for example H, halo, cyano, C 1-4 alkyl, C 1-4 aIkoxy or halo(C 1-4 )alkyl.
摘要翻译：本发明涉及式（I）吡啶并吡嗪的新型N-氧化物衍生物作为具有杀微生物活性，特别是杀真菌活性的活性成分：其中X为N + -O，Y为N; 或X为N且Y为N + O“; 或X和Y均为N + O-O“; R为例如H，卤素，氰基，C 1-6烷基或C 1-6烷基， R 1是任选取代的芳基或杂芳基; R 2是例如卤素，C 1-8烷基，C 1-4烷基，环烷基，芳基或杂芳基; R 3和R 4彼此独立地是例如H，C 1〜烷基，卤代（C 1-8）烷基，C 2-8链烯基，C 2-8炔基或芳基;或R 3， R 4和R 4与它们所连接的氮原子一起形成C 3-10亚烷基链或C 3-7亚烷基，任选被卤素取代的亚烯基链，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或R 3和R 3 与它们所连接的氮原子一起形成例如吗啉，硫代吗啉或硫代吗啉S-氧化物环;或R 3和R 4， SUP与它们所连接的氮原子一起形成a 双环环或稠环; R 7和R 8彼此独立地是例如H，卤素，氰基，C 1-4烷基，C 1 -C 4烷基， 1-4烷氧基或卤代（C 1-4烷基）烷基。

10. 发明申请

WO2006066874A1 NOVEL TRIAZOLOPYRIMIDINE DERIVATIVES 审中-公开
标题翻译：新型三唑并嘧啶衍生物
公开(公告)号：WO2006066874A1
公开(公告)日：2006-06-29
申请号：PCT/EP2005/013710
申请日：2005-12-20
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , WENDEBORN, Sebastian, Volker , LAMBERTH, Clemens , NEBEL, Kurt , CROWLEY, Patrick, Jelf
发明人： WENDEBORN, Sebastian, Volker , LAMBERTH, Clemens , NEBEL, Kurt , CROWLEY, Patrick, Jelf
IPC分类号： C07D487/04 , C07F7/18 , A01N43/90
CPC分类号： A01N55/00 , C07D487/04 , C07F7/0836 , C07F7/0898 , C07F7/1896
摘要： The present invention relates to novel triazolopyrimidine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein the substituents are as defined in claim 1.
摘要翻译：本发明涉及式（I）的新型三唑并嘧啶衍生物作为活性成分，其具有杀微生物活性，特别是杀真菌活性：其中取代基如权利要求1所定义。

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