专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明申请

US20050096406A1 Reactive diluents and alkyd resin coating compositions 审中-公开
标题翻译：活性稀释剂和醇酸树脂涂料组合物
公开(公告)号：US20050096406A1
公开(公告)日：2005-05-05
申请号：US10504239
申请日：2003-02-25
申请人： Roger Pretot , Andreas Muhlebach , Wolfgang Peter , Kurt Dietliker , Tunja Jung , Clemens Auschra , Hans Kirner , Paul Van Der Schaaf
发明人： Roger Pretot , Andreas Muhlebach , Wolfgang Peter , Kurt Dietliker , Tunja Jung , Clemens Auschra , Hans Kirner , Paul Van Der Schaaf
IPC分类号： C07C13/28 , C07C13/44 , C07C33/12 , C07C43/162 , C07C69/007 , C07C69/54 , C07C69/60 , C07C69/80 , C09D4/00 , C09D5/00 , C09D7/00 , C09D7/12 , C09D11/02 , C09D11/10 , C09D167/08 , C08G2/00
CPC分类号： C09D11/101 , C07C13/28 , C07C13/44 , C07C33/12 , C07C43/162 , C07C69/007 , C07C69/54 , C07C69/60 , C07C69/80 , C07C2601/08 , C07C2602/22 , C09D167/08
摘要： The invention relates to new reactive diluents of the formulae (Ia, Ib, Ic, Id, Ie) and to an alkyd coating composition comprising them. In a preferred embodiment R1 and R2 are hydrogen; R3 is (meth)acryloyloxy-methyl or phenyl para substituted by vinyl, R4 is phenyl or phenyl para substituted by vinyl or (meth)acryloyloxy; or a substituted phenyl residue of the formula —C6H4CH2—W, wherein W is (meth)acryloyloxy, or an aliphatic residue of the formula —CH2—Y-A, wherein Y is a bond, O—C1-C12alkylene, wherein the alkylene linker is linear or branched and may be interrupted once or more than once by oxygen, A is hydroxy, C1-C6alkoxy, acetoxy, (meth)acryloyloxy, or a phthalate- or maleate-residue; R5 is hydrogen; n is 1; X is —(CH2)—. The invention further relates to a solvent-based or water-based alkyd coating composition comprising 0.3 to 10 wt. % of a mono-, bis- or trisacylphosphinoxide photoinitiator, especially Irgacure 819.
摘要翻译：本发明涉及式（Ia，Ib，Ic，Id，Ie）的新型反应性稀释剂和包含它们的醇酸树脂涂料组合物。在优选的实施方案中，R 1和R 2是氢; R 3是（甲基）丙烯酰氧基 - 甲基或被乙烯基取代的对苯基，R 4是苯基或被乙烯基或（甲基）丙烯酰氧基取代的对苯基; 或式-C 6 H 2 CH 2 -W的取代的苯基，其中W是（甲基）丙烯酰氧基或脂族基式-CH 2 -YA的残基，其中Y是一个键，OC 1 -C 12亚烷基，其中亚烷基接头是直链的或分支，并且可以被氧中断一次或多于一次，A是羟基，C 1 -C 6烷氧基，乙酰氧基，（甲基）丙烯酰氧基或邻苯二甲酸酯 - 或马来酸盐残基; R 5是氢; n为1; X是 - （CH 2） - 。本发明还涉及一种溶剂型或水性醇酸涂料组合物，其包含0.3至10wt。％的单，双或三酰基次膦酰基光引发剂，特别是Irgacure 819。

2. 发明申请

US20050197404A1 Polymorphic forms of sertraline hydrochloride 失效
标题翻译：盐酸舍曲林的多形态
公开(公告)号：US20050197404A1
公开(公告)日：2005-09-08
申请号：US11101860
申请日：2005-04-08
申请人： Paul Van Der Schaaf , Franz Schwarzenbach , Hans Kirner , Martin Szelagiewicz , Claudia Marcolli , Andreas Burkhard
发明人： Paul Van Der Schaaf , Franz Schwarzenbach , Hans Kirner , Martin Szelagiewicz , Claudia Marcolli , Andreas Burkhard
IPC分类号： A61K31/135 , A61K31/137 , C07C211/42
CPC分类号： A61K31/137 , A61K31/135 , C07C211/42 , C07C2602/10
摘要： Sertraline hydrochloride polymorphic form II is conveniently prepared by adding hydrogen chloride to solution of sertraline free amine in a ketone. In preferred processes, the solution of sertraline free amine seeded with some crystals of polymorphic form II and/or the solution is heated before addition of the hydrogen chloride.
摘要翻译：盐酸舍曲林多晶型II通过将氯化氢加入酮中的舍曲林游离胺溶液方便地制备。在优选的方法中，在加入氯化氢之前加入接种有多晶型II和/或溶液的一些晶体的舍曲林游离胺溶液。

3. 发明申请

US20050043552A1 Process for the synthesis of amine ethers from secondary amino oxides 有权
标题翻译：从仲氨基氧化物合成胺醚的方法
公开(公告)号：US20050043552A1
公开(公告)日：2005-02-24
申请号：US10919776
申请日：2004-08-17
申请人： Andreas Hafner , Hans Kirner , Franz Schwarzenbach , Paul Van Der Schaaf , Peter Nesvadba
发明人： Andreas Hafner , Hans Kirner , Franz Schwarzenbach , Paul Van Der Schaaf , Peter Nesvadba
IPC分类号： B01J27/122 , C07B61/00 , C07D209/44 , C07D211/94 , C07D217/26 , C07D241/08 , C07D401/12 , C07D401/14 , C07D405/12 , C08F4/00 , C08K5/3412 , C08K5/3435 , C08L101/00 , C09K15/30 , C09K21/10 , C07D303/08 , C07C239/10
CPC分类号： C07D401/14 , C04B35/632 , C07D209/44 , C07D211/94 , C07D217/26 , C07D241/08 , C07D401/12 , C07D405/12 , C08K5/3412
摘要： An amine ether of formula A wherein a is 1 or 2; and when a is 1, E is E′; when a is 2, E is L; E′ is C1-C36 alkyl; C3-C18 alkenyl; C2-C18 alkinyl; C5-C18 cydoalkyl; C5-C18 cycloalkenyl; a radical of a saturated or unsaturated aliphatic bicyclic or tricyclic hydrocarbon of 7 to 12 carbon atoms; C2-C7alkyl or C3-C7alkenyl substituted by halogen; C7-C15 aralkyl or C7-C15 aralkyl substituted by C1-C4 alkyl or phenyl; or E′ is a radical of formula (VII) as explained in claim 1; T′ is tertiary C4-C18alkyl or phenyl, each of which are unsubstituted or substituted by halogen, OH, COOR21 or C(O)—R22; or T′ is C5-C12cycloalkyl; C5-C12 cycloalkyl which is interrupted by at least one O or —NR18—; a polycyclic alkyl radical having 7-18 carbon atoms, or the same radical which is interrupted by at least one O or —NR18—; or T′ is —C(G1)(G2)—T″; or C1-C18alkyl or C5-C12cycloalkyl substituted by T″ is hydrogen, halogen, NO2, cyano, or is a monovalent organic radical comprising 1-50 carbon atoms; or T″ and T′ together form a divalent organic linking group completing, together with the hindered amine nitrogen atom and the quaternary carbon atom substituted by G1 and G2, an optionally substituted five- or six-membered ring structure; and all other residues are as defined in claim 1, are obtained in good yield from the corresponding N-oxyl hindered amine precursor by reaction with a hydrocarbon E1—H or H—L—H in the presence of an organic hydroperoxide and a catalytic amount of copper or a copper compound. The products of present process find utility as polymerization regulators and/or light stabilizers for organic material.
摘要翻译：式A的胺醚，其中a为1或2; 当a为1时，E为E'; 当a为2时，E为L; E'是C 1 -C 36烷基; C3-C18烯基; C2-C18炔基; C5-C18环烷基; C5-C18环烯基; 7-12个碳原子的饱和或不饱和脂族二环或三环烃基团; C 2 -C 7烷基或被卤素取代的C 3 -C 7链烯基; 被C 1 -C 4烷基或苯基取代的C 7 -C 15芳烷基或C 7 -C 15芳烷基; 或E'是如权利要求1所述的式（VII）的基团; T'是叔C4-C18烷基或苯基，其各自为未取代的或被卤素，OH，COOR21或C（O）-R22取代; 或T'为C 5 -C 12环烷基; 被至少一个O或-NR 18 - 中断的C 5 -C 12环烷基; 具有7-18个碳原子的多环烷基或被至少一个O或-NR 18 - 中断的相同基团; 或T'为-C（G1）（G2）-T“; 或被T“取代的C 1 -C 18烷基或C 5 -C 12环烷基是氢，卤素，NO 2，氰基，或是包含1-50个碳原子的一价有机基团; 或T“和T'一起形成二价有机连接基团，与受阻胺氮原子和被G1和G2取代的季碳原子一起形成任选取代的五元或六元环结构; 并且所有其它残基如权利要求1中所定义，通过在有机氢过氧化物和催化量的铜或其盐的存在下与烃E1-H或HLH反应，由相应的N-氧基受阻胺前体以良好的产率获得铜化合物。本发明的产品可用作有机材料的聚合调节剂和/或光稳定剂。

4. 发明申请

US20050033086A1 Process for the preparation of 7-amino syn 3,5-dihydroxy heptanoic acid derivatives via 6-cyano syn 3,5-dihydroxy hexanoic acid derivatives 失效
标题翻译：通过6-氰基顺式3,5-二羟基己酸衍生物制备7-氨基顺式3,5-二羟基庚酸衍生物的方法
公开(公告)号：US20050033086A1
公开(公告)日：2005-02-10
申请号：US10481704
申请日：2002-07-02
申请人： Reinhold Ohrlein , Gabriele Baisch , Hans Kirner , Frank Bienewald , Stephan Burkhardt , Martin Studer
发明人： Reinhold Ohrlein , Gabriele Baisch , Hans Kirner , Frank Bienewald , Stephan Burkhardt , Martin Studer
IPC分类号： C07C67/307 , C07B53/00 , C07B61/00 , C07C67/30 , C07C67/31 , C07C69/67 , C07C69/675 , C07C69/708 , C07C69/716 , C07C69/732 , C07C69/738 , C07C227/06 , C07C227/16 , C07C227/32 , C07C229/22 , C07C231/02 , C07C235/06 , C07C235/74 , C07C247/12 , C07C253/30 , C07D207/34 , C12P7/62
CPC分类号： C07C69/67 , C07C69/716 , C07C69/732 , C07C69/738 , C07C227/32 , C07C229/22 , C07C235/06 , C07C235/74 , C12P7/62 , Y02P20/55
摘要： The invention relates to novel synthesis methods for the preparation of the intermediates, which are suitable for the preparation of statin derivatives, especially to novel synthesis methods of the intermediate of formula VI wherein Ra and Rc are each independently of the other hydrogen or a hydroxy-protecting group or together are a bridging hydroxy-protecting group, and Rb is a carboxy-protecting group, which methods are carried out by conversion of the intermediate of formula XIX wherein Ra and Rc are each independently of the other hydrogen or a hydroxy-protecting group, and Rb is a carboxy-protective group.
摘要翻译：本发明涉及适用于制备他汀类衍生物的中间体的新型合成方法，特别是式VI中间体的新合成方法，其中R a和R c各自独立地为氢或羟基 - 保护基或一起是桥接羟基保护基，Rb是羧基保护基，该方法通过式XIX的中间体转化而进行，其中R a和R c各自独立地为氢或羟基保护基基团，Rb是羧基保护基。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式