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1. 发明授权

US4861787A Nematicidal compositions 失效
标题翻译：杀线虫组合物
公开(公告)号：US4861787A
公开(公告)日：1989-08-29
申请号：US263961
申请日：1988-10-25
申请人： Ernst Beriger , Wolfgang Eckhardt , Robert Nyfeler
发明人： Ernst Beriger , Wolfgang Eckhardt , Robert Nyfeler
IPC分类号： A01N43/82 , A01N43/824 , C07D413/04 , C07D417/04
CPC分类号： C07D413/04 , A01N43/82 , C07D417/04
摘要： Novel compounds of the formula ##STR1## in which R' represents C.sub.1 -C.sub.5 -alkyl, halogen, trifluoromethyl or C.sub.1 -C.sub.3 -alkoxy;R" represents C.sub.1 -C.sub.5 -alkyl or halogen; andR"' represents C.sub.1 -C.sub.5 -alkyl that is unsubstituted or is substituted by from 1 to 6 halogen atoms, C.sub.1 -C.sub.5 -alkenyl that is unsubstituted or is substituted by from 1 to 6 halogen atoms, or C.sub.1 -C.sub.5 - alkynyl that is unsubstituted or is substituted by from 1 to 6 halogen atoms;m represents 0, 1, 2 or 3 andn represents 0 or 1; andX.sub.1 and X.sub.2 each represents, independently of the other, oxygen or sulphur,as active ingredients for controlling plant parasite nematodes and for preventing damage to cultivated plants caused by nematode attack.
摘要翻译：式中，R'表示C 1 -C 5 - 烷基，卤素，三氟甲基或C 1 -C 3 - 烷氧基的新化合物＆lt; IMAGE＆gt; R“表示C 1 -C 5烷基或卤素; 和R“'表示未被取代或被1至6个卤素原子取代的C1-C5-烷基，未被取代或被1至6个卤素原子取代的C1-C5-烯基或C1-C5-炔基未被取代或被1至6个卤素原子取代; m表示0,1,2或3，n表示0或1; X1和X2各自独立地表示作为控制植物寄生线虫的活性成分的氧或硫，并且用于防止由线虫攻击引起的对栽培植物的损害。

2. 发明授权

US4894380A 2-mercapto-5-pyridyl-1,3,4-oxadiazoles and 2-mercapto-5-pyridyl-1,3,4-thiadiazoles of the formula I 失效
标题翻译： 2-巯基-5-吡啶基-1,3,4-恶二唑和式I的2-巯基-5-吡啶基-1,3,4-噻二唑
公开(公告)号：US4894380A
公开(公告)日：1990-01-16
申请号：US176483
申请日：1988-03-25
申请人： Robert Nyfeler , Wolfgang Eckhardt , Ernst Beriger , Odd Kristiansen
发明人： Robert Nyfeler , Wolfgang Eckhardt , Ernst Beriger , Odd Kristiansen
IPC分类号： A01N43/82 , A01N43/824 , C07D413/04 , C07D417/04
CPC分类号： C07D413/04 , A01N43/82 , C07D417/04
摘要： The invention relates to 2-mercapto-5-pyridyl-1,3,4-oxadiazoles and 2-mercapto-5-pyridyl-1,3,4-thiadiazoles of the formula I ##STR1## wherein X is oxygen or sulfur,R' is C.sub.1 -C.sub.3 alkyl which is substituted by bromine, fluorine, C.sub.1 -C.sub.3 alkoxy or cyano; unsubstituted or halogen-substituted C.sub.3 -C.sub.7 alkenyl; unsubstituted or halogen-substituted C.sub.4 -C.sub.7 alkynyl,R is C.sub.1 -C.sub.3 alkyl, unsubstituted C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkoxy which is substituted by halogen or C.sub.1 -C.sub.3 alkoxy; unsubstituted or halogen-substituted C.sub.3 -C.sub.7 alkenyl; C.sub.3 -C.sub.7 alkynyl, C.sub.1 -C.sub.3 alkylthio, halogen, cyano, hydroxy, amino or amino which is substituted by one or two C.sub.1 -C.sub.3 alkyl groups; or is aminocarbonyl; andn is 0, 1, 2, 3 or 4,to the preparation of the compounds of formula I and to novel intermediates for the synthesis of these compounds. The compounds of formula I have nematicidal properties. The invention further relates to nematicidal compositions which contain at least one compound of formula I as active component, and to methods of using said compounds and of the compositions containing them for controlling nematodes.
摘要翻译：本发明涉及式I的2-巯基-5-吡啶基-1,3,4-恶二唑和2-巯基-5-吡啶基-1,3,4-噻二唑，其中X是氧或硫，R'是被溴，氟，C 1 -C 3烷氧基或氰基取代的C 1 -C 3烷基; 未取代或卤素取代的C 3 -C 7链烯基; 未取代的或卤素取代的C4-C7炔基，R是C1-C3烷基，未取代的C1-C3烷氧基或被卤素或C1-C3烷氧基取代的C1-C3烷氧基; 未取代或卤素取代的C 3 -C 7链烯基; 被一个或两个C 1 -C 3烷基取代的C 3 -C 7炔基，C 1 -C 3烷硫基，卤素，氰基，羟基，氨基或氨基; 或是氨基羰基; 和n为0,1,2,3或4，用于制备式I化合物和用于合成这些化合物的新中间体。式I的化合物具有杀线虫性质。本发明还涉及含有至少一种式I化合物作为活性组分的杀线虫组合物，以及使用所述化合物和含有它们的组合物控制线虫的方法。

3. 发明授权

US4861367A 2-Mercapto-5-pyrazinyl-1,3,4-oxadiazoles or 2-mercapto-5-pyrazinyl-1,3,4-thiadiazoles as nematicides 失效
标题翻译： 2-巯基-5-吡嗪基-1,3,4-恶二唑或2-巯基-5-吡嗪基-1,3,4-噻二唑作为杀线虫剂
公开(公告)号：US4861367A
公开(公告)日：1989-08-29
申请号：US172884
申请日：1988-03-25
申请人： Robert Nyfeler , Wolfgang Eckhardt , Ernst Beriger
发明人： Robert Nyfeler , Wolfgang Eckhardt , Ernst Beriger
IPC分类号： A01N43/82 , A01N43/824 , C07D413/04 , C07D417/04
CPC分类号： C07D413/04 , A01N43/82 , C07D417/04
摘要： 2-Mercapto-5-pyrazinyl-1,3,4-oxadiazoles and 2-mercapto-5-pyrazinyl-1,3,4-thiadiazoles of formula I ##STR1## wherein X is oxygen or sulfur,R' is C.sub.1 -C.sub.5 alkyl, unsubstituted or substituted by halogen, C.sub.1 -C.sub.3 alkoxy or cyano; unsubstituted or halogen-substituted C.sub.3 -C.sub.7 alkenyl; unsubstituted or halogen-substituted C.sub.3 -C.sub.7 alkynyl,R is C.sub.1 -C.sub.3 alkyl, unsubstituted C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkoxy which is substituted by halogen or C.sub.1 -C.sub.3 alkoxy; halogen, cyano, hydroxy, amino or amino which is substituted by one or two C.sub.1 -C.sub.3 alkyl groups; or is aminocarbonyl; andn is 0, 1, 2 or 3, the preparation thereof and novel intermediates for their synthesis are disclosed.The compounds of formula I have nematicidal properties. Nematicidal compositions which contain at least one compound of formula I as active ingredient, methods of using said compounds and of the compositions containing them for controlling nematodes are also disclosed.
摘要翻译： 2-巯基-5-吡嗪基-1,3,4-恶二唑和式I的2-巯基-5-吡嗪基-1,3,4-噻二唑其中X是氧或硫，R'是 C1-C5烷基，未取代或被卤素，C1-C3烷氧基或氰基取代; 未取代或卤素取代的C 3 -C 7链烯基; 未取代的或卤素取代的C3-C7炔基，R是C1-C3烷基，未取代的C1-C3烷氧基或被卤素或C1-C3烷氧基取代的C1-C3烷氧基; 卤素，氰基，羟基，氨基或被一个或两个C 1 -C 3烷基取代的氨基; 或是氨基羰基; 并且n为0,1,2或3，其制备及其合成的新中间体被公开。式I的化合物具有杀线虫性质。还公开了含有至少一种式I化合物作为活性成分的杀线虫剂组合物，使用所述化合物和含有它们的组合物用于控制线虫的方法。

4. 发明授权

US4849009A 2-arylmethyliminopyrazines pyrazines, compositions and method of combating undesirable plant growth and of regulating plant growth 失效
公开(公告)号：US4849009A
公开(公告)日：1989-07-18
申请号：US92257
申请日：1987-09-02
申请人： Helmut Zondler , Wolfgang Eckhardt , Robert Nyfeler
发明人： Helmut Zondler , Wolfgang Eckhardt , Robert Nyfeler
IPC分类号： A01N43/54 , A01N43/60 , C07D239/42 , C07D241/14 , C07D241/20 , C07D405/12
CPC分类号： C07D239/42 , A01N43/54 , A01N43/60 , C07D241/20 , C07D405/12
摘要： 2-Arylmethyliminopyrazines of the formula I ##STR1## in which R.sub.1 is SR.sub.2 ; OR.sub.2 ; O--CHR.sub.10 R.sub.2 ; N(R.sub.3)(CHR.sub.10 R.sub.4); N(R.sub.11)(CHR.sub.10 R.sub.4) or NR.sub.3 R.sub.4 ; R.sub.2 is C.sub.1 -C.sub.10 - alkyl which is unsubstituted or substituted by hydroxyl, mercapto, C.sub.1 -C.sub.4 -alkoxycarbonyl, mercaptoalkoxy, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylcarbonyl, mono- or di-C.sub.1 -C.sub.4 -alkylamino, C.sub.1 -C.sub.4 -haloalkoxy, tri-(C.sub.1 -C.sub.4 -alkoxy)-silyl, cyano, nitro or phenyl; C.sub.1 -C.sub.4 -haloalkyl; C.sub.3 -C.sub.8 -alkenyl; (3-methyl-oxetan-3-yl)methyl; C.sub.3 -C.sub.8 -alkynyl; or a radical from the group comprising phenyl, benzyl, C.sub.3 -C.sub.7 -cycloalkyl, furanyl or furfuryl which is unsubstituted or mono-, di- or trisubstituted by identical or different substituents from the group comprising halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkylcarbonyl, nitro, C.sub.1 -C.sub.4 -alkoxy and C.sub.1 -C.sub.4 -haloalkyl; R.sub.3 and R.sub.4 independently of one another are hydrogen; a phenyl or benzyl radical which is unsubstituted or mono-, di-, tri- or tetrasubstituted by identical or different substituents from the group comprising halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkylcarbonyl, nitro, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkylthio and C.sub.1 -C.sub.4 -haloalkylthio; C.sub.1 -C.sub.8 -alkyl; or C.sub.3 -C.sub.6 -cycloalkyl; or R.sub.3 and R.sub.4, together with the nitrogen atom, form a saturated 5- or 6-membered heterocyclic ring which contains up to two heteroatoms from the group comprising N, O and S and can be mono- or disubstituted by C.sub.1 -C.sub.4 -allkyl; R.sub.5 is hydrogen; halogen; C.sub.1 -C.sub.8 -alkyl; C.sub.1 -C.sub.4 -alkoxy; C.sub.1 -C.sub.4 -haloalkyl; nitro; cyano; C.sub.1 -C.sub.4 -haloalkoxy; phenylthio; di-C.sub.1 -C.sub.4 -alkylamino; phenyl; or is phenoxy which is unsubstituted or substituted by the radicals R.sub.8 and R.sub.9 ; and R.sub.6, R.sub.7, R.sub.8 and R.sub.9 independently of one another are hydrogen; halogen; C.sub.1 -C.sub.8 -alkyl; C.sub.1 -C.sub.4 -haloalkyl; C.sub.1 -C.sub.4 -alkoxy; C.sub.1 -C.sub.4 -haloalkoxy; nitro; cyano; or di-C.sub.1 -C.sub.4 -alkylamino; and R.sub.10 and R.sub.11 independently of one another are C.sub.1 -C.sub.4 -alkyl; and salts of compounds of the formula I with acids and bases, process for their preparation and herbicidal or plant growth-regulating compositions containing compounds of the formula I.

5. 发明授权

US4851028A Method of combating undesirable plant growth and of regulating plant growth 失效
标题翻译：打击不良植物生长和调节植物生长的方法
公开(公告)号：US4851028A
公开(公告)日：1989-07-25
申请号：US92252
申请日：1987-09-02
申请人： Helmut Zondler , Wolfgang Eckhardt , Robert Nyfeler , Hans-Georg Brunner
发明人： Helmut Zondler , Wolfgang Eckhardt , Robert Nyfeler , Hans-Georg Brunner
IPC分类号： A01N43/54 , A01N43/60 , C07D239/42 , C07D241/14 , C07D241/20 , C07D405/12
CPC分类号： C07D239/42 , A01N43/54 , A01N43/60 , C07D241/20 , C07D405/12
摘要： A method of combating undesirable plant growth and of regulating plant growth, which comprises allowing a herbicidal or plant-regulating amount of a compound of the formula I ##STR1## in which R.sub.1 is SR.sub.2 ; OR.sub.2 ; O--CHR.sub.10 R.sub.2 ; N(R.sub.3) (CHR.sub.10 R.sub.4); N(R.sub.11)(CHR.sub.10 R.sub.4) or NR.sub.3 R.sub.4 ; R.sub.2 is optionally substituted C.sub.1 -C.sub.10 -alkyl C.sub.1 -C.sub.4 -haloalkyl; C.sub.3 -C.sub.8 -alkenyl; (3-methyloxetan-3-yl)methyl; C.sub.3 -C.sub.8 -alkynyl; or an optionally substituted radical from the group comprising phenyl, benzyl, C.sub.3 -C.sub.7 -cycloalkyl, furanyl or furfuryl R.sub.3 and R.sub.4 independently of one another are hydrogen; an optionally substituted phenyl or benzyl radical; C.sub.1 -C.sub.8 -alkyl; or C.sub.3 -C.sub.6 -cycloalkyl; or R.sub.3 and R.sub.4, together with the nitrogen atom, form a saturaated 5- or 6-membered heterocyclic ring which contains up to two heteroatoms from the group comprising N, O and S and can be mono- or disubstituted by C.sub.1 -C.sub.4 -alkyl; R.sub.5 is hydrogen; halogen; C.sub.1 -C.sub.8 -alkyl; C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkyl; nitro; cyano; C.sub.1 -C.sub.4 -haloalkoxy; phenylthio; di-C.sub.1 -C.sub.4 - alkylamino; phenyl; or is optionally substituted phenoxy; and R.sub.6 and R.sub.7 independently of one another are hydrogen; halogen; C.sub.1 -C.sub.8 -alkyl; C.sub.1 -C.sub.4 -haloalkyl; C.sub.1 -C.sub.4 -alkoxy; C.sub.1 -C.sub.4 -haloalkoxy; nitro; cyano; or di-C.sub.1 -C.sub.4 -alkylamino, and R.sub.10 and R.sub.11 independently of one another are C.sub.1 -C.sub.4 -alkyl; and salts of compounds of the formula I with acids and bases, to act on the plants or on the environment of the plants, and novel compounds of the formula I' ##STR2## process for their preparation and herbicidal or plant growth-regulating compositions containing these novel compounds.
摘要翻译：一种防治不期望的植物生长和调节植物生长的方法，其包括允许除草或植物调节量的其中R 1为SR 2的式I化合物（I）; OR2; O-CHR10R2; N（R3）（CHR10R4）; N（R11）（CHR10R4）或NR3R4; R2是任选取代的C 1 -C 10 - 烷基C 1 -C 4 - 卤代烷基; C3-C8-烯基; （3-甲基氧杂环丁烷-3-基）甲基; C3-C8-炔基; 或由苯基，苄基，C 3 -C 7 - 环烷基，呋喃基或糠基R3和R4彼此独立地选自任意取代的基团是氢; 任选取代的苯基或苄基; C 1 -C 8 - 烷基; 或C 3 -C 6 - 环烷基; 或R3和R4与氮原子一起形成饱和的5或6元杂环，其含有至多两个来自包含N，O和S的基团的杂原子，并且可被C1-C4烷基单或二取代 ; R5是氢; 卤素; C 1 -C 8 - 烷基; C 1 -C 4 - 烷氧基，C 1 -C 4 - 卤代烷基; 硝基氰基; C 1 -C 4卤代烷氧基; 苯硫基二-C 1 -C 4烷基氨基; 苯基; 或任选取代的苯氧基; 且R 6和R 7彼此独立地为氢; 卤素; C 1 -C 8 - 烷基; C 1 -C 4 - 卤代烷基; C1-C4-烷氧基; C 1 -C 4卤代烷氧基; 硝基氰基; 或二-C 1 -C 4烷基氨基，R 10和R 11彼此独立地为C 1 -C 4 - 烷基; 和式I化合物与酸和碱的盐作用于植物或植物环境，以及式I'（I'）的新化合物，其制备和除草或植物生长过程含有这些新化合物的调节组合物。

6. 发明授权

US4259505A Process for the preparation of 1H-azole derivatives 失效
标题翻译：制备1H-唑衍生物的方法
公开(公告)号：US4259505A
公开(公告)日：1981-03-31
申请号：US127018
申请日：1980-03-04
申请人： Elmar Sturm , Wolfgang Eckhardt , Bernhard Gloor , Robert Nyfeler
发明人： Elmar Sturm , Wolfgang Eckhardt , Bernhard Gloor , Robert Nyfeler
IPC分类号： C07D405/06 , A61K31/41 , A61P31/04 , C07D521/00
CPC分类号： C07D231/12 , C07D233/56 , C07D249/08
摘要： An improved process for the preparation of 2-tert.-butyl-2-[1-phenoxy-1-(1H-azol-1-yl)]-methyl-ketales is disclosed, which process comprises reacting a 2-tert.-butyl-2-[1-phenoxy-1-halo]-methyl-ketale with a quaternary ammonium or phosphonium salt of an azole. The azoles used are 1H-1,2,4-triazole or 1H-imidazole.
摘要翻译：公开了制备2-叔丁基-2- [1-苯氧基-1-（1H-吡唑-1-基）] - 甲基 - 缩酮的改进方法，该方法包括使2-叔丁基-2- 丁基-2- [1-苯氧基-1-卤代] - 甲基 - 缩酮与唑的季铵盐或鏻盐。所用的唑类是1H-1,2,4-三唑或1H-咪唑。

7. 发明授权

US4767443A Antifungal and antibacterial diazine derivatives compositions, intermediates, and method of use therefor 失效
标题翻译：抗真菌和抗菌二嗪衍生物组合物，中间体及其使用方法
公开(公告)号：US4767443A
公开(公告)日：1988-08-30
申请号：US775972
申请日：1985-09-13
申请人： Helmut Zondler , Wolfgang Eckhardt , Robert Nyfeler
发明人： Helmut Zondler , Wolfgang Eckhardt , Robert Nyfeler
IPC分类号： A01N43/54 , C07D239/42 , C07D405/12
CPC分类号： C07D239/42 , A01N43/54 , C07D405/12
摘要： There are described novel, microbicidally active 5-(arylmethylimino)-pyrimidines of the formula I ##STR1## wherein R.sub.n --A-- is an unsubstituted or substituted phenyl, naphthyl, biphenyl, phenoxyphenyl or phenylthiophenyl, and R.sub.1 is an ether, thioether or amino function, these substances being produced according to the invention by substitution of the halogen atom in the claimed intermediates of the formula II ##STR2## The use of these substances in plant protection, and also further important intermediates, are likewise described.
摘要翻译：描述了式I（I）的新颖的杀微生物活性5-（芳基甲基亚氨基） - 嘧啶，其中Rn-A-是未取代或取代的苯基，萘基，联苯基，苯氧基苯基或苯硫基苯基，R1是醚，硫醚或氨基官能团，这些物质根据本发明通过取代所要求的式II的中间体中的卤素原子（II）而产生。这些物质在植物保护中的用途以及其它重要的中间体同样是描述。

8. 发明授权

US4690942A 1-aryl-2-fluoro-2-azolyl alkanones, alkanols, esters, and ethers, composition containing them, and use of them to control phytopathogenic microorganisms 失效
标题翻译： 1-芳基-2-氟-2-噻唑烷酮，链烷醇，酯和醚，含有它们的组合物，以及它们用于控制植物病原微生物
公开(公告)号：US4690942A
公开(公告)日：1987-09-01
申请号：US681989
申请日：1984-12-14
申请人： Willy Frick , Alfred Meyer , Robert Nyfeler
发明人： Willy Frick , Alfred Meyer , Robert Nyfeler
IPC分类号： C07D249/08 , A01N43/50 , A01N43/653 , C07C45/63 , C07C49/80 , C07D233/56 , C07D233/60 , C07D249/00 , C07D307/00 , C07D405/12 , C07D521/00
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07C45/63 , C07C49/80 , C07D233/56 , C07D249/08
摘要： The invention relates to 1-aryl-2-fluoro-2-azolyl alkanones, alkanols, esters and ethers of formula I ##STR1## wherein Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole;T is --C(O)--, --CH(OH)-- or one of the groups ##STR2## wherein R.sub.7 is C.sub.1 -C.sub.6 alkyl which is unsubstituted or substituted by C.sub.1 -C.sub.3 -alkoxy, halogen or cyano, or is C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl, C.sub.3 -C.sub.6 cycloalkyl, 2-furyl, 2-tetrahydrofuryl, or is phenyl or benzyl, each unsubstituted or substituted by halogen, nitro, C.sub.1 -C.sub.3 -alkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkyl and/or C.sub.1 -C.sub.3 haloalkoxy;R.sub.8, R.sub.9 and R.sub.10 are each independently hydrogen, nitro, halogen, cyano, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 haloalkoxy, --COO(C.sub.1 -C.sub.3 alkyl), NH.sub.2 or NHCOCH.sub.3 ;R is hydrogen or C.sub.1 -C.sub.6 alkyl;R.sub.1 and R.sub.2 are each independently hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 -alkoxy, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkoxy, nitro and/or cyano; andR.sub.3 is hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 haloalkoxy, nitro, cyano and/or the group ##STR3## wherein X is O, S, SO or SO.sub.2 ;R.sub.4, R.sub.5 and R.sub.6 are each independently hydrogen, halogen, cyano, nitro, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.1 -C.sub.6 haloalkyl and/or C.sub.1 -C.sub.6 haloalkoxy; and to the acid addition salts and metal complexes thereof.These compounds have microbicidal properties and can be used in particular against diseases occurring in rice.The invention also relates to the preparation and use of these compounds.
摘要翻译：本发明涉及式I的1-芳基-2-氟-2-噻唑烷酮，链烷醇，酯和醚其中Az是1H-1,2,4-三唑，4H-1,2， 4-三唑或1H-咪唑; T是-C（O） - ， - CH（OH） - 或其中一个基团，其中R 7是未被取代或被C 1 -C 3 - 烷氧基，卤素或氰基取代的C 1 -C 6烷基，或者是C 3 -C 6烯基硝基，C 1 -C 3烷基，C 1 -C 3烷氧基，C 1 -C 3卤代烷基和/或C 1 -C 3烷氧基，C 3 -C 6炔基，C 3 -C 6环烷基，2-呋喃基，2-四氢呋喃基，或者是苯基或苄基， C3卤代烷氧基; R8，R9和R10各自独立地为氢，硝基，卤素，氰基，C1-C3烷基，C1-C3烷氧基，C1-C3卤代烷氧基，-COO（C1-C3烷基），NH2或NHCOCH3; R是氢或C 1 -C 6烷基; R 1和R 2各自独立地为氢，卤素，C 1 -C 6烷基，C 1 -C 6 - 烷氧基，C 1 -C 6卤代烷基，C 1 -C 6卤代烷氧基，硝基和/或氰基; 并且R 3是氢，卤素，C 1 -C 6烷基，C 1 -C 6烷氧基，C 1 -C 6卤代烷基，C 1 -C 6卤代烷氧基，硝基，氰基和/或其中X是O，S，SO或SO 2; R4，R5和R6各自独立地为氢，卤素，氰基，硝基，C1-C6烷基，C1-C6烷氧基，C1-C6卤代烷基和/或C1-C6卤代烷氧基; 和其酸加成盐和金属络合物。这些化合物具有杀微生物的性质，特别可用于防治水稻中发生的疾病。本发明还涉及这些化合物的制备和用途。

9. 发明授权

US4567052A 3-Phenyl-4-cyanopyrrole derivatives, the preparation thereof, and method of use thereof as microbicides 失效
标题翻译： 3-苯基-4-氰基吡咯衍生物，其制备方法及其作为杀微生物剂的使用方法
公开(公告)号：US4567052A
公开(公告)日：1986-01-28
申请号：US618867
申请日：1984-06-08
申请人： Robert Nyfeler
发明人： Robert Nyfeler
IPC分类号： A23L3/3526 , A23L3/3544 , C07D207/34 , C07D405/12 , A23L3/34 , C07D207/30 , C07D307/02 , C07D407/00
CPC分类号： C07D405/12 , A23L3/3526 , A23L3/3544 , C07D207/34
摘要： The invention relates to novel N-alkylated 3-phenyl-4-cyanopyrrole derivatives of the formula I ##STR1## wherein R.sub.1 and R.sub.2, each independently of the other, are hydrogen, halogen, methoxy or methylthio,R.sub.3 is hydrogen or C.sub.1 -C.sub.8 haloalkyl,Y is hydroxy, halogen or the --O--C(O)--R.sub.4 group, andR.sub.4 is hydrogen, C.sub.1 -C.sub.8 alkyl, C.sub.1 -C.sub.8 haloalkyl, C.sub.2 -C.sub.6 alkenyl, 2-tetrahydrofuryl, 2-tetrahydropyranyl, C.sub.1 -C.sub.6 alkoxycarbonyl or the --CH(R.sub.5)--XR.sub.6 group, whereinX is oxygen or sulfur,R.sub.5 is hydrogen or C.sub.1 -C.sub.3 alkyl, andR.sub.6 is C.sub.1 -C.sub.6 alkyl, (C.sub.1 -C.sub.6 alkoxy)-C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 alkynyl, phenyl or phenyl which is substituted by halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy, or C.sub.1 -C.sub.6 alkoxycarbonyl.The invention also relates to the preparation of these compounds by N-alkylation of the starting pyrroles, as well as to microbicidal compositions which contain a compound of formula I as active ingredient. Also disclosed is a method of controlling phytopathogenic micro-organisms which comprises the use of the novel compounds.
摘要翻译：本发明涉及式I（I）的新型N-烷基化3-苯基-4-氰基吡咯衍生物，其中R 1和R 2各自独立地为氢，卤素，甲氧基或甲硫基，R 3为氢或 C1-C8卤代烷基，Y是羟基，卤素或-OC（O）-R4基团，R4是氢，C1-C8烷基，C1-C8卤代烷基，C2-C6链烯基，2-四氢呋喃基，2-四氢吡喃基，C1-C6烷氧基羰基或 -CH（R5）-XR6基，其中X是氧或硫，R5是氢或C1-C3烷基，R6是C1-C6烷基，（C1-C6烷氧基）-C1-C6烷基，C3-C6链烯基，C3-C6炔基，苯基或被卤素，C 1 -C 6烷基，C 1 -C 6烷氧基或C 1 -C 6烷氧基羰基取代的苯基。本发明还涉及通过起始吡咯的N-烷基化制备这些化合物，以及含有式I化合物作为活性成分的杀微生物剂组合物。还公开了一种控制植物病原微生物的方法，其包括使用该新化合物。

10. 发明授权

US5190928A Process and a composition for immunizing plants against diseases 失效
标题翻译：用于免疫植物以防止疾病的方法和组合物
公开(公告)号：US5190928A
公开(公告)日：1993-03-02
申请号：US683582
申请日：1991-04-10
申请人： Rolf Schurter , Walter Kunz , Robert Nyfeler
发明人： Rolf Schurter , Walter Kunz , Robert Nyfeler
IPC分类号： C07D417/12 , A01N43/82 , A01N43/828 , C07D285/14 , C07D413/06 , C07D413/12 , C07D521/00 , C07F7/08 , C07F7/10 , C07F9/32 , C07F9/6515 , C07F9/6518 , C07F9/6539 , C07F9/6541 , C07H13/08 , C07H13/10 , C07H17/00 , C07H17/02
CPC分类号： C07D285/14 , A01N43/82 , C07D231/12 , C07D233/56 , C07D249/08 , C07D413/06 , C07D413/10 , C07D413/12 , C07F7/0812 , C07F9/6541 , C07H13/10
摘要： A method and composition for the immunization of healthy useful plants against plant diseases containing as active ingredients compounds of formula ##STR1## in which: X is hydrogen, halogen, hydroxy, methyl, methoxy, HOOC or MOOC;Y is hydrogen, halogen, SO.sub.3 H, SO.sub.3 M, nitro, hydroxy or amino, M being the molar equivalent of an alkali metal or alkaline earth metal ion that is formed from a corresponding base or basic compound; andZ is cyano or --CO--A;A represents either --OH or --SH, the hydrogen atom of which may also be replaced by the molar equivalent of an inorganic or organic cationic residue,or wherein A represents any other organic residue which has a molecular weight of less than 900 and which may also contain one, or more than one, hetero atom, including the salts of the phytophysiologically tolerable 7-carboxylic acid or 7-thiocarboxylic acid with primary, secondary or tertiary amines or with inorganic bases.
摘要翻译：含有作为活性成分的式（I）化合物的健康有益植物免疫植物病害的方法和组合物，其中：X是氢，卤素，羟基，甲基，甲氧基，HOOC或MOOC; Y是氢，卤素，SO 3 H，SO 3 M，硝基，羟基或氨基，M是由相应的碱或碱化合物形成的碱金属或碱土金属离子的摩尔当量; 和Z是氰基或-CO-A; A表示-OH或-SH，其氢原子也可被无机或有机阳离子残基的摩尔当量代替，或其中A表示分子量小于900的任何其它有机残基，还含有一个或多于一个杂原子，包括植物生理学上可耐受的7-羧酸或7-硫代羧酸与伯胺，仲胺或叔胺或与无机碱的盐。

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