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1. 发明申请

US20050215797A1 Pyrazole derivatives and process for the production thereof 有权
标题翻译：吡唑衍生物及其制备方法
公开(公告)号：US20050215797A1
公开(公告)日：2005-09-29
申请号：US10521593
申请日：2003-07-31
申请人： Masao Nakatani , Minoru Ito , Masahiro Miyazaki
发明人： Masao Nakatani , Minoru Ito , Masahiro Miyazaki
IPC分类号： C07D231/20 , C07D231/22 , A61K31/4152 , C07D231/18
CPC分类号： C07D231/20 , C07D231/22
摘要： The present invention provides pyrazole derivatives useful as production intermediates for isoxazoline derivatives having an excellent herbicidal effect and selectivity between crops and weeds as well as processes for producing the same. The pyrazole derivatives or pharmaceutically acceptable salts thereof which are inventive compounds are represented by the general formula [I] or a salt thereof: wherein R1 represents a C1 to C6 alkyl group, R2 represents a C1 to C3 haloalkyl group, R3 represents a hydrogen atom, a C1 to C3 alkyl group which may be substituted with one or more substituents selected from the following substituent group α, or a formyl group, R4 represents a hydrogen atom or a C1 to C3 haloalkyl group, provided that R4 represents a C1 to C3 haloalkyl group in the case that R3 is a hydrogen or a formyl group, and R4 is a hydrogen group or a C1 to C3 haloalkyl group in the case that R3 is a C1 to C3 alkyl group which may be substituted with one or more substituents selected from the following substituent group α.
摘要翻译：本发明提供了可用作具有优异的除草效果和作物和杂草之间的选择性的异恶唑啉衍生物的生产中间体的吡唑衍生物及其制备方法。作为本发明化合物的吡唑衍生物或其药学上可接受的盐由通式[I]或其盐表示：其中R 1表示C 1至C 6烷基，R 2， / SUP>表示C1至C3卤代烷基，R 3表示氢原子，可被一个或多个选自以下取代基组α的取代基取代的C1至C3烷基，或甲酰基，R 4表示氢原子或C 1至C 3卤代烷基，条件是R 4表示C 1至C 3卤代烷基， 3是氢或甲酰基，R 4是氢或C1至C3卤代烷基，在R 3是C1的情况下可以被一个或多个选自以下取代基组α的取代基取代的C 3烷基。

2. 发明授权

US07256298B2 Pyrazole derivatives and process for the production thereof 有权
标题翻译：吡唑衍生物及其制备方法
公开(公告)号：US07256298B2
公开(公告)日：2007-08-14
申请号：US10521593
申请日：2003-07-31
申请人： Masao Nakatani , Minoru Ito , Masahiro Miyazaki
发明人： Masao Nakatani , Minoru Ito , Masahiro Miyazaki
IPC分类号： C07D231/18
CPC分类号： C07D231/20 , C07D231/22
摘要： The present invention provides pyrazole derivatives useful as production intermediates for isoxazoline derivatives having an excellent herbicidal effect and selectivity between crops and weeds as well as processes for producing the same.The pyrazole derivatives or pharmaceutically acceptable salts thereof which are inventive compounds are represented by the general formula [I] or a salt thereof: wherein R1 represents a C1 to C6 alkyl group, R2 represents a C1 to C3 haloalkyl group, R3 represents a hydrogen atom, a C1 to C3 alkyl group which may be substituted with one or more substituents selected from the following substituent group α, or a formyl group, R4 represents a hydrogen atom or a C1 to C3 haloalkyl group, provided that R4 represents a C1 to C3 haloalkyl group in the case that R3 is a hydrogen or a formyl group, and R4 is a hydrogen group or a C1 to C3 haloalkyl group in the case that R3 is a C1 to C3 alkyl group which may be substituted with one or more substituents selected from the following substituent group α.
摘要翻译：本发明提供了可用作具有优异的除草效果和作物和杂草之间的选择性的异恶唑啉衍生物的生产中间体的吡唑衍生物及其制备方法。作为本发明化合物的吡唑衍生物或其药学上可接受的盐由通式[I]或其盐表示：其中R 1表示C 1至C 6烷基，R 2， / SUP>表示C1至C3卤代烷基，R 3表示氢原子，可被一个或多个选自以下取代基组α的取代基取代的C1至C3烷基，或甲酰基，R 4表示氢原子或C 1至C 3卤代烷基，条件是R 4表示C 1至C 3卤代烷基， 3是氢或甲酰基，R 4是氢或C1至C3卤代烷基，在R 3是C1的情况下可以被一个或多个选自以下取代基组α的取代基取代的C 3烷基。

3. 发明授权

US07875606B2 Izoxazoline derivative and herbicide 有权
标题翻译：伊佐唑啉衍生物和除草剂
公开(公告)号：US07875606B2
公开(公告)日：2011-01-25
申请号：US10480376
申请日：2002-06-20
申请人： Masao Nakatani , Minoru Ito , Kyoko Kimijima , Masahiro Miyazaki , Makoto Fujinami , Ryohei Ueno , Satoru Takahashi
发明人： Masao Nakatani , Minoru Ito , Kyoko Kimijima , Masahiro Miyazaki , Makoto Fujinami , Ryohei Ueno , Satoru Takahashi
IPC分类号： A61K31/541 , A61K31/496 , C07D417/02 , C07D413/02
CPC分类号： C07D413/12 , A01N43/80 , A01N43/82 , A01N43/90
摘要： The present invention aims at providing an isoxazoline derivative and a pharmaceutically acceptable salt thereof, both having an excellent herbicidal effect and an excellent selectivity between crop and weed.The isoxazoline derivative of the present invention is represented by the following general formula: wherein R1 is a haloalkyl group; R2 is a hydrogen atom, an alkyl group, or the like; R3, R4, R5 and R6 are each a hydrogen atom, or the like; Y is a pyrrolyl group, a pyrazolyl group, an isothiazolyl group, an oxazolyl group, an imidazolyl group, a pyridazinyl group, a pyrimidinyl group, a pyrazinyl group, a triazinyl group, a triazolyl group, an oxadiazolyl group, or the like; and n is an integer of 0 to 2.
摘要翻译：本发明的目的在于提供一种异恶唑啉衍生物及其药学上可接受的盐，它们具有优异的除草效果和作物和杂草之间优异的选择性。本发明的异恶唑啉衍生物由以下通式表示：其中R1是卤代烷基; R2是氢原子，烷基等; R3，R4，R5和R6各自为氢原子等; Y是吡咯基，吡唑基，异噻唑基，恶唑基，咪唑基，哒嗪基，嘧啶基，吡嗪基，三嗪基，三唑基，恶二唑基等; n为0〜2的整数。

4. 发明申请

US20070249844A1 Pyrazole derivatives and process for the production thereof 审中-公开
公开(公告)号：US20070249844A1
公开(公告)日：2007-10-25
申请号：US11819965
申请日：2007-06-29
申请人： Masao Nakatani , Minoru Ito , Masahiro Miyazaki
发明人： Masao Nakatani , Minoru Ito , Masahiro Miyazaki
IPC分类号： C07D231/20
CPC分类号： C07D231/20 , C07D231/22
摘要： The present invention provides pyrazole derivatives useful as production intermediates for isoxazoline derivatives having an excellent herbicidal effect and selectivity between crops and weeds as well as processes for producing the same. The pyrazole derivatives or pharmaceutically acceptable salts thereof which are inventive compounds are represented by the general formula [I] or a salt thereof: wherein R1 represents a C1 to C6 alkyl group, R2 represents a C1 to C3 haloalkyl group, R3 represents a hydrogen atom, a C1 to C3 alkyl group which may be substituted with one or more substituents selected from the following substituent group α, or a formyl group, R4 represents a hydrogen atom or a C1 to C3 haloalkyl group, provided that R4 represents a C1 to C3 haloalkyl group in the case that R3 is a hydrogen or a formyl group, and R4 is a hydrogen group or a C1 to C3 haloalkyl group in the case that R3 is a C1 to C3 alkyl group which may be substituted with one or more substituents selected from the following substituent group α.

5. 发明授权

US07238689B2 Isoxazoline derivative and herbicide comprising the same as active ingredient 有权
标题翻译：异恶唑啉衍生物和除草剂，其与活性成分相同
公开(公告)号：US07238689B2
公开(公告)日：2007-07-03
申请号：US10250937
申请日：2002-02-07
申请人： Masao Nakatani , Ryotaro Kugo , Masahiro Miyazaki , Koichiro Kaku , Makoto Fujinami , Ryohei Ueno , Satoru Takahashi
发明人： Masao Nakatani , Ryotaro Kugo , Masahiro Miyazaki , Koichiro Kaku , Makoto Fujinami , Ryohei Ueno , Satoru Takahashi
IPC分类号： C07D417/02 , C07D413/02 , A61K31/541 , A61K31/5377 , A61K31/496
CPC分类号： C07D261/10 , A01N43/80 , A01N43/90 , A01N47/38 , C07D261/04 , C07D261/08 , C07D261/20 , C07D413/12 , C07D413/14 , C07D417/12
摘要： An isoxazoline derivative represented by the following general formula [I]: wherein R1 and R2 may be the same or different and are each an alkyl group; R3, R4, R5 and R6 are each a hydrogen atom; Y is an optionally substituted 5- to 6-membered aromatic heterocyclic group or fused aromatic heterocyclic group having a hetero atom selected from a nitrogen atom, a oxygen atom and a sulfur atom; and n is an integer: of 0 to 2. The isoxazoline derivative has an excellent herbicidal effect and an excellent selectivity between crop and weed.
摘要翻译：由以下通式[I]表示的异恶唑啉衍生物：其中R 1和R 2可以相同或不同，并且各自为烷基; R 3，R 4，R 5和R 6各自为氢原子; Y是具有选自氮原子，氧原子和硫原子的杂原子的任选取代的5至6元芳族杂环基或稠合芳族杂环基; n为0〜2的整数。异恶唑啉衍生物具有优良的除草效果，作物和杂草之间的选择性优异。

6. 发明授权

US06841519B1 Isoxazoline derivatives and herbicides containing the same as the active ingredient 有权
标题翻译：含有与活性成分相同的异恶唑啉衍生物和除草剂
公开(公告)号：US06841519B1
公开(公告)日：2005-01-11
申请号：US10049039
申请日：2000-08-09
申请人： Masao Nakatani , Kouichirou Kaku , Takumi Yoshimura , Masatoshi Tamaru , Hiroshi Kawasaki , Kazunori Kobayashi , Takeshige Miyazawa
发明人： Masao Nakatani , Kouichirou Kaku , Takumi Yoshimura , Masatoshi Tamaru , Hiroshi Kawasaki , Kazunori Kobayashi , Takeshige Miyazawa
IPC分类号： A01N43/80 , A01P13/00 , C07D261/04 , C07D261/20
CPC分类号： A01N43/80 , C07D261/04 , C07D261/20
摘要： The isoxazoline derivative of the present invention is represented by the following general formula [I]: [wherein Q is a group represented by —S(O)n—(CR5R6)m- (wherein n is an integer of 0 to 2, m is an integer of 1 to 3, and R5 and R6 are a hydrogen atom, a cyano group, an alkoxycarbonyl group, if an alkyl group or the like); R1 and R2 are a hydrogen atom, all optionally substituted alkyl group, an alkoxycarbonyl group, an optionally substituted phenyl group or the like; R3 and R4 are a hydrogen atom, an optionally substituted alkyl group, a cycloalkyl group or the like; Y is a hydrogen atom, an alkoxycarbonyl group, a carboxyl group, an alkenyl group, an optionally substituted alkyl group or an optionally substituted phenyl group]. The herbicide of the present invention contains the above isoxazoline derivative as the active ingredient.
摘要翻译：本发明的异恶唑啉衍生物由以下通式[I]表示：[其中Q为-S（O）n - （CR 5 R 6）m - （其中n为0〜2的整数，m 为1〜3的整数，R5，R6为氢原子，氰基，烷氧基羰基，烷基等）。 R1和R2是氢原子，全部任选取代的烷基，烷氧基羰基，任意取代的苯基等; R3和R4是氢原子，任选取代的烷基，环烷基等; Y是氢原子，烷氧基羰基，羧基，烯基，任意取代的烷基或任意取代的苯基]。本发明的除草剂含有上述异恶唑啉衍生物作为有效成分。

7. 发明授权

US5763463A Pyridine compounds which are useful as pesticides 失效
标题翻译：用作农药的吡啶化合物
公开(公告)号：US5763463A
公开(公告)日：1998-06-09
申请号：US849718
申请日：1997-06-25
申请人： Nobuo Takefuji , Masao Nakatani , Junko Suzuki , Masami Ozaki , Ryouhei Ueno , Hiroyuki Yano , Mieko Kawashima , Yutaka Kurihara , Tomonori Shimazu
发明人： Nobuo Takefuji , Masao Nakatani , Junko Suzuki , Masami Ozaki , Ryouhei Ueno , Hiroyuki Yano , Mieko Kawashima , Yutaka Kurihara , Tomonori Shimazu
IPC分类号： A01N43/40 , A01N47/20 , C07D213/75 , C07D213/84 , C07D213/85 , C07F7/08 , C07D213/71
CPC分类号： C07D213/75 , A01N43/40 , A01N47/20 , C07D213/84 , C07D213/85 , C07F7/0812
摘要： A pyridine derivative of the formula (I), or its oxide or salt: ##STR1## wherein R.sup.1 is a halogen atom, an alkyl group, etc., R.sup.2 is an alkenyl group, an alkynyl group, an alkoxycarbonyl group, an alkenyloxycarbonyl group, etc., R.sup.3 is a hydrogen atom, etc., R.sup.4 is a halogen atom, a cyano group, a haloalkyl group, etc., each of R.sup.5 and R.sup.6 is a hydrogen atom, etc., Q is a methine group or a nitrogen atom, m is 0 or 1, n is 1 or 2 and r is 1 or 2. Such a compound is useful as a pesticide. The compound of the present invention is a pyridine derivative which is capable of killing or controlling various pests without adversely affecting crop plants and which is readily decomposable and presents no substantial acute toxity to mammals.
摘要翻译： PCT No.PCT / JP96 / 01096 Sec。 371日期：1997年6月25日 102（e）日期1996年6月25日PCT提交1996年4月23日PCT公布。第WO96 / 33975号公报日期：1996年10月31日一种式（I）的吡啶衍生物或其氧化物或盐：其中R1是卤素原子，烷基等，R2是链烯基，炔基，烷氧基羰基，链烯氧基羰基等，R3为氢原子等，R4为卤素原子，氰基，卤代烷基等，R5和R6分别为氢原子等。 Q为次甲基或氮原子，m为0或1，n为1或2，r为1或2.这种化合物可用作农药。本发明的化合物是能够杀死或控制各种害虫而不会不利影响作物的吡啶衍生物，其易于分解并且对哺乳动物没有显着的急性毒性。

8. 发明申请

US20090042917A1 Aminopyrimidine Derivative and Plant Disease Control Agent for Agricultural or Horticultural Use 审中-公开
标题翻译：氨基嘧啶衍生物和农业或园艺用途的植物病害防治剂
公开(公告)号：US20090042917A1
公开(公告)日：2009-02-12
申请号：US12087003
申请日：2007-01-18
申请人： Junichiro Bessho , Masao Nakatani , Yuuki Hirano , Hirokazu Arai , Atsushi Kogure , Norihisa Yonekura , Ryo Hanai
发明人： Junichiro Bessho , Masao Nakatani , Yuuki Hirano , Hirokazu Arai , Atsushi Kogure , Norihisa Yonekura , Ryo Hanai
IPC分类号： A01N43/56
CPC分类号： C07D403/04 , A01N43/56 , C07D401/14 , C07D403/14
摘要： A plant disease control agent contains, as an active ingredient, at least one aminopyrimidine derivatives represented by General Formula [I]: wherein R is a C2-10 alkyl group; R1 and R2 are each independently a hydrogen atom or a substituent such as an optionally substituted C1-10 alkyl group; X is hydrogen or a substituent selected from a predefined substituent group; Y is a substituent selected from a predefined substituent group; and m is an integer from 0 to 3, and agriculturally acceptable salts thereof.
摘要翻译：植物病害防治剂含有至少一种由通式[I]表示的氨基嘧啶衍生物作为活性成分：其中R是C2-10烷基; R 1和R 2各自独立地为氢原子或取代基，例如任选取代的C 1-10烷基; X是氢或选自预定义的取代基的取代基; Y是选自预定义的取代基的取代基; m为0〜3的整数，以及农业上可接受的盐。

9. 发明授权

US06458748B1 Di- or tri-fluoromethanesulfonyl anilide derivatives, process for the preparation of them and herbicides containing them as the active ingredient 有权
标题翻译：二 - 或三氟甲磺酰苯胺衍生物，其制备方法和含有它们作为活性成分的除草剂
公开(公告)号：US06458748B1
公开(公告)日：2002-10-01
申请号：US09744209
申请日：2001-01-22
申请人： Takumi Yoshimura , Masao Nakatani , Masatoshi Tamaru , Takeshi Danjo , Yukimasa Ono , Katsutada Yanagisawa
发明人： Takumi Yoshimura , Masao Nakatani , Masatoshi Tamaru , Takeshi Danjo , Yukimasa Ono , Katsutada Yanagisawa
IPC分类号： C07D23952
CPC分类号： A01N43/54 , A01N47/02 , C07D239/52
摘要： The present invention provides a novel compound which is effective for the removal of a wide variety of weeds including difficult-to-control weeds emerging in paddy field and which is safe to mammals; a process for production thereof; a herbicide containing the compound as an active ingredient; and novel raw material compounds used in said process. The present invention relates to a di- or trifluoromethanesulfonyl anilide derivative represented by the following general formula: (wherein R1 is a hydrogen atom, an alkyl group or an alkoxyalkyl group; and R2 is a hydrogen atom when R1 is a hydrogen atom or an alkyl group, and is a hydrogen atom or a fluorine atom when R1 is an alkoxyalkyl group), or a salt thereof, both of said derivative and said salt having a herbicidal activity.
摘要翻译：本发明提供了一种新颖的化合物，其有效去除各种杂草，包括难以控制的稻田中出现的杂草，对哺乳动物是安全的; 其生产方法; 含有该化合物作为活性成分的除草剂; 和所述方法中使用的新型原料化合物。本发明涉及由以下通式表示的二 - 或三氟甲磺酰苯胺衍生物：其中R1是氢原子，烷基或烷氧基烷基; R2是氢当R 1为氢原子或烷基时为原子，当R 1为烷氧基烷基时为氢原子或氟原子）或其盐，所述衍生物和所述盐都具有除草活性。

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