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1. 发明申请

US20120065154A1 Pyrazolo Pyrimidine Derivatives and Methods of Use Thereof 审中-公开
标题翻译：吡唑并嘧啶衍生物及其使用方法
公开(公告)号：US20120065154A1
公开(公告)日：2012-03-15
申请号：US13016957
申请日：2011-01-28
申请人： Masahiro Tanaka , Chao Zhang , Kevan M. Shokat , Alma L. Burlingame , Kirk Hansen , Raynard L. Bateman , Stephen G. DiMagno
发明人： Masahiro Tanaka , Chao Zhang , Kevan M. Shokat , Alma L. Burlingame , Kirk Hansen , Raynard L. Bateman , Stephen G. DiMagno
IPC分类号： A61K31/704 , A61K31/519 , A61K31/52 , A61P35/00 , C12Q1/18 , A61P29/00 , A61P3/00 , A61P3/10 , A61P3/04 , C07D487/04 , A61P35/02
CPC分类号： C07D487/04
摘要： This invention generally relates to pyrazolo pyrimidine derivatives useful as, inter alia, inhibitors of short chain dehydrogenase/reductase (SDR) family of NAD(P)(H) dependent oxido-reductases. More specifically, the invention relates to pyrazolo pyrimidine derivatives, including derivatives and analogs of SDR inhibitors, pharmaceutical compositions containing derivatives and analogs of SDR inhibitors, methods of making derivatives and analogs of SDR inhibitors and methods of use thereof.
摘要翻译：本发明一般涉及用作特别是NAD（P）（H）依赖性氧化还原酶的短链脱氢酶/还原酶（SDR）家族的抑制剂的吡唑并嘧啶衍生物。更具体地，本发明涉及吡唑并嘧啶衍生物，包括SDR抑制剂的衍生物和类似物，含有SDR抑制剂的衍生物和类似物的药物组合物，制备SDR抑制剂的衍生物和类似物的方法及其使用方法。

2. 发明申请

US20090181988A1 Pyrazolo Pyrimidine Derivatives and Methods of Use Thereof 审中-公开
标题翻译：吡唑并嘧啶衍生物及其使用方法
公开(公告)号：US20090181988A1
公开(公告)日：2009-07-16
申请号：US12194469
申请日：2008-08-19
申请人： Masahiro Tanaka , Chao Zhang , Kevan M. Shokat , Alma L. Burlingame , Kirk Hansen , Raynard L. Bateman , Stephen G. DiMagno
发明人： Masahiro Tanaka , Chao Zhang , Kevan M. Shokat , Alma L. Burlingame , Kirk Hansen , Raynard L. Bateman , Stephen G. DiMagno
IPC分类号： A61K31/522 , C12Q1/02 , C07D473/34 , A61K31/519 , C07D473/30 , A61K31/52 , C07D487/04 , A61P35/00
CPC分类号： C07D487/04
摘要： This invention generally relates to pyrazolo pyrimidine derivatives useful as, inter alia, inhibitors of short chain dehydrogenase/reductase (SDR) family of NAD(P)(H) dependent oxido-reductases. More specifically, the invention relates to pyrazolo pyrimidine derivatives, including derivatives and analogs of SDR inhibitors, pharmaceutical compositions containing derivatives and analogs of SDR inhibitors, methods of making derivatives and analogs of SDR inhibitors and methods of use thereof.
摘要翻译：本发明一般涉及用作特别是NAD（P）（H）依赖性氧化还原酶的短链脱氢酶/还原酶（SDR）家族的抑制剂的吡唑并嘧啶衍生物。更具体地，本发明涉及吡唑并嘧啶衍生物，包括SDR抑制剂的衍生物和类似物，含有SDR抑制剂的衍生物和类似物的药物组合物，制备SDR抑制剂的衍生物和类似物的方法及其使用方法。

3. 发明授权

US07429596B2 1H-pyrrolo [2,3-D] pyrimidine derivatives and methods of use thereof 有权
标题翻译： 1H-吡咯并[2,3-D]嘧啶衍生物及其使用方法
公开(公告)号：US07429596B2
公开(公告)日：2008-09-30
申请号：US10871732
申请日：2004-06-18
申请人： Masahiro Tanaka , Chao Zhang , Kevan M. Shokat , Alma L. Burlingame , Kirk Hansen , Raynard L. Bateman , Stephen G. DiMagno
发明人： Masahiro Tanaka , Chao Zhang , Kevan M. Shokat , Alma L. Burlingame , Kirk Hansen , Raynard L. Bateman , Stephen G. DiMagno
IPC分类号： C07D487/04 , C07D413/06 , A61K31/519 , A61K31/675 , A61K31/662 , A61K31/497 , A61K31/5355 , C07F9/38 , A61P35/04 , A61P35/02
CPC分类号： C07D487/04
摘要： This invention generally relates to pyrazolo pyrimidine derivatives useful as inhibitors of short chain dehydrogenase/reductase (SDR) family of NAD(P)(H) dependent oxido-reductases. The invention further relates to pharmaceutical compositions and methods of preventing or treating disease with 1H-Pyrrolo[2.3-d]pyrimidine derivatives. More specifically, the invention relates to a 1H-Pyrrolo[2.3-d]pyrimidine which is a compound of Formula I or II: or a pharmaceutically-acceptable salt or prodrug thereof; wherein: Y is N or CR5; Z is NR3R4, halo, H, OH, alkyl, alkyloxy, or haloalkyl; and R1a is indolyl, thiazolyl, benzyl, biphenylyl, thiophenyl, pyrrolyl, or phenyl, wherein said phenyl is substituted with at least one of OH, —NR3R4, —C(═O)NR6R7, —CN, NO2—C(═O)OH, —C(═O)O-alkyl, (C1-C4)alkyl, halo, haloalkyl or haloaryl; and wherein said indolyl, thiazolyl, benzyl, biphenylyl, thiophenyl, or pyrrolyl is optionally substituted with OH, —NR3R4, —C(═O)NR6R7, —CN, NO2, —C(═O)O—R3, (C1-C4)alkyl, halo, haloalkyl or haloaryl.
摘要翻译：本发明一般涉及可用作NAD（P）（H）依赖性氧化还原酶的短链脱氢酶/还原酶（SDR）家族的抑制剂的吡唑并嘧啶衍生物。本发明还涉及用1H-吡咯并[2,3-d]嘧啶衍生物预防或治疗疾病的药物组合物和方法。更具体地，本发明涉及作为式I或II化合物的1H-吡咯并[2,3-d]嘧啶或其药学上可接受的盐或前药; 其中：Y是N或CR 5; Z是NR 3 R 4，卤素，H，OH，烷基，烷氧基或卤代烷基; 并且R 1a是吲哚基，噻唑基，苄基，联苯基，噻吩基，吡咯基或苯基，其中所述苯基被OH，-NR 3 R 3中的至少一个取代， -C（-O）NR 6 R 7，-CN，NO 2 -C（-O（O））OH，-C（-O）O-烷基，（C 1 -C 4 -C 4）烷基，卤素，卤代烷基或卤代芳基; 并且其中所述吲哚基，噻唑基，苄基，联苯基，噻吩基或吡咯基任选被OH，-NR 3 R 4，-C（ - ）NR -C（O）OR 3，-C（-O）OR 3，（C 1 -C 6） C 1 -C 4烷基，卤素，卤代烷基或卤代芳基。

4. 发明申请

US20050085472A1 Pyrazolo pyrimidine derivatives and methods of use thereof 有权
标题翻译：吡唑并嘧啶衍生物及其使用方法
公开(公告)号：US20050085472A1
公开(公告)日：2005-04-21
申请号：US10871732
申请日：2004-06-18
申请人： Masahiro Tanaka , Chao Zhang , Kevan Shokat , Alma Burlingame , Kirk Hansen , Raynard Bateman , Stephen DiMagno
发明人： Masahiro Tanaka , Chao Zhang , Kevan Shokat , Alma Burlingame , Kirk Hansen , Raynard Bateman , Stephen DiMagno
IPC分类号： A61K20060101 , A61K31/519 , A61K31/5377 , A61P35/00 , C07D487/02 , C07D487/04
CPC分类号： C07D487/04
摘要： This invention generally relates to pyrazolo pyrimidine derivatives useful as, inter alia, inhibitors of short chain dehydrogenase/reductase (SDR) family of NAD(P)(H) dependent oxido-reductases. More specifically, the invention relates to pyrazolo pyrimidine derivatives, including derivatives and analogs of SDR inhibitors, pharmaceutical compositions containing derivatives and analogs of SDR inhibitors, methods of making derivatives and analogs of SDR inhibitors and methods of use thereof.
摘要翻译：本发明一般涉及用作特别是NAD（P）（H）依赖性氧化还原酶的短链脱氢酶/还原酶（SDR）家族的抑制剂的吡唑并嘧啶衍生物。更具体地，本发明涉及吡唑并嘧啶衍生物，包括SDR抑制剂的衍生物和类似物，含有SDR抑制剂的衍生物和类似物的药物组合物，制备SDR抑制剂的衍生物和类似物的方法及其使用方法。

5. 发明申请

US20140232536A1 INTRUSION DETECTION DEVICE 有权
标题翻译：入侵检测装置
公开(公告)号：US20140232536A1
公开(公告)日：2014-08-21
申请号：US14009090
申请日：2012-04-02
申请人： Ryuzo Uda , Toyohiro Tani , Kazushi Goto , Tomoyuki Funayama , Takeo Endo , Masahiro Tanaka
发明人： Ryuzo Uda , Toshimasa Takagi , Toyohiro Tani , Kazushi Goto , Tomoyuki Funayama , Takeo Endo , Masahiro Tanaka
IPC分类号： B60R25/30
CPC分类号： B60R25/30 , B60R25/10 , B60R25/1009 , G01S15/523 , G08B13/04 , G08B13/1618 , G08B13/1645
摘要： In an intrusion detection device of the embodiment, a determining unit allows a transmission unit to stop transmitting ultrasonic waves until a level of a Doppler signal exceeds a predetermined threshold (threshold for detecting destruction of a window glass), and allows the transmission unit to transmit the ultrasonic waves when the level of the Doppler signal exceeds said threshold. Therefore, if the destruction of the window glass is not detected, it is possible to reduce power consumption through allowing the transmission unit to stop the transmission. Further, because processing for detecting intrusion is performed after the destruction of the window glass has been detected, it is possible to reduce erroneous detection of an intruder resulting from a movement of an object (e.g., falling of papers, a sunshade, or the like that is leaned against the interior wall) other than a human.
摘要翻译：在本实施例的入侵检测装置中，确定单元允许发送单元停止发送超声波，直到多普勒信号的电平超过预定阈值（用于检测窗玻璃的破坏的阈值），并且允许发送单元发送当多普勒信号的电平超过所述阈值时的超声波。因此，如果没有检测到窗玻璃的破坏，则可以通过允许传输单元停止传输来降低功耗。此外，由于在检测到窗玻璃的破坏之后执行用于检测入侵的处理，可以减少由于物体的移动导致的入侵者的错误检测（例如，纸张的下落，遮阳等等这是靠在内墙上），而不是一个人。

6. 发明申请

US20130292860A1 HOLLOW FIBER MEMBRANE SPINNING NOZZLE, AND METHOD FOR MANUFACTURING HOLLOW FIBER MEMBRANE 审中-公开
标题翻译：中空纤维膜纺丝喷嘴及制造中空纤维膜的方法
公开(公告)号：US20130292860A1
公开(公告)日：2013-11-07
申请号：US13988697
申请日：2011-11-24
申请人： Hiroyuki Fujiki , Toshinori Sumi , Yasuo Hiromoto , Osamu Maehara , Masahiro Tanaka , Masashi Teramachi
发明人： Hiroyuki Fujiki , Toshinori Sumi , Yasuo Hiromoto , Osamu Maehara , Masahiro Tanaka , Masashi Teramachi
IPC分类号： D01D5/247
CPC分类号： B01D69/085 , B01D69/087 , B01D2323/42 , B29C48/11 , B29C48/29 , B29L2031/755 , D01D1/09 , D01D4/02 , D01D4/06 , D01D5/24 , D01D5/247
摘要： A hollow fiber membrane-spinning nozzle that spins a hollow fiber membrane having a porous membrane layer and a support is provided in which the nozzle includes a resin flow channel through which a membrane-forming resin solution forming the porous membrane layer flows, the resin flow channel includes a liquid storage section that stores the membrane-forming resin solution and a shaping section that shapes the membrane-forming resin solution in a cylindrical shape and satisfies at least one of conditions (a) to (c): (a) the resin flow channel is disposed to cause the membrane-forming resin solution to branch and merge; (b) a delay means for delaying the flow of the membrane-forming resin solution is disposed in the resin flow channel; and (c) the liquid storage section or the shaping section includes branching and merging means for the membrane-forming resin solution therein.
摘要翻译：提供一种中空纤维膜纺丝喷嘴，其旋转具有多孔膜层和支撑体的中空纤维膜，其中，喷嘴包括树脂流路，形成多孔膜层的成膜树脂溶液通过该树脂流路流动，树脂流通道包括储存膜形成树脂溶液的液体储存部分和成形部分，其将成膜树脂溶液成形为圆柱形并满足条件（a）至（c）中的至少一个：（a）树脂设置流路使膜成形树脂溶液分支合并; （b）在树脂流动通道中设置用于延迟成膜树脂溶液的流动的延迟装置; 和（c）液体储存部分或成形部分包括其中的成膜树脂溶液的分支和合并装置。

7. 发明授权

US08432950B2 Radio control transmitter and method for communication in the same 有权
标题翻译：无线电控制发射机和通信方法相同
公开(公告)号：US08432950B2
公开(公告)日：2013-04-30
申请号：US12883855
申请日：2010-09-16
申请人： Masahiro Tanaka , Eiichi Nishizawa
发明人： Masahiro Tanaka , Eiichi Nishizawa
IPC分类号： H04B1/69 , H04B1/707 , H04B1/713
CPC分类号： A63H30/04 , G08C17/02
摘要： A maneuvering signal for controlling a radio-controlled object is transmitted using 2.4 GHz band frequency hopping techniques. In a trainer mode, an instructor's radio control transmitter is configured to transmit the maneuvering signal and receive a trainer signal in each of frame periods by which a frequency is switched in accordance with the frequency hopping scheme. A trainee's radio control transmitter is configured to transmit the trainer signal for each of the frame periods by which a frequency is switched in accordance with the frequency hopping scheme.
摘要翻译：用于控制无线电控制对象的操纵信号使用2.4GHz频带跳频技术传输。在训练器模式中，教师的无线电控制发射机被配置为发送操纵信号，并且在根据跳频方案切换频率的每个帧周期中接收训练器信号。受训者的无线电控制发射机被配置为根据跳频方案发送频率切换的每个帧周期的训练器信号。

8. 发明申请

US20130076494A1 Controlling Communication Device, Controlled Body Communication Device And Controlling Communication System 审中-公开
标题翻译：控制通信设备，受控体通信设备和控制通信系统
公开(公告)号：US20130076494A1
公开(公告)日：2013-03-28
申请号：US13612141
申请日：2012-09-12
申请人： Takahiro Isono , Kota Toyotomi , Yasutaka Koike , Masahiro Tanaka
发明人： Takahiro Isono , Kota Toyotomi , Yasutaka Koike , Masahiro Tanaka
IPC分类号： G05B11/01
CPC分类号： A63H30/04 , G05B19/042
摘要： In a controlling communication device, parameter of a device mounted in an airframe is modified remotely from a transmitting side without a personal computer or a dedicated setting box. The communication device is operable to select an operation mode and a parameter mode, and includes a controlling communication device (a transmitter) having a display, a controlled body communication device (a receiver) connected to a device mounted in the airframe. In the parameter mode, the parameter signal is transmitted to the receiver by operation of the transmitter, and the parameter of the device is modified remotely by radio while seeing the display. The parameter signal by return from the receiver notifies results of the modification. Even if the device is made plurally in types or in number, it is unnecessary to detach the device from the controlled communication device, so as to readily modify the parameter.
摘要翻译：在控制通信设备中，安装在机身中的设备的参数在没有个人计算机或专用设置箱的情况下远离发送侧被修改。通信装置可操作以选择操作模式和参数模式，并且包括具有显示器的控制通信设备（发射机），连接到安装在机身中的设备的被控体通信设备（接收机）。在参数模式下，通过发射机的操作将参数信号发送给接收机，同时在看到显示器的同时通过无线电远程修改设备的参数。从接收器返回的参数信号通知修改的结果。即使该装置的数量多种多样，也不需要从受控通信装置中分离装置，从而容易地修改参数。

9. 发明申请

US20130038429A1 Wireless Communication System 审中-公开
标题翻译：无线通信系统
公开(公告)号：US20130038429A1
公开(公告)日：2013-02-14
申请号：US13564801
申请日：2012-08-02
申请人： Yasutaka Koike , Masahiro Tanaka
发明人： Yasutaka Koike , Masahiro Tanaka
IPC分类号： G08C19/16
CPC分类号： A63H30/04
摘要： A servo device 30 includes: a control portion 31 for driving and controlling a drive mechanism 32 by receiving a control signal from a transmitter 10, and by transforming the control signal into a drive signal corresponding to characteristic data previously stored in a memory portion 35. The control portion 31 includes: a signal processing portion 33 for discriminating whether the control signal is a maneuver signal or a characteristic data signal; and the memory portion for updating and storing the characteristic data based on the received characteristic data signal when the control signal is discriminated as the characteristic data signal.
摘要翻译：伺服装置30包括：控制部分31，用于通过接收来自发射器10的控制信号来驱动和控制驱动机构32，并且通过将控制信号变换成与先前存储在存储部分35中的特征数据相对应的驱动信号。控制部分31包括：信号处理部分33，用于鉴别控制信号是操纵信号还是特征数据信号; 以及存储器部分，用于当控制信号被鉴别为特征数据信号时，基于接收到的特征数据信号来更新和存储特征数据。

10. 发明授权

US08344613B2 Organic electroluminescence display device 有权
公开(公告)号：US08344613B2
公开(公告)日：2013-01-01
申请号：US12216788
申请日：2008-07-10
申请人： Masahiro Tanaka
发明人： Masahiro Tanaka
IPC分类号： H01J1/62
CPC分类号： H01L51/5088 , H01L51/5052
摘要： The invention provides an organic electroluminescence display device that makes it possible to obtain a highly reliable display. The organic electroluminescence display device has an organic electroluminescence element that includes a first layer (3) that contains a first substance that exhibits electron transport properties, and a second substance that exhibits electron-donating properties with respect to the first substance; a second layer (4) that is composed of a third substance that exhibits hole transport properties; a third layer (light-emitting layer (5) that contains a light-emitting substance; and a fourth layer (6) that is formed from a substance that exhibits electron transport properties.

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