会员体验
专利管家(专利管理)
工作空间(专利管理)
风险监控(情报监控)
数据分析(专利分析)
侵权分析(诉讼无效)
联系我们
交流群
官方交流:
QQ群: 891211   
微信请扫码    >>>
现在联系顾问~
热词
    • 7. 发明公开
    • ISOXAZOLINE DERIVATIVES AND HERBICIDES
    • ISOXAZOLINDERIVATE UND HERBIZIDE
    • EP1405853A1
    • 2004-04-07
    • EP02743670.8
    • 2002-06-20
    • KUMIAI CHEMICAL INDUSTRY CO., LTD.IHARA CHEMICAL INDUSTRY CO., LTD.
    • NAKATANI, Masao, K.I Chemical Res. Inst. Co. Ltd.ITO, Minoru, K.I Chemical Res. Inst. Co. Ltd.KIMIJIMA, KyokoMIYAZAKI, Masahiro, K.I Chem. Res. Inst. Co. Ltd.FUJINAMI, MakotoUENO, RyoheiTAKAHASHI, Satoru
    • C07D413/12A01N43/80
    • C07D413/12A01N43/80A01N43/82A01N43/90
    • The present invention aims at providing an isoxazoline derivative and a pharmaceutically acceptable salt thereof, both having an excellent herbicidal effect and an excellent selectivity between crop and weed.
      The isoxazoline derivative of the present invention is represented by the following general formula:
      wherein R 1 is a haloalkyl group; R 2 is a hydrogen atom, an alkyl group, or the like; R 3 , R 4 , R 5 and R 6 are each a hydrogen atom, or the like; Y is a pyrrolyl group, a pyrazolyl group, an isothiazolyl group, an oxazolyl group, an imidazolyl group, a pyridazinyl group, a pyrimidinyl group, a pyrazinyl group, a triazinyl group, a triazolyl group, an oxadiazolyl group, or the like; and n is an integer of 0 to 2.
    • 3-巯基 - 异恶唑啉衍生物(I)是新的。 式(I)的3-巯基 - 异恶唑啉衍生物及其盐是新的。 [图像] R 11-4C卤代烷基; R 2H,1-6C烷基,R 1,3-8C环烷基或3-8C环烷基1-3C烷基; R 3,R 4H,1-6C烷基或3-8C环烷基; 或R 3 + R 43-7C螺烷基; 或R 2 + R 35-8元环; R 5,R 6H或1-6C烷基; Y:吡咯基,吡唑基,异噻唑基,恶唑基,咪唑基,哒嗪基,嘧啶基,吡嗪基,三嗪基,三唑基,恶二唑基,苯并噻吩基,吲哚基,苯并恶唑基,苯并咪唑基,苯并异恶唑基,苯并异噻唑基,吲唑基,“哒嗪基”,喹喔啉基,喹唑啉基,噌啉基或苯并三唑基 任选地被1-6个Q取代并任选地与5-8元环稠合(任选被1-4个卤素取代); n:0-2; Q:OH,卤素,1-6C烷基(任选被Q 1单取代),R 1,3-8C环烷基,OA 1,OR 1,O-3-8C环烷基,3-8C环烷基1-3C烷氧基,SA 1,SR1,2-6C烯基,2-6C炔基,2-6C烯氧基,2-6C炔氧基,SO-1-6C烷基,SO2A 1,SOR1,SO2R 1,OSO2-1-6C烷基 ,OSO 2R1,1-6C酰基,COR1,COOH,COO-1-6C烷基,CN,CONH2(任选被1-6C烷基或Ph 1取代),1-6C酰氧基,OCOR 1,NO 2, 氨基(任选被1-6C烷基,Ph 1,1-6C酰基,COR 1,COCH 2 Ph,COPh,SO 2-1-6C烷基,SO 2 R 1,SO 2 CH 2 Ph或SO 2 Ph)或任选取代的Ph取代, OPh,SPh,Het,OHet,SHet,SOPh,SO 2 Ph,SOHet,SO 2 Het,OSO 2 Ph,COPh,COCH 2 Ph,COOPh或COOCH 2Ph; Q 1 OH,3-8C环烷基(任选被卤素或1-6C烷基取代),O-1-6C烷基,S-1-6C烷基,SO 2-1-6C烷基,COO-1-6C烷基, 6C卤代链烯基,氨基(任选被1-6C烷基,2-6C酰基,COR 1,SO 2 - C 1-6烷基或SO 2 R 1取代),CONH 2(任选被1-6C烷基或Ph取代),2- 6C酰基,COR 1,= N(O-1-6C烷基),CN,Ph 1或OPh 1; C 2 COO-1-6C烷基,CN,CONH 2,CONH-1-6C烷基,CON(1-6C烷基)2或任选取代的Ph或Het; 11-6C烷基(任选被Q 2单取代); Het:芳族杂环基; Ph 1取代Ph。活性:除草剂。 在试验中,3-(5-氯-1-甲基-3-三氟甲基-1H-吡唑-4-基甲基磺酰基)-5-氯甲基-5-甲基-2-异恶唑啉(Ia)(1000g / ha)得到大于 稗草和阴道阴茎90%的控制。 行动机制:无给予。