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1. 发明授权

EP0207563B1 A method for controlling weeds 失效
标题翻译：一种防治杂草的方法
公开(公告)号：EP0207563B1
公开(公告)日：1991-07-31
申请号：EP86201098.0
申请日：1986-06-24
申请人： JANSSEN PHARMACEUTICA N.V.
发明人： Lutz, William R. , van Lommen, Guy Rosalia Eugène , van Gestel, Jozef Frans Elisabetha
IPC分类号： A01N43/50 , C07D233/90 , C07D401/04 , C07D405/04 , C07D409/04
CPC分类号： C07D401/04 , A01N43/50 , C07D233/90 , C07D405/04 , C07D409/04

2. 发明公开

EP0277384A3 1H-imidazole-5-carboxylic acid derivatives 失效
标题翻译： 1H-咪唑-5-羧酸衍生物
公开(公告)号：EP0277384A3
公开(公告)日：1990-05-23
申请号：EP87202601.8
申请日：1987-12-22
申请人： JANSSEN PHARMACEUTICA N.V.
发明人： De Bruyn, Marcel F.L. , Van Lommen, Guy R.E. , Lutz, William R.
IPC分类号： C07D233/90 , A01N43/50 , C07D401/04 , C07D401/06 , C07D403/04 , C07D405/04 , C07D405/14 , C07D409/04 , C07D413/04 , C07D413/14 , A01N43/40
CPC分类号： C07D233/64 , A01N43/50 , A01N43/52 , A01N43/60 , A01N43/713 , A01N43/76 , A01N43/82 , A01N45/02 , A01N57/24 , C07D233/90 , C07D401/04 , C07D401/06 , C07D403/04 , C07D405/04 , C07D405/14 , C07D409/04 , C07D413/04 , C07D413/14 , C07F7/0812 , C07F9/65062
摘要： A method of controlling weeds by applying thereto or to the locus thereof of an imidazole derivative of formula
wherein
R 1 is hydrogen or mercapto; L is cyano or a radical of formula X is 1-indanyl, 1-tetrahydronaphthalenyl, 5-benzocycloheptanyl, 4-tetrahydrobenzothienyl, 4-tetrahydroben- zofuryl, 5-tetrahydroquinolyl, 5-tetrahydroisoquinolyl, 8-tetrahydroquinolyl, 8-tetrahydroisoquinolyl, 9,10-dihydro-9-antracenyl, 9H-fluoren-9-yl, 5-dibenzo[a,d]-cycloheptenyl, 5-dibenzo[a,d]cycloheptanyl or 1-dihydronaphthalenyl each unsubstituted or substituted; or X is a group
or a group -
; wherein n is 0, 1 or 2 or two; A is hydrogen, optionally substituted C 3 -C 7 cycloalkyl or pyridinyl, pyrimidinyl, naphthalenyl, f6ranyt and thienyl, each unsubstituted or substituted; Z is naphthalenyl, thienyl, furanyl, pyrimidinyl, phenyl or pyridinyl, each unsubstituted or substituted; a salt or stereoisomeric form thereof, novel compounds for use in said method; herbicidal compositions containing such compounds as active ingredient and methods of preparing said compounds.

3. 发明公开

EP0273531A1 1-Methyl-1h-imidazole-5-carboxylic acid derivatives 失效
标题翻译：衍生1-甲基-1H-咪唑-5-羧酸。
公开(公告)号：EP0273531A1
公开(公告)日：1988-07-06
申请号：EP87202612.5
申请日：1987-12-23
申请人： JANSSEN PHARMACEUTICA N.V. , CIBA-GEIGY AG
发明人： Lutz, William R. , Van Lommen, Guy R.E. , Sipido, Victor , Verschueren, Wim G.
IPC分类号： C07D233/90 , C07D233/64 , C07D233/66 , C07D403/04 , C07D413/04 , C07D417/04 , A01N43/50 , A01N43/707 , A01N43/713 , A01N43/76 , A01N43/78
CPC分类号： C07D233/90 , A01N43/50
摘要： Novel 1-methyl-1H-imidazole-5-carboxylic acid derivatives of formula

R 1 is hydrogen or mercapto;
R 2 is hydrogen, C 1 -C 7 alkyl, C 3 -C 7 alkenyl, C 3 -C 7 alkynyl, C 3 -C 7 cycloalkyl, C 5 -C 7 cycloalkenyl; said C 1 -C 7 alkyl, C 3 -C 7 alkenyl, C 3 -C 7 alkynyl, C 3 -C 7 cycloalkyl, C 5 -C 7 cycloalkenyl being optionally substituted;
R 3 is C 4 -C 13 alkyl, C 3 -C 7 cycloalkyl, or C 5 -C 7 cycloalkenyl each unsubstituted or substituted;
L is cyano, -COOR 4 ,

or a group -C( = G)-D-R 6 ;
a salt or stereoisomeric form thereof, which compounds are herbicidals; compositions containing such compounds as active ingredient and methods of preparing said compounds and compositions.
摘要翻译：式 R 1的新颖的1-甲基-1H-咪唑-5-羧酸衍生物是氢或巯基; R 2是氢，C 1 -C 7烷基，C 3 -C 7链烯基，C 3 -C 7炔基，C 3 -C 7环烷基，C 5 -C 7环烯基; 所述C 1 -C 7烷基，C 3 -C 7链烯基，C 3 -C 7炔基，C 3 -C 7环烷基，任选取代的C 5 -C 7环烯基; R 3是未取代或取代的C 4 -C 13烷基，C 3 -C 7环烷基或C 5 -C 7环烯基; L是氰基，-COOR 4，CHEM或基团-C（= G）-D-R 6; 其盐或立体异构形式，该化合物为除草剂; 含有这些化合物作为活性成分的组合物和制备所述化合物和组合物的方法。

4. 发明公开

EP0207563A3 A method for controlling weeds 失效
标题翻译：一种控制肥料的方法
公开(公告)号：EP0207563A3
公开(公告)日：1987-10-14
申请号：EP86201098
申请日：1986-06-24
申请人： JANSSEN PHARMACEUTICA N.V.
发明人： Lutz, William R. , van Lommen, Guy Rosalia Eugène , van Gestel, Jozef Frans Elisabetha
IPC分类号： A01N43/50 , C07D233/90 , C07D401/04 , C07D405/04 , C07D409/04
CPC分类号： C07D401/04 , A01N43/50 , C07D233/90 , C07D405/04 , C07D409/04
摘要： Method of controlling weeds by using a 5-imidazolecarboxylic acid of formula
wherein X is 1-indanyl, 1-tetrahydronaphthalenyl, 5-benzocycloheptanyl, 4-tetrahydrobenzothienyl, 4-tetrahydrobenzofuryl, 5-tetrahydroquinolyl, 5-tetrahydroisoquinolyl, 8-tetrahydroquinolyl, 8-tetrahydroisoquinolyl, 9,10-dihydro-9-antracenyl, 9H-fluoren-9-yl, 5-dibenzo[a,d]cycloheptenyl, 5-dibenzo[a,d]cycloheptanyl or 1-dihydronaphthalenyl each unsubstituted or substituted; and whereby the compounds with X other than unsubstituted 1-indanyl or 1-tetrahydronaphthalenyl are novel; compositions containing such agents as an active ingredient and methods of preparing said compositions and novel compounds.

5. 发明授权

EP0240050B1 A method for controlling weeds 失效
标题翻译：一种控制肥料的方法
公开(公告)号：EP0240050B1
公开(公告)日：1991-06-26
申请号：EP87200390.0
申请日：1987-03-04
申请人： JANSSEN PHARMACEUTICA N.V.
发明人： Van Gestel, Jozef Frans Elisabetha , Lutz, William R. , Van Lommen, Guy Rosalia Eugène , Fischer, Hanspeter , Schroven, Marc Francis Josephine , Thummel, Rudolph C.
IPC分类号： A01N43/50 , C07D233/90 , C07D401/06 , C07D403/06 , C07D405/06 , C07D409/06
CPC分类号： C07D401/06 , A01N43/50 , C07D233/90 , C07D403/06 , C07D405/06 , C07D409/06

6. 发明公开

EP0289066A1 1,5-Substituted 1H-imidazoles 失效
标题翻译： 1,5- Substituierte -1H-咪唑。
公开(公告)号：EP0289066A1
公开(公告)日：1988-11-02
申请号：EP88200586.1
申请日：1988-03-29
申请人： JANSSEN PHARMACEUTICA N.V. , CIBA-GEIGY AG
发明人： De Bruyn, Marcel Frans Leopold , Van Lommen, Guy Rosalia Eugène , Lutz, William R.
IPC分类号： C07D233/84 , C07D233/60 , C07D233/61 , C07D401/06 , C07D405/04 , C07D405/14 , C07D409/04 , C07D401/04 , A01N43/50 , A01N43/36 , A01N43/16
CPC分类号： C07D233/64 , A01N43/50 , C07D233/84 , C07D401/04 , C07D401/06 , C07D403/04 , C07D405/04 , C07D405/14 , C07D409/04
摘要： Novel 1,5-substituted 1H-imidazoles of formula
or a stereochemically isomeric form thereof, or a salt thereof, wherein R 1 is hydrogen or mercapto; L is
wherein X is 1-indanyl, 1-tetrahydronaphthalenyl, 5-benzocycloheptanyl, 4-tetrahydrobenzothienyl, 4-tetrahydrobenzofuryl, 5-tetrahydroquinolyl, 5-tetrahydroisoquinolyl, 8-tetrahydroquinolyl, 8-tetrahydroisoquinolyl, 9,10-dihydro-9-antracenyl, 9H-fluoren-9-yl, 5-dibenzo[a,d]cycloheptenyl, 5-dibenzo[a,d]cycloheptanyl or 1-dihydronaphthalenyl each unsubstituted or substituted, or X is a radical of formula
said compounds possessing herbicidal activity. Compositions containing said compounds as active ingredient. Processes for preparing said compouds and compositions. Methods of controlling weeds.
摘要翻译：新颖的式“CHEM”的1,5-取代的1H-咪唑或其立体化学异构形式或其盐，其中R 1是氢或巯基; 其中X是1-二氢化茚基，1-四氢萘基，5-苯并环庚烯基，4-四氢苯并噻吩基，4-四氢苯并呋喃基，5-四氢喹啉基，5-四氢异喹啉基-8-四氢喹啉基，8-四氢异喹啉基，9,10-二氢-9- 蒽基-9H-芴-9-基，5-二苯并[a，d]环庚烯基，5-二苯并[a，d]环庚基或每个未取代或取代的1-二氢萘基，或X是式CHEM的基团所述化合物具有除草活性。含有所述化合物作为活性成分的组合物。制备所述组合物和组合物的方法。控制杂草的方法

7. 发明公开

EP0277384A2 1H-imidazole-5-carboxylic acid derivatives 失效
标题翻译： 1H-咪唑-5-Kohlensäurederivate。
公开(公告)号：EP0277384A2
公开(公告)日：1988-08-10
申请号：EP87202601.8
申请日：1987-12-22
申请人： JANSSEN PHARMACEUTICA N.V.
发明人： De Bruyn, Marcel F.L. , Van Lommen, Guy R.E. , Lutz, William R.
IPC分类号： C07D233/90 , A01N43/50 , C07D401/04 , C07D401/06 , C07D403/04 , C07D405/04 , C07D405/14 , C07D409/04 , C07D413/04 , C07D413/14 , A01N43/40
CPC分类号： C07D233/64 , A01N43/50 , A01N43/52 , A01N43/60 , A01N43/713 , A01N43/76 , A01N43/82 , A01N45/02 , A01N57/24 , C07D233/90 , C07D401/04 , C07D401/06 , C07D403/04 , C07D405/04 , C07D405/14 , C07D409/04 , C07D413/04 , C07D413/14 , C07F7/0812 , C07F9/65062
摘要： A method of controlling weeds by applying thereto or to the locus thereof of an imidazole derivative of formula
wherein

R 1 is hydrogen or mercapto;
L is cyano or a radical of formula

X is 1-indanyl, 1-tetrahydronaphthalenyl, 5-benzocycloheptanyl, 4-tetrahydrobenzothienyl, 4-tetrahydroben- zofuryl, 5-tetrahydroquinolyl, 5-tetrahydroisoquinolyl, 8-tetrahydroquinolyl, 8-tetrahydroisoquinolyl, 9,10-dihydro-9-antracenyl, 9H-fluoren-9-yl, 5-dibenzo[a,d]-cycloheptenyl, 5-dibenzo[a,d]cycloheptanyl or 1-dihydronaphthalenyl each unsubstituted or substituted; or X is a group
or a group -
; wherein
n is 0, 1 or 2 or two; A is hydrogen, optionally substituted C 3 -C 7 cycloalkyl or pyridinyl, pyrimidinyl, naphthalenyl, f6ranyt and thienyl, each unsubstituted or substituted; Z is naphthalenyl, thienyl, furanyl, pyrimidinyl, phenyl or pyridinyl, each unsubstituted or substituted;
a salt or stereoisomeric form thereof, novel compounds for use in said method; herbicidal compositions containing such compounds as active ingredient and methods of preparing said compounds.
摘要翻译：通过向其施加式（CHEM）的咪唑衍生物或其基团的位置来控制杂草的方法，其中R 1是氢或巯基; L是氰基或式 X的基团是1-茚满基，1-四氢萘基，5-苯并环庚烯基，4-四氢苯并噻吩基，4-四氢苯并呋喃基，5-四氢喹啉基，5-四氢异喹啉基，8-四氢喹啉基，8-四氢异喹啉基，，10-二苯并[a，d] - 环庚烯基，5-二苯并[a，d]环庚烷基或1-二氢萘基，各自未取代或取代; 或X为基团或基团-H-Z; 其中n为0,1或2或2; A是氢，任选取代的C 3 -C 7环烷基或吡啶基，嘧啶基，萘基，呋喃基和噻吩基，各自未取代或取代; Z是萘基，噻吩基，呋喃基，嘧啶基，苯基或吡啶基，各自未取代或取代; 其盐或立体异构形式，用于所述方法的新化合物; 含有这些化合物作为活性成分的除草组合物和制备所述化合物的方法。

8. 发明公开

EP0240050A1 A method for controlling weeds 失效
标题翻译： Verfahren zur Beherrschung von Unkraut。
公开(公告)号：EP0240050A1
公开(公告)日：1987-10-07
申请号：EP87200390.0
申请日：1987-03-04
申请人： JANSSEN PHARMACEUTICA N.V.
发明人： Van Gestel, Jozef Frans Elisabetha , Lutz, William R. , Van Lommen, Guy Rosalia Eugène , Fischer, Hanspeter , Schroven, Marc Francis Josephine , Thummel, Rudolph C.
IPC分类号： A01N43/50 , C07D233/90 , C07D401/06 , C07D403/06 , C07D405/06 , C07D409/06
CPC分类号： C07D401/06 , A01N43/50 , C07D233/90 , C07D403/06 , C07D405/06 , C07D409/06
摘要： Method of controlling weeds by using a 5-imidazolecarboxylic acid of formula
or a stereochemically isomeric form thereof, or a salt thereof, or a quatemised form thereof, or a N-oxide thereof, wherein

A is hydrogen; C 3 -C 7 cycloalkyl optionally substituted with one or two C 1 -C 5 alkyl radicals; C 1 -C 7 alkyl optionally substituted with C 1 -C 7 alkyloxy or with an Ar radical; or C 1 -C 7 alkyl substituted with both a a C 1 -C 7 alkyloxy and an Ar radical; or a radical selected from pyridinyl, pyrimidinyl, naphthalenyl, furanyl and thienyl, each unsubstituted or substituted; said radical Ar being unsubstituted or substituted phenyl, pyridinyl, pyrimidinyl, naphthalenyl, furanyl or thienyl;
Z is naphthalenyl, thienyl, furanyl, pyrimidinyl, phenyl or pyridinyl, each unsubstituted or substituted; novel compounds of formula (I); compositions containing such agents as an active ingredient and methods of preparing said compositions and novel compounds.
摘要翻译：通过使用式CHEM的5-咪唑甲酸或其立体化学异构形式或其盐或其季铵化形式或其N-氧化物控制杂草的方法，其中A为氢; 任选被一个或两个C 1 -C 5烷基取代的C 3 -C 7环烷基; 任选被C 1 -C 7烷氧基或Ar基团取代的C 1 -C 7烷基; 或被C 1 -C 7烷氧基和Ar基团二取代的C 1 -C 7烷基; 或选自吡啶基，嘧啶基，萘基，呋喃基和噻吩基的基团，各自未取代或取代; 所述基团Ar为未取代或取代的苯基，吡啶基，嘧啶基，萘基，呋喃基或噻吩基; Z是萘基，噻吩基，呋喃基，嘧啶基，苯基或吡啶基，各自未取代或取代; 式（I）的新化合物; 含有作为活性成分的试剂的组合物和制备所述组合物和新化合物的方法。

9. 发明授权

EP0234656B1 1H-imidazole-5-carboxylic acid derivatives 失效
标题翻译： 1H-咪唑-5-羧酸衍生物
公开(公告)号：EP0234656B1
公开(公告)日：1992-04-22
申请号：EP87200265.4
申请日：1987-02-19
申请人： JANSSEN PHARMACEUTICA N.V.
发明人： Van Lommen, Guy Rosalia Eugène , Lutz, William R. , Van Gestel, Jozef Franz Elisabetha
IPC分类号： C07D405/04 , C07D409/04 , C07D401/04 , C07D403/04 , A01N43/50
CPC分类号： C07D401/04 , A01N43/50 , C07D403/04 , C07D405/04 , C07D409/04

10. 发明公开

EP0234656A2 1H-imidazole-5-carboxylic acid derivatives 失效
标题翻译： 1H-咪唑-5-carbonsäurederivate。
公开(公告)号：EP0234656A2
公开(公告)日：1987-09-02
申请号：EP87200265.4
申请日：1987-02-19
申请人： JANSSEN PHARMACEUTICA N.V.
发明人： Van Lommen, Guy Rosalia Eugène , Lutz, William R. , Van Gestel, Jozef Franz Elisabetha
IPC分类号： C07D405/04 , C07D409/04 , C07D401/04 , C07D403/04 , A01N43/50
CPC分类号： C07D401/04 , A01N43/50 , C07D403/04 , C07D405/04 , C07D409/04
摘要： Novel 1H-imidazole-5-carboxylic acid derivatives of formula
wherein Y is a group -CH 2 -S(O) m , -CH 2 -O-, -CH 2 -N(E)-, or -CH=N-, wherein the heteroatom is linked to the carbon atom of the benzene ring and wherein m is zero, one or two;

E is hydrogen, C 1 -C 5 alkyl, C 1 -C 5 alkanoyl, or 4-methylphenylsulfonyl;
the salts, stereochemically isomeric forms, N-oxides and quaternised forms thereof, which compounds are herbicidal agents; compositions containing such compounds as an active ingredient; processes for preparing said compounds and pharmaceutical compositions; and methods for controlling weeds.
摘要翻译： 1-苯并杂环基-1H-咪唑-3-羧酸衍生物。的式（I）化合物及其盐和季铵盐。 derivs。和它们的N-氧化物是新的。式中R1 = H或SH; R2 = H，1-7C烷基，3-7C烯基，3-7C炔基，3-7C环烷基，（1-7C）烷氧基 - （1-7C）烷基或芳基 - （1-5C）烷基; n = 0,1或2; Y = S（O）m-CH 2，O-CH 2，N（E）-CH 2或N = CH，杂原子与苯环的C原子连接; m = 0,1或2; E = H，1-5C烷基，1-5C烷酰基或对甲基C 6 H 4 SO 2; R 3 -R 6 = H，1-6C烷基，单 - 或二 - 芳基 - （1-5C）烷基，1-6C烷氧基，卤素，3-7C烯基1-5C烷基或1-5C烷氧基。含1-3个卤素或芳基; 或R3 + R4 =稠合苯环选择的残基。 substd。 1或2 H，1-5C烷基，1-5C烷氧基，卤素，1-5C烷基或1-5C烷氧基。 1-3个卤素，NO2，NH2或NH-CPG; 或者当R3 + R4被取代时，它们形成3-7C螺环C环; R7，R8 = H，1-5C烷基，1-5C烷氧基，卤素，1-5C烷基或1-5C烷氧基。通过1-3个卤素，CN，NO 2 NH 2，单 - 或二 - （1-5C）烷基氨基或NH-COG; G = 1-6C烷基; 芳基= Ph opt substd。 1-3个卤素，1-5C烷基或1-5C烷氧基。 R3-R6可以存在于双环的Y-contg.part的任何C原子上，包括CH 2或CH gps。的（CH 2）n，S-CH 2，O-CH 2，N（E）-CH 2或N = CH。

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