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1. 发明授权

US3542779A New 4-quinazolone derivatives and process for the preparation thereof 失效
标题翻译：新的四氮杂萘酮衍生物及其制备方法
公开(公告)号：US3542779A
公开(公告)日：1970-11-24
申请号：US3542779D
申请日：1968-02-23
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , KOSA ILDIKO
IPC分类号： C07D239/92 , C07D51/48
CPC分类号： C07D239/92

2. 发明授权

US3920651A Quaternary ammonium compounds 失效
标题翻译：季铵化合物
公开(公告)号：US3920651A
公开(公告)日：1975-11-18
申请号：US30023372
申请日：1972-10-24
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , HERMANN NEE VOROS JUDIT , VOROS NEE , TOROK ZOLTAN , DVORCSAK PETER
IPC分类号： C07D239/26 , C07D239/30 , C07D239/42
CPC分类号： C07D239/30 , C07D239/42
摘要： A quaternary ammonium compound of the formula: WHEREIN R10 is propyl, R2 is hydrogen, halogen, hydroxy, alkoxy or amino, R3, R4 and R5 are each aryl, aralkyl, heteroaralkyl or alkyl and Y is an acid or hydroxyl anion. The compound has superior coccidiostatic properties.
摘要翻译：下式的季铵化合物：

3. 发明授权

US3485874A Ortho and para bromophenyl isopropyl methylamines 失效
标题翻译： ORTHO和PARA BROMOPHENYL异丙基甲基胺
公开(公告)号：US3485874A
公开(公告)日：1969-12-23
申请号：US3485874D
申请日：1966-05-04
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , KNOLL JOZSEF , KOSA ILDIKO , SANDOR ILDIKO , SOMFAI EVA , TOROK SANDOR
IPC分类号： A61K31/135 , C07C87/28 , A61K27/00
CPC分类号： A61K31/135

4. 发明授权

US3663610A Amidine derivatives with spasmolytic,psychostimulant and anorexigenic properties 失效
标题翻译：具有弹性，精神分裂和异构性质的氨基衍生物
公开(公告)号：US3663610A
公开(公告)日：1972-05-16
申请号：US3663610D
申请日：1968-07-08
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , KOSA ILDIKO , KNOLL JOZSEF
IPC分类号： A61K31/155 , A61P3/04 , A61P25/26 , C07C67/00 , C07C239/00 , C07C257/10 , C07D213/16 , C07D213/81 , C07D265/22 , C07C101/54
CPC分类号： C07D265/22 , A61K31/155 , C07D213/16 , C07D213/81
摘要： PSYCHOSTIMULANT, ANOREXIGENIC AND SPASMOLYTIC COMPOUNDS OF THE GENERAL FORMULA

1-(R2-N(-R3)-C(-R1)=N-),2-(HOOC-),R4,R5-BENZENE

WHEREIN

R1 IS A MEMBER SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ALKYL, SUBSTITUTED ALKYL, ARYL, SUBSTITUTED ARYL AND HETEROCYCLIC RADICAL, R2 IS A MEMBER SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ALKYL, SUBSTITUTED ALKYL, ARYL, SUBSTITUTED ARYL AND HETEROCYCLIC RADICAL, R3 IS A MEMBER SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ALKYL, SUBSTITUTED ALKYL, ARYL, SUBSTITUTED ARYL AND HETEROCYCLIC RADICAL, R4 IS A MEMBER SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, HALOGEN, NITRO, AMINO, ACYLAMINO, HYDROXY AND ALKOXY, R5 IS A MEMBER SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, HALOGEN, NITRO, AMINO, ACYLAMINO, HYDROXY AND ALKOXY.

5. 发明授权

US3496195A D-o-bromo-phenyl-isopropyl-methylpropinylamine and its salts 失效
标题翻译： D-O-溴 - 苯基 - 异丙基 - 甲基丙烯酰胺及其盐
公开(公告)号：US3496195A
公开(公告)日：1970-02-17
申请号：US3496195D
申请日：1966-05-11
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , KOSA ILDIKO , KNOLL JOZSEF , SOMFAI EVA
IPC分类号： C07C87/28 , C07C91/00
CPC分类号： C07D307/33

6. 发明专利

FI78457C FOERFARANDE FOER FRAMSTAELLNING AV PROPARGYLAMMONIUMKLORIDER. 未知
公开(公告)号：FI78457C
公开(公告)日：1989-08-10
申请号：FI832538
申请日：1983-07-12
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , SOMFAI EVA , HERMANN NEE VOEROES JUDIT , NAGY LAJOS , SZABO GABOR , ORBAN OTTO , ARVAI LASZLO
IPC分类号： C07C67/00 , C07C209/00 , C07C209/08 , C07C211/63 , C07C87/30 , C07C85/145

7. 发明专利

FI78457B 未知
公开(公告)号：FI78457B
公开(公告)日：1989-04-28
申请号：FI832538
申请日：1983-07-12
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , SOMFAI EVA , HERMANN NEE VOEROES JUDIT , NAGY LAJOS , SZABO GABOR , ORBAN OTTO , ARVAI LASZLO
IPC分类号： C07C67/00 , C07C209/00 , C07C209/08 , C07C211/63 , C07C87/30 , C07C85/145

8. 发明专利

AT38621T 未知
公开(公告)号：AT38621T
公开(公告)日：1988-12-15
申请号：AT84308751
申请日：1984-12-14
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： KNOLL JOZSEF , BIRKMAYER WALTER , KALLOY KATALIN , MARTON JENO , ECSERY ZOLTAN
IPC分类号： A61K31/195 , C07C211/48

9. 发明专利

CA1215394A PROCESS FOR THE PREPARATION OF PROPARGYL-AMINES 未知
公开(公告)号：CA1215394A
公开(公告)日：1986-12-16
申请号：CA432358
申请日：1983-07-13
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , SOMFAI EVA , HERMANN JUDIT NEE VOROS , NAGY LAJOS , SZABO GABOR , ORBAN OTTO , ARVAI LASZLO
IPC分类号： C07C67/00 , C07C209/00 , C07C209/08 , C07C211/63 , C07C85/04 , C07C87/28
摘要： NEW PROCESS FOR THE PREPARATION OF PROPARGYL AMINES The invention relates to a new process for the preparation of propargyl ammonium chlorides of the general Formula I /I/ by alkaline decomposition of the d-tartarate of the 1-isomer of an amine of the general Formula II /II/ and subsequent reaction of the amine of the general Formula II with a halide of the general Formula III X - CH2 - C ? CH /III/ in the presence of an organic solvent, alkali and water /in which general Formulae n is 1 or 0 and X stands for halogen/ which comprises reacting the d-tartarate of the 1-isomer of an amine of the general Formula II in aqueous suspension with an alkali, dissolving the base of the general Formula II, thus set free without isolation in a water non-miscible organic solvent and reacting the same in the said phase with a halide of the general Formula III, and thereafter - preferably after separating the aqueous layer - reacting the mixture which contains the amines of the general Formulae II and IV /IV/ in the organic phase in the presence of water with an organic acid or a solution which has a pH value of 1.5-6 and consists of an inorganic acid and water, thus dissolving in the two-phase mixture formed the salt of the amine of the general Formula II in the aqueous layer and selectively separating the amine of the general Formula II from the amine of the general Formula IV, and thereafter adding after the separation of the phases hydrogen chloride to the amine of the general Formula IV being in the organic phase and thus precipitating the salt of the general Formula I. The compounds of the general Formula I are known pharmaceutical active ingredients. The advantage of the process of the present invention that it is highly economical and enables the recovery of the starting materials on large scale production too.

10. 发明专利

DK45786D0 未知
公开(公告)号：DK45786D0
公开(公告)日：1986-01-30
申请号：DK45786
申请日：1986-01-30
申请人： CHINOIN GYOGYSZER ES VEGYESZET
发明人： ECSERY ZOLTAN , KNOLL JOZSEF , SOMFAI EVA , TOEROEK ZOLTAN , SZINNYEI EVA , MOZSOLICS KAROLY
IPC分类号： A61K31/135 , A01N33/04 , A61K20060101 , A61K31/13 , A61K31/137 , A61K31/37 , A61P13/02 , A61P15/00 , A61P25/00 , A61P25/02 , A61P25/24 , A61P25/26 , A61P25/28 , A61P43/00 , C07C20060101 , C07C67/00 , C07C209/00 , C07C209/04 , C07C209/08 , C07C209/16 , C07C209/22 , C07C209/24 , C07C209/28 , C07C209/52 , C07C209/60 , C07C209/68 , C07C209/74 , C07C209/84 , C07C209/88 , C07C211/00 , C07C211/03 , C07C211/27 , C07C211/29 , C07C211/48 , C07F13/00 , C07C
摘要： The invention relates to the new N-[2-/4-fluorophenyl/-1-methyl]-ethyl-N-methyl-N-propynyl amine of the Formula I (I) and isomers and salts thereof. The compound of the formula I is useful as a selective MAO inhibitor.

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