会员体验
专利管家(专利管理)
工作空间(专利管理)
风险监控(情报监控)
数据分析(专利分析)
侵权分析(诉讼无效)
联系我们
交流群
官方交流:
QQ群: 891211   
微信请扫码    >>>
现在联系顾问~
热词
    • 6. 发明申请
    • RESORCINE DERIVATIVES AND THEIR USE AS PESTICIDES
    • RESORCINE衍生物及其作为杀虫剂的用途
    • WO2007054558A2
    • 2007-05-18
    • PCT/EP2006068329
    • 2006-11-10
    • BASF AGPUHL MICHAELKORDES MARKUSPOHLMAN MATTHIASGOETZ NORBERTRACK MICHAELLANGEWALD JUERGENSCHNEIDER FELIXANSPAUGH DOUGLAS DCULBERTSON DEBORAH LOLOUMI-SADEGHI HASSANKUHN DAVID G
    • PUHL MICHAELKORDES MARKUSPOHLMAN MATTHIASGOETZ NORBERTRACK MICHAELLANGEWALD JUERGENSCHNEIDER FELIXANSPAUGH DOUGLAS DCULBERTSON DEBORAH LOLOUMI-SADEGHI HASSANKUHN DAVID G
    • C07D213/64C07D277/34C07D307/80
    • This invention relates to resorcine derivatives of formula (I) wherein R 1 is phenyl or a 5- to 6-membered heteroaromatic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the heteroaromatic ring may be fused to a ring selected from phenyl and a 5- to 6-membered saturated, partially unsaturated or aromatic heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the 5- to 6-membered heteroaromatic ring or the respective fused ring systems may be unsubstituted or substituted by any combination of 1 to 6 optionally substituted groups R 3 , wherein R 3 is halogen, cyano, nitro, hydroxy, mercapto, amino, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, halocycloalkyl, halocycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, haloalkenyloxy, haloalkynyloxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, haloalkenylthio, haloalkynylthio, alkylamino, alkenylamino, alkynylamino, dialkylamino, dialkenylamino, dialkynylamino, alkyl-alkenylamino, alkyl-alkynylamino, alkenyl- alkynylamino, trialkylsilyl, or phenyl or a 5-to 7-membered saturated or partially unsaturated heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen or a 5- to 6-membered heteraromatic ring system which may contain 1 to 4 heteroatoms selected from oxygen, nitrogen and sulfur, which phenyl and which heteroaromatic ring may be bonded via an oxygen or a sulfur atom, or -C(=G)Ra, -C(=G)ORa, -C(=G)NRa2, -C(=G)[N=SRa2], -C(=NORa)Ra, -C(=NORa)NRa2, -C(=NNRa2)Ra , -OC(=G)-OC(=G)ORa, N=SRa2, -NRaC(=G)Ra, -N[C(=G)Ra]2, - NRaC(=G)ORa, -C(=G)NRa-NRa2, -C(=G)NRa-NRa [C(=G)Ra], -NRa-C(=G)NRa2, -NRa-NRaC(=G)Ra, -NRa-N[C(=G)Ra]2, -N[(C=G)Ra]-NRa2, -NRa-NRa[(C=G)GRa], -NRa[(C=G)NRa2, -NRa[C=NRa]Ra, -NRa(C=NRa)NRa2, -O-NRa2, -O-NRa(C=G)Ra, - SO2NRa2, -NRaSO2Ra, -S(=O)Ra, -S(=O)2Ra, -SO2ORa, or -OSO2Ra, wherein G is oxygen or sulfur and Ra is as defined in the description, R 2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, alkoxy, or haloalkoxy, x is 2, 3, 4, 5, 6, or 7, or the diastereomers, enantiomers, salts or N-oxides thereof, with the proviso that R 1 is not 5-chloro-2,2,-dimethyl-2,3-dihydrobenzo[b]furan-7-yl when R 2 is hydrogen and x is 3 or 4, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.
    • 本发明涉及其中R 1为苯基或可含有1-3个选自氧,氮和硫的杂原子的5至6元杂芳环的式(I)的间苯二酚衍生物,其中苯基 或杂芳环可以与选自苯基和5-至6-元饱和,部分不饱和或芳族杂环的环稠合,所述杂环可以含有1-3个选自氧,氮和硫的杂原子,其中苯基或5- 至6元杂芳环或相应的稠环体系可以是未取代的或被1至6个任选取代的基团R 3 3的任何组合取代,其中R 3是卤素, 氰基,硝基,羟基,巯基,氨基,烷基,烯基,炔基,环烷基,环烯基,卤代烷基,卤代烯基,卤代炔基,卤代环烷基,卤代环烯基,烷氧基,烯氧基,炔氧基,卤代烷氧基,卤代烯氧基,卤代炔氧基,烷硫基,烯硫基,炔硫基,卤代烷硫基, H 烯基氨基,炔基氨基,二烷基氨基,二链烷基氨基,二炔基氨基,烷基 - 链烯基氨基,烷基 - 炔基氨基,烯基 - 炔基氨基,三烷基甲硅烷基或苯基或5至7元饱和或部分不饱和的杂环, 至3个选自氧,硫和氮的杂原子或5至6元杂芳环体系,其可以含有1至4个选自氧,氮和硫的杂原子,该苯基和杂芳环可以通过氧或 硫原子或-C(= G)R a,-C(= G)OR a,-C(= G)NR a 2,-C(= G)[N = SR a 2] (= NORa)NRa2,-C(= NNRa2)Ra,-OC(= G)-OC(= G)ORa,N = SRa2,-NRaC(= G)Ra,-N [C(= G)Ra] 2,-NR a C(= G)OR a,-C(= G)NR a -NR a 2,-C(= G)NR a -NR a [C(= G)R a] -NRaC(= G)Ra,-NRa-N [C(= G)Ra] 2,-N [(C = G)Ra] -NRa2,-NRa-NRa [(C = G) [(C = G)NRa2,-NRa [C = NRa] Ra,-NRa(C = NRa)NRa2,-O-NRa2,-O-NRa(C = G)Ra,-SO2NRa2,-NRaSO2Ra,-S (= O)R a,-S(= O)2 R a,-SO 2 OR a或-O SO 2 R a,其中G是氧或硫,Ra如说明书中所定义,R 2是氢,卤素,氰基,烷基,卤代烷基,烯基,卤代烯基,炔基,卤代炔基,烷氧基或卤代烷氧基, x是2,3,4,5,6或7,或其非对映异构体,对映异构体,盐或N-氧化物,条件是R 1不是5-氯-2,2 ,当R 2是氢并且x是3或4时,制备化合物I的方法和中间体,使用化合物I,其中R 1,R 2,R 3, 用于防治昆虫,螨虫或线虫,以及用化合物I治疗,控制,预防或保护动物免受寄生虫侵袭或感染的方法。
    • 8. 发明申请
    • PESTICIDAL MIXTURES
    • 农药混合物
    • WO2007122163A3
    • 2008-02-07
    • PCT/EP2007053791
    • 2007-04-18
    • BASF AGLANGEWALD JUERGENVAN TUYL COTTER HENRYCULBERTSON DEBORAH LOLOUMI-SADEGHI HASSAN
    • LANGEWALD JUERGENVAN TUYL COTTER HENRYCULBERTSON DEBORAH LOLOUMI-SADEGHI HASSAN
    • A01N37/34A01N43/56A01N43/88A01N43/90A01N47/02A01N47/06A01N47/22A01N47/30A01N47/34A01N47/38A01N47/40A01N51/00A01N53/00A01N57/12A01N57/14
    • A01N37/34A01N47/02A01N43/22A01N43/88A01N51/00A01N63/00A01N47/30A01N2300/00
    • Pesticidal mixtures comprising, as active components, 1) a malonodinitrile compound selected from compounds I-1 to I-8 CF 2 HCF 2 CF 2 CF 2 CH 2 C(CN) 2 CH 2 CH 2 CF 3 (compound I-1; name: 2-(2,2,3,3,4,4,5,5- octafluoro-pentyl)-2-(3,3,3-trifluoro-propyl)-malononitrile); CF 3 (CH 2 ) 2 C(CN) 2 CH 2 (CF 2 ) 5 CF 2 H (compound I-2; name: 2-(2,2,3,3,4,4,5,5,6,6,7,7- dodecafluoro-heptyl)-2-(3,3,3-trifluoro-propyl)-malononitrile); CF 3 (CH 2 ) 2 C(CN) 2 (CH 2 ) 2 C(CF 3 ) 2 F (compound I-3; name: 2-(3,4,4,4-tetrafluoro-3- trifluoromethyl-butyl)-2-(3,3,3-trifluoro-propyl)-malononitrile); CF 3 (CH 2 ) 2 C(CN) 2 (CH 2 ) 2 (CF 2 ) 3 CF 3 (compound I-4; name: 2-(3,3,4,4,5,5,6,6,6- nonafluoro-hexyl)-2-(3,3,3-trifluoro-propyl)-malononitrile); CF 2 H(CF 2 ) 3 CH 2 C(CN) 2 CH 2 (CF 2 ) 3 CF 2 H (compound I-5; name: 2,2-bis-(2,2,3,3,4,4,5,5- octafluoro-pentyl)-malononitrile); CF 3 (CH 2 ) 2 C(CN) 2 CH 2 (CF 2 ) 3 CF 3 (compound I-6; name: 2-(2,2,3,3,4,4,5,5,5-nonafluoro- pentyl)-2-(3,3,3-trifluoro-propyl)-malononitrile); CF 3 (CF 2 ) 2 CH 2 C(CN) 2 CH 2 (CF 2 ) 3 CF 2 H (compound I-7; name: 2-(2,2,3,3,4,4,4- heptafluoro-butyl)-2-(2,2,3,3,4,4,5,5-octafluoro-pentyl)-malononitrile); or CF 3 CF 2 CH 2 C(CN) 2 CH 2 (CF 2 ) 3 CF 2 H (compound I-8; name: 2-(2,2,3,3,4,4,5,5-octafluoro- pentyl)-2-(2,2,3,3,3-pentafluoro-propyl)-malononitrile); and 2) one or more compounds II selected from group A consisting of organo(thio)- phosphates, carbamates, pyrethroids, growth regulators, nicotinic receptor agonists/antagonists compounds, GABA antagonist compounds, macrocyclic lactone insecticides, METI I acaricides, METI II and III compounds, uncoupler compounds, oxida- tive phosphorylation inhibitor compounds, mixed function oxidase inhibitor compounds, sodium channel blocker compounds and others, all as defined in the description, in synergistically effective amounts, use of these mixture for combating insects, arachnids or nematodes in and on plants and for the protection of seeds, and for treating, controlling, preventing or protecting a warm-blooded animal or a fish against infestation or infection by parasites.
    • 作为活性组分的包含1)选自化合物I-1至I-8的丙二腈化合物的杀虫混合物CF 2 CO 2 C 2 CF 2 CF 2 CH 2 C(CN) 2 CH 2 CH 2 CF < (化合物I-1;名称:2-(2,2,3,3,4,4,5,5-八氟 - 戊基)-2-(3,3,3-三氟 - 丙基) - 丙二腈); CF 3 (CH 2 2 C(CN) 2 CH 2 ( CF 2 H 2(化合物I-2;名称:2-(2,2,3,3,4,4 ,5,5,6,6,7,7-十二氟 - 庚基)-2-(3,3,3-三氟 - 丙基) - 丙二腈); CF 3 (CH 2 2 C(CN) 2 (CH 2 )(C 3 CF 3)2 F(化合物I-3;名称:2-(3,4,4,4-四氟 -3-三氟甲基 - 丁基)-2-(3,3,3-三氟 - 丙基) - 丙二腈); CF 3 (CH 2 2 C(CN) 2 (CH 2 (CF 2)3(化合物I-4);名称:2-(3, 3,4,4,5,5,6,6,6-九氟己基)-2-(3,3,3-三氟丙基) - 丙二腈); CF 2 H(CF 2 3 CH 2 C(CN) 2 CH 2(CF 2)2 CH 2(化合物I-5;名称:2,2-二甲基-2- (2,2,3,3,4,4,5,5-八氟 - 戊基) - 丙二腈); CF 3 (CH 2 2 C(CN) 2 CH 2 ( (化合物I-6;名称:2-(2,2,3,3,4,4,..., 5,5 - 九氟 - 戊基)-2-(3,3,3-三氟 - 丙基) - 丙二腈); CF 3 (CF 2 2 CH 2 C(CN) 2 CH (化合物I-7;名称:2-(2,2,2-三氟乙基) 2,3,3,4,4,4-七氟丁基)-2-(2,2,3,3,4,4,5,5-八氟 - 戊基) - 丙二腈); 或CF 3 CH 2 CH 2 C(CN)2 CH 2((C 1 -C 2) CF 2 H 2(化合物I-8;名称:2-(2,2,3,3,4,...) ,5,5-八氟 - 戊基)-2-(2,2,3,3,3-五氟 - 丙基) - 丙二腈); 和2)选自有机(硫代) - 磷酸酯,氨基甲酸酯,拟除虫菊酯,生长调节剂,烟碱受体激动剂/拮抗剂化合物,GABA拮抗剂化合物,大环内酯杀虫剂,METI I杀螨剂,METI II和 III化合物,非偶联剂化合物,氧化磷酸化抑制剂化合物,混合功能氧化酶抑制剂化合物,钠通道阻断剂化合物和其他,如描述中所定义的,协同有效量的这些混合物用于防治昆虫,蜘蛛或线虫 植物和保护种子,以及治疗,控制,预防或保护温血动物或鱼类免受寄生虫感染或感染。