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1. 发明申请

WO2008092851A3 PESTICIDAL COMPOSITIONS COMPRISING 3 -ACETYL-I- PHENYLPYRAZOLE COMPOUNDS 审中-公开
公开(公告)号：WO2008092851A3
公开(公告)日：2008-08-07
申请号：PCT/EP2008/051026
申请日：2008-01-29
申请人： BASF SE , KORADIN, Christopher , LANGEWALD, Jürgen , ANSPAUGH, Douglas D. , COTTER, Henry Van Tuyl
发明人： KORADIN, Christopher , LANGEWALD, Jürgen , ANSPAUGH, Douglas D. , COTTER, Henry Van Tuyl
IPC分类号： A01N43/56 , A01N47/02 , A01P7/04
摘要： The present invention relates to pesticidal compositionscomprising as active componentsat least one 3-acetyl-1-phenylpyrazole compound of the formula (I) or a salt thereof: wherein X is N or C-R 5 ; R 1 is C 1 -C 4 -alkyl or C 1 -C 4 -haloalkyl; R 2 is NR 6 R 7 or S(O) n R 8 ; R 3 is halogen, C 1 -C 4 -haloalkyl, C 1 -C 4 -haloalkoxy, SF 5 or S(O) p R 9 ; R 4 is hydrogen or halogen; R 5 is halogen; R 6 is hydrogen, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl,C(O)R 10 , S(O) q CF 3 ; R 7 is hydrogen or C 1 -C 4 -alkyl, or R 6 and R 7 are joined so as together form a C 4 - C 6 -alkylene moiety, wherein one CH 2 -group may be replaced by oxygen or a radical N-R 11 ; R 8 , R 9 , R 10 , R 11 are each independently hydrogen, C 1 -C 4 -alkylorC 1 -C 4 -haloalkyl; m, n, p and q are each independently 0, 1 or 2; and at least one further pesticidally active compound II, selected from A.1GABA-gated chloride channel antagonists; A.2Nicotinic acetylcholine receptor agonists/antagonists A.3Juvenile hormone mimics; A.4Compounds affecting the oxidative phosphorylation; A.5Inhibitors of the chitin biosynthesis; A.6Moulting disruptors; A.7Mitochondrial electron transport inhibitors;. A.8Voltage-dependent sodium channel blockers; A.9Inhibitors of the lipid synthesis; and A.10group of various compounds.

2. 发明申请

WO2008092851A2 PESTICIDALLY ACTIVE COMPOSITIONS COMPRISING 3-ACETYL-1-PHENYLPYRAZOLE COMPOUNDS 审中-公开
标题翻译：包含3-乙酰基-1-苯基甲基吡唑化合物的农药活性组合物
公开(公告)号：WO2008092851A2
公开(公告)日：2008-08-07
申请号：PCT/EP2008051026
申请日：2008-01-29
申请人： BASF SE , KORADIN CHRISTOPHER , LANGEWALD JUERGEN , ANSPAUGH DOUGLAS D , COTTER HENRY VAN TUYL
发明人： KORADIN CHRISTOPHER , LANGEWALD JUERGEN , ANSPAUGH DOUGLAS D , COTTER HENRY VAN TUYL
CPC分类号： A01N43/56 , A01N47/02 , A01N43/58 , A01N43/80 , A01N51/00 , A01N2300/00
摘要： The present invention relates to pesticidal compositionscomprising as active componentsat least one 3-acetyl-1-phenylpyrazole compound of the formula (I) or a salt thereof: wherein X is N or C-R 5 ; R 1 is C 1 -C 4 -alkyl or C 1 -C 4 -haloalkyl; R 2 is NR 6 R 7 or S(O) n R 8 ; R 3 is halogen, C 1 -C 4 -haloalkyl, C 1 -C 4 -haloalkoxy, SF 5 or S(O) p R 9 ; R 4 is hydrogen or halogen; R 5 is halogen; R 6 is hydrogen, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl,C(O)R 10 , S(O) q CF 3 ; R 7 is hydrogen or C 1 -C 4 -alkyl, or R 6 and R 7 are joined so as together form a C 4 - C 6 -alkylene moiety, wherein one CH 2 -group may be replaced by oxygen or a radical N-R 11 ; R 8 , R 9 , R 10 , R 11 are each independently hydrogen, C 1 -C 4 -alkylorC 1 -C 4 -haloalkyl; m, n, p and q are each independently 0, 1 or 2; and at least one further pesticidally active compound II, selected from A.1GABA-gated chloride channel antagonists; A.2Nicotinic acetylcholine receptor agonists/antagonists A.3Juvenile hormone mimics; A.4Compounds affecting the oxidative phosphorylation; A.5Inhibitors of the chitin biosynthesis; A.6Moulting disruptors; A.7Mitochondrial electron transport inhibitors;. A.8Voltage-dependent sodium channel blockers; A.9Inhibitors of the lipid synthesis; and A.10group of various compounds.
摘要翻译：本发明涉及具有式（I）的至少一种3-乙酰基-1-苯基吡唑化合物或其盐的活性成分的杀虫组合物：其中X是N或C-R 5; R 1是C 1 -C 4 - 烷基或C 1 -C 4 - （C 1 -C 4）烷基或C 1 -C 4 - > - 卤代烷基; R 2是NR 6 R 7或S（O）n R 8， ; R 3是卤素，C 1 -C 4 - 卤代烷基，C 1 -C 4烷基， / SO 2 - 烷基，SF 5或S（O）n R 9。 R 4是氢或卤素; R 5是卤素; R 6是氢，C 1 -C 4 - 烷基，C 1 -C 4 - C（O）R 10，S（O）q CF 3 3， R 7是氢或C 1 -C 4 - 烷基，或R 6和R 7 连接在一起形成C 4 -C 6亚烷基部分，其中一个CH 2 - 亚基可以被取代通过氧或自由基NR 11; R 9，R 9，R 10，R 11，各自独立地为氢，C 1〜 / SUB> -C _{4 -alkylorC _{1 -C _{4 - 卤代烷基; m，n，p和q各自独立地为0,1或2; 和至少一种另外的选自A.1GABA门控氯化物通道拮抗剂的杀虫活性化合物II; A.2烟碱乙酰胆碱受体激动剂/拮抗剂A.3避孕激素模拟物; A.4影响氧化磷酸化的化合物; A.5壳多糖生物合成抑制剂 A.6造成破坏者 A.7线粒体电子传递抑制剂 A.8电压依赖性钠通道阻滞剂; A.9脂质合成抑制剂; 和A.10组各种化合物。}}}

3. 发明申请

WO2008074686A1 SUBSTITUTED 1-(AZOLIN-2-YL)-AMINO-1,2-HETEROCYCLYL-ETHANE COMPOUNDS FOR COMBATING PESTS 审中-公开
标题翻译：取代的1-（亚氨基-2-YL） - 氨基-1,2-杂环化合物 - 乙炔化合物
公开(公告)号：WO2008074686A1
公开(公告)日：2008-06-26
申请号：PCT/EP2007/063654
申请日：2007-12-11
申请人： BASF SE , KORDES, Markus , VEZOUET, Ronan Le , KORADIN, Christopher , BAUMANN, Ernst , CULBERTSON, Deborah L.
发明人： KORDES, Markus , VEZOUET, Ronan Le , KORADIN, Christopher , BAUMANN, Ernst , CULBERTSON, Deborah L.
IPC分类号： C07D401/06 , C07D405/06 , C07D409/06 , C07D417/12 , C07D417/14 , A01N43/78
CPC分类号： C07D409/06 , A01N43/50 , A01N43/76 , A01N43/78 , C07D401/06 , C07D405/06 , C07D417/12 , C07D417/14
摘要： The present invention relates to 1-(Azolin-2-yl)-amino-1,2-heterocyclyl-ethane compounds, which are useful for combating insects, arachnids and nematodes. The present invention also relates to methods for combating animal pests and to compositions for combating animal pests. It has been found that animal pests can be combated by 1-(Azolin-2-yl)-amino-1,2- heterocyclyl-ethane compounds of the general formula (I): wherein A is a radical of the formulae A 1 or A 2 : and wherein X is sulfur, oxygen or NR 7 , and Het A , Het B and R 1 to R 7 are defined as in the description.
摘要翻译：本发明涉及1-（唑啉-2-基） - 氨基-1,2-杂环基 - 乙烷化合物，其可用于防治昆虫，蜘蛛和线虫。本发明还涉及用于对抗动物害虫的方法和用于对抗动物害虫的组合物。已经发现，可以通过通式（I）的1-（氮杂-2-基） - 氨基-1,2-杂环基 - 乙烷化合物来对抗动物害虫：其中A是式A

4. 发明申请

WO2007104726A1 QUINOLINE DERIVATIVES AND THEIR USE AS PESTICIDES 审中-公开
标题翻译：喹啉衍生物及其作为杀虫剂的用途
公开(公告)号：WO2007104726A1
公开(公告)日：2007-09-20
申请号：PCT/EP2007/052262
申请日：2007-03-12
申请人： BASF AKTIENGESELLSCHAFT , PUHL, Michael , GRAMMENOS, Wassilios , RHEINHEIMER, Joachim , LOHMANN, Jan Klaas , RACK, Michael , PARRA RAPADO, Liliana , KORADIN, Christopher , LANGEWALD, Jürgen , CULBERTSON, Deborah, L. , ANSPAUGH, Douglas, D. , OLOUMI-SADEGHI, Hassan , VAN TUYL COTTER, Henry , KUHN, David, G.
发明人： PUHL, Michael , GRAMMENOS, Wassilios , RHEINHEIMER, Joachim , LOHMANN, Jan Klaas , RACK, Michael , PARRA RAPADO, Liliana , KORADIN, Christopher , LANGEWALD, Jürgen , CULBERTSON, Deborah, L. , ANSPAUGH, Douglas, D. , OLOUMI-SADEGHI, Hassan , VAN TUYL COTTER, Henry , KUHN, David, G.
IPC分类号： C07D215/12 , C07D215/60 , A01N43/42
CPC分类号： C07D215/12 , C07D215/60
摘要： This invention relates to quinoline derivatives of formula (I) wherein R 1 , R 2 , R 3 are each independently halogen, hydroxy, cyano, amino, nitro, C 1 - C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 3 -C 7 -cycloalkyl-C 1 -C 4 -alkyl, C 1 -C 6 -alkoxy, C 2 -C 6 -alkenyloxy, C 2 -C 6 -alkynyloxy, C 1 -C 4 -alkoxy-C 1 -C 4 -alkoxy, C 3 -C 7 - cycloalkyl-C 1 -C 4 -alkoxy, C(OH)(CF 3 ) 2 , C 1 -C 6 -haloalkyl, C 1 -C 6 -haloalkoxy, C 1 -C 6 - alkylthio, C 1 -C 6 -haloalkylthio, C 1 -C 6 -alkylsulfinyl, C 1 -C 6 -haloalkylsulfinyl, C 1 -C 6 - alkylsulfonyl, C 1 -C 6 -haloalkylsulfonyl, C(R a )=O, C(R a )=NOR b , C(=O)OR x , or C(=O)NR x R y ; R a is hydrogen or C 1 -C 4 -alkyl; R b is hydrogen, C 1 -C 4 -alkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -alkynyl, C 1 -C 4 -haloalkyl, or C 2 -C 4 - haloalkenyl; R x , R y are each independently hydrogen, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy-C 1 - C 4 -alkyl, C 1 -C 4 -thioalkyl-C 1 -C 4 -alkyl, C 1 -C 4 -alkyl-S(=O)C 1 -C 4 -alkyl, C 1 -C 4 -alkyl- S(=O) 2 C 1 -C 4 -alkyl, C 3 -C 6 -cyloalkyl, C 1 -C 4 -alkyl-C 3 -C 6 -cycloalkyl, C 3 -C 6 -alkenyl, C 3 -C 6 - alkinyl; R 4 , R 5 , R 6 , R 7 are each independently hydrogen, halogen, cyano, amino, nitro, hydroxy, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkyl, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, C 1 -C 6 - haloalkylthio, C 1 -C 6 -alkylsulfinyl, C 1 -C 6 -haloalkylsulfinyl, C 1 -C 6 -alkylsulfonyl, C 1 -C 6 - haloalkylsulfonyl, or C(=O)OR c ; R c is hydrogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, or C 2 -C 6 -alkinyl; m and n are each independently 1, 2, 3, 4, or 5; p is 0, 1, 2, 3, 4, or 5; and the N-oxides, enantiomers, diastereomers and salts thereof, processes and intermediates for the preparation of compounds (I), use of compounds (I) for combating insects, acarids, or nematodes and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds (I).
摘要翻译：本发明涉及式（I）的喹啉衍生物，其中R 1，R 2，R 3，3各自独立地为卤素，羟基，氰基，氨基，硝基，C 1 -C 6 - 烷基，C 2 -C 6 - 烯基，C 1 -C 6 - C 2 -C 6 - 炔基，C 3 -C 7 - 环烷基，C 3

5. 发明申请

WO2006125748A1 1-(IMIDAZOLIN-2-YL)AMINO-1,2-DIPHENYLETHANE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
标题翻译： 1-（咪唑烷-2-基）氨基-1,2-二苯醚化合物，用于组合动物乳剂
公开(公告)号：WO2006125748A1
公开(公告)日：2006-11-30
申请号：PCT/EP2006/062419
申请日：2006-05-18
申请人： BASF AKTIENGESELLSCHAFT , KORDES, Markus , GÖTZ, Norbert , RACK, Michael , KORADIN, Christopher , TEDESCHI, Livio , CULBERTSON, Deborah L.
发明人： KORDES, Markus , GÖTZ, Norbert , RACK, Michael , KORADIN, Christopher , TEDESCHI, Livio , CULBERTSON, Deborah L.
IPC分类号： C07D233/48 , A01N43/54
CPC分类号： A01N43/50 , C07D233/48
摘要： The present invention relates to 1-(imidazolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and their agriculturally acceptable salts, wherein A is a radical of the formula A 1 or A 2 . The invention relates also to agricultural compositions and to seed comprising at least one compound I and/or a salt thereof, as well as a method of combating animal pests, a method for protecting crops from attack or infestation by animal pests and a method for protecting non-living materials from attack or infestation by animal pests, a method for the protection of seeds from animal pests and of the seedlings' roots and shoots from animal pests by applying a pesticidally effective amount of at least one 1-(imidazolin-2-yl)amino-1 ,2- diphenylethane compound I and/or a salt thereof.
摘要翻译：本发明涉及式I的1-（咪唑啉-2-基）氨基-1,2-二苯基乙烷化合物及其农业上可接受的盐，其中A是式A 1或 A ^{2 。本发明还涉及农业组合物和包含至少一种化合物I和/或其盐的种子，以及防治动物害虫的方法，用于保护作物免受动物害虫侵袭或侵染的方法和保护方法通过施用杀虫有效量的至少一种1-（咪唑啉-2-酮）的动物害虫的攻击或感染的非生物材料，动物害虫的种子保护方法和来自动物害虫的幼苗的根和芽，吡啶-2-基）氨基-1,2-二苯基乙烷化合物I和/或其盐。}

6. 发明申请

WO2009133179A3 METHOD FOR THE PRODUCTION OF HALOGEN-SUBSTITUTED 2-(AMINOMETHYLIDENE)-3- OXOBUTYRIC ACID ESTERS 审中-公开
标题翻译：用于生产方法卤素取代的2-（氨基亚甲基）-3-氧代丁酸
公开(公告)号：WO2009133179A3
公开(公告)日：2010-02-25
申请号：PCT/EP2009055285
申请日：2009-04-30
申请人： BASF SE , ZIERKE THOMAS , MAYWALD VOLKER , RACK MICHAEL , SMIDT SEBASTIAN PEER , KEIL MICHAEL , WOLF BERND , KORADIN CHRISTOPHER
发明人： ZIERKE THOMAS , MAYWALD VOLKER , RACK MICHAEL , SMIDT SEBASTIAN PEER , KEIL MICHAEL , WOLF BERND , KORADIN CHRISTOPHER
IPC分类号： C07D231/14 , C07D295/145
CPC分类号： C07D295/145 , C07D231/14
摘要： The present invention relates to a method for producing 2- (aminomethylidene)-4,4dihalo-3-oxobutyric acid esters of the formula (I), where R1, R2, R3 are C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C3-C10-cycloalkyl or benzyl and/or R2 together with R3 and the nitrogen atom, to which both radicals are bound, are a heterocyclic radical, wherein a corresponding 3-aminoacrylic acid ester is reacted with a halogen-substituted acetyl fluoride in the presence of at least one alkali or earth alkali metal fluoride. The invention also relates to the further reaction of halogen-substituted 2-(aminomethylidene)-3-oxobutyric acid esters of the formula (1) into halomethyl-substituted pyrazole-4-ylcarboxylic acids and the esters thereof.
摘要翻译：本发明涉及2-（氨基 - 亚甲基）的制备方法中，式-4,4-二卤代-3-氧代丁酸酯（I）其中R1，R2，R3是C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C3-C10环烷基或与R 3苄基和/或R 2在一起并到两个基团连接的氮原子代表的杂环基团，其中一个相应的3-氨基丙烯酸酯是具有卤乙酰氟取代反应是在至少一种碱金属或碱土金属氟化物的存在; 和卤素 - 取代的2-（氨基亚甲基）-3-氧代丁酸的式（I）的酯的进一步反应卤代甲基取代的吡唑-4-基甲酸和它们的酯。

7. 发明申请

WO2009133178A1 VERFAHREN ZUR HERSTELLUNG VON 2-(AMINOMETHYLIDEN)-4,4-DIFLUOR-3-OXOBUTTERSÄUREESTERN 审中-公开
标题翻译：用于生产2-（氨基亚甲基）-4,4-二氟-3-氧代丁酸酯
公开(公告)号：WO2009133178A1
公开(公告)日：2009-11-05
申请号：PCT/EP2009/055283
申请日：2009-04-30
申请人： BASF SE , ZIERKE, Thomas , MAYWALD, Volker , RACK, Michael , SMIDT, Sebastian Peer , KEIL, Michael , WOLF, Bernd , KORADIN, Christopher
发明人： ZIERKE, Thomas , MAYWALD, Volker , RACK, Michael , SMIDT, Sebastian Peer , KEIL, Michael , WOLF, Bernd , KORADIN, Christopher
IPC分类号： C07C227/16 , C07C229/30 , C07D231/14
CPC分类号： C07D231/14 , C07C229/30 , C07D295/145
摘要： Die vorliegende Erfindung betrifft ein Verfahren zur Herstellung von difluormethylsubsti- tuierten Pyrazol4-ylcarbonsäuren und deren Ester, 2-(Aminomethyliden)-4,4-difluor-3- oxobuttersäureester der Formel (I), worin R 1 , R 2 und R 3 unabhängig voneinander für C 1 -C 6 -Alkyl, C 1 -C 6 -Haloalkyl, C 2 -C 6 -Alkenyl, C 3 -C 10 -Cycloalkyl oder Benzyl steht oder NR 2 R 3 für einen 5- bis 10-gliedrigen heterocyclischen Rest steht, ein Verfahren zur Herstellung von Verbindungen der Formel (I), bei dem man einen entsprechenden 3-Aminoacrylsäureester mit Difluoracetylfluorid umsetzt sowie die Verwendung von Verbindungen der Formel (I) in dem Verfahren zur Herstellung von difluormethylsubstituierten Pyrazol- 4-ylcarbonsäuren und deren Ester.
摘要翻译：本发明涉及一种用于difluormethylsubsti的制备 - 取代的吡唑基甲酸及其酯，2-（氨基亚甲基）的式（I）的-4,4-二氟-3-氧代丁酸乙酯，其特征在于R1，R2和R3各自独立地为C1 C6烷基，C1-C6卤代烷基，C2-C6链烯基，C3-C10环烷基或苄基或NR2R3表示5至10元杂环基团，为式I化合物的制备方法（I），该方法包括用二氟乙酰氟一个相应的3-氨基丙烯酸酯，以及用于制备吡唑difluormethylsubstituierten唑-4-基甲酸和它们的酯的使用过程中的式（I）的化合物的反应。

8. 发明申请

WO2009106619A1 Process for preparing alkyl 2-alkoxymethylene-4,4-difluoro-3-oxobutyrates 审中-公开
标题翻译：制备2-烷氧基亚甲基-4,4-二氟-3-氧代丁酸烷基酯的方法
公开(公告)号：WO2009106619A1
公开(公告)日：2009-09-03
申请号：PCT/EP2009/052378
申请日：2009-02-27
申请人： BASF SE , Maywald, Volker , Smidt, Sebastian Peer , Wolf, Bernd , Koradin, Christopher , Zierke, Thomas , Rack, Michael , Keil, Michael
发明人： Maywald, Volker , Smidt, Sebastian Peer , Wolf, Bernd , Koradin, Christopher , Zierke, Thomas , Rack, Michael , Keil, Michael
IPC分类号： C07C67/343 , C07C69/72
CPC分类号： C07D231/14 , C07C67/343 , C07C69/72
摘要： A process for preparing alkyl 2-alkoxymethylene-4,4-difluoro-3-oxobutyrates (VI) where R is methyl or ethyl, from crude reaction mixtures of alkyl 4,4-difluoroacetoacetates (I) by a) reacting alkyl acetate (II), RO M alkoxide (III), where M is a sodium or potassium ion, and alkyl difluoroacetate (IV), without additional solvent to form an enolate (V), b) releasing the corresponding alkyl 4,4-difluoroacetoacetate (I) from the enolate (V) by means of acid, c) removing the salt formed from cation M and acid anion as a solid and d) converting (I), without isolation from the crude reaction mixture, to the alkyl 2-alkoxymethylene-4,4-difluoro-3-oxobutyrate (VI), and the use of (VI) for preparing 1-methyl-3-difluoromethyl-pyrazol-3-ylcarboxyates (VII).
摘要翻译：由烷基4,4-二氟乙酰乙酸酯（I）的粗反应混合物制备R为甲基或乙基的2-烷氧基亚甲基-4,4-二氟-3-氧代丁酸烷基酯（VI）的方法，通过以下步骤a）使乙酸烷基酯），RO M醇盐（III），其中M是钠或钾离子，和二氟乙酸烷基酯（IV），没有另外的溶剂以形成烯醇化物（V），b）释放相应的4,4-二氟乙酰乙酸烷基酯（I）从烯醇化物（V）通过酸，c）除去由阳离子M和酸阴离子形成的盐作为固体，以及d）将（I）从粗反应混合物转化成2-烷基亚甲基-4 ，4-二氟-3-氧代丁酸（VI），以及（VI）用于制备1-甲基-3-二氟甲基 - 吡唑-3-基羧酸酯（VII）的用途。

9. 发明申请

WO2009004032A1 1-(AZOLIN-2-YL)AMINO-1,2-DIPHENYLETHANE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
标题翻译： 1-（AZOLIN-2-YL）氨基-1,2-二苯醚化合物，用于组合动物饲料
公开(公告)号：WO2009004032A1
公开(公告)日：2009-01-08
申请号：PCT/EP2008/058517
申请日：2008-07-02
申请人： BASF SE , KORDES, Markus , KORADIN, Christopher , LE VEZOUET, Ronan , BAUMANN, Ernst , CULBERTSON, Deborah L. , ANSPAUGH, Douglas D. , OLOUMI-SADEGHI, Hassan , EBUENGA, Cecile
发明人： KORDES, Markus , KORADIN, Christopher , LE VEZOUET, Ronan , BAUMANN, Ernst , CULBERTSON, Deborah L. , ANSPAUGH, Douglas D. , OLOUMI-SADEGHI, Hassan , EBUENGA, Cecile
IPC分类号： C07D233/48 , C07D263/28 , C07D277/18 , C07D417/12 , C07D417/06 , A01N43/50 , A01N43/76 , A01N43/78
CPC分类号： C07D263/28 , A01N43/50 , A01N43/76 , A01N43/78 , A01N47/12 , A01N47/16 , C07D233/48 , C07D277/18 , C07D417/06 , C07D417/12
摘要： The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the formula I and to their salts which are useful for combating animal pests. The invention also relates to a method for controlling animal pests by using these compounds, to seed and to an agricultural and veterinary composition comprising said compounds, wherein A is a radical of formulae A.1 or A.2 wherein # denotes the bond to the remaining compound of formula I, X is selected from O, S and NR x , R 1 is selected from the group consisting of -OR A , -NR B1 R B2 , -C(=O)-R C , -C(=O)-OR D , -C(=O)-SR E , -C(=O)-NR B1 R B2' , -C(=S)-R C' , -C(=S)-OR D' , -C(=S)-SR E' , -C(=S)-NR B1 R B2 , -C(=NR 1a )-R C' , -C(=NR 1b )-OR D' , -C(=NR 1c )-SR E' , -C(=NR 1d )-NR B1 R B2 , -S(=O)-R F , -S(=O) 2 -R G , -S(=O) 2 -NR B1 R B2' , -P(=O)R H1 R H2 , -P(=S)R H1 R H2 , -B-C(=O)-R I , -B-O-C(=O)-R I , -B-S-C(=O)-R I , -B-N(R J )-C(=O)-R K , -B-C(=S)-R K , -B-O-C(=S)-R K , -B-S-C(=S)-R K , -B-N(R J )-C(=S)-R K , C 1 -C 8 -alkenyl, C 1 -C 8 -alkynyl, C 3 -C 8 -cycloalkyl, which is unsubstituted or may carry 1 to 4 substituents R 1e , naphthyl, which is unsubstituted or may carry 1 to 4 substituents R 1f , a saturated or partially unsaturated heterocycle, which is unsubstituted or may carry 1 to 4 substituents R 1g , hetaryl, which is unsubstituted or may carry 1 to 4 substituents R 1h , and C 1 -C 6 -alkyl, which carries a radical selected from the group consisting of -NR 1i R 1j , C 1 -C 4 -alkoxycarbonyl, C 3 -C 8 -cycloalkyl, aryl, aryloxy, arylthio, heterocyclyl, heterocyclyloxy and heterocyclylthio, R 2 , R 3 , R 4 , R 5 , R 6 and R 7 are each independently hydrogen, halogen, OH, SH, NH 2 , SO 3 H, COOH, cyano, nitro, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -alkylamino etc.
摘要翻译：本发明涉及式I的1-（吡唑-2-基）氨基-1,2-二苯基乙烷化合物及其盐，其可用于防治动物害虫。本发明还涉及通过使用这些化合物，种子和包含所述化合物的农业和兽医组合物来控制动物害虫的方法，其中A是式A.1或A.2的基团，其中＃表示与剩余的式I化合物，X选自O，S和NR x，R1选自-ORA，-NRB1RB2，-C（= O）-RC，-C（= O）-OR，-C （= O）-SRE，-C（= O）-NRB1RB2'，-C（= S）-RC'，-C（= S）-OR'，-C（= S）-SRE' =（NR1c）-SR'，-C（= NR1d）-NRB1RB2，-S（= O））-RF，-S（= O）2 -RG，-S（= O）2 -NRB 1 R B 2'，-P（= O）RH1RH 2，-P（= S）RH1RH 2，-BC（= O） -BOC（= O）-RI，-BSC（= O）-RI，-BN（RJ）-C（= O）-RK，-BC（= S）-RK，-BOC（= S）-RK， -BSC（= S）-RK，-BN（RJ）-C（= S）-RK，C1-C8-烯基，C1-C8-炔基，C3-C8-环烷基，其未被取代或可携带1至4 取代基R 1e，萘基，其是未取代的或可以携带1至4个取代基R 1f，饱和或部分不饱和的杂环，其为未制备的或可以携带1至4个未取代的或可以携带1至4个取代基R 1h的取代基R 1g，杂芳基，其中C 1 -C 6 - 烷基带有选自以下的基团：-NR 1 1 R 1，C 1 -C 4 - 烷氧基羰基， C 3 -C 8 - 环烷基，芳基，芳氧基，芳硫基，杂环基，杂环基氧基和杂环硫基，R 2，R 3，R 4，R 5，R 6和R 7各自独立地为氢，卤素，OH，SH，NH 2，SO 3 H，COOH，氰基，硝基， C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，C 1 -C 6烷基氨基等

10. 发明申请

WO2008000834A1 SUBSTITUTED 1-(AZOLIN-2-YL)-AMINO-2-ARYL-1-HETARYL-ETHANE COMPOUNDS 审中-公开
标题翻译：取代的1-（AZOLIN-2-YL） - 氨基-2-芳基-1-乙基 - 乙炔化合物
公开(公告)号：WO2008000834A1
公开(公告)日：2008-01-03
申请号：PCT/EP2007/056604
申请日：2007-06-29
申请人： BASF AKTIENGESELLSCHAFT , KORDES, Markus , BREUNINGER, Delphine , LE VEZOUET, Ronan , KORADIN, Christopher , TEDESCHI, Livio , PUHL, Michael , CULBERTSON, Deborah, L.
发明人： KORDES, Markus , BREUNINGER, Delphine , LE VEZOUET, Ronan , KORADIN, Christopher , TEDESCHI, Livio , PUHL, Michael , CULBERTSON, Deborah, L.
IPC分类号： C07D213/50 , C07D231/12 , C07D307/52 , C07D333/20 , C07D413/12 , C07D417/12 , A01N43/76 , A01N43/78 , A61P33/14
CPC分类号： C07D333/20 , C07D213/40 , C07D231/12 , C07D307/52 , C07D413/12 , C07D417/12
摘要： The present invention relates to 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane compounds (I) and 1-(aminothiocarbonylamino)-2-aryl-1-hetaryl-ethane compounds (II) and their salts which are useful for combating animal pest, in particular insects, arachnids and nematodes. Furthermore, the present invention relates to a method for combating animal pests selected from insects, arachnids and nematodes, and to agricultural compositions for combating animal pests. Furthermore, the present invention relates to veterinary compositions for combating animal pests.
摘要翻译：本发明涉及1-（吡唑啉-2-基） - 氨基-2-芳基-1-杂芳基 - 乙烷化合物（I）和1-（氨基硫代羰基氨基）-2-芳基-1-杂芳基 - 乙烷化合物（II）和它们的盐可用于对抗动物害虫，特别是昆虫，蜘蛛和线虫。此外，本发明涉及一种对抗从昆虫，蜘蛛和线虫中选出的动物害虫的方法以及用于对抗动物害虫的农业组合物。此外，本发明涉及用于对抗动物害虫的兽用组合物。

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