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    • 9. 发明授权
    • 1-heteroaryl-4-aryl-pyrazole microbicides
    • 1-杂芳基-4-芳基 - 吡唑杀微生物剂
    • US4806540A
    • 1989-02-21
    • US99928
    • 1987-09-23
    • Klaus SasseGerd HansslerHans-Georg SchmittWilfried Paulus
    • Klaus SasseGerd HansslerHans-Georg SchmittWilfried Paulus
    • A01N43/40A01N43/56A01N47/06A01N47/16A01N47/22C07D401/04C07D403/04C07D405/14A61K31/44A61K31/47A61K31/505C07D215/20C07D215/36C07D215/38
    • C07D401/04A01N43/56A01N47/06A01N47/16A01N47/22C07D403/04C07D405/14
    • Novel microbicidally active 1-heteroaryl-4-arylpyrazole derivatives of the formulae (I) and/or (1A) ##STR1## in which R represents hydrogen or alkyl,R.sup.1 represents halogen, hydroxyl, optionally substituted alkyl, optionally substituted alkoxy, a radical --S(O).sub.p -alkyl which is optionally substituted in the alkyl part, nitro or optionally substituted amino, or represents a fused-on carbocyclic or heterocyclic radicalp represents the integer 0, 1 or 2,n represents an integer from 0 to 5,X represents .dbd.CH--, or represents a nitrogen atom,Y represents CO or SO.sub.2 andR.sup.2 represents hydrogen, in each case optionaly substituted alkyl, cycloalkyl or aryl or a heterocyclic radical, or represents OR.sup.3, or also represents SR.sup.3, if Y is CO,whereinR.sup.3 represents optionally substituted alkyl or aryl, orR.sup.2 represents a radical ##STR2## wherein R.sup.4 represents hydrogen or saturated or unsaturated optionally substituted alkyl and optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aryl or an optionally substituted heterocyclic radical, orR.sup.4 and R.sup.5, together with the nitrogen atom on which they are located, form a heterocyclic ring which optionally contains further hetero atoms and can optionally be mono- or polysubstituted by identical or different substituents.
    • 式(I)和/或(1A)的新型杀微生物活性1-杂芳基-4-芳基吡唑衍生物其中R表示氢或烷基,R 1表示卤素,羟基,任选地 取代的烷基,任选取代的烷氧基,在烷基部分任选取代的-S(O)对 - 烷基,硝基或任选取代的氨基,或表示稠合的碳环或杂环基p表示整数0,1或 2,n表示0〜5的整数,X表示= CH-,或表示氮原子,Y表示CO或SO2,R2表示氢,各自为任选取代的烷基,环烷基或芳基或杂环基,或表示 OR 3,或者也表示SR 3,如果Y是CO,其中R 3表示任选取代的烷基或芳基,或R 2表示基团,其中R 4表示氢或饱和或不饱和的任选取代的烷基和任选取代的烷基,任选取代的环烷 或任选取代的芳基或任选取代的杂环基,或者R 4和R 5与它们所位于的氮原子一起形成任选含有其它杂原子的杂环,并且可任选地被相同或不同的单取代或多取代 取代基。