专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明授权

US08853414B2 Process for producing pyripyropene derivatives 有权
标题翻译：生产拟南芥衍生物的方法
公开(公告)号：US08853414B2
公开(公告)日：2014-10-07
申请号：US13581857
申请日：2010-11-10
申请人： Yoshimasa Fukuda , Takashi Ando , Kimihiko Goto , Nozomu Nakanishi , Takashi Watanabe , Kenichi Kurihara , Nobuto Minowa , Masaaki Mitomi
发明人： Yoshimasa Fukuda , Takashi Ando , Kimihiko Goto , Nozomu Nakanishi , Takashi Watanabe , Kenichi Kurihara , Nobuto Minowa , Masaaki Mitomi
IPC分类号： C07D401/04 , C07D493/04
CPC分类号： C07D493/04
摘要： Disclosed is a process for efficiently producing pyripyropene derivatives having acyloxy at the 1-position and 11-position and hydroxyl at the 7-position. The process comprises selectively acylating hydroxyl at the 1-position and 11-position of a compound represented by formula B1 through one to three steps with an acylating agent in the presence or absence of a base.
摘要翻译：公开了一种有效生产在1-位和11位上具有酰氧基并在7-位具有羟基的吡啶并苯衍生物的方法。该方法包括在存在或不存在碱的情况下用酰化剂选择性地将式B1化合物的1位和11位羟基选择性酰化1至3个步骤。

2. 发明授权

US08759529B2 Process for producing pyripyropene derivatives and intermediates for the production thereof 有权
标题翻译：生产拟南芥衍生物的方法及其生产用中间体
公开(公告)号：US08759529B2
公开(公告)日：2014-06-24
申请号：US13572971
申请日：2012-08-13
申请人： Kimihiko Goto , Kazumi Yamamoto , Masayo Sakai , Masaaki Mitomi , Takashi Ando
发明人： Kimihiko Goto , Kazumi Yamamoto , Masayo Sakai , Masaaki Mitomi , Takashi Ando
IPC分类号： C07D493/04
CPC分类号： C07D493/04 , Y02P20/55
摘要： A process for producing compound C represented by formula C is disclosed: wherein R′ represents substituent groups as described herein. The process can produce pyripyropene derivatives that have acyloxy groups at the 1- and 11-positions and a hydroxyl group at the 7-position and are useful as insect pest control agents at a high yield.
摘要翻译：公开了制备由式C表示的化合物C的方法：其中R'表示如本文所述的取代基。该方法可以产生在1-位和11位上具有酰氧基并且在7-位上具有羟基并且以高产率用作害虫防治剂的吡哆烯衍生物。

3. 发明授权

US08263778B2 Process for producing pyripyropene derivatives and intermediates for the production thereof 有权
标题翻译：生产拟南芥衍生物的方法及其生产用中间体
公开(公告)号：US08263778B2
公开(公告)日：2012-09-11
申请号：US12733113
申请日：2008-08-13
申请人： Kimihiko Goto , Kazumi Yamamoto , Masayo Sakai , Masaaki Mitomi , Takashi Ando
发明人： Kimihiko Goto , Kazumi Yamamoto , Masayo Sakai , Masaaki Mitomi , Takashi Ando
IPC分类号： C07D493/04
CPC分类号： C07D493/04 , Y02P20/55
摘要： Disclosed is a process for producing compound C represented by formula C: wherein R′ represents straight chain, branched chain, or cyclic C2-6 alkylcarbonyl, wherein R1b is used as a protective group for hydroxyl at the 7-position of compound C. R1b represents formyl; optionally substituted straight chain C1-4 alkylcarbonyl; optionally substituted benzyl; group —SiR3R4R5 optionally substituted by halogen atom wherein R3, R4, and R5 each independently represent straight chain or branched chain C1-6 alkyl or phenyl; C1-6 alkyloxy-C1-6 alkyl optionally substituted by halogen atom; C1-6 alkylthio-C1-6 alkyl optionally substituted by halogen atom; straight chain, branched chain, or cyclic C1-4 alkyl optionally substituted by halogen atom, provided that, when alkyl in the C1-4 alkyl group is of a branched chain or cyclic type, the alkyl group is C3-4 alkyl; C2-6 alkenyl optionally substituted by halogen atom; C2-6 alkynyl optionally substituted by halogen atom; or an optionally substituted saturated or unsaturated five- or six-membered heterocyclic group. The process can produce pyripyropene derivatives that have acyloxy groups at the 1- and 11-positions and a hydroxyl group at the 7-position and are useful as insect pest control agents at a high yield.
摘要翻译：公开了一种制备由式C表示的化合物C的方法：其中R'表示直链，支链或环状C 2-6烷基羰基，其中R 1b用作化合物C的7-位羟基保护基。R1b 代表甲酰基; 任选取代的直链C 1-4烷基羰基; 任选取代的苄基; 基团-SiR 3 R 4 R 5任选被卤素原子取代，其中R 3，R 4和R 5各自独立地表示直链或支链C 1-6烷基或苯基; 任选被卤素原子取代的C 1-6烷氧基-C 1-6烷基; 任选被卤素原子取代的C 1-6烷硫基-C 1-6烷基; 直链，支链或任选被卤素原子取代的环状C 1-4烷基，条件是当C 1-4烷基中的烷基为支链或环状时，该烷基为C 3-4烷基; 任选被卤素原子取代的C 2-6烯基; 任选被卤素原子取代的C 2-6炔基; 或任选取代的饱和或不饱和的五元或六元杂环基。该方法可以产生在1-位和11位上具有酰氧基并且在7-位上具有羟基并且以高产率用作害虫控制剂的吡哆烯衍生物。

4. 发明申请

US20060281780A1 Pest control agents 有权
标题翻译：害虫控制剂
公开(公告)号：US20060281780A1
公开(公告)日：2006-12-14
申请号：US11443299
申请日：2006-05-31
申请人： Kimihiko Goto , Ryo Horikoshi , Mariko Tsuchida , Kazuhiko Oyama , Satoshi Omura , Hiroshi Tomoda , Toshiaki Sunazuka
发明人： Kimihiko Goto , Ryo Horikoshi , Mariko Tsuchida , Kazuhiko Oyama , Satoshi Omura , Hiroshi Tomoda , Toshiaki Sunazuka
IPC分类号： A01N43/42 , A01N43/40
CPC分类号： A01N43/90
摘要： There is provided a pest control agent comprising a compound represented by formula (I) as active ingredient.
摘要翻译：提供了包含由式（I）表示的化合物作为活性成分的害虫防治剂。

5. 发明授权

US09169504B2 Method for producing pyripyropene 有权
标题翻译：生产拟南芥的方法
公开(公告)号：US09169504B2
公开(公告)日：2015-10-27
申请号：US13575159
申请日：2011-01-19
申请人： Hiroyuki Anzai , Kentaro Yamamoto , Kazuhiko Oyama , Mariko Tsuchida , Kimihiko Goto , Masaaki Mitomi
发明人： Hiroyuki Anzai , Kentaro Yamamoto , Kazuhiko Oyama , Mariko Tsuchida , Kimihiko Goto , Masaaki Mitomi
IPC分类号： C12P17/18 , C12N9/02 , C12N9/10 , C12N9/88 , C12N9/00 , C12N15/52
CPC分类号： C12P17/181 , C12N9/0071 , C12N9/1025 , C12N9/1029 , C12N9/88 , C12N9/93 , C12N15/52 , C12Y114/13008 , C12Y114/14001 , C12Y203/00 , C12Y203/01 , C12Y205/01 , C12Y406/01 , C12Y602/01
摘要： There is provided a method for culturing a microorganism in which a particular polynucleotide or a recombinant vector comprising it/them is introduced with an intermediate compound necessary for biosynthesis of pyripyropene A. The method of the present invention allows for the production of pyripyropene.
摘要翻译：提供了一种培养微生物的方法，其中特定的多核苷酸或包含它们的重组载体被引入与生物合成拟南芥A所必需的中间体化合物。本发明的方法允许产生吡啶并吡喃。

6. 发明授权

US08367707B2 Pest control agents 有权
公开(公告)号：US08367707B2
公开(公告)日：2013-02-05
申请号：US12903624
申请日：2010-10-13
申请人： Kimihiko Goto , Ryo Horikoshi , Mariko Tsuchida , Kazuhiko Oyama , Satoshi Omura , Hiroshi Tomoda , Toshiaki Sunazuka
发明人： Kimihiko Goto , Ryo Horikoshi , Mariko Tsuchida , Kazuhiko Oyama , Satoshi Omura , Hiroshi Tomoda , Toshiaki Sunazuka
IPC分类号： A01N43/40 , A61K31/44 , C07D211/34
CPC分类号： A01N43/90
摘要： Disclosed is a composition for use as a pest control agent, comprising a compound represented by formula (I) or an agriculturally and horticulturally acceptable salt thereof as active ingredient and an agriculturally and horticulturally acceptable carrier:

7. 发明授权

US07838538B2 Pest control agents 有权
标题翻译：害虫控制剂
公开(公告)号：US07838538B2
公开(公告)日：2010-11-23
申请号：US12318232
申请日：2008-12-23
申请人： Kimihiko Goto , Ryo Horikoshi , Mariko Tsuchida , Kazuhiko Oyama , Satoshi Omura , Hiroshi Tomoda , Toshiaki Sunazuka
发明人： Kimihiko Goto , Ryo Horikoshi , Mariko Tsuchida , Kazuhiko Oyama , Satoshi Omura , Hiroshi Tomoda , Toshiaki Sunazuka
IPC分类号： A61K31/44 , A01N43/40 , C07D405/00
CPC分类号： A01N43/90
摘要： Disclosed is a composition for use as a pest control agent, comprising a compound represented by formula (I) or an agriculturally and horticulturally acceptable salt thereof as active ingredient and an agriculturally and horticulturally acceptable carrier:
摘要翻译：公开了一种用作害虫控制剂的组合物，其包含式（I）表示的化合物或其农业和园艺可接受的盐作为活性成分和农业和园艺可接受的载体：

8. 发明申请

US20130060042A1 PROCESS FOR PRODUCING PYRIPYROPENE DERIVATIVES 有权
标题翻译：生产吡啶衍生物的方法
公开(公告)号：US20130060042A1
公开(公告)日：2013-03-07
申请号：US13581857
申请日：2010-11-10
申请人： Yoshimasa Fukuda , Takashi Ando , Kimihiko Goto , Nozomu Nakanishi , Takashi Watanabe , Kenichi Kurihara , Nobuto Minowa , Masaaki Mitomi
发明人： Yoshimasa Fukuda , Takashi Ando , Kimihiko Goto , Nozomu Nakanishi , Takashi Watanabe , Kenichi Kurihara , Nobuto Minowa , Masaaki Mitomi
IPC分类号： C07D493/04
CPC分类号： C07D493/04
摘要： Disclosed is a process for efficiently producing pyripyropene derivatives having acyloxy at the 1-position and 11-position and hydroxyl at the 7-position. The process comprises selectively acylating hydroxyl at the 1-position and 11-position of a compound represented by formula B1 through one to three steps with an acylating agent in the presence or absence of a base.
摘要翻译：公开了一种有效生产在1-位和11位上具有酰氧基并在7-位具有羟基的吡啶并苯衍生物的方法。该方法包括在存在或不存在碱的情况下用酰化剂选择性地将式B1化合物的1位和11位羟基选择性酰化1-3步。

9. 发明申请

US20130023017A1 METHOD FOR PRODUCING PYRIPYROPENE 有权
标题翻译：生产吡啶的方法
公开(公告)号：US20130023017A1
公开(公告)日：2013-01-24
申请号：US13575159
申请日：2011-01-19
申请人： Hiroyuki Anzai , Kentaro Yamamoto , Kazuhiko Oyama , Mariko Tsuchida , Kimihiko Goto , Masaaki Mitomi
发明人： Hiroyuki Anzai , Kentaro Yamamoto , Kazuhiko Oyama , Mariko Tsuchida , Kimihiko Goto , Masaaki Mitomi
IPC分类号： C12P17/18 , C12N15/53 , C12N1/19 , C12N15/63 , C12N1/21 , C12N1/15 , C12P17/16 , C12N15/54
CPC分类号： C12P17/181 , C12N9/0071 , C12N9/1025 , C12N9/1029 , C12N9/88 , C12N9/93 , C12N15/52 , C12Y114/13008 , C12Y114/14001 , C12Y203/00 , C12Y203/01 , C12Y205/01 , C12Y406/01 , C12Y602/01
摘要： There is provided a method for culturing a microorganism in which a particular polynucleotide or a recombinant vector comprising it/them is introduced with an intermediate compound necessary for biosynthesis of pyripyropene. A. The method of the present invention allows for the production of pyripyropene.
摘要翻译：提供了一种培养微生物的方法，其中将特定的多核苷酸或其包含的重组载体与生物合成吡啶并苯所必需的中间体化合物引入。 A.本发明的方法允许生产吡啶并苯。

10. 发明申请

US20120330022A1 METHOD FOR PRODUCING PYRIPYROPENE DERIVATIVES BY THE ENZYMATIC METHOD 审中-公开
标题翻译：通过酶法制备吡啶衍生物的方法
公开(公告)号：US20120330022A1
公开(公告)日：2012-12-27
申请号：US13575171
申请日：2011-01-19
申请人： Kentaro Yamamoto , Mariko Tsuchida , Kazuhiko Oyama , Kimihiko Goto , Masaaki Mitomi
发明人： Kentaro Yamamoto , Mariko Tsuchida , Kazuhiko Oyama , Kimihiko Goto , Masaaki Mitomi
IPC分类号： C12P17/18 , C07D493/04
CPC分类号： C07D403/04 , C07D403/08 , C12P17/181
摘要： There is provided a method for producing a pyripyropene derivative represented by the following formula A by an enzyme method. The production method of the present invention allows for production of a pyripyropene derivative under simpler conditions and in shorter steps. [wherein R represents a linear, branched or cyclic C2-6 alkylcarbonyl group (when the alkyl moiety of this group is branched or cyclic, C3-6 alkyl carbonyl group)].
摘要翻译：提供了通过酶法制备由下式A表示的嘧啶衍生物的方法。本发明的制备方法允许在更简单的条件下和较短的步骤中生产吡啶并苯衍生物。 [其中R表示直链，支链或环状C 2-6烷基羰基（当该基团的烷基部分为支链或环状时，为C 3-6烷基羰基）]。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式