专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明专利

IL216132A Diamino heterocyclic carboxamide compounds, use thereof and pharmaceutical compositions and inhibitors comprising them 未知
公开(公告)号：IL216132A
公开(公告)日：2015-10-29
申请号：IL21613211
申请日：2011-11-03
申请人： KOTOBUKI PHARMACEUTICAL CO LTD , SHIMADA ITSURO , KUROSAWA KAZUO , MATSUYA TAKAHIRO , IIKUBO KAZUHIKO , KONDOH YUTAKA , KAMIKAWA AKIO , TOMIYAMA HIROSHI , IWAI YOSHINORI , ASTELLAS PHARMA INC
发明人： SHIMADA ITSURO , KUROSAWA KAZUO , MATSUYA TAKAHIRO , IIKUBO KAZUHIKO , KONDOH YUTAKA , KAMIKAWA AKIO , TOMIYAMA HIROSHI , IWAI YOSHINORI
IPC分类号： A61K20060101 , A61P20060101 , C07D20060101
摘要： Provided is the compound 6-ethyl-3-({3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}amino)-5-(tetrahydro-2H-pyran-4-ylamino)pyrazine-2-carboxamide or a salt thereof for use in a method for preventing and/or treating acute myelocytic leukemia or atypical chronic myelocytic leukemia.

2. 发明专利

IL216132D0 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND 未知
公开(公告)号：IL216132D0
公开(公告)日：2012-01-31
申请号：IL21613211
申请日：2011-11-03
申请人： ASTELLAS PHARMA INC , KOTOBUKI PHARMACEUTICAL CO LTD , SHIMADA ITSURO , KUROSAWA KAZUO , MATSUYA TAKAHIRO , IIKUBO KAZUHIKO , KONDOH YUTAKA , KAMIKAWA AKIO , TOMIYAMA HIROSHI , IWAI YOSHINORI
IPC分类号： C07D20060101
摘要： Provided is the compound 6-ethyl-3-({3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}amino)-5-(tetrahydro-2H-pyran-4-ylamino)pyrazine-2-carboxamide or a salt thereof for use in a method for preventing and/or treating acute myelocytic leukemia or atypical chronic myelocytic leukemia.

3. 发明申请

WO1993020053A1 PYRIDYLSERINE DERIVATIVE 审中-公开
标题翻译：吡啶衍生物
公开(公告)号：WO1993020053A1
公开(公告)日：1993-10-14
申请号：PCT/JP1993000356
申请日：1993-03-25
申请人： YAMANOUCHI PHARMACEUTICAL CO., LTD. , SAKAMOTO, Shuichi , NODA, Ichio , KONDOH, Yutaka , KOSHIYA, Kazuo , HIDAKA, Kazuyuki
发明人： YAMANOUCHI PHARMACEUTICAL CO., LTD.
IPC分类号： C07D213/55
CPC分类号： C07D249/08 , C07D213/55 , C07D231/12 , C07D233/56 , C07D401/06 , C07D401/12 , Y02P20/55
摘要： A pyridylserine derivative represented by general formula (I) or a pharmaceutically acceptable salt thereof, wherein R represents hydrogen or an amino-protecting group, R represents hydrogen or a carboxyl-protecting group, A represents a single bond or lower alkylene, B represents -NR R , or mercapto which may be substituted by lower alkyl or cycloalkyl, R and R may be the same or different from each other and each represents hydrogen; a lower alkyl group which may be substituted by amino, lower alkylamino or carbocyclic aryl; an acyl group which may be substituted by amino; an aminocarbonyl group which may be substituted by lower alkyl or cycloalkyl; lower alkoxycarbonyl; cycloalkylcarbonyl; a nitrogenous heterocyclic group; or alternatively, R and R may be combined together to represent a nitrogenous heterocyclic group, a fused nitrogenous heterocyclic group or a cross-linked nitrogenous heterocyclic group. It has an anti-PCP effect and is useful as a psychotropic.
摘要翻译：由通式（I）表示的吡啶基丝氨酸衍生物或其药学上可接受的盐，其中R 1表示氢或氨基保护基，R 2表示氢或羧基保护基，A表示单键或低级亚烷基，B表示-NR 3 R 4或可被低级烷基或环烷基取代的巯基，R 3和R 4可以彼此相同或不同，各自表示氢; 可被氨基，低级烷基氨基或碳环芳基取代的低级烷基; 可被氨基取代的酰基; 可被低级烷基或环烷基取代的氨基羰基; 低级烷氧基羰基; 环烷基; 含氮杂环基; 或者R 3和R 4可以组合在一起以表示含氮杂环基，稠合杂环基或交联的含氮杂环基。它具有抗PCP作用，可作为精神药物使用。

4. 发明申请

WO1996014173A1 METHOD OF RECOVERING METAL MATERIALS FROM GAS GENERATOR FOR AIR BAG 审中-公开
标题翻译：从气囊发电机回收金属材料的方法
公开(公告)号：WO1996014173A1
公开(公告)日：1996-05-17
申请号：PCT/JP1995002251
申请日：1995-11-06
申请人： DAICEL CHEMICAL INDUSTRIES, LTD. , TOYOTA, JIDOSHA, KABUSHIKI, KAISHA , FUKABORI, Mitsuhiko , NAKAZATO, Yuzaburo , FUJIMOTO, Osamu , KONDOH, Yutaka , MIYAJI, Masahiro
发明人： DAICEL CHEMICAL INDUSTRIES, LTD. , TOYOTA, JIDOSHA, KABUSHIKI, KAISHA
IPC分类号： B09B05/00
CPC分类号： C22B7/001 , B09B5/00 , B60R21/26 , C22B1/005 , C22B7/003 , C22B7/005 , F23G2900/7001 , Y02P10/214
摘要： A method for easily taking out a gas generator from a scrapped car and efficiently recovering metal materials from the gas generator. This method comprises the steps of: a) pulverizing a scrapped car having an air bag apparatus mounted thereto by pulverizing means adjusted so that the size of the shreds is substantially equal that of the gas generator, and separating the gas generator as a single substantially-unpulverized body from the air bag device, b) taking out the gas generator from the shreds of the scrapped car, c) charging the gas generator taken out into a melting furnace, and d) recovering the metal materials of the gas generator from the melting furnace.
摘要翻译：一种用于从废弃汽车中轻松取出气体发生器并有效地从气体发生器回收金属材料的方法。该方法包括以下步骤：a）通过调节粉碎装置对安装有气囊装置的废弃汽车进行粉碎，使粉碎物的尺寸与气体发生器的尺寸基本相同，来自气囊装置的未熔化体，b）从废弃车辆的碎片中取出气体发生器，c）将取出的气体发生器装入熔炉中，d）从熔化中回收气体发生器的金属材料炉。

5. 发明申请

WO1992011246A1 NOVEL BENZODIAZEPINE DERIVATIVE 审中-公开
标题翻译：新的苯二甲酸衍生物
公开(公告)号：WO1992011246A1
公开(公告)日：1992-07-09
申请号：PCT/JP1991001720
申请日：1991-12-17
申请人： YAMANOUCHI PHARMACEUTICAL CO., LTD. , SATOH, Masato , KONDOH, Yutaka , OKAMOTO, Yoshinori , NISHIDA, Akito , HONDA, Kazuo , SAITO, Masayuki
发明人： YAMANOUCHI PHARMACEUTICAL CO., LTD.
IPC分类号： C07D243/24
CPC分类号： C07D401/06 , B65D83/0847 , B65H35/10 , B65H2701/11231 , C07D243/24 , C07D403/04 , C07D409/06
摘要： A novel benzodiazepine derivative represented by general formula (I), a pharmaceutically acceptable salt thereof, a pharmaceutical composition thereof, and a process for producing the same. In formula (I), R represents optionally substituted aryl, five-membered monocyclic group, six-membered monocyclic group or aromatic heterocyclic group comprising five-membered and six-membered rings; and R represents optionally substituted aryl. The compound (I) has a CCK-B receptor antagonism and an action of inhibiting pentagastrin-stimulated gastric secretion and hence is useful in treating and preventing the diseases wherein a CCK-B receptor and a gastrin receptor participate.
摘要翻译：由通式（I）表示的新型苯并二氮杂衍生物，其药学上可接受的盐，其药物组合物及其制备方法。在式（I）中，R 1表示任选取代的芳基，五元单环基，六元单环基或包含五元和六元环的芳族杂环基; 且R 2表示任选取代的芳基。化合物（I）具有CCK-B受体拮抗作用和抑制五肽胃泌素刺激的胃分泌的作用，因此可用于治疗和预防CCK-B受体和胃泌素受体参与的疾病。

6. 发明申请

WO2005047253A1 MELANOCORTIN RECEPTOR AGONISTS 审中-公开
标题翻译：梅兰康汀受体激动剂
公开(公告)号：WO2005047253A1
公开(公告)日：2005-05-26
申请号：PCT/KR2004/002930
申请日：2004-11-12
申请人： LG LIFE SCIENCES LTD. , YAMANOUCHI PHARMACEUTICAL CO., LTD. , LEE, Koo , PARK, Heui-Sul , AHN, In-Ae , YOO, Hyun-Ju , CHOI, Sung-Pil , CHOI, Deog-Young , YIM, Hyeon-Joo , KWON, O-Hwan , KONDOH, Yutaka
发明人： LEE, Koo , PARK, Heui-Sul , AHN, In-Ae , YOO, Hyun-Ju , CHOI, Sung-Pil , CHOI, Deog-Young , YIM, Hyeon-Joo , KWON, O-Hwan , KONDOH, Yutaka
IPC分类号： C07D211/34
CPC分类号： C07D401/04 , C07D211/22 , C07D211/26 , C07D211/32 , C07D211/34 , C07D211/58 , C07D401/14
摘要： The present invention relates a compound of formula 1, and pharmaceutically acceptable salt, hydrate, solvate, or isomer thereof effective as agonist of melanocortin receptor, and an agonistic composition of melanocortin receptor comprising the same as active ingredient.
摘要翻译：本发明涉及有效作为黑皮质素受体激动剂的式1化合物及其药学上可接受的盐，水合物，溶剂化物或异构体，以及包含与活性成分相同的黑皮质素受体激动剂组合物。

7. 发明申请

WO2005047251A1 MELANOCORTIN RECEPTOR AGONISTS 审中-公开
标题翻译：黑色素受体激动剂
公开(公告)号：WO2005047251A1
公开(公告)日：2005-05-26
申请号：PCT/KR2004/002929
申请日：2004-11-12
申请人： LG LIFE SCIENCES LTD. , YAMANOUCHI PHARMACEUTICAL CO., LTD. , LEE, Koo , PARK, Heui-Sul , AHN, In-Ae , YOO, Hyun-Ju , KIM, Jong-Yup , CHOI, Deog-Young , YIM, Hyeon-Joo , CHUNG, Kyung-Ha , SHIM, Dong-Sup , LEE, Sang-Kyun , KONDOH, Yutaka , HIRABAYASHI, Ryoji , HONDA, Shugo , KAKU, Hidetaka , SHISHIKURA, Jun-Ichi , ITO, Hiroyuki , KURAMA, Takeshi
发明人： LEE, Koo , PARK, Heui-Sul , AHN, In-Ae , YOO, Hyun-Ju , KIM, Jong-Yup , CHOI, Deog-Young , YIM, Hyeon-Joo , CHUNG, Kyung-Ha , SHIM, Dong-Sup , LEE, Sang-Kyun , KONDOH, Yutaka , HIRABAYASHI, Ryoji , HONDA, Shugo , KAKU, Hidetaka , SHISHIKURA, Jun-Ichi , ITO, Hiroyuki , KURAMA, Takeshi
IPC分类号： C07D207/16
CPC分类号： C04B35/632 , C07D205/04 , C07D207/14 , C07D211/58 , C07D401/12 , C07D403/12 , C07D405/12
摘要： The present invention relates a compound of formula 1, and pharmaceutically acceptable salt, hydrate, solvate, or isomer thereof effective as agonist of melanocortin receptor, and an agonistic composition of melanocortin receptor comprising the same as active ingredient.
摘要翻译：本发明涉及作为黑皮质素受体激动剂有效的式1化合物及其药学上可接受的盐，水合物，溶剂化物或异构体，以及包含其作为活性成分的黑皮质素受体激动剂组合物

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式