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61. 发明申请

US20120010195A1 IMIDAZOLE DERIVATIVES 审中-公开
标题翻译：咪唑衍生物
公开(公告)号：US20120010195A1
公开(公告)日：2012-01-12
申请号：US13256074
申请日：2010-02-08
申请人： Raphael Dumeunier , Clemens Lamberth , Stephan Trah
发明人： Raphael Dumeunier , Clemens Lamberth , Stephan Trah
IPC分类号： A01N43/46 , A01P3/00 , C07D403/04
CPC分类号： C07D233/88
摘要： The present invention relates to novel imidazole derivatives of formula (I) having microbiocidal, in particular fungicidal, activity, to processes for their preparation and intermediates used in their preparation, to agrochemical compositions comprising them and to the use in agriculture or horticulture for controlling or preventing infestation of plants, harvested food crops, seeds or non-living materials by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的新型咪唑衍生物，其具有杀微生物，特别是杀真菌活性，其制备方法和用于其制备的中间体，包含它们的农用化学组合物以及在农业或园艺中用于控制或通过植物病原微生物，优选真菌预防植物，收获的食物作物，种子或非生物材料的侵染。

62. 发明申请

US20110224252A1 NOVEL IMIDAZOLE DERIVATIVES 审中-公开
标题翻译：新咪唑衍生物
公开(公告)号：US20110224252A1
公开(公告)日：2011-09-15
申请号：US12739863
申请日：2008-10-24
申请人： Raphael Dumeunier , Clemens Lamberth , Stephan Trah , Sebastian Wendeborn
发明人： Raphael Dumeunier , Clemens Lamberth , Stephan Trah , Sebastian Wendeborn
IPC分类号： A01N43/42 , C07D233/68 , A01N43/50 , C07D401/04 , A01N43/40 , C07D409/04 , C07D401/02 , A01P3/00
CPC分类号： C07D401/04 , A01N43/50 , C07D233/28 , C07D401/14 , C07D409/14
摘要： The present invention relates to novel imidazole derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is halogen, C1-C4alkyl or C1-C4haloalkyl; R2 is an optionally substituted aryl or heteroaryl; R3 is halogen; R4 is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; R5 is halogen; X is N or C(R); and R is hydrogen, halogen, C1-C4alkyl, C1-C4haloalkyl, C1-C4alkoxy, C1-C4haloalkoxy or cyano; or an agrochemically usable salt form thereof; provided that when X is C(R), R2 cannot be an optionally substituted aryl.
摘要翻译：本发明涉及式（I）的新咪唑衍生物作为具有杀微生物活性，特别是杀真菌活性的活性成分：其中R1是卤素，C1-C4烷基或C1-C4卤代烷基; R2是任选取代的芳基或杂芳基; R3是卤素; R4是氢，卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基或氰基; R5是卤素; X是N或C（R）; 且R为氢，卤素，C 1 -C 4烷基，C 1 -C 4卤代烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷氧基或氰基; 或其农业化学可用的盐形式; 条件是当X是C（R）时，R 2不能是任选取代的芳基。

63. 发明申请

US20100113464A1 NOVEL PYRIDAZINE DERIVATIVES 审中-公开
标题翻译：新的吡咯烷酮衍生物
公开(公告)号：US20100113464A1
公开(公告)日：2010-05-06
申请号：US12373906
申请日：2007-07-16
申请人： Stephan Trah , Clemens Lamberth , Sebastian Volker Wendeborn
发明人： Stephan Trah , Clemens Lamberth , Sebastian Volker Wendeborn
IPC分类号： A61K31/50 , C07D401/04 , C07D405/04 , C07D409/04
CPC分类号： C07D401/04 , A01N43/58 , A01N43/60 , A01N43/78 , A01N43/80 , A01N43/82 , C07D403/04 , C07D405/04 , C07D407/04 , C07D409/04 , C07D413/04 , C07D417/04
摘要： The present invention relates to novel pyridazine derivatives of formula I as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is an optionally substituted heteroaryl; R3 is an optionally substituted aryl; and R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, (VCehaloalkoxy, hydroxy or cyano; or an agrochemically usable salt form thereof.
摘要翻译：本发明涉及式I的新的哒嗪衍生物作为具有杀微生物活性，特别是杀真菌活性的活性成分，其中R1是氢，C1-C6烷基，C1-C6卤代烷基或C3-C6环烷基; R2是任选取代的杂芳基; R3是任选取代的芳基; 和R 4是氢，卤素，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基，（C 5卤代烷氧基，羟基或氰基）或其农业上可用的盐形式。

64. 发明申请

US20100022526A1 PYRIDAZINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES 审中-公开
标题翻译：吡咯烷酮衍生物，其制备方法及其作为防腐剂的使用
公开(公告)号：US20100022526A1
公开(公告)日：2010-01-28
申请号：US12524096
申请日：2008-01-21
申请人： Clemens Lamberth , Sebastian Volker Wendeborn , Stephan Trah , Raphael Dumeunier
发明人： Clemens Lamberth , Sebastian Volker Wendeborn , Stephan Trah , Raphael Dumeunier
IPC分类号： A01N43/58 , C07D237/02 , A01N43/84 , A01P3/00
CPC分类号： C07D237/12 , A01N43/58 , C07D237/14 , C07D237/16 , C07D237/24 , C07D401/04 , C07D403/04 , C07D405/04 , C07D409/04
摘要： The present invention relates to compounds of formula (I) wherein R1, R2, R3 and R4 are as defined in claim 1, which are useful as fungicides.
摘要翻译：本发明涉及式（I）化合物，其中R 1，R 2，R 3和R 4如权利要求1中所定义，其可用作杀真菌剂。

65. 发明申请

US20100016339A1 FUNGICIDAL COMPOUNDS AND COMPOSITIONS 审中-公开
标题翻译：杀真菌化合物和组合物
公开(公告)号：US20100016339A1
公开(公告)日：2010-01-21
申请号：US12375839
申请日：2007-07-30
申请人： Jeremy Godwin , Stephan Trah , Clemens Lamberth , Sebastian Volker Wendeborn
发明人： Jeremy Godwin , Stephan Trah , Clemens Lamberth , Sebastian Volker Wendeborn
IPC分类号： A01N43/90 , C07D237/02 , A01N43/58 , A01P3/00
CPC分类号： C07D237/12 , A01N43/58
摘要： The present invention relates, inter alia, to a compound having the formula (I):—wherein (R)n is selected from the group consisting of 4-Br, 4-OCH2CH3, 4-OCH2CF3, 2-CH3-4-Cl, 2-CH3-4-OCH3, 2-CH3-4-OCF3, 2-F-4-Br, 2-F-4-CF3, 3-CH3-4-Br, 3-F-4-Cl, 3-F-4-CH3, 3-F-4-Br, 3-F-4-OCH3 and 3-F-4-F. The present invention further relates to a fungicidal composition comprising a compound having the formula (I)—and also to fungicidal compositions comprising compounds having the formula (II) and/or (III): Furthermore, the present invention relates to methods for controlling pathogenic organisms using the compositions.
摘要翻译：本发明特别涉及具有式（I）的化合物：其中（R）n选自4-Br，4-OCH2CH3,4-OCH2CF3,2-CH3-4-Cl ，2-CH3-4-OCH3,2-CH3-4-OCF3,2-F-4-Br，2-F-4-CF3,3-CH3-4-Br，3-F-4-Cl，3 -F-4-CH 3，3-F-4-Br，3-F-4-OCH 3和3-F-4-F。本发明还涉及包含具有式（I）的化合物的杀真菌组合物，还涉及包含具有式（II）和/或（III）的化合物的杀真菌组合物：此外，本发明涉及控制致病性的方法使用组合物的生物体。

66. 发明申请

US20090298816A1 PESTICIDES CONTAINING A BICYCLIC BISAMIDE STRUCTURE 失效
标题翻译：含有双相BISAMIDE结构的杀虫剂
公开(公告)号：US20090298816A1
公开(公告)日：2009-12-03
申请号：US12278807
申请日：2007-02-14
申请人： Olivier Loiseleur , Patricia Durieux , Stephan Trah , Andrew Edmunds , Andre Jeanguenat , Andre Stoller , David John Hughes
发明人： Olivier Loiseleur , Patricia Durieux , Stephan Trah , Andrew Edmunds , Andre Jeanguenat , Andre Stoller , David John Hughes
IPC分类号： A01N43/58 , C07D401/14 , A01N43/42 , A61K31/44 , C07D401/04 , A01N43/54 , C07D498/04
CPC分类号： C07D401/14 , A01N43/56 , A01N43/60 , A01N43/78 , A01N43/82 , A01N43/86 , C07D409/14 , C07D413/14 , C07D417/14
摘要： Compounds of formula (I), wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula I can be used as agrochemical active ingredients and can be prepared in a manner known per se.
摘要翻译：式（I）的化合物，其中取代基如权利要求1中所定义，以及式I化合物的农业化学上可接受的盐和所有立体异构体和互变异构形式可用作农业化学活性成分，并且可以以已知的方式制备 se。

67. 发明授权

US07332518B2 Carboxamides as fungicides in agriculture 失效
公开(公告)号：US07332518B2
公开(公告)日：2008-02-19
申请号：US10470069
申请日：2002-01-24
申请人： Harald Walter , Stephan Trah
发明人： Harald Walter , Stephan Trah
IPC分类号： A61K31/415 , A61K31/38 , C07D231/10 , C07D333/22 , C07D307/34
CPC分类号： C07D207/34 , C07D231/14 , C07D277/56
摘要： The invention concerns novel carboxamides of formula (I) wherein A is (A1), (A2), (A3), (A4), (A5); Q is (Q1), (Q2), (Q3), (Q4), (Q5), (Q6); R1 is CH2 R2, CH2CH═CHR2, CH═C═CHR2 or COR3; R2 is hydrogen, C1-C6alkyl, C1-C6haloalkyl, C2-C6alkenyl, C2-C6alkynyl, C3-C7cycloalkyl, COOC1-C4alkyl, COOC3-C6alkenyl, COOC3-C6alkynyl or CN; R3 is C1-C6alkyl, C1-C6alkyl substituted by halogen, C1-C6alkoxy or C1-C6haloalkoxy; or is C1-C6alkylthio, C1-C6haloalkylthio, C1-C6alkoxy, C1-C6haloalkoxy; C3-C6alkenyloxy or C3-C6haloalkenyloxy; C3-C6haloalkenyloxy; C3-C6alkynyloxy or C3-C6haloalkynyloxy; R4 is methyl, CF2Cl, CF3, CF2H, CFH2, Cl or Br, R5 is methyl, CF3, CH2OCH3 or CH2OCF3; R6 is hydrogen, fluoro, CF3 or methyl; R7 is hydrogen, methyl or halogen; and Z is phenyl, halophenyl, C5-C7cycloalkyl, C5-C7cycloalkyl substituted by C1-C3alkyl, C1C3haloalkyl or halogen, or a group of the form —CHR8—CH2—CHR9R10 wherein R8, R9 and R10 are independently of each other C1-C3alkyl. The novel compounds have plant-protective properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms, in particular fungi.

68. 发明申请

US20070281930A1 Novel Insecticides 有权
公开(公告)号：US20070281930A1
公开(公告)日：2007-12-06
申请号：US10598041
申请日：2005-03-02
申请人： David Hughes , James Peace , Suzanna Riley , Sally Russell , Joseph Swanborough , Roger Hall , Andre Jeanguenat , Olivier Loiseleur , Peter Renold , Stephan Trah , Jean Wenger
发明人： David Hughes , James Peace , Suzanna Riley , Sally Russell , Joseph Swanborough , Roger Hall , Andre Jeanguenat , Olivier Loiseleur , Peter Renold , Stephan Trah , Jean Wenger
IPC分类号： C07D401/04 , A01N43/42 , A01N43/56 , A01N43/80 , A01N43/84 , A01P7/00 , A01P7/02 , C07D498/00 , C07D413/00 , C07D215/38 , C07D265/12 , C07D275/02 , C07D275/04 , C07D401/00
CPC分类号： C07D401/04 , A01N37/46 , A01N43/40 , A01N43/56 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14 , C07D491/04 , C07D493/08 , C07D495/04 , C07D513/04
摘要： Compounds of the formula in which Z1 is an oxygen atom; or a sulfur atom; Z2 is an oxygen atom; or a sulfur atom; R1 is an aryl or heteroaryl group, which is unsubstituted or substituted; R2 is hydrogen; or an organic substituent; R3 is hydrogen; or an organic substituent; R4 is hydrogen; or an organic substituent; or R3 and R4, taken together, form, together with the nitrogen atom, to which they are attached, a ring, which is unsubstituted or substituted; R5 is hydrogen; or an unsubstituted or substituted alkyl group; or forms, taken together with R8 or with a monovalent substituent attached to that atom of R6, via which atom R6 is directly connected with the carbon atom, shown in the formula I, which carries R5, one additional bond; R6 and R7, taken together, form, together with the two carbon atoms, shown in the formula I, to which atoms they are attached, a bicyclic ring system, which ring system is carbocyclic or heterocyclic, which ring system is substituted, in the manner shown in the formula I, by the four substituents —N(R2)—C(=Z1)—R1, —C(=Z2)-N(R3)—R4, R5 and R8, and which ring system is optionally further substituted; and R8 is hydrogen; or an unsubstituted or substituted alkyl group; or forms, taken together with R5 or with a monovalent substituent attached to that atom of R7, via which atom R7 is directly connected with the carbon atom, shown in the formula I, which carries R8, one additional bond, and, where appropriate, tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.

69. 发明授权

US07109150B2 Trifluoromethylpyrrolecarboxamides and trifluoromethylpyrrolethioamides as fungicides 失效
标题翻译：三氟甲基吡咯酰胺和三氟甲基吡咯硫酰胺作为杀真菌剂
公开(公告)号：US07109150B2
公开(公告)日：2006-09-19
申请号：US10785836
申请日：2004-02-24
申请人： Harald Walter , Stephan Trah , Hermann Schneider
发明人： Harald Walter , Stephan Trah , Hermann Schneider
IPC分类号： A01N43/40 , C07D401/12
CPC分类号： C07D401/12 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/60 , A01N43/713 , A01N43/80 , A01N43/88 , C07D207/34 , C07D401/14 , C07D403/12 , C07D405/12 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12 , C07D417/14
摘要： Novel pyrrole derivatives of formula I wherein X is oxygen or sulfur; R1 is hydrogen, C1–C4alkyl unsubstituted or substituted, or halogen; R2 is C1–C4alkyl unsubstituted or substituted; and A is orthosubstituted aryl; orthosubstituted heteroaryl; bicycloaryl unsubstituted or substituted; or bicycloheteroaryl unsubstituted or substituted. The novel compounds have plant-protective properties and are suitable for protecting plants against infestations by phytopathogenic microorganisms.
摘要翻译：式I的新型吡咯衍生物，其中X是氧或硫; R 1是氢，C 1 -C 4烷基未取代或取代的或卤素; R 2是未取代或取代的C 1 -C 4烷基; 和A是邻位取代的芳基; 邻位取代的杂芳基; 未取代或取代的双环芳基; 或双环杂芳基未取代或取代。新化合物具有植物保护性质，适用于通过植物病原微生物保护植物免受侵袭。

70. 发明授权

US06646151B1 Process for the preparation of pesticides 失效
标题翻译：农药制备工艺
公开(公告)号：US06646151B1
公开(公告)日：2003-11-11
申请号：US09670147
申请日：2000-09-26
申请人： Saleem Farooq , Stephan Trah , Hugo Ziegler , René Zurflüh
发明人： Saleem Farooq , Stephan Trah , Hugo Ziegler , René Zurflüh
IPC分类号： C07C24904
CPC分类号： C07C249/12 , C07C251/48 , C07C251/60
摘要： The invention relates to a process for the preparation of compounds of the formula or, if appropriate, a tautomer thereof, in each case in the free form or in salt form, in which A, X, Y, Z, R2, R3, R4, R5, R7, R9 and n are as defined in claim 1 and the C═N double bond marked with E has the E configuration, which comprises a1) reacting either a compound of the formula (II) mentioned above with a compound of the formula (III) mentioned above, in which X1 is a leaving group, or a2) a compound of the formula (IV) mentioned above, if appropriate in the presence of a base, with a compound of the formula (V) mentioned above, or b1) reacting a compound of the formula (VI) mentioned above with a compound of the formula R7—A—X2 (VII), in which X2 is a leaving group, and either further reacting the compound thus obtainable, of the formula (IV), for example according to method a2), or b2) reacting it with hydroxylamine or a salt thereof, if appropriate in the presence of a basic or acid catalyst, and further reacting the compound thus obtainable, of the formula (II), for example according to method a1), or c) reacting a compound of the formula (VIII), mentioned above with a C1-C6alkyl nitrite and further reacting the compound thus obtainable, of the formula (VI), for example according to method b), the E isomers of the compounds of the formulae (II), (IV) and (VI), a process for their preparation and their use for the preparation of compounds of the formula (I).
摘要翻译：本发明涉及一种制备式的化合物的方法，如果合适，其合适的是其互变异构体，其各自为游离形式或盐形式，其中A，X，Y，Z，R 2，R 3，R 4， R5，R7，R9和n如权利要求1中所定义，并且用E标记的C = N双键具有E构型，其包括a）使上述式（II）的化合物与式（II） III），其中X1是离去基团，ora2）如果合适的话，在碱的存在下，上述式（Ⅳ）的化合物与上述式（Ⅴ）的化合物相同，反应1）使上述式（Ⅵ）化合物与式R7-A-X2（Ⅶ）化合物反应，其中X 2为离去基团，并进一步使由此得到的式（Ⅳ）化合物与根据方法a2）的示例，orb2）如果合适，在碱性或酸性催化剂存在下，使其与羟胺或其盐反应，以及进一步使由式（II）得到的化合物，例如按照方法a1）进行反应，或者使上述式（Ⅷ）化合物与亚硝酸C 1 -C 6烷基酯反应，并进一步使由此得到的化合物，式（Ⅵ）化合物的方法，例如根据方法b），式（II），（Ⅳ）和（Ⅵ）化合物的E异构体，其制备方法及其制备方法式（I）。

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