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1. 发明申请

WO2011101402A1 ISOXAZOLINE DERIVATIVES AS INSECTICIDES 审中-公开
标题翻译：异辛唑衍生物作为杀虫剂
公开(公告)号：WO2011101402A1
公开(公告)日：2011-08-25
申请号：PCT/EP2011/052336
申请日：2011-02-17
申请人： SYNGENTA PARTICIPATIONS AG , PITTERNA, Thomas , EL QACEMI, Myriem , CASSAYRE, Jérôme Yves , RENOLD, Peter , BOBOSIK, Vladimir
发明人： PITTERNA, Thomas , EL QACEMI, Myriem , CASSAYRE, Jérôme Yves , RENOLD, Peter , BOBOSIK, Vladimir
IPC分类号： C07D261/04 , C07D413/12 , A01N43/80
CPC分类号： C07D261/04 , A01N43/80 , C07D413/10 , C07D413/12 , C07D417/12
摘要： The present invention relates to compounds formula (I), wherein P is P1, P2, heterocyclyl or heterocyclyl substituted by one to five Z; and wherein A 1 , A 2 , A 3 , A 4 , G 1 , R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 17 , R 18 , R 19 and R 20 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.
摘要翻译：本发明涉及式（I）化合物，其中P为P1，P2，被1至5个Z取代的杂环基或杂环基; 并且其中A1，A2，A3，A4，G1，R1，R2，R3，R4，R5，R6，R17，R18，R19和R20如权利要求1中所定义; 或其盐或N-氧化物。此外，本发明涉及制备式（I）化合物的方法和中间体，其包含式（I）化合物的杀虫，杀螨，杀线虫和杀软体动物的组合物和使用式（I）化合物控制的方法昆虫，螨虫，线虫和软体动物害虫。

2. 发明申请

WO2011154555A1 PROCESS FOR THE PREPARATION OF DIHYDROPYRROLE DERIVATIVES 审中-公开
标题翻译：制备二氢衍生物衍生物的方法
公开(公告)号：WO2011154555A1
公开(公告)日：2011-12-15
申请号：PCT/EP2011/059823
申请日：2011-06-14
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , EL QACEMI, Myriem , SMITS, Helmars , CASSAYRE, Jérôme Yves , MULHOLLAND, Nicholas Phillip , RENOLD, Peter , GODINEAU, Edouard , PITTERNA, Thomas
发明人： EL QACEMI, Myriem , SMITS, Helmars , CASSAYRE, Jérôme Yves , MULHOLLAND, Nicholas Phillip , RENOLD, Peter , GODINEAU, Edouard , PITTERNA, Thomas
IPC分类号： C07D413/12 , C07D413/14 , C07D417/14 , A01N43/80 , C07D207/20 , C07D401/04 , C07D403/04 , C07D409/12 , C07D409/14 , A01N43/36 , A01N43/40 , C07C1/32
CPC分类号： C07D207/46 , A01N43/36 , C07D207/20 , C07D401/04 , C07D413/12 , C07D413/14 , C07D417/14
摘要： The present invention provides stereoselective processes for the preparation of compounds of formula (I) wherein P is phenyl, naphthyl, a 6-membered heteroaryl group containing one or two nitrogen atoms as ring members, or a 10-membered bicyclic heteroaryl group containing one or two nitrogen atoms as ring members, and wherein the phenyl, naphthyl and heteroaryl groups are optionally substituted; R 1 is chlorodifluoromethyl or trifluoromethyl; R 2 is optionally substituted aryl or optionally substituted heteroaryl; n is 0 or 1; including the process comprising (a-i) reacting a compound of formula II wherein P, R 1 and R 2 are as defined for the compound of formula I; with nitromethane in the presence a chiral catalyst to give a compound of formula III Wherein P, R 1 and R 2 are as defined for the compound of formula I; and (a-ii) reductively cyclising the compound of formula III to give the compound of formula I. The invention also provides intermediates useful for processes for the synthesis of compounds of formula (I).
摘要翻译：本发明提供了制备式（I）化合物的立体选择性方法，其中P是苯基，萘基，含有一个或两个氮原子作为环成员的6元杂芳基或含有一个或多个氮原子的10元双环杂芳基两个氮原子作为环成员，并且其中苯基，萘基和杂芳基任选被取代; R1是氯二氟甲基或三氟甲基; R2是任选取代的芳基或任选取代的杂芳基; n为0或1; 包括（a-i）使式II化合物与式Ⅰ化合物反应的方法，其中P，R 1和R 2如对式I化合物所定义; 在硝基甲烷中存在手性催化剂，得到式III化合物，其中P，R 1和R 2如式I化合物所定义; 和（a-ii）还原性环化式III化合物以得到式I化合物。本发明还提供了可用于合成式（I）化合物的方法的中间体。

3. 发明申请

WO2010084067A2 INSECTICIDAL COMPOUNDS 审中-公开
标题翻译：杀虫化合物
公开(公告)号：WO2010084067A2
公开(公告)日：2010-07-29
申请号：PCT/EP2010/050358
申请日：2010-01-13
申请人： SYNGENTA PARTICIPATIONS AG , RENOLD, Peter , CASSAYRE, Jérôme Yves , PABBA, Jagadish , EL QACEMI, Myriem , PITTERNA, Thomas , SYNGENTA LIMITED
发明人： RENOLD, Peter , CASSAYRE, Jérôme Yves , PABBA, Jagadish , EL QACEMI, Myriem , PITTERNA, Thomas
IPC分类号： C07D413/12 , C07D413/14 , C07D417/14 , A01N43/80
CPC分类号： C07D413/12 , A01N43/80 , A01N43/82 , C07D413/14 , C07D417/14
摘要： A compound of Formula (I): wherein A 1 , A 2 , A 3 , A 4 , A 5 , G 1 , R 1 , R 2 , R 3 and R 4 are as defined in claim 1; or a salt or N- oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising them and to methods of using them to combat and control insect, acarine, nematode and mollusc pests.
摘要翻译：式（I）的化合物：其中A 1，A 2，A 3，A 4，A 5，G 1，R 1，R 2，R R 3和R 4如权利要求1所定义; 或其盐或N-氧化物。此外，本发明涉及制备式（I）化合物的方法和中间体，包含它们的杀虫，杀螨，杀线虫和杀软体动物组合物，以及使用它们来对抗和控制昆虫，螨，线虫和软体动物害虫的方法。 / p>

4. 发明申请

WO2010025998A1 INSECTICIDAL COMPOUNDS 审中-公开
标题翻译：杀虫剂化合物
公开(公告)号：WO2010025998A1
公开(公告)日：2010-03-11
申请号：PCT/EP2009/059560
申请日：2009-07-24
申请人： SYNGENTA PARTICIPATIONS AG , RENOLD, Peter , CASSAYRE, Jérôme Yves , EL QACEMI, Myriem , PITTERNA, Thomas
发明人： RENOLD, Peter , CASSAYRE, Jérôme Yves , EL QACEMI, Myriem , PITTERNA, Thomas
IPC分类号： C07D413/12 , A01N43/80
CPC分类号： A01N43/80 , C07D413/12
摘要： A compoundof Formula (I): where A 1 , A 2 , A 3 , A 4 , A 5 , A 6 , G 1 , L, R 1 , R 2 , R 3 , R 4 , Y 1 , Y 2 and Y 3 are as defined in claim 1; or a saltor N-oxidethereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising compounds of formula (I) and to methods of using compounds of formula (I) to combat and control insect, acarine, mollusc and nematode pests.
摘要翻译：式（I）的化合物：其中A1，A2，A3，A4，A5，A6，G1，L，R1，R2，R3，R4，Y1，Y2和Y3如权利要求1所定义; 或一个盐氧化物N-氧化物。此外，本发明涉及制备式（I）化合物的方法和中间体，其包含式（I）化合物的杀虫，杀螨，杀软体动物和杀线虫组合物，以及使用式（I）化合物来对抗和控制的方法昆虫，螨虫，软体动物和线虫害虫。

5. 发明申请

WO2013026930A1 PROCESS FOR THE PREPARATION OF THIETANE DERIVATIVES 审中-公开
标题翻译：制备衍生物的方法
公开(公告)号：WO2013026930A1
公开(公告)日：2013-02-28
申请号：PCT/EP2012/066552
申请日：2012-08-24
申请人： SYNGENTA PARTICIPATIONS AG , CASSAYRE, Jérôme Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
发明人： CASSAYRE, Jérôme Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
IPC分类号： C07D331/04 , C07D409/12 , C07D413/12 , A01N43/36 , A01N43/80
CPC分类号： C07D413/12 , A01N43/36 , A01N43/80 , C07D331/04 , C07D409/12
摘要： The present invention relates to processes for the preparation of thietane derivatives of the formula (IA) and thietane derivatives of the formula (IB) wherein R 1 , R 2 , A 1 , A 2 , A 3 , A 4 , B, and n are as defined in the claims. The invention also relates to intermediates useful in the processes, as well as the compounds of formula (IA) and (IB) and their use as pesticides.
摘要翻译：本发明涉及制备式（IA）的硫杂环丁烷衍生物和式（IB）的硫杂环丁烷衍生物的方法，其中R1，R2，A1，A2，A3，A4，B和n如权利要求中所定义。本发明还涉及可用于该方法的中间体以及式（IA）和（IB）的化合物及其作为农药的用途。

6. 发明申请

WO2013026695A1 ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS 审中-公开
标题翻译：异辛唑衍生物作为杀虫剂化合物
公开(公告)号：WO2013026695A1
公开(公告)日：2013-02-28
申请号：PCT/EP2012/065421
申请日：2012-08-07
申请人： SYNGENTA PARTICIPATIONS AG , CASSAYRE, Jérôme Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
发明人： CASSAYRE, Jérôme Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
IPC分类号： C07D331/04 , C07D409/12 , C07D413/12 , A01N43/36 , A01N43/80
CPC分类号： C07D331/04 , A01N43/80 , C07D413/12
摘要： The present invention provides compounds of formula (I) wherein G 1 is oxygen; R 1 is hydrogen; R 2 is group P, L is a bond, methylene or ethylene; one of A 1 and A 2 is S, SO or SO 2 and the other is -C(R 4 )R 4 -; R 3 is hydrogen or methyl; each R 4 is independently hydrogen or methyl; Y 1 , Y 2 and Y 3 are independently CH or nitrogen; wherein no more than two of Y 1 , Y 2 and Y 3 are nitrogen and wherein Y 2 and Y 3 are not both nitrogen; R 5 is chloro, bromo, fluoro; X 2 is C-X 6 or nitrogen; Χ 1 , Χ 3 and X 6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X 1 , X 3 and X 6 are not hydrogen; X 4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also relates to methods of using the compounds to control insects, acarines, nematodes or molluscs, as well as intermediates usefor the the sysnthesis of the compounds.
摘要翻译：本发明提供其中G1是氧的式（I）化合物; R1是氢; R2为基团P，L为键，亚甲基或亚乙基; A1和A2之一是S，SO或SO2，另一个是-C（R 4）R 4 - ; R3是氢或甲基; 每个R 4独立地是氢或甲基; Y1，Y2和Y3独立地为CH或氮; 其中Y1，Y2和Y3中不超过两个是氮，并且其中Y2和Y3不都是氮; R5是氯，溴，氟; X2是C-X6或氮; α1，β3和X6独立地为氢，卤素或三卤代甲基，其中X1，X3和X6中的至少两个不是氢; X4是三氟甲基，二氟甲基或氯二氟甲基。本发明还涉及使用这些化合物来控制昆虫，螨虫，线虫或软体动物的方法，以及用于化合物系统的中间体。

7. 发明申请

WO2010108733A1 INSECTICIDAL COMPOUNDS 审中-公开
标题翻译：杀虫剂化合物
公开(公告)号：WO2010108733A1
公开(公告)日：2010-09-30
申请号：PCT/EP2010/052056
申请日：2010-02-18
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , RENOLD, Peter , PITTERNA, Thomas , CASSAYRE, Jérôme Yves , EL QACEMI, Myriem
发明人： RENOLD, Peter , PITTERNA, Thomas , CASSAYRE, Jérôme Yves , EL QACEMI, Myriem
IPC分类号： C07D413/12 , C07D409/12 , C07D413/14 , C07D417/14 , A01N43/80 , C07D261/02 , C07D417/12
CPC分类号： C07D413/12 , A01N43/80 , A01N43/82 , A01N43/84 , C07D261/02 , C07D417/12
摘要： A compound of formula (I): wherein A 1 , A 2 , A 3 , A 4 , G 1 , R 1 , R 2 , R 3 , R 4 , R 5a , R 5b and R 6 are as defined in claim 1; or a salt or N -oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.
摘要翻译：式（I）化合物：其中A1，A2，A3，A4，G1，R1，R2，R3，R4，R5a，R5b和R6如权利要求1中所定义; 或其盐或N-氧化物。此外，本发明涉及制备式（I）化合物的方法和中间体，其包含式（I）化合物的杀虫，杀螨，杀线虫和杀软体动物的组合物和使用式（I）化合物控制的方法昆虫，螨虫，线虫和软体动物害虫。

8. 发明申请

WO2013026933A1 ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS 审中-公开
标题翻译：异辛唑衍生物作为杀虫剂化合物
公开(公告)号：WO2013026933A1
公开(公告)日：2013-02-28
申请号：PCT/EP2012/066556
申请日：2012-08-24
申请人： SYNGENTA PARTICIPATIONS AG , CASSAYRE, Jérôme Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
发明人： CASSAYRE, Jérôme Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
IPC分类号： A01N43/50 , C07D331/04 , C07D409/12 , C07D413/12 , C07D413/14
CPC分类号： A01N43/80 , A01N37/42 , A01N37/50 , A01N43/20 , A01N43/40 , A01N43/42 , C07D413/12 , C07D413/14 , C07F7/1856
摘要： The present invention provides compounds of formula (I) wherein G 1 is oxygen; R 1 is hydrogen; R 2 is group (P) L is a bond, methylene or ethylene; one of A 1 and A 2 is S, SO or SO 2 and the other is -C(R 4 )R 4 -; R 3 is hydrogen or methyl; each R 4 is independently hydrogen or methyl; Y 2 and Y 3 are independently CH or nitrogen, wherein Y 2 and Y 3 are not both nitrogen; X 2 is C-X 6 or nitrogen; X 1 , X 3 and X 6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X 1 , X 3 and X 6 are not hydrogen; X 4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).
摘要翻译：本发明提供其中G1是氧的式（I）化合物; R1是氢; R2是基团（P），L是键，亚甲基或亚乙基; A1和A2之一是S，SO或SO2，另一个是-C（R 4）R 4 - ; R3是氢或甲基; 每个R 4独立地是氢或甲基; Y2和Y3独立地是CH或氮，其中Y2和Y3不都是氮; X2是C-X6或氮; X1，X3和X6独立地为氢，卤素或三卤代甲基，其中X 1，X 3和X 6中的至少两个不是氢; X4是三氟甲基，二氟甲基或氯二氟甲基。本发明还提供了可用于制备式（I）化合物的中间体，以及使用式（I）化合物控制昆虫，螨虫，线虫或软体动物的方法。

9. 发明申请

WO2013026929A1 DIHYDROPYRROLE DERIVATIVES AS INSECTICIDAL COMPOUNDS 审中-公开
标题翻译：作为杀虫剂化合物的二氢衍生物衍生物
公开(公告)号：WO2013026929A1
公开(公告)日：2013-02-28
申请号：PCT/EP2012/066550
申请日：2012-08-24
申请人： SYNGENTA PARTICIPATIONS AG , CASSAYRE, Jérôme Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
发明人： CASSAYRE, Jérôme Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
IPC分类号： C07D409/12 , A01N43/36
CPC分类号： C07D409/12
摘要： The present invention provides compounds of formula (I), wherein G 1 is oxygen; R 1 is hydrogen; R 2 is group P L is a bond, methylene or ethylene; one of A 1 and A 2 is S, SO or S0 2 and the other is -C(R 4 )R 4 - R 3 is hydrogen or methyl; each R 4 is independently hydrogen or methyl; Y 1 is C-R 6 , CH or nitrogen; Y 2 and Y 3 are independently CH or nitrogen; wherein no more than two of Y 1 , Y 2 and Y 3 are nitrogen and wherein Y 2 and Y 3 are not both nitrogen; R 5 is hydrogen, halogen, cyano, nitro, NH 2 , -C 2 alkyl, C 3 -C 2 haloalkyl, C 3 -C 5 cycloalkyl, C 3 - C 5 halocycloalkyl, C 1 -C 2 alkoxy, C 1 -C 2 haloalkoxy; R 6 together with R 5 forms a -CH=CH-CH=CH- bridge; X 2 is C-X 6 or nitrogen; X1, X 3 and X 6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X 1 , X 3 and X 6 are not hydrogen; X 4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula I, as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula I.
摘要翻译：本发明提供式（I）化合物，其中G1是氧; R1是氢; R2是基团P L是键，亚甲基或亚乙基; A1和A2之一是S，SO或SO 2，另一个是-C（R 4）R 4 -R 3是氢或甲基; 每个R 4独立地是氢或甲基; Y1是C-R6，CH或氮; Y2和Y3独立地是CH或氮; 其中Y1，Y2和Y3中不超过两个是氮，并且其中Y2和Y3不都是氮; R5是氢，卤素，氰基，硝基，NH2，-C2烷基，C3-C2卤代烷基，C3-C5环烷基，C3-C5卤代环烷基，C1-C2烷氧基，C1-C2卤代烷氧基; R6与R5一起形成-CH = CH-CH = CH-桥; X2是C-X6或氮; X1，X3和X6独立地为氢，卤素或三卤代甲基，其中X 1，X 3和X 6中的至少两个不是氢; X4是三氟甲基，二氟甲基或氯二氟甲基。本发明还提供了可用于制备式I化合物的中间体，以及使用式I化合物控制昆虫，螨虫，线虫或软体动物的方法。

10. 发明申请

WO2011101229A1 DIHYDROFURAN DERIVATIVES AS INSECTICIDAL COMPOUNDS 审中-公开
标题翻译： DIHYDROFURAN衍生物作为杀虫剂化合物
公开(公告)号：WO2011101229A1
公开(公告)日：2011-08-25
申请号：PCT/EP2011/051284
申请日：2011-01-31
申请人： SYNGENTA PARTICIPATIONS AG , EL QACEMI, Myriem , CASSAYRE, Jérôme Yves , TOUEG, Julie Clementine , RENOLD, Peter , PITTERNA, Thomas
发明人： EL QACEMI, Myriem , CASSAYRE, Jérôme Yves , TOUEG, Julie Clementine , RENOLD, Peter , PITTERNA, Thomas
IPC分类号： C07D307/20 , C07D307/28 , C07D307/30 , C07D307/32 , C07D307/58 , C07D405/04 , C07D405/10 , C07D407/12 , C07D409/12 , C07D409/14 , C07D413/12 , A01N43/08
CPC分类号： C07D307/28 , C07D307/52 , C07D307/58 , C07D405/04 , C07D405/10 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D413/12 , C07D413/14 , C07D417/14
摘要： The present invention relates to compounds of formula (I) wherein Q is Q1 or Q2 P is P1, heterocyclylor heterocyclyl substituted by one to five Z; and wherein A 1 , A 2 , A 3 , A 4 , G 1 , Y 1 , Z, R 1 , R 2 , R 3 and R 4 are as defined in claim 1; or a salt or N -oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.
摘要翻译：本发明涉及式（I）的化合物，其中Q是Q 1或Q 2是P 1，被1至5个Z取代的杂环基杂环基; 并且其中A1，A2，A3，A4，G1，Y1，Z，R1，R2，R3和R4如权利要求1中所定义; 或其盐或N-氧化物。此外，本发明涉及制备式（I）化合物的方法和中间体，其包含式（I）化合物的杀虫，杀螨，杀线虫和杀软体动物的组合物和使用式（I）化合物控制的方法昆虫，螨虫，线虫和软体动物害虫。

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