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    • 8. 发明申请
    • PALATABLE MICRO-CAPSULES
    • 可口微胶囊
    • WO2004045588A1
    • 2004-06-03
    • PCT/GB2003/004941
    • 2003-11-14
    • MICAP PLCNELSON, GordonDUCKHAM, Stephen, CraigROUND, Andrew, Edward
    • NELSON, GordonDUCKHAM, Stephen, CraigROUND, Andrew, Edward
    • A61K9/50
    • A61K9/5068
    • A formulation comprising at least one active or at least one ingredient, and a plurality of micro-capsules formed from a plurality of micro-organisms and having at least one flavouring encapsulated and passively retained within said micro-capsules, said flavouring not being a natural constituent of said micro-organisms, said micro-capsules having: (a) an at least substantially intact cell wall; and (b) an intact cell membrane; wherein said at least one active or said at least one ingredient is foul-tasting and said at least one flavouring masks, disguises or neutralises the foul-taste of said at least one active or said at least one ingredient, preventing a patient to whom said formulation is orally administered from tasting said foul-tasting active, or causing the flavour of said foul-tasting at least one active or ingredient to be reduced such that it is more palatable. Also disclosed are methods of manufacturing said formulations.
    • 包含至少一种活性成分和至少一种成分的制剂以及由多种微生物形成并具有至少一种包封并被动地保留在所述微胶囊内的调味剂的微胶囊,所述调味剂不是天然的 所述微型胶囊具有:(a)至少基本完整的细胞壁; 和(b)完整的细胞膜; 其中所述至少一种活性物质或所述至少一种成分是不合格的,并且所述至少一种调味剂掩盖,伪装或中和所述至少一种活性物质或所述至少一种成分的污点,防止所述至少一种活性物质或所述至少一种成分 制剂通过品尝所述污点活性物质口服施用,或引起所述污迹的风味至少一种活性成分或成分被还原,使得其更可口。 还公开了制造所述制剂的方法。