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1. 发明申请

WO2010128528A9 PIPERIDINE DERIVATIVES USEFUL FOR TREATMENT OF DIEBETES 审中-公开
标题翻译：用于治疗糖尿病的哌啶衍生物
公开(公告)号：WO2010128528A9
公开(公告)日：2011-03-03
申请号：PCT/IN2010000295
申请日：2010-05-06
申请人： TORRENT PHARMACEUTICALS LTD , DUTT CHAITANYA , CHAUTHAIWALE VIJAY , GUPTA RAMESH CHANDRA , PATEL MANISH , KOTECHA JIGNESH , LATAD SACHIN , ABRAHAM JAYA , SRIVASTAVA SANJAY , RODE MILIND , DESHPANDE SHAILESH , CHAUDHARY ANITA , KESARWANI AMIT KUMAR
发明人： DUTT CHAITANYA , CHAUTHAIWALE VIJAY , GUPTA RAMESH CHANDRA , PATEL MANISH , KOTECHA JIGNESH , LATAD SACHIN , ABRAHAM JAYA , SRIVASTAVA SANJAY , RODE MILIND , DESHPANDE SHAILESH , CHAUDHARY ANITA , KESARWANI AMIT KUMAR
IPC分类号： C07D211/56 , A61K31/4535 , A61K31/454 , A61P3/06 , C07D211/60 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04
CPC分类号： C07D409/06 , C07D211/56 , C07D211/60 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/14 , C07D417/04
摘要： The present invention relates to a new class of heterocyclic compounds and pharmaceutically acceptable salts thereof, process for preparing the same, pharmaceutical composition containing these compounds and to their use in treatment of diseases caused due to formation and accumulation of AGEs (Advanced Glycation endproducts). The compounds of the present invention are useful for the treatment of diabetic and aging-related complications caused by formation and accumulation of AGEs, such as neuropathy, nephropathy, microangiopathy, retinopathy, hypertension, heart failure, atherosclerosis, Alzheimer's disease & dermatological disorders.
摘要翻译：本发明涉及一类新的杂环化合物及其药学上可接受的盐，其制备方法，含有这些化合物的药物组合物及其用于治疗由于AGEs的形成和积累引起的疾病（高级糖化终产物）。本发明的化合物可用于治疗由AGEs的形成和积累引起的糖尿病和老化相关并发症，例如神经病，肾病，微血管病变，视网膜病变，高血压，心力衰竭，动脉粥样硬化，阿尔茨海默病和皮肤病。

2. 发明申请

WO2008134742A1 CUSTOMIZABLE MEDIA CHANNELS 审中-公开
标题翻译：可定制的媒体渠道
公开(公告)号：WO2008134742A1
公开(公告)日：2008-11-06
申请号：PCT/US2008/062058
申请日：2008-04-30
申请人： GOOGLE INC. , GOSSWEILER, III, Richard C. , SAHAMI, Mehran , PATEL, Manish G. , BLACKBURN, John , BROWN, David A. , GUPTA, Neha , TAYLOR, Thomas H.
发明人： GOSSWEILER, III, Richard C. , SAHAMI, Mehran , PATEL, Manish G. , BLACKBURN, John , BROWN, David A. , GUPTA, Neha , TAYLOR, Thomas H.
IPC分类号： G06F17/00 , H04N5/445 , H04N7/08
CPC分类号： H04N21/4532 , G06F3/0486 , G06F17/30864 , G06Q10/10 , H04H60/72 , H04N5/44543 , H04N7/17318 , H04N21/254 , H04N21/4147 , H04N21/4227 , H04N21/4334 , H04N21/4828 , H04N21/6543
摘要： A computer-implemented method includes receiving an identification of a media program from a broadcast channel on an electronic program guide for inclusion in a personalized channel, adding the identified program to a personalized channel at a first time, and adding one or more additional programs to the personalized channel at times other than the first time.
摘要翻译：计算机实现的方法包括从电子节目指南上的广播频道接收媒体节目的标识以包含在个性化频道中，将所识别的节目在第一时间添加到个性化频道，并将一个或多个附加节目添加到个性化频道在第一时间以外的时间。

3. 发明申请

WO2008134736A1 MOMENTARY ELECTRONIC PROGRAM GUIDE 审中-公开
标题翻译：动画电子节目指南
公开(公告)号：WO2008134736A1
公开(公告)日：2008-11-06
申请号：PCT/US2008/062050
申请日：2008-04-30
申请人： GOOGLE INC. , GOSSWEILER, Richard, C., III , SAHAMI, Mehran , BROWN, David, A. , PATEL, Manish, G. , BLACKBURN, John , TAYLOR, Thomas, H. , GUPTA, Neha
发明人： GOSSWEILER, Richard, C., III , SAHAMI, Mehran , BROWN, David, A. , PATEL, Manish, G. , BLACKBURN, John , TAYLOR, Thomas, H. , GUPTA, Neha
IPC分类号： H04N5/445 , G06F17/00 , H04N7/173
CPC分类号： H04N5/44543 , H04N21/44016 , H04N21/4532 , H04N21/472 , H04N21/4826
摘要： A computer-implemented method includes determining a time relative to a playing media program to insert a user notification, automatically generating a suggestion regarding a media program other than the playing media program to be presented to an audience member of the playing media program, providing, in a format for presentation on a user-related media player, the generated suggestion at the location in the playing media program, and causing the generation of a control that, when selected, performs an action related to the non-playing media program.
摘要翻译：计算机实现的方法包括：确定相对于播放媒体程序插入用户通知的时间，自动生成关于要呈现给播放媒体节目的观众的播放媒体节目之外的媒体节目的建议，以用于在用户相关的媒体播放器上呈现的格式，在播放媒体节目中的位置处产生的建议，并且产生当被选择时执行与非播放媒体节目有关的动作的控制。

4. 发明申请

WO2008083013A1 SYSTEM AND METHOD FOR DISPLAYING MULTIMEDIA EVENTS SCHEDULING INFORMATION 审中-公开
标题翻译：用于显示多媒体事件调度信息的系统和方法
公开(公告)号：WO2008083013A1
公开(公告)日：2008-07-10
申请号：PCT/US2007/088246
申请日：2007-12-19
申请人： GOOGLE INC. , GOSSWEILER, Richard, Carl, III. , BAUER, Marisa , BLACKBURN, John , BROWN, David, A. , GUPTA, Neha , HEILMAN, Timothy, Dharma , PATEL, Manish, Gordhan , REISS, David, Scott , SAHAMI, Mehran , SCOTT, Maricia , TAYLOR, Thomas, H. , TULL, Alice , WAGNER, Mark , ZHANG, Lucy, Congyun , ZIGMOND, Daniel, John
发明人： GOSSWEILER, Richard, Carl, III. , BAUER, Marisa , BLACKBURN, John , BROWN, David, A. , GUPTA, Neha , HEILMAN, Timothy, Dharma , PATEL, Manish, Gordhan , REISS, David, Scott , SAHAMI, Mehran , SCOTT, Maricia , TAYLOR, Thomas, H. , TULL, Alice , WAGNER, Mark , ZHANG, Lucy, Congyun , ZIGMOND, Daniel, John
IPC分类号： G06F17/30
CPC分类号： G06F17/3084 , G06F17/30817 , H04N5/44543 , H04N5/44591 , H04N7/163 , H04N21/4438 , H04N21/482 , H04N21/8453
摘要： A system for displaying information may include memory, one or more processors, and one or more modules stored in memory. The one or more modules are configured for execution by the one or more processors and may include instructions for: presenting a subset of a collection of data on a first grid having a first axis corresponding to units of time and a second axis, the collection of data comprising data representing time-bounded events; presenting a second grid having, first and second axes corresponding to the first and second axes of the first grid, the second grid corresponding to a larger portion of the collection of data than the subset presented on the first grid; and presenting a user moveable window for selecting a portion of the second grid, and selecting the subset presented on the first grid in accordance with a current position of the window.
摘要翻译：用于显示信息的系统可以包括存储器，一个或多个处理器以及存储在存储器中的一个或多个模块。一个或多个模块被配置为由一个或多个处理器执行，并且可以包括以下指令：用于在具有对应于时间单位和第二轴的第一轴线的第一网格上呈现数据集合的子集，数据包括表示时间有限事件的数据; 呈现第二网格，具有对应于第一网格的第一和第二轴的第一和第二轴，第二网格对应于数据集合的大部分，而不是呈现在第一网格上的子集; 以及呈现用户可移动窗口，用于选择第二格子的一部分，以及根据窗口的当前位置选择呈现在第一格栅上的子集。

5. 发明申请

WO2008055317A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PROSTATE CANCER 审中-公开
标题翻译：用于治疗前列腺癌的组合物和方法
公开(公告)号：WO2008055317A1
公开(公告)日：2008-05-15
申请号：PCT/AU2007/001726
申请日：2007-11-09
申请人： THE UNIVERSITY OF SYDNEY , DONG, Qihan , PATEL, Manish
发明人： DONG, Qihan , PATEL, Manish
IPC分类号： A61K31/192 , A61K31/427 , A61P35/00 , A61K31/353 , A61K31/635
CPC分类号： A61K31/192 , A61K31/353 , A61K31/427 , A61K31/635 , A61K45/06 , A61K2300/00
摘要： A pharmaceutical composition for inhibiting the proliferation of prostate cancer cells, said composition comprising a synergistic combination of a therapeutically effective amount of at least one COX inhibitor, and either one or both of: (a) at least one LOX inhibitor (b) at least one cPLA 2 -α inhibitor.
摘要翻译：一种用于抑制前列腺癌细胞增殖的药物组合物，所述组合物包含治疗有效量的至少一种COX抑制剂与以下之一或两者的协同组合：（a）至少一种LOX抑制剂（b）至少一个cPLA 2 -a抑制剂。

6. 发明申请

WO2008007388A1 NOVEL PROCESS FOR THE PREPARATION OF TELITHROMYCIN 审中-公开
标题翻译：用于制备紫杉醇的新方法
公开(公告)号：WO2008007388A1
公开(公告)日：2008-01-17
申请号：PCT/IN2006/000488
申请日：2006-12-08
申请人： ALEMBIC LIMITED , DESHPANDE, Pandurang, Balwant , LUTHRA, Parven, Kumar , PATEL, Manish, Kanchanbbai , DHAMELIYA, Kalpesh, Haribhai
发明人： DESHPANDE, Pandurang, Balwant , LUTHRA, Parven, Kumar , PATEL, Manish, Kanchanbbai , DHAMELIYA, Kalpesh, Haribhai
IPC分类号： C07H17/00
CPC分类号： C07H17/00
摘要： The present invention relates to the process for the preparation of compounds of formula (I) or its pharmaceutically acceptable salts; wherein R is formula (A).
摘要翻译：本发明涉及制备式（I）化合物或其药学上可接受的盐的方法; 其中R是式（A）。

7. 发明申请

WO2007116240A1 AN IMPROVED PROCESS FOR THE MANUFACTURE OF MONTELUKAST SODIUM 审中-公开
标题翻译：改进的MONTELUKAST SODIUM制造工艺
公开(公告)号：WO2007116240A1
公开(公告)日：2007-10-18
申请号：PCT/IB2006/002690
申请日：2006-09-28
申请人： GLADE ORGANICS PRIVATE LIMITED , CHAWLA, Harmander, Pal, Singh , CHOWDHARY, Anil, Shankar , PATEL, Ajay, Mangubhai , PATEL, Manish, Popatlal
发明人： CHAWLA, Harmander, Pal, Singh , CHOWDHARY, Anil, Shankar , PATEL, Ajay, Mangubhai , PATEL, Manish, Popatlal
IPC分类号： C07D215/18
CPC分类号： C07D215/18
摘要： Process for the manufacture of 1-[[[(1R)-1-[3-[(1E)-2-(7-chloro-2-quinolinyl)ethenyl]phenyl]-3-[2-(1-hydroxy-1-methylethyl)phenyl]propyl]thio]methyl]cyclopropane acetic acid, sodium salt [montelukast sodium (I)] consisting of: i. Converting methyl 1-(mercaptomethyl)-cyclopropaneacetate to a metal salt (X) using a metal hydroxide, ii. Subjecting the metal salt (X) to monometallation to provide a dimetallide (XI). iii. Converting a diol of formula (II) to a mesylate of formula (III) and reacting (III) in situ with (XI) affordin the metal salt of 1-[[[(1R)-1-[3-[(1E)-2-(7-chloro-2-quinolinyl)ethenyl]phenyl]-3-[2-(1-hydroxy-1-methylethyl)phenyl]propyl]thio]methyl]cyclopropane acetic acid. iv. Reacting the metal salt in-situ with a base and purifying to afford an amine salt (XII). v. Treating (XII) with a sodium base and precipitating out montelukast sodium (I).
摘要翻译：制备1 - [[（1R）-1- [3 - [（1E）-2-（7-氯-2-喹啉基）乙烯基]苯基] -3- [2-（1-羟基 - 1-甲基乙基）苯基]丙基]硫基]甲基]环丙烷乙酸钠盐[孟鲁司特钠（I）]由以下组成：i。使用金属氢氧化物将1-（巯基甲基） - 环丙烷甲酸甲酯转化为金属盐（X），ii。使金属盐（X）进行单金属化以提供二叠氮化物（XI）。 III。将式（II）的二醇转化为式（III）的甲磺酸酯并与（XI）原位反应，得到1 - [[（1R）-1- [3 - [（1E） -2-（7-氯-2-喹啉基）乙烯基]苯基] -3- [2-（1-羟基-1-甲基乙基）苯基]丙基]硫基]甲基]环丙烷乙酸。 IV。用碱反应金属盐并纯化得到胺盐（Ⅻ）。 v。用钠碱处理（XII）并沉淀孟鲁司特钠（I）。

8. 发明申请

WO2007039914A3 NOVEL POLYMORPHS OF TELITHROMYCIN 审中-公开
标题翻译： TELITHROMYCIN的新型多聚体
公开(公告)号：WO2007039914A3
公开(公告)日：2007-06-21
申请号：PCT/IN2006000242
申请日：2006-07-10
申请人： ALEMBIC LTD , DESHPANDE PANDURANG BALWANT , LUTHRA PARVEN KUMAR , PATEL MANISH KANCHANBHAI , DAVADRA MAHESH PRAVINCHANDRA
发明人： DESHPANDE PANDURANG BALWANT , LUTHRA PARVEN KUMAR , PATEL MANISH KANCHANBHAI , DAVADRA MAHESH PRAVINCHANDRA
IPC分类号： C07H17/08
CPC分类号： C07H17/08
摘要： The present invention relates to novel polymorphs of Telithromycin designated as Form I, II and III and its process for preparation. Also it provides Telithromycin with at least 99% purity.
摘要翻译：本发明涉及被称为I型，II型和III型的泰利霉素的新型多晶型物及其制备方法。此外，它提供至少99％纯度的泰利霉素。

9. 发明申请

WO2007039914A2 NOVEL POLYMORPHS OF ERYTHROMYCIN COMPOUND 审中-公开
标题翻译：红霉素化合物的新型聚合物
公开(公告)号：WO2007039914A2
公开(公告)日：2007-04-12
申请号：PCT/IN2006/000242
申请日：2006-07-10
申请人： ALEMBIC LIMITED , DESHPANDE, Pandurang, Balwant , LUTHRA, Parven, Kumar , PATEL, Manish, Kanchanbhai , DAVADRA, Mahesh, Pravinchandra
发明人： DESHPANDE, Pandurang, Balwant , LUTHRA, Parven, Kumar , PATEL, Manish, Kanchanbhai , DAVADRA, Mahesh, Pravinchandra
IPC分类号： C07H17/08
CPC分类号： C07H17/08
摘要： The present invention relates to novel polymorphs of Telithromycin designated as Form I, II and III and its process for preparation. Also it provides Telithromycin with at least 99% purity.
摘要翻译：本发明涉及被称为I型，II型和III型的泰利霉素的新型多晶型物及其制备方法。此外，它提供至少99％纯度的泰利霉素。

10. 发明申请

WO2005105821A3 PROCESS FOR THE PREPARATION OF TELITHROMYCIN 审中-公开
标题翻译：制备紫杉醇的方法
公开(公告)号：WO2005105821A3
公开(公告)日：2006-04-27
申请号：PCT/IN2005000125
申请日：2005-04-25
申请人： ALEMBIC LTD , SOHANI SUHAS , DEODHAR MANDAR , PATEL NISHANT , PATEL MANISH , DAVADRA MAHESH , KANSAL VINODKUMAR
发明人： SOHANI SUHAS , DEODHAR MANDAR , PATEL NISHANT , PATEL MANISH , DAVADRA MAHESH , KANSAL VINODKUMAR
IPC分类号： C07H17/00 , C07H17/08
CPC分类号： C07H17/00 , C07H17/08
摘要： The present invention relates to the process for the preparation of compounds of formula (I) or its pharmaceutically acceptable salts.The novel compounds (i) 10,11-Anhydro-2',4"-di-O-benzoyl-12-O-imidazolylcarbonyl-6-O-methylerythromycin A of formula (Xa) (ii) 2',4"-di-O-benzoyl-11-amino-11-N-[4-[4-(3-pyridyl)imidazol-1-yl]butyl]-11-deoxy-6-O- methylerythromycin A 11,12-cyclic carbamate of formula (XIa) (iii) 2'-O-benzoyl-11-amino-11-N-[4-[4-(3-pyridyl)imidazol-1-yl]butyl]-11-deoxy-5-O-desosaminyl- 6-O-methylerythronolide A 11,12-cyclic carbamate of formula (XIIa) (iv) 2'-benzoyl-11-amino-11-N-[4-[4-(3-pyridyl)imidazol-1-yl]butyl]-11-deoxy-5-O- desosaminyl-6-O-methylerythronolide A 11,12-cyclic carbamate of formula (XIIa) and their use as intermediates in formation of compound of Formula (I). Also the process of preparation of compound of formula (XIIIa).
摘要翻译：本发明涉及制备式（I）化合物或其药学上可接受的盐的方法。新化合物（i）10,11-脱氢-2'，4“ - 二-O-苯甲酰基-12-O （Xa）（ⅱ）2'，4“ - 二-O-苯甲酰基-11-氨基-11-N- [4- [4-（3-吡啶基）咪唑-2-基] - 咪唑基羰基-6-O-甲基红霉素A 哌啶-1-基]丁基] -11-脱氧-6-O-甲基红霉素将式（XIa）（iii）的11,12-环状氨基甲酸酯2'-O-苯甲酰基-11-氨基-11-N- [4- [ 4-（3-吡啶基）咪唑-1-基]丁基] -11-脱氧-5-O-二十一烷基-6-O-甲基红霉内酯将式（Ⅻa）（ⅳ）的11,12-环状氨基甲酸酯（ⅳ） -11-氨基-11-N- [4- [4-（3-吡啶基）咪唑-1-基]丁基] -11-脱氧-5-O-氨基甲酰基-6-O-甲基红霉素A 11,12-环（XIIa）的氨基甲酸酯及其作为形成式（I）化合物的中间体的用途。还有式（XIIIa）化合物的制备方法。

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