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    • 1. 发明申请
    • PYRIDYLOXYALKANOIC ACID AMIDE DERIVATIVES USEFUL AS FUNGICIDES
    • 作为杀菌剂有用的吡咯烷酮酸酰胺衍生物
    • WO2003048128A1
    • 2003-06-12
    • PCT/GB2002/005303
    • 2002-11-25
    • SYNGENTA LIMITEDSYNGENTA PARTICIPATIONS AGWHITTINGHAM, William, GuyLAWSON, Kevin, RobertWORTHINGTON, Paul, AnthonyRUSSELL, Charles, AdamSALMON, RogerMAY, Leslie, FrancisJORG, MarioPACHLATKO, Johannes, Paul
    • WHITTINGHAM, William, GuyLAWSON, Kevin, RobertWORTHINGTON, Paul, AnthonyRUSSELL, Charles, AdamSALMON, RogerMAY, Leslie, FrancisJORG, MarioPACHLATKO, Johannes, Paul
    • C07D213/65
    • C07D213/70A01N43/40C07D213/65C07D213/68C07D213/80C07D213/82C07D213/85
    • Fungicidal compounds of the general formula (I): wherein X and Y are independently H, halo, C 1-8 alkyl, C 3-6 cycloalkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 alkoxy, C 1-8 alkylthio, nitro, amino, mono- or di-(C 1-6 )alkylamino, mono- or di-(C 2-6 )alkenylamino, mono- or di-(C 2-6 )alkynylamino, formylamino, C 1-4 alkyl(formyl)amino, C 1-4 alkylcarbonylamino, C 1-4 alkyl(C 1-4 alkylcarbonyl)amino, cyano, formyl, C 1-4 alkylcarbonyl, C 1-4 alkoxycarbonyl, aminocarbonyl, mono- or di-(C 1-4 )alkylaminocarbonyl, carboxy, C 1-4 alkylcarbonyloxy, aryl(C 1-4 )alkylcarbonyloxy, C 1-4 alkylsulphinyl, C 1-4 alkylsulphonyl, C 1-4 alkylsulphonyloxy, aryl, heteroaryl, aryloxy, arylthio, heteroaryloxy or heteroarylthio wherein any of the foregoing alkyl, cycloalkyl, alkenyl, alkynyl, aryl, heteroaryl, groups or moieties are optionally substituted; R 1 is phenyl, cyano, C 1-4 alkyl, C 2-4 alkenyl or C 2-4 alkynyl in which the alkyl, alkenyl and alkynyl groups are optionally substituted on their terminal carbon atom with one, two or three halogen atoms, with a cyano group, with a C 1-4 alkylcarbonyl group, with a C 1-4 alkoxycarbonyl group or with a hydroxy group, or R 1 is alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl or alkylsulphonylalkyl in which the total number of carbon atoms is 2 or 3; R 2 is H, C 1-4 alkyl, C 1-4 alkoxymethyl or benzyloxymethyl in which the phenyl ring of the benzyl moiety is optionally substituted with C 1-4 alkoxy; R 3 and R 4 are independently H, C 1-3 alkyl, C 2-3 alkenyl or C 2-3 alkynyl provided that both are not H and that when both are other than H their combined total of carbon atoms does not exceed 4, or R 3 and R 4 join with the carbon atom to which they are attached to form a 3 or 4 membered carbocyclic ring optionally containing one O, S or N atom and optionally substituted with halo or C 1-4 alkyl; and R 5 is halo, C 1-4 alkyl or C 3-4 cycloalkyl in which the alkyl or cycloalkyl group is optionally substituted with halo, hydroxy, C 1-6 alkoxy, C 1-6 alkylthio, cyano, C 1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di(C 1-4 )alkylaminocarbonyloxy, or tri(C 1-4 )alkylsilyloxy. The compounds and compositions containing them are especially useful for combating fungal infections of plants.
    • 通式(I)的杀真菌化合物:其中X和Y独立地为H,卤素,C 1-8烷基,C 3-6环烷基,C 2-8链烯基,C 2-8 炔基,C> 1-8 <烷氧基,C 1-8烷基硫基,硝基,氨基,单 - 或二 - (C 1-6)烷基氨基,单 - 或二 - (C 2-6) 链烯基氨基,单 - 或二 - (C 2-6)炔基氨基,甲酰氨基,C 1-4烷基(甲酰基)氨基,C 1-4烷基羰基氨基,C 1-4烷基(C 1 -4 <烷基羰基)氨基,氰基,甲酰基,C 1-4烷基羰基,C 1-4烷氧基羰基,氨基羰基,一或二 - (C 1-4)烷基氨基羰基,羧基, 4 <烷基羰基氧基,芳基(C 1-4)烷基羰基氧基,C 1-4烷基亚磺酰基,C 1-4烷基磺酰基,C 1-4烷基磺酰氧基,芳基,杂芳基,芳氧基,芳硫基,杂芳氧基或杂芳硫基 其中任何前述烷基,环烷基,烯基,炔基,芳基,杂芳基,基团或部分任选被取代; R 1是苯基,氰基,C 1-4烷基,C 2-4链烯基或C 2-4炔基,其中烷基,烯基和炔基在其末端碳原子上任选被一个,两个或三个卤素原子取代, 具有C 1-4烷基羰基,C 1-4烷氧基羰基或羟基的氰基,或者R 1是烷基烷基或烷基磺酰基烷基,其中总碳原子数为2或3的烷氧基烷基,烷硫基烷基,烷基亚磺酰基烷基或烷基磺酰基烷基 ; R 2是H,C 1-4烷基,C 1-4烷氧基甲基或苄氧基甲基,其中苄基部分的苯环任选被C 1-4烷氧基取代; R 3和R 4独立地是H,C 1-3烷基,C 2-3烯基或C 2-3炔基,条件是两者都不是H,当两者都不是H时,它们的总碳原子数不超过 4或R 3和R 4与它们所连接的碳原子一起形成任选含有一个O,S或N原子并任选被卤素或C 1-4烷基取代的3或4元碳环 ; 羟基,C 1-6烷氧基,C 1-6烷硫基,氰基,C 1-4烷基羰基氧基,氨基羰基氧基,C 1-4烷氧基,C 1-4烷氧基, ,单或二(C 1-4)烷基氨基羰基氧基或三(C 1-4)烷基甲硅烷氧基。 含有它们的化合物和组合物特别可用于防治植物的真菌感染。