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1. 发明申请

WO1991011443A1 PROCESS FOR PRODUCING ISOXAZOLE DERIVATIVE 审中-公开
标题翻译：生产异噻唑衍生物的方法
公开(公告)号：WO1991011443A1
公开(公告)日：1991-08-08
申请号：PCT/JP1991000064
申请日：1991-01-22
申请人： TAIHO PHARMACEUTICAL COMPANY, LIMITED , TANAKA, Motoaki , HAGIWARA, Yuichi , KAJITANI, Makoto , YASUMOTO, Mitsugi
发明人： TAIHO PHARMACEUTICAL COMPANY, LIMITED
IPC分类号： C07D261/08
CPC分类号： C07D261/08
摘要： A process for producing an isoxazole derivative of general formula (II), wherein R?1 and R2¿ may be the same or different from each other and each represents hydrogen or lower alkoxy, and R3 represents cyano or alkoxycarbonyl, by oxidizing an α,β-unsaturated ketoxime derivative of general formula (I), wherein R?1, R2 and R3¿ are as defined above. The isoxazole derivative (II) is useful as an intermediate for the production of (3,4-diaryl-isoxazol-5-yl)acetic acid derivatives useful as an antiinflammatory, analgesic and antipyretic.

2. 发明申请

WO1991007374A1 'alpha','beta'-UNSATURATED KETONE AND KETOXIME DERIVATIVE 审中-公开
标题翻译：（ALPHA），（BETA） - 饱和酮和酮替代衍生物
公开(公告)号：WO1991007374A1
公开(公告)日：1991-05-30
申请号：PCT/JP1990001512
申请日：1990-11-19
申请人： TAIHO PHARMACEUTICAL COMPANY, LIMITED , TANAKA, Motoaki , HAGIWARA, Yuichi , KAJITANI, Makoto , YASUMOTO, Mitsugi
发明人： TAIHO PHARMACEUTICAL COMPANY, LIMITED
IPC分类号： C07C69/738
CPC分类号： C07C69/738 , C07C251/48 , C07C255/40 , C07C255/64
摘要： An α,β-unsaturated ketone and ketoxime derivatives thereof represented by general formula (I), wherein Y is an oxygen atom or a hydroxyimino group, Z is a cyano group or an alkoxycarbonyl group, R?1 and R2¿ which may be the same or different are each a hydrogen atom or a lower alkoxy group. They are useful as an intermediate for a (3,4-diarylisoxazol-5-yl)acetate derivative useful as an anti-inflammatory agent, an analgesic and an antifebrile.

3. 发明申请

WO1997026242A1 3-(BIS-SUBSTITUTED-PHENYLMETHYLENE)OXINDOLE DERIVATIVES 审中-公开
标题翻译： 3-（双 - 取代 - 苯基甲基）氧化衍生物
公开(公告)号：WO1997026242A1
公开(公告)日：1997-07-24
申请号：PCT/JP1997000066
申请日：1997-01-16
申请人： TAIHO PHARMACEUTICAL CO., LTD. , SATO, Atsushi , ASAO, Tetsuji , HAGIWARA, Yuichi , KITADE, Makoto , YAMAZAKI, Yasundo
发明人： TAIHO PHARMACEUTICAL CO., LTD.
IPC分类号： C07D209/34
CPC分类号： C07D401/06 , C07D209/34 , C07D401/14 , C07D471/04
摘要： Oxindole derivatives represented by general formula (1) and drugs containing the same, wherein R represents methyl or methoxy. Because of having excellent effects of inhibiting granulation with little hepatic toxicity, these compounds are useful as drugs and usable in the prevention and treatmeent of articular rheumatism, arterial sclerosis, hepatic cirrhosis, arthrosis deformans, psoriasis, gout, nephritis, angiitis, inflammatory enteral diseases (ulcerative colitis, Crohn's disease), bronchitis, arthritis, chronic granulomatous disease, etc.
摘要翻译：由通式（1）表示的羟吲哚衍生物和含有它们的药物，其中R表示甲基或甲氧基。由于具有抑制肉毒毒性极小的效果，这些化合物可用作药物，可用于预防和治疗关节风湿病，动脉硬化，肝硬化，变形性关节炎，牛皮癣，痛风，肾炎，血管炎，炎性肠内疾病（溃疡性结肠炎，克罗恩病），支气管炎，关节炎，慢性肉芽肿病等

4. 发明申请

WO1997025986A1 INTIMAL THICKENING INHIBITORS 审中-公开
标题翻译：最终增稠抑制剂
公开(公告)号：WO1997025986A1
公开(公告)日：1997-07-24
申请号：PCT/JP1997000065
申请日：1997-01-16
申请人： TAIHO PHARMACEUTICAL CO., LTD. , SATO, Atsushi , ASAO, Tetsuji , HAGIWARA, Yuichi , KITADE, Makoto , YAMAZAKI, Yasundo
发明人： TAIHO PHARMACEUTICAL CO., LTD.
IPC分类号： A61K31/40
CPC分类号： C07D401/06 , C07D209/34 , C07D401/14 , C07D471/04
摘要： Intimal thickening inhibitors containing as the active ingredient oxyindole derivatives represented by general formula (1) or salts thereof (wherein R represents hydrogen, phenyl optionally substituted by lower alkyl, lower alkoxy, lower alkylaminoalkoxy, hydroxy, amino, lower alkylamino or halogeno, or pyridyl optionally substituted by lower alkyl, lower alkoxy, lower alkylaminoalkoxy, hydroxy, amino, lower alkylamino, halogeno, lower alkoxycarbonyl or carboxy; R represents optionally substituted phenyl, or pyridyl optionally substituted by lower alkyl, lower alkoxy, lower alkylamino-alkoxy, hydroxy, amino, lower alkylamino, halogeno, lower alkoxycarbonyl or carboxy; R represents hydrogen, optionally substituted lower alkyl, benzyl or benzenesulfonyl, or acyl; R represents hydrogen, lower alkoxy, halogeno, amino, lower alkylamino, carboxy, lower alkoxycarbonyl, optionally substituted phenylcarbamoyl, or trifluoromethyl; X represents CH or N; n represents the number of the substituents ranging from 0 to 4; and the double line composed of dotted and solid lines means that this bond is either a single or a double bond). These drugs show excellent effects of inhibiting intimal thickening and thus useful in preventing, treating and relieving proliferative vascular lesions such as vascular reconstriction after percutaneous transluminal coronary recanalization, arterial sclerosis, peripheral embolism and angiitis.
摘要翻译：含有作为活性成分的由通式（1）表示的氧吲哚衍生物或其盐（其中R 1表示氢，任选被低级烷基，低级烷氧基，低级烷基氨基烷氧基，羟基，氨基，低级烷基氨基或卤素取代的苯基）的内增稠抑制剂或任选被低级烷基，低级烷氧基，低级烷基氨基烷氧基，羟基，氨基，低级烷基氨基，卤代，低级烷氧基羰基或羧基取代的吡啶基; R 2表示任选取代的苯基，或任选被低级烷基，低级烷氧基，低级烷基氨基 - 烷氧基，羟基，氨基，低级烷基氨基，卤代，低级烷氧基羰基或羧基; R 3表示氢，任选取代的低级烷基，苄基或苯磺酰基或酰基; R 4表示氢，低级烷氧基，，低级烷基氨基，羧基，低级烷氧基羰基，任选取代的苯基氨基甲酰基或三氟甲基; X表示CH或N; n表示取代基为0至4; 并且由虚线和实线组成的双线意味着该键是单键或双键）。这些药物显示出优异的抑制内膜增厚的效果，因此可用于预防，治疗和缓解经皮冠状动脉冠状动脉再通，动脉硬化，周围栓塞和血管炎等增殖性血管病变如血管再狭窄。

5. 发明申请

WO1995025387A1 TRANSCEIVER WITH ANTENNA 审中-公开
标题翻译：天线收发器
公开(公告)号：WO1995025387A1
公开(公告)日：1995-09-21
申请号：PCT/JP1994001621
申请日：1994-09-29
申请人： FUJITSU LIMITED , MINOWA, Yoshiaki , KUMAHARA, Kazuo , HAGIWARA, Yuichi , KOBAYASHI, Toshimitsu , KANEKO, Masahiko
发明人： FUJITSU LIMITED
IPC分类号： H04B01/38
CPC分类号： H04B1/38 , H01Q13/00 , H01Q19/13 , H01Q23/00
摘要： A small and light transceiver with an antenna, which is mainly installed outdoors, used for transmission and reception of radio signals, and manufactured from a small number of parts by a process of reduced man-hours. The transceiver is provided with an enclosure (5) having an opening (5B) in one end face and an antenna fitting surface (5A) on the other end face and incorporating a transmitting receiving function section (13) including a waveguide circuit section (8), high-frequency electric circuit section (2), and intermediate-frequency electric circuit section (3), antenna (7) fitted to the other end face of the enclosure (5) and connected to the section (13), and cover member (6) which closes the opening (5B). The circuit sections (8 and 2) constitute a first unit (10); the circuit section (3) constitutes a second unit (11). The units (10 and 11) are installed in the enclosure (5) in a stacked state.
摘要翻译：一个主要安装在户外的天线小型收发器用于发射和接收无线电信号，并通过减少工时的方法从少数部分制造。收发器设置有在一个端面中具有开口（5B）的壳体（5）和在另一端面上的天线配合表面（5A），并且包括发射接收功能部分（13），包括波导电路部分（8）），高频电路部（2）和中频电路部（3），安装在壳体（5）的另一端面并与该部分（13）连接的天线（7）关闭开口（5B）的构件（6）。电路部分（8和2）构成第一单元（10）; 电路部分（3）构成第二单元（11）。单元（10和11）以堆叠状态安装在外壳（5）中。

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