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1. 发明申请

WO2012153260A1 MIXTURE OF STERICALLY HINDERED AMINES FOR POLYMER STABILIZATION 审中-公开
标题翻译：用于聚合物稳定化的混合异构胺的混合物
公开(公告)号：WO2012153260A1
公开(公告)日：2012-11-15
申请号：PCT/IB2012/052271
申请日：2012-05-08
申请人： 3V SIGMA S.P.A. , DEL SORDO, Simone , MALANCHINI, Claudio , BERTE', Ferruccio , MAESTRI, Francesco
发明人： DEL SORDO, Simone , MALANCHINI, Claudio , BERTE', Ferruccio , MAESTRI, Francesco
IPC分类号： C08G73/06 , C08K5/00
CPC分类号： C08G73/0644 , C08G73/0273 , C08K5/34 , C08K2201/014
摘要： The present invention relates to mixtures of polypiperidine compounds, which are able to impart to the polymeric materials of different nature a high stability towards oxidative action and photodegradation.
摘要翻译：本发明涉及多哌啶化合物的混合物，其能够赋予不同性质的聚合物材料对氧化作用和光降解的高稳定性。

2. 发明申请

WO2011080264A1 NEW TERTIARY 8-HYDROXYQUINOLINE-7-CARBOXAMIDE DERIVATIVES AND USES THEREOF 审中-公开
标题翻译：新型8-羟基喹啉-7-羧酰胺衍生物及其用途
公开(公告)号：WO2011080264A1
公开(公告)日：2011-07-07
申请号：PCT/EP2010/070790
申请日：2010-12-28
申请人： POLICHEM S.A. , GAGLIARDI, Stefania , DEL SORDO, Simone , MAILLAND, Federico , LEGORA, Michela
发明人： GAGLIARDI, Stefania , DEL SORDO, Simone , MAILLAND, Federico , LEGORA, Michela
IPC分类号： C07D215/48 , C07D401/06 , C07D401/12 , C07D407/06 , C07D407/12 , C07D417/06 , C07D491/113 , A61K31/4709 , A61P31/10
CPC分类号： C07D215/48 , C07D401/06 , C07D401/12 , C07D407/06 , C07D407/12 , C07D417/06 , C07D491/113
摘要： New tertiary 8-hydroxyquinoiine-7-carboxamide derivatives of general formula (I) and pharmaceutically acceptable salts thereof are disclosed. These compounds are useful as antifungal agents. Specifically, these compounds were tested against Tricophyton Rubrum, Tricophyton Mentagrophytes, Aspergillus Niger and Scopulariopsis Brevicaulis. These compounds are also active against Candida species such as Candida Albicans and Candida Glabrata.
摘要翻译：公开了通式（I）的新的8-羟基喹喔啉-7-甲酰胺衍生物及其药学上可接受的盐。这些化合物可用作抗真菌剂。具体地说，这些化合物被测试针对红纹枯菌（Tricophyton Rubrum），三孢球菌（Tricophyton Mentagrophytes），黑曲霉（Aspergillus Niger）和Scopulariopsis Brevicaulis（Scopulariopsis Brevicaulis）。这些化合物对假丝酵母属（Candida albicans）和假丝酵母（Candida Glabrata）也是有活性的。

3. 发明申请

WO2011080266A1 NEW SECONDARY 8-HYDROXYQUINOLINE-7-CARBOXAMIDE DERIVATIVES. 审中-公开
标题翻译：新的二次8-羟基喹啉-7-羧酰胺衍生物。
公开(公告)号：WO2011080266A1
公开(公告)日：2011-07-07
申请号：PCT/EP2010/070793
申请日：2010-12-28
申请人： POLICHEM S.A. , GAGLIARDI, Stefania , DEL SORDO, Simone , MAILLAND, Federico , LEGORA, Michela
发明人： GAGLIARDI, Stefania , DEL SORDO, Simone , MAILLAND, Federico , LEGORA, Michela
IPC分类号： C07D215/48 , C07D401/12 , C07D407/12 , C07D409/12 , C07D413/12 , C07D417/12 , A61K31/4709 , A61P31/10
CPC分类号： C07D417/12 , C07D215/48 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12
摘要： The present invention provides new secondary 8-hydroxyquinoline-7-carboxamide derivatives of general formula (I) and pharmaceutically acceptable salts thereof. These compounds are useful as antifungal agents. Specifically, these compounds were tested against Tricophyton Rubrum, Tricophyton Mentagrophytes, Aspergillus Niger and Scopuiariopsis Brevicaulis. Many of these compounds are active against Candida species such as Candida Albicans and Candida Glabrata.
摘要翻译：本发明提供了通式（I）的新的仲羟基喹啉-7-甲酰胺衍生物及其药学上可接受的盐。这些化合物可用作抗真菌剂。具体地说，这些化合物被测试针对红纹枯菌（Tricophyton Rubrum），三孢球菌（Tricophyton Mentagrophytes），黑曲霉（Aspergillus Niger）和Scopuiariopsis Brevicaulis（Scopuiariopsis Brevicaulis）。这些化合物中的许多对假丝酵母属（Candida Albicans）和念珠菌（Candida Glabrata）是有活性的。

4. 发明申请

WO2012055965A1 NEW STERICALLY HINDERED POLYMERIC AMINES AND THEIR USE AS POLYMER STABILIZERS 审中-公开
标题翻译：新型异质聚合物及其作为聚合物稳定剂的用途
公开(公告)号：WO2012055965A1
公开(公告)日：2012-05-03
申请号：PCT/EP2011/068867
申请日：2011-10-27
申请人： 3V SIGMA S.P.A. , MAESTRI, Francesco , DEL SORDO, Simone , BERTE', Ferruccio
发明人： MAESTRI, Francesco , DEL SORDO, Simone , BERTE', Ferruccio
IPC分类号： C07D401/14 , C08K5/3492 , C09K15/30
CPC分类号： C08K5/3492 , C07D401/14 , C07D413/14 , C08K5/34926 , C09K15/30
摘要： The present invention relates to polypiperidine compounds of polymeric type which are capable of conferring to the polymeric materials, particularly to polyolefins, a high stability against photodegradation and oxidative action of air, belong to the HALS category and have general formula (I): wherein p is from 3 to 20; n is from 2 to 12; R and R 1 , which are the same or different, are selected in the group consisting of hydrogen, linear and branched C 1 -C 12 alkyl groups, alkenyl groups having 3 to 8 carbon atoms and aralkyl groups having 7 to 19 carbon atoms; X and X 1 , which are the same or different, are selected in the group consisting of oxygen and groups of formula (II) wherein R 2 is selected in the group consisting of hydrogen, linear and branched C 1 -C 12 alkyl groups, cycloalkyl groups having 5 to 12 carbon atoms and aralkyl groups having 7 to 12 carbon atoms; A represents a –(CH 2 ) a – group wherein a is from 2 to 12, with the proviso that a is different from n; Z is selected in the group consisting of C 1 -C 18 alkyl groups, groups of formula (III) wherein n, X, X 1 , R and R 1 are as above defined, and groups of formula (IV) wherein R is as above defined; Y represents a substituent selected in the group consisting of the groups of general formula (V) the groups O-R4 and S-R4, wherein R 3 and R 4 , which may be the same or different, represent hydrogen, a linear and branched C 1 -C 18 alkyl group, a cycloakyl group having 5 to 12 carbon atoms, an aralkyl group having 7 to 12 carbon atoms, an aryl group having 6 to 12 carbon atoms or may form, together with the nitrogen atom to which they are linked, a heterocycle containing 5 to 7 carbon atoms; and the piperidine group (VI) wherein R and X are as above defined. The invention further relates to the processes for preparation of the compounds according to the invention.
摘要翻译：本发明涉及能够赋予聚合物材料，特别是赋予聚烯烃，对光降解和空气氧化作用的高稳定性的聚合型聚哌啶化合物，属于HALS类别，并具有通式（I）：其中p 从3到20; n为2至12; R和R 1相同或不同，选自氢，直链和支链C 1 -C 12烷基，具有3至8个碳原子的烯基和具有7至19个碳原子的芳烷基; X和X 1相同或不同，选自氧和式（II）基团，其中R 2选自氢，直链和支链C 1 -C 12烷基，环烷基具有5 至12个碳原子和具有7至12个碳原子的芳烷基; A表示 - （CH 2）a - 基团，其中a为2至12，条件是a不同于n; Z选自C 1 -C 18烷基，其中n，X，X 1，R和R 1如上所定义的式（III）基团和式（Ⅳ）基团，其中R如上所定义; Y表示选自通式（Ⅴ）基团O-R4和S-R4的取代基，其中R3和R4可以相同或不同，表示氢，直链和支链C1- C18烷基，碳原子数5〜12的环烷酰基，碳原子数7〜12的芳烷基，碳原子数6〜12的芳基，可以与它们所连结的氮原子一起形成杂环含有5至7个碳原子; 和其中R和X如上所定义的哌啶基（Ⅵ）。本发明还涉及本发明化合物的制备方法。

5. 发明申请

WO2005005411A1 SUBSTITUTED INDOLE LIGANDS FOR THE ORL-1 RECEPTOR 审中-公开
标题翻译：替代ORL-1受体的替代配体
公开(公告)号：WO2005005411A1
公开(公告)日：2005-01-20
申请号：PCT/EP2004/007294
申请日：2004-07-01
申请人： GLAXOSMITHKLINE S.P.A. , CONSONNI, Alessandra , DEL SORDO, Simone , FARINA, Carlo , GAGLIARDI, Stefania , RONZONI, Silvano , VALLESE, Stefania
发明人： CONSONNI, Alessandra , DEL SORDO, Simone , FARINA, Carlo , GAGLIARDI, Stefania , RONZONI, Silvano , VALLESE, Stefania
IPC分类号： C07D401/06
CPC分类号： C07D409/14 , C07D401/06 , C07D401/14 , C07D405/14
摘要： New ligands for the ORL-1 receptor are described, useful for modulating the activity of said receptors in a patient in need thereof, and for preventing and treating illnesses dependent on the stimulation of this receptor. The new compounds conform to structural formula (I), wherein Q is a moiety of formula (II) and R, R 0 , R 1 , R 2 , R 3 , R 4 , R 5 , R 6 are further defined in the description.
摘要翻译：描述了ORL-1受体的新配体，可用于调节有需要的患者中所述受体的活性，以及用于预防和治疗依赖于该受体刺激的疾病。新化合物符合结构式（I），其中Q是式（II）的部分，R 1，R 2，R 1，R 2，R 3，R 4，R 4， <5>，R 6在说明书中进一步限定。

6. 发明申请

WO2011080265A1 SECONDARY 8-HYDROXYQUINOLINE-7-CARBOXAMIDE DERIVATIVES FOR USE AS ANTIFUNGAL AGENTS 审中-公开
标题翻译：用作抗真菌剂的二级8-羟基喹啉-7-羧酰胺衍生物
公开(公告)号：WO2011080265A1
公开(公告)日：2011-07-07
申请号：PCT/EP2010/070791
申请日：2010-12-28
申请人： POLICHEM S.A. , GAGLIARDI, Stefania , DEL SORDO, Simone , MAILLAND, Federico , LEGORA, Michela
发明人： GAGLIARDI, Stefania , DEL SORDO, Simone , MAILLAND, Federico , LEGORA, Michela
IPC分类号： C07D215/48 , C07D401/12 , C07D407/12 , C07D409/12 , C07D413/12 , C07D417/12 , A61K31/4709 , A61P31/10
CPC分类号： C07D401/12 , C07D215/48 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12
摘要： The present invention provides secondary 8-hydroxyquinoiine-7-carboxamide derivatives of general formula (I) and pharmaceutically acceptable salts thereof. These compounds are useful as antifungal agents. Specifically, these compounds were tested against Tricophyton Rubrum, Tricophyton Mentagrophytes, Aspergillus Niger and Scopulahopsis Brevicaulis. These compounds are active against Candida species such as Candida Albicans and Candida Glabrata.
摘要翻译：本发明提供通式（I）的第二8-羟基喹啉-7-甲酰胺衍生物及其药学上可接受的盐。这些化合物可用作抗真菌剂。具体地说，对这些化合物进行了针对红壤菌（Tricophyton Rubrum），嫩枝菌（Tricophyton Mentagrophytes），黑曲霉（Aspergillus Niger）和禾本科（Scopulahopsis Brevicaulis）的试验。这些化合物对假丝酵母属（Candida albicans）和念珠菌（Candida Glabrata）有活性。

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