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1. 发明申请

WO1998022462A1 8-AZABICYCLO[3.2.1]OCTANE-, 8-AZABICYCLO[3.2.1]OCT-6-ENE-, 9-AZABICYCLO[3.3.1]NONANE-, 9-AZA-3-OXABICYCLO[3.3.1]NONANE-, 9-AZA-3-THIABICYCLO[3.3.1]NONANE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INSECTICIDES 审中-公开
标题翻译： 8-亚氨基双环[3.2.1]十八烷，8-亚氨基二环[3.2.1] OCT-6-ENE-，9-异亚氨基[3.3.1] NONANE-，9-亚氨基-3-氧代羰基[3.3.1] NONANE - ，9-AZA-3-THIABICYCLO [3.3.1] NONANE DORIVATIVES，其制备及其作为杀虫剂的用途
公开(公告)号：WO1998022462A1
公开(公告)日：1998-05-28
申请号：PCT/GB1997002987
申请日：1997-10-30
申请人： ZENECA LIMITED , BISHOP, Nigel, Douglas , URCH, Christopher, John , LEWIS, Terence , SUNLEY, Raymond, Leo , SALMON, Roger , GODFREY, Christopher, Richard, Ayles
发明人： ZENECA LIMITED
IPC分类号： C07D451/02
CPC分类号： C07D519/00 , A01N43/90 , A01N47/38
摘要： A compound of formula (I): P-R -Q, where each of P and Q is, independently, a group of formula (B), wherein J is a bidentate group of formula -CH2-X-CH2- (wherein X is methylene, sulfur or oxygen), X'C=CY or X'WC-CYZ (wherein X', W, Y and Z are independently hydrogen, hydroxy, acyloxy, alkoxy, alkylsilyloxy or halogen); R is an optionally substituted phenyl or 5- or 6-membered heterocyclic ring system containing from 1 to 3 heteroatoms individually selected from nitrogen, oxygen and sulfur atoms, and at least one unsaturation (double bond) between adjacent atoms in the ring, said heterocyclic ring being optionally fused to a benzene ring, wherein the substituents, if present, are selected from halogen atoms, cyano, alkyl, alkenyl, alkynyl, alkoxy, haloalkyl, haloalkenyl, alkylthio and alkyl amino groups, any of which groups contain up to six carbon atoms; R is a bidentate linking group and is a substituted or unsubstituted alkylene, alkylenearyl, alkyleneheteroaryl, alkenylene, alkylenylarylalkynlenyl, carbonyl or diacyl group, provided that when R is alkenylene or alkylenylarylalkylenyl, said group does not have an unsaturated carbon atom bonding directly to the ring nitrogen of formula (B); R is hydrogen, cyano, hydroxy, alkyl, alkoxy, amino, nitro, isocyanato, acylamino, hydroxyalkyl, optionally substituted heteroaryl, alkoxyalkyl, haloalkyl, halohydroxyalkyl, aralkyloxyalkyl, acyloxyalkyl, amidoximido, sulfonyloxyalkyl, aminoalkyl, alkoxycarbonylamino, acylaminoalkyl, cyanoalkyl, imino, formyl, acyl or carboxylic acid or an ester or amide thereof, or alkenyl or alkynyl either of which is optionally substituted by halogen, alkoxy, cycloalkyl, optionally substituted aryl, optionally substituted heteroaryl or cyano; or an acid addition salt, quaternary ammonium salt or N -oxide derived therefrom; an insecticidal, acaricidal or nematicidal composition comprising a compound of formula (I) and a suitable carrier or diluent therefor; a method of combating and controlling insect, acarine or nematode pests at a locus which comprises treating the pests or the locus of the pests with an effective amount of a compound of formula (I) or a composition as hereinbefore described.
摘要翻译：式（I）的化合物：PR 2 -Q，其中P和Q各自独立地是式（B）的基团，其中J是式-CH 2 -X-CH 2 - 的双齿基团（其中 X是亚甲基，硫或氧），X'C = CY或X'WC-CYZ（其中X'，W，Y和Z独立地是氢，羟基，酰氧基，烷氧基，烷基甲硅烷氧基或卤素）; R 1是任选取代的苯基或5-或6-元杂环体系，其含有1-3个分别选自氮，氧和硫原子的杂原子，以及环中相邻原子之间的至少一个不饱和键（双键）所述杂环任选地与苯环稠合，其中所述取代基（如果存在的话）选自卤原子，氰基，烷基，烯基，炔基，烷氧基，卤代烷基，卤代烯基，烷硫基和烷基氨基，最多6个碳原子; R 2是二齿连接基团，并且是取代或未取代的亚烷基，亚烷基硬脂基，亚烷基杂芳基，亚烯基，亚烷基芳基烯烃基，羰基或二酰基，条件是当R 2是亚烯基或亚烷基芳基亚烷基时，所述基团不具有不饱和碳原子直接键合到式（B）的环氮上; R 3是氢，氰基，羟基，烷基，烷氧基，氨基，硝基，异氰酸根合，酰氨基，羟基烷基，任选取代的杂芳基，烷氧基烷基，卤代烷基，卤代羟烷基，芳烷氧基烷基，酰氧基烷基，酰氨基亚氨基，磺酰氧基烷基，氨基烷基，烷氧基羰基氨基，酰基氨基烷基，酰基或羧酸或其酯或酰胺，或任选被卤素，烷氧基，环烷基，任选取代的芳基，任选取代的杂芳基或氰基取代的链烯基或炔基; 或由其衍生的酸加成盐，季铵盐或N，N-氧化物; 杀虫杀螨或杀线虫组合物，其包含式（I）化合物及其合适的载体或稀释剂; 一种防治昆虫，螨虫或线虫害虫的方法，包括用有效量的式（I）化合物或上述组合物处理害虫或害虫的场所。

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