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51. 发明申请

WO2007113322A2 SUBSTITUTED 5-HETARYLPYRIMIDINES 审中-公开
标题翻译：取代的5 HETARYLPYRIMIDINE
公开(公告)号：WO2007113322A2
公开(公告)日：2007-10-11
申请号：PCT/EP2007053332
申请日：2007-04-04
申请人： BASF AG , RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , ULMSCHNEIDER SARAH
发明人： RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , ULMSCHNEIDER SARAH
CPC分类号： C07D401/04 , A01N43/54
摘要： The invention relates to 5-hetaryl-4-pyrimidines of formula (I) and to their salts and plant protection agents which contain at least one compound of said type as an active component, wherein W represents oxygen, sulphur, a group S=O or S(=O) 2 ; R 1 represents optionally substituted C 1 -C 8 -alkyl, C 3 -C 8 -cycloalkyl, C 5 -C 10 -bicycloalkyl, C 2 -C 8 -alkenyl, C 4 -C 10 -alkadienyl, C 3 -C 6 -cycloalkenyl, C 2 -C 8 -alkynyl, phenyl, naphthyl, or a C-bound five- or six-membered saturated, partially unsaturated or aromatic heterocycle containing one, two, three or four heteroatoms from the groups O, N or S as ring members; R 2 represents halogen, cyano, hydroxy, mercapto, N 3 , C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 1 C 6 -halogenalkyl, C 1 C 6 -alkoxy, C 3 -C 8 -alkenyloxy, C 3 -C 8 -alkynyloxy, C 1 C 6 -halogenalkoxy, C 1 -C 6 -alkylthio, C 3 -C 8 -alkenylthio, C 3 -C 8 -alkynylthio, C 1 -C 6 -halogenalkylthio, or a radical of formulae C(=Z)OR 21 , C(=Z)NR 22 R 23 , C(=Z)NR 24 -NR 22 R 23 , C(=Z)R 25 , CR 26 R 27 -OR 28 , CR 26 R 27 -NR 22 R 23 , ON(=CR 29 R 30 ), O-C(=Z)R 25 , NR 22 R 23a , NR 31 (C(=Z)R 25 ), NR 31 (C(=Z)OR 21 ), NR 31 (C(=Z)-NR 22 R 23 ), NR 32a (N=CR 29 R 30 ), NR 32 NR 22 R 23 , NR 32 OR 21 , or C(=N-Z'-R 25 )SR 21 ; or a cyclic radical; R3 represents hydrogen, OH, halogen, cyano, NR 37 R 38 , C 1 -C--alkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylsulfinyl, C 1 -C--alkylsulfonyl, C 2 -C 8 -alkenyl or C 2 -C 8 -alkinyl, whereby the seven latter radicals can be partially or totally halogenated and/or optionally can support one, two or three substitutes, selected among nitro, cyano, OH, C 1 -C 2 -alkoxy, C 1 -C 4 -alkoxycarbonyl, amino, C 1 -C 4 -alkylamino and Di-C 1 -C 4 -alkylamino, Het represents a substituted C- or N-bound, 5-or 6-membered aromatic heterocycle which comprises 1, 2, 3 or 4 heteroatoms as ring members selected among nitrogen, oxygen and sulphur. The invention also relates to the use of 5-hetaryl-4-pyrimidines of formula (I) and there salts for combating plant pathogenic fungi.
摘要翻译：本发明涉及式（I）的包含至少一种这样的化合物作为有效成分的5-杂芳基-4-嘧啶和它们的盐和杀虫剂。其中W = O或S（= O）_{2 表示氧，硫，基团S; [R ^{1 表示任选subsitituiert.esç_{1 -C _{8 烷基，C _{3 -C _{8 环烷基，C _{5 -C _{10 双环，C _{2 -C _{8 - 烯基，C _{4 -C _{10 链二烯基，C _{3 -C _{6 环烯基，C _{2 -C _{8 是炔基，苯基，萘基或C-连接的五元或六元饱和，部分不饱和或芳族的含有一个，两个，三个或四个杂原子的从杂环包含基团的O，N或S作为环成员; [R ^{2 表示卤素，氰基，羟基，巯基，N _{3 ，C _{1 -C _{6 烷基， ç_{2 -C _{8 烯基，C _{2 -C _{8 - 炔基，C _{1 < / SUB> C _{6 卤代烷基，C _{1 C _{6 烷氧基，C _{3 -C _{8 烯，C _{3 -C _{8 炔氧基，C _{1 C _{6 卤代烷氧基，C _{1 -C _{6 烷硫基，C _{3 -C _{8 烯，C _{3 -C _{8 炔硫基，C _{1 -C _{6 卤代烷硫基，或一个基团，式C（= Z） OR ^{21 ，C（= Z）NR ^{22 - [R ^{23 ，C（= Z）NR ^{24 -NR ^{22 - [R ^{23 ，C（= Z）R ^{25 ，CR ^{26 - [R ^{27 -OR ^{28 ，CR ^{26 - [R ^{27 -NR ^{22 - [R ^{23 ， ON（= CR ^{29 - [R ^{30 ），OC（= Z）R ^{25 ，NR ^{22 - [R ^{图23A ，NR ^{31 （C（= Z）R ^{25 ），NR ^{31 （C（= Z）OR < SUP> 21 ）NR ^{31 （ C（= Z）-NR ^{22 - [R ^{23 ），NR ^{32A （N = CR ^{29 - [R ^{30 ），NR ^{32 NR ^{22 - [R ^{23 ，NR ^{32 OR ^{21 ，或C（= N-Z'-R ^{25 ）SR ^{21 ; 或环状基团; R 3是氢，OH，卤素，氰基，NR ^{37 - [R ^{38 ，C _{1 -C - 烷基，C _{1 -C _{8 烷氧基，C _{1 -C _{8 烷硫基，C _{1 -C _{8 烷基亚磺酰基，C _{1 -C - 烷基磺酰基，C _{2 -C _{8 链烯基或C _{2 -C _{8 炔基，其中所述7最后提到的基团可以部分或完全卤化和/或选自硝基一个，两个或三个取代基，氰基，OH，C _{1 -C _{2 烷氧基，C _{1 -C _{4 烷氧基羰基，氨基，C _{1 -C _{4 烷基氨基和二C _{1 -C _{4可携带>烷基氨基，}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}}

52. 发明申请

WO2006114405A2 USE OF 5-ALKYL-6-PHENYLALKYL-7-AMINO-AZOLOPYRIMIDINES, NOVEL AZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THE SAME 审中-公开
标题翻译：使用5-烷基-6-苯基 - 7-氨基AZOLOPYRIMIDINEN，NEW azolopyrimidines，METHOD用于生产和AGENTS CONTAINING THE SAME
公开(公告)号：WO2006114405A2
公开(公告)日：2006-11-02
申请号：PCT/EP2006061786
申请日：2006-04-24
申请人： BASF AG , DIETZ JOCHEN , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , LOHMANN JAN KLAAS , MUELLER BERND , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA
发明人： DIETZ JOCHEN , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , LOHMANN JAN KLAAS , MUELLER BERND , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA
IPC分类号： A01N43/90
CPC分类号： A01N43/90 , C07D487/04
摘要： The invention relates to the use of 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines of formula I for controlling phytopathogenic fungi. The variables in formula I have the following designations: Y represents alkylene, alkenylene or alkinylene, optionally substituted by alkyl groups; R 1 represents halogen, cyano, nitro, hydroxy, mercapto, alkyl, halogenalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, halogenalkoxy, alkenyloxy, alkinyloxy, alkylthio, NR A R B , alkylcarbonyl, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; R A , R B represent hydrogen, alkyl and alkylcarbonyl; n represents 0, 1, 2, 3 or 4; R 2 represents alkyl, alkenyl, cycloalkyl, alkoxyalkyl and alkylthioalkyl; R 3 represents hydrogen, halogen, cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, or alkyl-S(O) m- ; m represents 0, 1 or 2; A represents N and C-R a ; and R a represents hydrogen and alkyl. The carbon atoms in Y, R 1 , R 2 , R 3 and Ra can be substituted according to the description. The invention also relates to novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, to methods for producing said compounds, and to agents containing the same.
摘要翻译：式的5-烷基-6-苯基-7-氨基azolopyrimidinen的使用I：其中各变量具有以下含义：Y是任选被烷基取代的亚烷基，亚烯基或亚炔基; [R ^{1 为卤素，氰基，硝基，羟基，巯基，烷基，卤代烷基，链烯基，环烷基，环烯基，烷氧基，卤代烷氧基，烯氧基，炔氧基，烷硫基，NR ^{一 - [R < SUP>乙，烷基羰基，苯基，萘基或五 - 或六元饱和环，其包含选自一至四个杂原子的部分不饱和或罗马杂环O，N或S; [R ^{一，R ^{乙是氢，烷基和烷基羰基; n是零，1，2，3或4; [R ^{2 烷基，烯基，环烷基，烷氧基烷基和烷硫基烷基; [R ^{3 为氢，卤素，氰基，NR ^{一 - [R ^{乙，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基，环烷硫基，羧基，甲酰基，烷基羰基，烷氧基羰基，烯氧基羰基，炔氧基羰基，苯基，苯氧基，苯硫基，苄氧基，苄硫基，烷基-S（O）_{米 - ; m是0，1或2; A N和C-R ^{一; [R ^{一氢和烷基; 其中Y中的碳原子，R ^{1 ，R ^{2 ，R ^{3 和R a可以按照该描述被取代; 防治植物病原性有害真菌; 新5-烷基-6-苯基-7- aminoazolopyrimidines，处理用于制备这些化合物和含有它们的组合物。}}}}}}}}}}}}}}

53. 发明申请

WO2006097489A8 BIPHENYL-N-(4-PYRIDYL) METHYLSUFONAMIDES 审中-公开
标题翻译：二苯基-N-（4-吡啶基）甲基磺酰胺
公开(公告)号：WO2006097489A8
公开(公告)日：2007-03-08
申请号：PCT/EP2006060753
申请日：2006-03-15
申请人： BASF AG , GRAMMENOS WASSILIOS , RHEINHEIMER JOACHIM , LOHMANN JAN KLAAS , GROTE THOMAS , PUHL MICHAEL , KORADIN CHRISTOPHER , BAUMANN ERNST , DEYN WOLFGANG VON , LANGEWALD JUERGEN , GOETZ NORBERT , CULBERTSON DEBORAH L , ANSPAUGH DOUGLAS D , OLOUMI-SADEGHI HASSAN , COTTER HENRY VAN TUYL , KUHN DAVID G
发明人： GRAMMENOS WASSILIOS , RHEINHEIMER JOACHIM , LOHMANN JAN KLAAS , GROTE THOMAS , PUHL MICHAEL , KORADIN CHRISTOPHER , BAUMANN ERNST , VON DEYN WOLFGANG , LANGEWALD JUERGEN , GOETZ NORBERT , CULBERTSON DEBORAH L , ANSPAUGH DOUGLAS D , OLOUMI-SADEGHI HASSAN , COTTER HENRY VAN TUYL , KUHN DAVID G
IPC分类号： A01N43/40 , C07D213/42
CPC分类号： A01N43/40 , C07D213/42
摘要： Biphenylsulfonamides of the formula (I) and the N-oxides and the agriculturally acceptable salts and the veterinarily acceptable salts of the compounds I, a process for preparing these compounds, compositions comprising them, their use for controlling phytopathogenic harmful fungi and harmful arthropodes, a method for combating arthropodal pests, a method for protecting crops from attack or infestation of arthropodal pests, a method for protecting seed and non-living materials from infestation by arthropodal pests, a method for protecting non-living materials from attack or infestation by arthropodal pests and seed comprising the compounds I.
摘要翻译：式（I）的联苯磺酰胺和化合物I的N-氧化物和农业上可接受的盐和兽医学上可接受的盐，制备这些化合物的方法，包含它们的组合物，其用于控制植物病原性有害真菌和有害的节肢动物的用途防治节肢动物害虫的方法，保护作物免受节肢动物害虫侵袭或侵扰的方法，保护种子和非生物材料免受节肢动物害虫侵扰的方法，保护非生物材料免受节肢动物害虫侵袭或侵袭的方法和包含化合物I的种子。

54. 发明申请

WO2006092428A2 2-SUBSTITUTED 7-AMINO-AZOLOPYRIMIDINE, A METHOD FOR THE PRODUCTION AND USE THEREOF FOR CONTROLLING PATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUND 审中-公开
标题翻译： 2-取代的7- aminoazolopyrimidines，METHOD用于生产和它们用于防治有害真菌和代理含
公开(公告)号：WO2006092428A2
公开(公告)日：2006-09-08
申请号：PCT/EP2006060399
申请日：2006-03-02
申请人： BASF AG , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , LOHMANN JAN KLAAS , MUELLER BERND , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHWOEGLER ANJA , RACK MICHAEL
发明人： GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , LOHMANN JAN KLAAS , MUELLER BERND , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHWOEGLER ANJA , RACK MICHAEL
IPC分类号： C07D487/04 , A01N43/90
CPC分类号： C07D487/04
摘要： The invention relates to 2-substituted 7-amino-azolopyrimidine of formula (I), wherein substituents have the following meanings: R 1 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, Cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or akoxyalkinyl; R 2 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, wherein a carbon chain in R 1 and/or R 2 are substitutable according to a description; R 3 is halogen, Cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phe- nylthio, benzyloxy, benzylthio, alkyl-S(O) m- ; A N and CR x ; R x is hydrogen or one of above groups for R 3 . A method and intermediate products for producing said compounds, agents containing said compounds and the use thereof for combating plant-pathogen fungi are also disclosed.
摘要翻译： 2-取代的式（I）其中取代基具有以下含义的7-氨基azolopyrimidines：R t ^{1 为氢，卤素，氰基，烷基，卤代烷基，烯基，炔基，环烷基，烷氧基，烷氧基烷基， benzyloxyalkyl，烷氧基烯基或alkoxyalkynyl; [R ^{2 为氢，卤素，氰基，烷基，卤代烷基，烯基，炔基，环烷基，烷氧基，烷氧基烷基和烷硫基烷基，其中在R中的碳链^{1 和/或R ^{2 可以根据描述被取代; [R ^{3 为卤素，氰基，NR ^{一 - [R ^{乙，羟基，巯基，烷基，卤代烷基，环烷基，烷氧基，烷硫基，环烷氧基，环烷硫基，羧基，甲酰基，烷基羰基，烷氧基羰基，烯氧基羰基，炔氧基羰基，苯基，苯氧基，苯丙氨酸nylthio，苄氧基，苄硫基，烷基-S（O）_{米 - ; A N和CR ^{X ; ，R 3 基^{X 是氢或其中R ^{称作; 的方法和中间体制备这些化合物，含有它们和它们在防治植物病原性有害真菌的组合物。}}}}}}}}}}}

55. 发明申请

WO2007116011A3 SUBSTITUTED TRIAZOLOPYRIMIDINES, METHOD FOR THE PRODUCTION THEREOF, USE THEREOF FOR CONTROLLING HARMFUL FUNGI, AND SUBSTANCES CONTAINING THE SAME 审中-公开
标题翻译：取代的三唑并嘧啶类化合物，其制备方法及其用于控制受损蘑菇的用途以及含有该化合物的培养基
公开(公告)号：WO2007116011A3
公开(公告)日：2007-12-21
申请号：PCT/EP2007053355
申请日：2007-04-05
申请人： BASF AG , DIETZ JOCHEN , GROTE THOMAS , GRAMMENOS WASSILIOS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH
发明人： DIETZ JOCHEN , GROTE THOMAS , GRAMMENOS WASSILIOS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH
IPC分类号： C07D487/04 , A01N43/90
CPC分类号： C07D487/04
摘要： Disclosed are compounds of formula (I), wherein X, Y, and Z are defined as indicated in the description, methods and intermediate products for producing said compounds, substances containing the same, and the use thereof for controlling plant pathogenic fungi.
摘要翻译：其中X，Y和Z如所述定义的式（I）化合物，用于制备这些化合物的方法和中间体，含有它们的试剂及其用于防治植物病原性有害真菌的用途。

56. 发明申请

WO2006079556A2 SUBSTITUTED 5-PHENYL PYRIMIDINES I IN THERAPY 审中-公开
标题翻译：取代的5-苯基吡啶在治疗中
公开(公告)号：WO2006079556A2
公开(公告)日：2006-08-03
申请号：PCT/EP2006000774
申请日：2006-01-30
申请人： BASF AG , RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , NAVE BARBARA , SCHIEWECK FRANK , SCHWOEGLER ANJA , JABS THORSTEN , BLETTNER CARSTEN
发明人： RHEINHEIMER JOACHIM , GROTE THOMAS , MUELLER BERND , NAVE BARBARA , SCHIEWECK FRANK , SCHWOEGLER ANJA , JABS THORSTEN , BLETTNER CARSTEN
IPC分类号： A61K31/506 , A61K31/505 , C07D239/42 , C07D239/48 , C07D401/04 , C07D403/04 , C07D417/04
CPC分类号： C07D239/48 , C07D239/42 , C07D401/04 , C07D403/04 , C07D417/04
摘要： The present invention relates to substituted 5-phenyl pyrimidines I, which carry a radical X in the 4-position of the pyrimidine ring, a radical Y in the 6-position of the pyrimidine ring, the radical X denoting a group of the formula NR 1 R 2 , OR 1a or SR 1a , in which R 1 , R 2 , independently of each other, denote hydrogen, C 1 -C 10 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 1 -C 10 -haloalkyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 -halocycloalkyl, phenyl, or 5- or 6-membered heteroaryl or 5- or 6-membered heterocyclyl, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which radicals may be unsubstituted or may carry 1, 2, 3 or 4 radicals R a1 ; or the radical NR 1 R 2 may also form a 5- or 6-membered optionally substituted heterocyclic ring, containing 1, 2, 3 or 4 nitrogen atoms or 1, 2 or 3 nitrogen atoms and one sulfur or oxygen atom as ring members, which are non-adjacent to the nitrogen of NR 1 R 2 , in which two adjacent C atoms or one N atom and one adjacent C atom can be linked by a C 1 -C 4 -alkylene chain and wherein the heterocyclic ring may be unsubstituted or may carry 1, 2, 3 or 4 radicals R a1 as defined in claim 1, R 1a has one of the meanings given for R 1 except for hydrogen; the radical Y being selected from the group consisting of halogen, cyano, C 1 -C 4 -alkyl, C 2 -C 4 -alkenyl, C 2 -C 4 -alkynyl, C 3 -C 6 -cycloalkyl, C 1 -C 4 -alkoxy, C 3 -C 4 -alkenyloxy, C 3 -C 4 -alkynyloxy, C 1 -C 6 -alkylthio, di-(C 1 -C 6 -alkyl)amino or C 1 -C 6 -alkylamino, where the alkyl, alkenyl and alkynyl radicals of Y may be substituted by halogen, cyano, nitro, C 1 -C 2 -alkoxy or C 1 -C 4 -alkoxycarbonyl; and wherein the pyrimidine radical may also carry a radical different from hydrogen in the 2-position and wherein the phenyl ring in the 5-position of the pyrimidine ring may be unsubstituted or carry 1, 2, 3, 4 or 5 radicals L which are different from hydrogen, and the pharmaceutically acceptable salts substituted 5-phenyl pyrimidines for use in therapy, in particular in therapy or treatment of cancerous diseases.
摘要翻译：本发明涉及取代的5-苯基嘧啶I，其在嘧啶环的4-位上携带基团X，嘧啶环的6-位的基团Y，基团X表示式NR的基团其中R 1，R 2，R 2，R 1，R 2， R 2彼此独立地表示氢，C 1 -C 10 - 烷基，C 2 - C 6 - 烯基，C 2 -C 6 - 炔基，C 1 -C 10 - C 1 -C 3烷基，C 3 -C 8 - 环烷基，C 3 -C 8 - 卤代烷基，C 3 -C 8 - 苯基或含有1,2,3或4个氮原子或1,2或3个氮原子和一个硫或氧原子作为环成员的5-或6-元杂芳基或5-或6-元杂环基，该基团可以未被取代或可以携带1,2,3或4个基团R a1a; 或自由基NR 1 R 2还可以形成含有1,2,3或4个氮原子或1,2或2个氮原子的5或6元任选取代的杂环或3个氮原子和一个硫或氧原子作为环成员，其与NR 1 R 2 O 2的氮不相邻，其中两个相邻的C原子或一个 N原子和一个相邻的C原子可以通过C 1 -C 4 - 亚烷基链连接，并且其中杂环可以是未取代的或可以携带1,2,3 或如权利要求1所定义的4个基团R a1，其中R 1a除了氢之外具有R 1给出的含义之一; 基团Y选自卤素，氰基，C 1 -C 4 - 亚烷基，C 2 -C 3 - 烷基， 4 - 烯基，C 2 -C 4 - 炔基，C 3 -C 6 - 环烷基，C 1 -C 4 - 烷氧基，C 3 -C 4 - 炔基氧基，C 1 -C 4 - 3-C 4 - 炔基氧基，C 1 -C 6 - 烷硫基，二 - （C 1 -C 6） C 1 -C 6 - 烷基）氨基或C 1 -C 6 - 烷基氨基，其中Y的烷基，烯基和炔基可以被卤素，氰基，硝基取代，C 1 -C 2 - 烷氧基或C 1 -C 4 - - 烷氧基; 并且其中嘧啶基团还可以携带2-位上与氢不同的基团，其中嘧啶环的5-位上的苯环可以是未取代的或携带1,2,3,4或5个基团L，其为不同于氢，以及用于治疗，特别是治疗或治疗癌性疾病的药学上可接受的盐取代的5-苯基嘧啶。

57. 发明申请

WO2008012234A2 AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME 审中-公开
标题翻译： Azolylmethyloxiranes，及其用于防治病原真菌植物及代理人含
公开(公告)号：WO2008012234A2
公开(公告)日：2008-01-31
申请号：PCT/EP2007057353
申请日：2007-07-17
申请人： BASF AG , DIETZ JOCHEN , GROTE THOMAS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH , GLAETTLI ALICE
发明人： DIETZ JOCHEN , GROTE THOMAS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH , GLAETTLI ALICE
IPC分类号： C07D405/14 , A01N43/707 , C07D409/14
CPC分类号： C07D405/14 , A01N43/653 , C07D409/14
摘要： The invention relates to azolylmethyloxiranes of general formula (I), wherein A or B is benzodioxolyl which is optionally substituted by between one and five of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, said substituents being optionally substituted by between one and three of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio. The invention also relates to the plant-tolerant acid addition salts or metal salts of said compounds, to the use of the compounds of formula (I) for controlling plant-pathogenic fungi, and to agents containing the same.
摘要翻译：本发明涉及通式（I），其中A或B是苯并二的azolylmethyloxirane其任选地被一个取代以下substi- tuenten卤素，CN，NO _{2 ，氨基，C <五 SUB> 1 -C _{4 烷基，C _{1 -C _{4 烷氧基，C _{1 -C _{4 - 卤代烷基，C _{1 -C 4卤代烷，C _{1 -C _{4 烷基氨基， ç_{1 -C _{4 二烷基氨基，硫代，或C _{1 -C _{4 是烷硫基，被取代的，和各其他取代基A或B为苯基或5元或6元杂芳基，所述取代基任选地被1-3个下列取代基取代：卤素，CN，NO _{2 ，氨基，C < SUB> 1 -C _{4 烷基，C _{1 -C _{4 烷氧基，C _{1 -C _{4 卤代烷基，C _{1 -C _{4 - 卤代烷氧基，C _{1 -C _{4 - 烷基氨基，C _{1 -C _{4 二烷基氨基，巯基或C _{1 -C _{4 - 烷硫基，被取代的，和它们的植物耐受的酸加成盐或金属盐，使用式（I）的用于控制植物病原真菌包含它们的化合物和试剂。}}}}}}}}}}}}}}}}}}}}}}}}}}}

58. 发明申请

WO2008152138A3 METHOD FOR PRODUCING DIFLUOROMETHYL-SUBSTITUTED PYRAZOLE COMPOUNDS 审中-公开
标题翻译：用于生产二氟吡唑
公开(公告)号：WO2008152138A3
公开(公告)日：2009-05-28
申请号：PCT/EP2008057506
申请日：2008-06-13
申请人： BASF SE , NETT MARKUS , GROTE THOMAS , LOHMANN JAN KLAAS , DIETZ JOCHEN , SMIDT SEBASTIAN PEER , RACK MICHAEL , ZIERKE THOMAS
发明人： NETT MARKUS , GROTE THOMAS , LOHMANN JAN KLAAS , DIETZ JOCHEN , SMIDT SEBASTIAN PEER , RACK MICHAEL , ZIERKE THOMAS
IPC分类号： C07D231/12 , C07D231/14
CPC分类号： C07D231/12 , C07D231/14
摘要： The invention relates to a method for producing 3-difluoromethyl-substituted pyrazole compounds of formula (I), wherein R1 represents H, halogen, nitro, C1-C8 alkyl, C1-C8 haloalkyl, C3-C8 cycloalkyl, phenyl, naphthyl, hetaryl, cyano, -C(=O)-OR1a, -C(=O)-NR1bR1c, -C(=O)-SR1d or -C(=S)-SR1 e; R2 represents H, C1-C4 alkyl, benzyl or phenyl; R3 represents H, halogen, C1-C8 alkoxy, C1-C8 haloalkoxy, C3-C8 cycloalkoxy, C2-C8 alkenyloxy, C1-C8 alkylthio, C1-C8 haloalkylthio, C3-C8 cycloalkylthio or C2-C8 alkenylthio; to compounds of formula (II.a) or (II.b), wherein R1 and R3 have one of the above definitions; R4 represents halogen, -OR4a, -SR4a , -O-SO2-R4a or a group -NR4bR4c; R5 and R6 represent C1-C8 alkyl, C1-C8 haloalkyl, C3-C8 cycloalkyl, benzyl or phenyl or together with the nitrogen atom to which they are bound represent a 3- to 8-membered heterocycle; to Lewis acid adducts of compounds of formula (II.b); to the use of compounds of formula (II.a) or (II.b) and of the Lewis acid adducts thereof for producing compounds of formula (I) or (VI); and to a method for converting said compounds to the corresponding 3-difluoromethylpyrazole-4-yl carboxylic acids.
摘要翻译：本发明涉及一种用于制备式-3-二氟甲基吡唑（I）化合物其中R1是H，卤素，硝基，C1-C8烷基，C1-C8卤代烷基，C3-C8环烷基，苯基，萘基，杂芳基，氰基，-C（= O）-OR1a，-C（= O）-NR1bR1c，-C（= O）-SR1d或-C（= S）-SR1e基; R2是H，C1-C4烷基，苄基或苯基; R 3为H，卤素，C1-C8烷氧基，C1-C8卤代烷氧基，C3-C8环烷氧基，C2-C8链烯氧基，C1-C8烷硫基，C1-C8卤代烷硫基，C3-C8-环烷硫基或C 2 -C C8-烯硫基;式（二.a）或（二.b）的化合物，其中R 1和R 3具有以上给出的含义之一; R 4是卤素，-OR4a，-SR4a，-O-SO2-R4A或一组-NR4bR4c基; R5和R6是C1-C8烷基，C1-C8卤代烷基，C3-C8环烷基，苄基或苯基或一起与氮原子到它们所键合的，代表3-至8-元杂环; 式（二.b）化合物的路易斯酸加合物;使用（二.a）或（二.b）和路易斯酸加合物，式I化合物的对式（I）或（VI）的化合物的制备方法; 并且这些化合物转变成相应的3-二氟甲基吡唑-4-基甲磺酸的方法。

59. 发明申请

WO2010102980A8 PROCESS FOR PREPARING SUBSTITUTED 2-NITROBIPHENYLS 审中-公开
标题翻译：制备取代的2-硝基苯酚的方法
公开(公告)号：WO2010102980A8
公开(公告)日：2010-11-18
申请号：PCT/EP2010052914
申请日：2010-03-08
申请人： BASF SE , KORTE ALEXANDER , LOHMANN JAN KLAAS , GROTE THOMAS , EBEL KLAUS , ZIERKE THOMAS , MAYER HORST , WAZULEK RALF
发明人： KORTE ALEXANDER , LOHMANN JAN KLAAS , GROTE THOMAS , EBEL KLAUS , ZIERKE THOMAS , MAYER HORST , WAZULEK RALF
IPC分类号： C07C205/09 , C07C205/10 , C07C205/11
CPC分类号： C07C205/11 , C07C205/09 , C07C205/10 , C07C2601/16
摘要： The present invention relates to a process for preparing substituted 2-nitrobiphenyls and to specific 2-nitrobiphenyls. The invention further relates to a process for preparing 2-aminobiphenyls from such 2-nitrobiphenyls and to a process for preparing (het)arylamides of such 2-aminobiphenyls.
摘要翻译：本发明涉及一种制备取代的2-硝基联苯和特定2-硝基联苯的方法。本发明还涉及从这种2-硝基联苯制备2-氨基联苯的方法和制备这种2-氨基联苯的（het）芳基酰胺的方法。

60. 发明申请

WO2009077443A3 AZOLYLMETHYLOXIRANES, USE THEREOF AND AGENTS CONTAINING THE SAME 审中-公开
标题翻译： Azolylmethyloxiranes，用途及含代理
公开(公告)号：WO2009077443A3
公开(公告)日：2010-02-25
申请号：PCT/EP2008067394
申请日：2008-12-12
申请人： BASF SE , DIETZ JOCHEN , GROTE THOMAS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH , GLAETTLI ALICE , VRETTOU MARIANNA
发明人： DIETZ JOCHEN , GROTE THOMAS , MUELLER BERND , LOHMANN JAN KLAAS , RENNER JENS , ULMSCHNEIDER SARAH , GLAETTLI ALICE , VRETTOU MARIANNA
IPC分类号： A01N43/653 , A61K31/4025 , A61P31/00 , C07D303/08 , C07D303/12 , C07D303/36 , C07D407/06 , C07D407/14 , C07F9/40
CPC分类号： A01N43/653 , C07D303/08 , C07D303/12 , C07D303/16 , C07D303/36 , C07D403/06
摘要： The invention relates to the triazolylmethyloxiranes of formula (I), wherein variables A, B and D have the meanings as defined in the description and the claims.
摘要翻译：本发明涉及式（I）的triazolylmethyloxiranes其中如在权利要求和说明书中描述的变量A，B和D的含义。

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