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1. 发明申请

US20080194498A1 Avermectins and Avermectin Monosacharides Substituted in the 4'-and 4" Position Having Pesticidal Properties 有权
标题翻译：在4'和4“位置具有农药性质的阿维菌素和阿维菌素单糖
公开(公告)号：US20080194498A1
公开(公告)日：2008-08-14
申请号：US10568715
申请日：2004-08-27
申请人： Fiona Murphy Kessabi , Thomas Pitterna , Peter Maienfisch , Jerome Cassayre , Laura Quaranta , Pierre Jung , Ottmar Franz Hueter
发明人： Fiona Murphy Kessabi , Thomas Pitterna , Peter Maienfisch , Jerome Cassayre , Laura Quaranta , Pierre Jung , Ottmar Franz Hueter
IPC分类号： A01N43/90 , C07H17/08 , A01P17/00
CPC分类号： A01N43/90 , C07H19/01
摘要： Described is a compound of the formula (1) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.
摘要翻译：描述了式（1）的化合物，其中碳原子22和23之间的键是单键或双键; m为0或1; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 3 -C 12烷基，C 3 -C 12烷基，C 3 -C 12烷基， >环烷基或C 2 -C 12 - 烯基; （A）R 2是-N（R 3）R 4，和（1）X是0，其中R _{3是例如氢，未取代的或一至五取代的C 1 -C 12烷基，R 4是氢，是例如一至五取代的C 1 -C 12烷基，未取代或单取代或五取代的C 3 -C 12烷基， 12环烷基; 或（2）X是S，其中R 3是例如氢，未取代的或一至五取代的C 1 -C 12 - 烷基和R 4是例如氢，未取代的或一至五取代的C 1 -C 12烷基; 或（3）X为0或S，其中R 3和R 4一起为例如三至七元亚烷基或四至七元亚烷基，多元亚烯基桥; 或（B）R 2是OR 5，X是0或S，其中R 5是例如C 1 C 1 -C 12烷基，一至五取代C 1 -C 12烷基; 或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下都是游离形式或盐形式; 这种化合物显示出杀虫活性。}

2. 发明授权

US08017589B2 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position 有权
标题翻译：在4“ - 或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物
公开(公告)号：US08017589B2
公开(公告)日：2011-09-13
申请号：US12768280
申请日：2010-04-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A61K31/70 , C07H17/04
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

3. 发明申请

US20100210574A1 AVERMECTIN B1 AND AVERMECTIN B1 MONOSACCHARIDE DERIVATIVES HAVING AN ALKOXYMETHYL SUBSTITUENT IN THE 4"-OR 4'-POSITION 有权
标题翻译：在4“-OR 4'-位置具有烷氧基取代基的AVERMECTIN B1和AVERMECTIN B1单糖衍生物
公开(公告)号：US20100210574A1
公开(公告)日：2010-08-19
申请号：US12768280
申请日：2010-04-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A01N43/16 , C07H17/08 , A01P17/00
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

4. 发明授权

US07632820B2 Avermectin and avemectin monosaccharide derivatives substituted in the 4″- or 4′-position having pesticidal properties 有权
标题翻译：在4“或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物
公开(公告)号：US07632820B2
公开(公告)日：2009-12-15
申请号：US10543638
申请日：2004-01-30
申请人： Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Pierre Jung
发明人： Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Pierre Jung
IPC分类号： A01N43/04 , A61K31/40 , A61K31/335 , A61K31/70 , A61K31/397 , A61K31/445 , A61K31/44 , A01N43/38
CPC分类号： A01N43/90 , C07H17/08
摘要： Disclosed are compounds of the formulain which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —SO2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.
摘要翻译：公开了n为0或1的甲醛化合物; X-Y是-CH-CH-或-CH 2 -CH 2 - ; Z是-C（-O） - ， - C（-S） - 或-SO 2 - ; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R2为R3-Z-，R3-O-Z-，R4或-Z-N（R6）（R7）; Q是O或-N-R5; R 3和R 4例如是H，C 1 -C 12烷基，C 2 -C 12烯基，C 2 -C 12炔基，C 3 -C 12环烷基，C 5 -C 12环烯基，芳基或杂环基; R5是例如H，C1-C8烷基，羟基-C1-C8烷基，C3-C8环烷基，C2-C8链烯基，C2-C8炔基，苯基或苄基; R 6和R 7为例如未取代的或未被取代的一价或五价取代的C 1 -C 12烷基，未被取代的或一至五取代的C 2 -C 12链烯基或（如果合适的话）E / Z异构体，E / Z异构体混合物和/或其互变异构体，在每种情况下以游离形式或盐形式，都可用作农药。

5. 发明申请

US20060166824A1 Avermectin and avemectin monosaccharide derivatives substituted in the 4"-or 4'-position having pesticidal properties 有权
标题翻译：在4“ - 或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物
公开(公告)号：US20060166824A1
公开(公告)日：2006-07-27
申请号：US10543638
申请日：2004-01-30
申请人： Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Pierre Jung
发明人： Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Pierre Jung
IPC分类号： A01N43/04 , A61K31/7048
CPC分类号： A01N43/90 , C07H17/08
摘要： Disclosed are compounds of the formula in which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —S02—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.
摘要翻译：公开了下式的化合物，其中n为0或1; X-Y是-CH-CH-或-CH 2 -CH 2 - 。 Z是-C（-O） - ， - C（-S） - 或-SO 2 - 。 R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 1 -C 12烷基，C 3 -C 12烷基，环烷基或C 2 -C 12 - 烯基; 和R 2是R 3 -Z-，R 3 -OZ-，R 4或-ZN（ R 6）（R 7）; Q是O或-N-R 5; R 3和R 4是例如H，C 1 -C 12烷基，C 2， C 1 -C 12亚烷基，C 2 -C 12炔基，C 3 -C 12链烯基，C 2 -C 12亚炔基，C 3 -C 12亚烷基， 12个环烷基，C 5 -C 12环烯基，芳基或杂环基; R 5是例如H，C 1 -C 8烷基，羟基-C 1 -C 3 C 1 -C 8烷基，C 3 -C 8环烷基，C 2 -C 8链烯基，C 1 -C 8烷基， C 2 -C 8炔基，苯基或苄基; R 6和R 7是例如H，未取代的或一至五取代的C 1 -C 12 - 烷基，未取代的或一至五取代的C 2 -C 12链烯基，或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体，在每种情况下以游离形式或盐形式，都可用作农药。

6. 发明授权

US08263566B2 Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4″-or 4′-position 有权
标题翻译：在4“ - 或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物
公开(公告)号：US08263566B2
公开(公告)日：2012-09-11
申请号：US13117292
申请日：2011-05-27
申请人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
发明人： Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre , Laura Quaranta , Thomas Pitterna , Ottmar Franz Hueter , Pierre Jung
IPC分类号： A61K31/70 , C07H17/04
CPC分类号： C07H17/08 , A61K31/7042
摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基，卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基，芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

7. 发明授权

US07678740B2 Avermectin and avermectin monosaccharide derivatives substituted in the 4″-or 4′-position having pesticidal properties 有权
标题翻译：在4“ - 或4”位取代的具有杀虫性的阿维菌素和阿维菌素单糖衍生物
公开(公告)号：US07678740B2
公开(公告)日：2010-03-16
申请号：US10543637
申请日：2004-01-30
申请人： Thomas Pitterna , Fiona Murphy Kessabi , Peter Maienfisch , Jerome Cassayre , Laura Quaranta , Pierre Jung
发明人： Thomas Pitterna , Fiona Murphy Kessabi , Peter Maienfisch , Jerome Cassayre , Laura Quaranta , Pierre Jung
IPC分类号： A01N25/26 , A01N43/02 , A01N43/04 , C07H17/08
CPC分类号： A01N43/90 , C07H17/08
摘要： What is described are a compound of the formula (I) Wherein U is —N(R2)OR3 or —N+(O−)═C(RE)RZ); n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 are, for example; independently from each other, —Q, —C(═O)—Z—Q or —CN; RZ and RE are, independently from each other, —Q, —C(═O)—Z—Q or —CN; or RZ and RE together are a three- to seven membered alkylene or alkenylene bridge, which is unsubstituted or mono- to tri-substituted; Z is a bond, O or —NR4—; Q is H, C1-C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12-Cycloalkyl, C5-C12-cycloalkenyl, aryl, or heterocyclyl, which are unsubstituted or mono- to pentasubstituted; R4 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl or C2-C8alkenyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions.
摘要翻译：描述的是式（I）的化合物，其中U是-N（R 2）OR 3或-N +（O-）= C（RE）R Z）; n为0或1; X-Y是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R2和R3例如是：独立地为-Q，-C（= O）-Z-Q或-CN; RZ和RE彼此独立地为-Q，-C（= O）-Z-Q或-CN; 或RZ和RE一起是三至七元的亚烷基或亚烯基桥，其是未取代的或一至三取代的; Z是O或-NR4-键; Q是未被取代或被一取代或五取代的H，C 1 -C 12烷基，C 2 -C 12烯基，C 2 -C 12炔基，C 3 -C 12环烷基，C 5 -C 12 - 环烯基，芳基或杂环基， R4是例如H，C1-C8烷基，羟基-C1-C8烷基，C3-C8环烷基或C2-C8链烯基; 或者，如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体; 制备这些化合物，其异构体和互变异构体的方法以及这些化合物，其异构体和互变异构体的用途; 活性化合物选自这些化合物及其互变异构体的杀虫组合物; 用于制备所述式（I）化合物的中间体，式（I）化合物的制备方法和使用这些组合物来控制害虫的方法。

8. 发明申请

US20060094600A1 Avermectins and avermectin monosaccharides substituted in the 4'-and 4"-position having pesticidal properties 审中-公开
标题翻译：在4'和4“位具有杀虫性质的阿维菌素和阿维菌素单糖被取代
公开(公告)号：US20060094600A1
公开(公告)日：2006-05-04
申请号：US10544281
申请日：2004-02-03
申请人： Laura Quaranta , Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre
发明人： Laura Quaranta , Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Jerome Cassayre
IPC分类号： A01N43/04 , A01N25/26 , C07H17/08
CPC分类号： C07H17/08 , A01N43/90
摘要： What is described are a compound of the formula (I) wherein the bond of atoms C22 and C23 is a single or double bond; m is 0 or 1; n is 0, 1 or 2; p is 0 or 1; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12alkenyl; R2 is for example H, C1-C12-alkyl, C1-C12-haloalkyl or C1-C12-hydroxyalkyl; or together with R4 form with the carbon to which they are bound for example a three- to seven-membered ring; R3 is for example H, C1-C12-alkyl, halogen, halo-C1-C2alkyl, CN, NO2 or C3-C8-cycloalkyl; R4 has the same meanings as R2; R5 and R6 independently of each other are for example H, C1-C12-alkyl, CN, NO2, OH, SH, halogen, halo-C1-C2alkyl or C3-C8cycloalkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译：描述的是式（I）的化合物，其中原子C 22和C 23的键是单键或双键; m为0或1; n为0,1或2; p为0或1; R 1是C 1 -C 12 - 烷基，C 3 -C 8亚烷基，C 3 -C 12 - 烷基，C 3 -C 12 - 环烷基或C 2 -C 12链烯基; R 2是例如H，C 1 -C 12 - 烷基，C 1 -C 3 - 12个 - 卤代烷基或C 1 -C 12 - 羟基烷基; 或与R 4 S形成的碳与它们所键合的碳例如为三至七元环; R 3是例如H，C 1 -C 12 - 烷基，卤素，卤素-C 1 - C 2 -C 12烷基，CN，NO 2或C 3 -C 8 - 环烷基; R 4具有与R 2'相同的含义; R 5和R 6彼此独立地是例如H，C 1 -C 12 - 烷基， CN，NO 2，OH，SH，卤素，卤代-C 1 -C 2烷基或C 3 - -C 8环烷基; 或者如果适用，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下以游离形式或盐形成用于制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

9. 发明授权

US07378399B2 Avermectins substituted in the 4″ and 4′-positions having pesticidal properties 有权
标题翻译：在4“和4”位取代的阿维菌素具有杀虫特性
公开(公告)号：US07378399B2
公开(公告)日：2008-05-27
申请号：US10544274
申请日：2004-02-03
申请人： Jerome Cassayre , Hans Tobler , Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Laura Quaranta , Ottmar Franz Hueter
发明人： Jerome Cassayre , Hans Tobler , Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Laura Quaranta , Ottmar Franz Hueter
IPC分类号： A01N43/04 , A01N43/00 , A01N43/40 , A01N43/02 , A01N43/16 , A61K31/40 , A61K31/38 , A61K31/335 , A61K31/35 , A61K31/70 , A61K31/397 , A61K31/445 , A61K31/44 , A01N43/38 , A01N31/40
CPC分类号： C07H17/08
摘要： What is described are a compound of the formula (I) Wherein A-B is —CH═CH— or —CH2—CH2—; n is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 for instance are either, (i) independently from each other for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; or (ii) together form with the nitrogen atom to which they are bound a three- to seven-membered ring, (iii) together are ═C(R4)R5; R4 and R5 are, independently from each other, for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; Y is O or S; Q is for instance H or unsubstituted or mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions
摘要翻译：描述的是式（I）的化合物，其中A-B是-CH-CH-或-CH 2 -CH 2 - 。 n为0或1; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 3 -C 12烷基，C 3 -C 12烷基，C 3 -C 12烷基， >环烷基或C 2 -C 12 - 烯基; 例如，R 2和R 3是（i）彼此独立地例如-Q，-C（-Y）-Q或-C（ - Y）-OQ; 或（ii）与其结合的氮原子一起形成三至七元环，（iii）一起为-C（R 4）R 5 >; R 4和R 5各自独立地为例如-Q，-C（-Y）-Q或-C（-Y）-O-Q; Y为O或S; Q是例如H或未被取代或单取代或未取代的C 1 -C 12烷基; 或者，如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体; 制备这些化合物，其异构体和互变异构体的方法以及这些化合物，其异构体和互变异构体的用途; 活性化合物选自这些化合物及其互变异构体的杀虫组合物; 用于制备所述式（I）化合物的中间体，式（I）化合物的制备方法和使用这些组合物来控制害虫的方法

10. 发明申请

US20060205595A1 Avermectin monosaccharide derivatives having pesticidal properties 审中-公开
标题翻译：具有杀虫性的阿维菌素单糖衍生物
公开(公告)号：US20060205595A1
公开(公告)日：2006-09-14
申请号：US10543643
申请日：2004-01-30
申请人： Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Hans Tobler , Jerome Cassayre , Laura Quaranta
发明人： Thomas Pitterna , Peter Maienfisch , Fiona Murphy Kessabi , Hans Tobler , Jerome Cassayre , Laura Quaranta
IPC分类号： A01N43/04 , C07H17/08
CPC分类号： C07H17/08
摘要： A compound of the general formula (I) pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I)m methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions.
摘要翻译：通式（I）杀虫组合物的化合物，其活性化合物选自这些化合物及其互变异构体; 用于制备所述式（I）化合物的中间体m制备式（I）化合物的方法和使用这些组合物来控制害虫的方法。

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