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1. 发明申请

US20070074967A1 Photodegradable protective group 审中-公开
标题翻译：可光降解防护组
公开(公告)号：US20070074967A1
公开(公告)日：2007-04-05
申请号：US11366464
申请日：2006-03-03
申请人： Tetsuo Nagano , Yasuteru Urano , Tomonori Kobayashi , Noriyuki Suzuki
发明人： Tetsuo Nagano , Yasuteru Urano , Tomonori Kobayashi , Noriyuki Suzuki
IPC分类号： C07C209/68 , C07C39/04 , C07C209/00
CPC分类号： C07D311/82 , Y02P20/55
摘要： A photodegradable protective group comprising a benzyl group which is bound with a light capturing moiety that can absorb light of around 470 nm and having one or more nitro groups on the benzene ring.
摘要翻译：包含与可吸收约470nm的光并且在苯环上具有一个或多个硝基的光捕获部分结合的苄基的光可降解保护基。

2. 发明申请

US20060174147A1 Electronic equipment, sensor, method and program for controlling electronic equipment 审中-公开
标题翻译：用于控制电子设备的电子设备，传感器，方法和程序
公开(公告)号：US20060174147A1
公开(公告)日：2006-08-03
申请号：US11271303
申请日：2005-11-10
申请人： Kensuke Uehara , Tomonori Kobayashi , Wataru Takahashi , Mikiko Arima
发明人： Kensuke Uehara , Tomonori Kobayashi , Wataru Takahashi , Mikiko Arima
IPC分类号： G06F1/26
CPC分类号： G06F1/3203 , G06F1/3231 , G06F21/34 , G06F21/83 , Y02D10/173
摘要： Electronic equipment includes two or more operating modes including a normal mode and a security mode and/or power saving mode. The electronic equipment comprises input devices which input information into the electronic equipment by a person performing an operation which is external to the electronic equipment, a sensor which is disposed in a rest portion of the input devices and which generates a predetermined signal in response to a detection that a part of the body of the person performing the operation rests on the rest portion, and a signal generator which generates a signal to instruct the electronic equipment not to shift to the security mode and/or power savings mode based on the predetermined signal generated by the sensor.
摘要翻译：电子设备包括两种或多种操作模式，包括正常模式和安全模式和/或省电模式。电子设备包括输入设备，其通过执行电子设备外部的操作的人员将信息输入到电子设备中;传感器，设置在输入设备的休息部分中，并且响应于一个检测到执行操作的人的身体的一部分依赖于休息部分，以及信号发生器，其基于预定信号产生指示电子设备不转移到安全模式和/或省电模式的信号由传感器产生。

3. 发明申请

US20100056497A1 AMIDE DERIVATIVE 审中-公开
公开(公告)号：US20100056497A1
公开(公告)日：2010-03-04
申请号：US12524921
申请日：2008-01-30
申请人： Hiroyuki Nakahira , Yohei Ikuma , Nobuhisa Fukuda , Tomonori Kobayashi , Shinya Tosaki
发明人： Hiroyuki Nakahira , Yohei Ikuma , Nobuhisa Fukuda , Tomonori Kobayashi , Shinya Tosaki
IPC分类号： A61K31/4462 , C07D211/56 , C07D207/14 , C07D223/12 , C07D401/12 , C07D413/12 , A61P9/12 , A61K31/40 , A61K31/55 , A61K31/4545 , A61K31/5377
CPC分类号： C07D207/14 , C07D211/56 , C07D221/22 , C07D223/12
摘要： The present invention relates to a compound of the formula (I) being useful as a renin inhibitor, or a pharmaceutically acceptable salt thereof. wherein R1a is a hydrogen atom, an optionally substituted C1-6 alkyl, etc.; R1b is an optionally substituted C1-6 alkoxy, etc.; R1c is a hydrogen atom, an optionally substituted C1-6 alkoxy, etc.; R2 is a hydrogen atom, an optionally substituted C1-6 alkyl, etc.; R3a, R3b, R3c and R3d are independently the same or different, and each is a group of the formula: -A-B (in which A is a single bond, —(CH2)sO—, —(CH2)sN(R4)CO—, etc., B is a hydrogen atom, an optionally substituted C1-6 alkyl, etc.), etc.; R4 is a hydrogen atom, an optionally substituted C1-6 alkyl, etc.; s is 0, etc.; and n is 1, etc.
摘要翻译：本发明涉及可用作肾素抑制剂的式（I）化合物或其药学上可接受的盐。其中R 1a是氢原子，任选取代的C 1-6烷基等; R1b是任选取代的C 1-6烷氧基等; R1c是氢原子，任选被取代的C 1-6烷氧基等; R2是氢原子，任选取代的C 1-6烷基等; R3a，R3b，R3c和R3d独立地相同或不同，并且各自为下式基团：其中A为单键， - （CH2）sO-， - （CH2）sN（R4）CO - 等等，B是氢原子，任选取代的C 1-6烷基等）等; R4是氢原子，任意取代的C 1-6烷基等; s为0等 n为1等

4. 发明申请

US20070105890A1 Novel condensed imidazole derivative 审中-公开
标题翻译：新型稠合咪唑衍生物
公开(公告)号：US20070105890A1
公开(公告)日：2007-05-10
申请号：US10580321
申请日：2004-11-24
申请人： Hiroyuki Nakahira , Hidenori Kimura , Tomonori Kobayashi , Hitoshi Hochigai
发明人： Hiroyuki Nakahira , Hidenori Kimura , Tomonori Kobayashi , Hitoshi Hochigai
IPC分类号： A61K31/4745 , C07D471/02
CPC分类号： C07D471/14 , C07D471/04 , C07D491/14 , C07D495/14
摘要： Disclosed is a compound represented by the formula (1) below which has a high DPP-IV inhibitory activity and is improved in safety, toxicity and the like. Also disclosed is a prodrug of such a compound and pharmaceutically acceptable salts of them. (In the formula, R1 represents a hydrogen atom, an optionally substituted alkyl group or the like; R2 and R3 independently represent a hydrogen atom, an optionally substituted alkyl group or the like; R4 and R5 independently represent a hydrogen atom, an optionally substituted alkyl group or the like: R6 represents a hydrogen atom, an optionally substituted aryl group or the like; and —Y—NH2, represents a group represented by the following formula (A): (wherein m is 0, 1 or 2; and R7 may not exist or one or two R7 may exist and independently represent an optionally substituted alkyl group or the like) or the like.]
摘要翻译：公开了由下式（1）表示的化合物，其具有高的DPP-IV抑制活性，并且其安全性和毒性等得到改善。还公开了这种化合物的前药和它们的药学上可接受的盐。（式中，R 1表示氢原子，任选取代的烷基等; R 2和R 3独立地表示氢原子，氢原子，任选取代的烷基等; R 4和R 5独立地表示氢原子，任选取代的烷基等： 6表示氢原子，任选取代的芳基等; -Y-NH 2表示由下式（A）表示的基团：（其中m为0 ，1或2; R 7可以不存在或一个或两个R 7可以存在并且独立地表示任选取代的烷基等）。

5. 发明申请

US20070082908A1 Bicycle pyrazole derivative 审中-公开
标题翻译：自行车吡唑衍生物
公开(公告)号：US20070082908A1
公开(公告)日：2007-04-12
申请号：US10595125
申请日：2004-08-25
申请人： Hiroyuki Nakahira , Hitoshi Hochigai , Tatsuya Takeda , Tomonori Kobayashi , William Hume
发明人： Hiroyuki Nakahira , Hitoshi Hochigai , Tatsuya Takeda , Tomonori Kobayashi , William Hume
IPC分类号： A61K31/53 , A61K31/498 , C07D487/04
CPC分类号： C07D487/04
摘要： A compound represented by the following formula (I), a prodrug thereof, or a pharmaceutically acceptable salt of either. These are compounds having high DPP-IV inhibitory activity and improved in safety, nontoxicity, etc. (I) [In the formula, R1 represents hydrogen, optionally substituted alkyl, etc.; the solid line and dotted line between A1 and A2 indicate a double bond (A1=A2), etc.; A1 represents a group represented by the formula C(R2), etc.; A2 represents a group represented by the formula C(R4), etc.; R2 represents hydrogen, optionally substituted alkyl, etc.; R4 represents hydrogen, optionally substituted alkyl, etc.; R6 represents hydrogen, optionally substituted aryl, etc.; and —Y represents, e.g.; a group represented by the formula (A): (A) (wherein m1 is 0, 1, 2, or 3; and R7 is absent, or one or two R7's are present and each independently represents optionally substituted alkyl, etc.).]
摘要翻译：由下式（I）表示的化合物，其前药或其药学上可接受的盐。这些是具有高DPP-IV抑制活性和安全性，无毒性等改善的化合物。（I）[式中，R 1表示氢，任选取代的烷基等; A 1和A 2之间的实线和虚线表示双键（A 1 SUP 1 = A 2））等 A ^{1表示由式C（R 2 O 2）表示的基团等; A <2>表示由式C（R 4）表示的基团等。 R 2表示氢，任选取代的烷基等; R 4表示氢，任选取代的烷基等; R 6表示氢，任选取代的芳基等; -Y表示例如由式（A）表示的基团：（A）（其中m1为0,1,2或3; R 7为不存在，或一个或两个R 7为氢， SUP'是存在的，各自独立地表示任选取代的烷基等）。}

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