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1. 发明授权

US07947697B1 8-(3-pentylamino)-2-methyl-3-(2-chloro-4-methoxyphenyl)-6,7-dihydro-5H-cyclopenta[d] pyrazolo[1,5-a]pyrimidine methanesulfonate as a CRF antagonist 有权
标题翻译： 8-（3-戊基氨基）-2-甲基-3-（2-氯-4-甲氧基苯基）-6,7-二氢-5H-环戊二烯并[d]吡唑并[1,5-a]嘧啶甲磺酸盐，为CRF拮抗剂
公开(公告)号：US07947697B1
公开(公告)日：2011-05-24
申请号：US10561214
申请日：2004-06-24
申请人： Tomoyuki Hasegawa , Toshiaki Matsui , Hiroshi Araki , Tetsuji Saito , Tetsuo Obitsu , Masaki Okamoto , Yuichi Gemba , Yutaka Mikami
发明人： Tomoyuki Hasegawa , Toshiaki Matsui , Hiroshi Araki , Tetsuji Saito , Tetsuo Obitsu , Masaki Okamoto , Yuichi Gemba , Yutaka Mikami
IPC分类号： C07D487/04 , A61K31/519 , A61P25/28 , A61P25/24 , A61P3/04 , A61P25/22
CPC分类号： C07D487/04
摘要： 8-(3-pentylamino)-2-methyl-3-(2-chloro-4-methoxyphenyl)-6,7-dihydro-5H-cyclopenta[d]pyrazolo[1,5-a]pyrimidine methanesulfonate of the structural formula (I) has Corticotropin Releasing Factor (CRF) antagonist activity and is useful in treating neuropsychiatric and digestive system diseases.
摘要翻译：具有结构式的8-（3-戊基氨基）-2-甲基-3-（2-氯-4-甲氧基苯基）-6,7-二氢-5H-环戊并[d]吡唑并[1,5-a]嘧啶甲磺酸盐（I）具有促肾上腺皮质激素释放因子（CRF）拮抗剂活性，可用于治疗神经精神和消化系统疾病。

2. 发明授权

US07629369B2 N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for its preparation 失效
标题翻译： N-苯基芳基磺酰胺化合物，包含该化合物作为活性成分的药物组合物，该化合物的合成中间体及其制备方法
公开(公告)号：US07629369B2
公开(公告)日：2009-12-08
申请号：US11239406
申请日：2005-09-30
申请人： Atsushi Naganawa , Tetsuji Saito , Kaoru Kobayashi , Takayuki Maruyama , Yoshihiko Nakai , Shinsuke Hashimoto
发明人： Atsushi Naganawa , Tetsuji Saito , Kaoru Kobayashi , Takayuki Maruyama , Yoshihiko Nakai , Shinsuke Hashimoto
IPC分类号： C07D285/08 , C07D271/06 , C07D257/04 , A61K31/41
CPC分类号： C07D213/70 , C07D277/36 , C07D307/64 , C07D401/12 , C07D405/12 , C07D413/12 , C07D417/12
摘要： An N-phenylarylsulfonylamide compound of formula (I) (R1 is COOH etc.; R2 is hydrogen, methyl, etc.; R3 and R4 are a combination of methyl and methyl, etc.; R5 is isopropyl etc.; Ar is thiazolyl, pyridyl, 5-methyl-2-furyl each optionally substituted with methyl; n is zero or 1), a synthetic intermediate for the compound and a process for its preparation. The compound of formula (I) binds to a prostaglandin E2 receptor, especially an EP1 subtype receptor, and antagonizes it. It is less affected by protein binding, so it has a satisfactory in vivo activity. Therefore, it is considered to be useful as an analgesic, an antipyretic agent, an agent for the treatment of pollakiuria (frequent urination) and/or lower urinary tract disease syndrome or an antineoplastic agent.
摘要翻译：式（I）的N-苯基芳基磺酰胺化合物（R1是COOH等; R2是氢，甲基等; R3和R4是甲基和甲基的组合等; R5是异丙基等; Ar是噻唑基，吡啶基，5-甲基-2-呋喃基，各自任选被甲基取代; n为0或1），化合物的合成中间体及其制备方法。式（I）化合物结合前列腺素E2受体，特别是EP1亚型受体，并拮抗它。蛋白质结合的影响较小，因此具有令人满意的体内活性。因此，认为可用作止痛剂，解热剂，治疗尿频（尿频）和/或下尿路疾病综合征或抗肿瘤药物的药剂。

3. 发明申请

US20090244306A1 IMAGE RECORDING AND REPRODUCING APPARATUS 有权
标题翻译：图像记录和再现设备
公开(公告)号：US20090244306A1
公开(公告)日：2009-10-01
申请号：US12415894
申请日：2009-03-31
申请人： Tetsuji Saito
发明人： Tetsuji Saito
IPC分类号： H04N5/225
CPC分类号： H04N1/2166 , H04N1/212 , H04N1/2129 , H04N1/2137 , H04N1/215 , H04N2101/00 , H04N2201/214 , H04N2201/3277
摘要： An image recording and reproducing apparatus that records and reproduces image data shot at a frame rate higher than a normal reproduction rate employed during reproduction of a moving image can generate a still image by attaching still image recording information to at least one frame image included in the recorded image data and combining a plurality of frame images of the recorded image data in accordance with the still image recording information.
摘要翻译：记录和再现以比运动图像再现期间采用的正常再现速率更高的帧速率拍摄的图像数据的图像记录和再现装置可以通过将静止图像记录信息附加到包含在运动图像中的至少一个帧图像来生成静止图像记录图像数据，并根据静止图像记录信息组合记录图像数据的多个帧图像。

4. 发明申请

US20080205306A1 COMMUNICATION APPARATUS AND CONTROL METHOD THEREOF 失效
标题翻译：通信装置及其控制方法
公开(公告)号：US20080205306A1
公开(公告)日：2008-08-28
申请号：US12038713
申请日：2008-02-27
申请人： Tetsuji Saito
发明人： Tetsuji Saito
IPC分类号： H04L5/16
CPC分类号： H04L5/16 , G09G5/006 , G09G2370/047 , G09G2370/12 , H04N5/765 , H04N21/43632
摘要： There is provided a communication apparatus that includes: a data communication unit which performs half-duplex communication of video frame data with an external device on a video frame-by-video frame basis, a switching unit which switches a transmission direction in which the data communication unit transmits the video frame data, a first control unit which controls the data communication unit to include a start command in the video frame data and send the video frame data, as well as controls the switching unit to switch the transmission direction in response to completion of the sending of the video frame data that includes the start command, and a second control unit which controls the switching unit to switch the transmission direction in response to completion of the reception of the video frame data that includes the start command.
摘要翻译：提供了一种通信装置，其包括：数据通信单元，其以视频帧为基础，与外部设备进行视频帧数据的半双工通信;切换单元，切换传输方向，其中数据通信单元发送视频帧数据，控制数据通信单元以在视频帧数据中包括开始命令并发送视频帧数据的第一控制单元，并且控制切换单元响应于完成包括开始命令的视频帧数据的发送;以及第二控制单元，其响应于包括开始命令的视频帧数据的接收完成而控制切换单元切换发送方向。

5. 发明申请

US20050124672A1 N-phenylarylsulfonamide compound drug containing the compound as active ingredient intermediate for the compound and processes for producing the same 有权
标题翻译：含有化合物作为化合物的活性成分中间体的N-苯基芳基磺酰胺化合物药物及其制备方法
公开(公告)号：US20050124672A1
公开(公告)日：2005-06-09
申请号：US10471673
申请日：2002-03-11
申请人： Atsushi Naganawa , Tetsuji Saito , Kaoru Kobayashi , Takayuki Maruyama , Yoshihiko Nakai , Shinsuke Hashimoto
发明人： Atsushi Naganawa , Tetsuji Saito , Kaoru Kobayashi , Takayuki Maruyama , Yoshihiko Nakai , Shinsuke Hashimoto
IPC分类号： C07D307/64 , A61K31/34 , A61K31/341 , A61K31/41 , A61K31/4245 , A61K31/426 , A61K31/427 , A61K31/4402 , A61K31/4406 , A61K31/4439 , A61P1/04 , A61P13/00 , A61P13/02 , A61P29/00 , A61P35/00 , A61P43/00 , C07D213/70 , C07D213/71 , C07D277/20 , C07D277/36 , C07D401/12 , C07D405/12 , C07D413/12 , C07D417/12
CPC分类号： C07D213/70 , C07D277/36 , C07D307/64 , C07D401/12 , C07D405/12 , C07D413/12 , C07D417/12
摘要： An N-phenylarylsulfonylamide compound of formula (I) (R1 is COOH etc.; R2 is hydrogen, methyl, etc.; R3 and R4 are a combination of methyl and methyl, etc.; R5 is isopropyl etc.; Ar is thiazolyl, pyridyl, 5-methyl-2-furyl each optionally substituted with methyl; n is zero or 1), a synthetic intermediate for the compound and a process for its preparation. The compound of formula (I) binds to a prostaglandin E2 receptor, especially an EP1 subtype receptor, and antagonizes it. It is less affected by protein binding, so it has a satisfactory in vivo activity. Therefore, it is considered to be useful as an analgesic, an antipyretic agent, an agent for the treatment of pollakiuria (frequent urination) and/or lower urinary tract disease syndrome or an antineoplastic agent.
摘要翻译：式（I）的N-苯基芳基磺酰胺化合物（R 1）是COOH等; R 2是氢，甲基等; R 3 O >和R 4是甲基和甲基等的组合; R 5是异丙基等; Ar是噻唑基，吡啶基，5-甲基-2-呋喃基任选被甲基取代; n为0或1），化合物的合成中间体及其制备方法。式（I）化合物与前列腺素E 2受体结合，特别是EP 1亚型受体，并拮抗它。蛋白质结合的影响较小，因此具有令人满意的体内活性。因此，认为可用作止痛剂，解热剂，治疗尿频（尿频）和/或下尿路疾病综合征或抗肿瘤药物的药剂。

6. 发明授权

US07235667B2 N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for its preparation 有权
标题翻译： N-苯基芳基磺酰胺化合物，包含该化合物作为活性成分的药物组合物，该化合物的合成中间体及其制备方法
公开(公告)号：US07235667B2
公开(公告)日：2007-06-26
申请号：US10471673
申请日：2002-03-11
申请人： Atsushi Naganawa , Tetsuji Saito , Kaoru Kobayashi , Takayuki Maruyama , Yoshihiko Nakai , Shinsuke Hashimoto
发明人： Atsushi Naganawa , Tetsuji Saito , Kaoru Kobayashi , Takayuki Maruyama , Yoshihiko Nakai , Shinsuke Hashimoto
IPC分类号： C07D277/04 , A61K31/425
CPC分类号： C07D213/70 , C07D277/36 , C07D307/64 , C07D401/12 , C07D405/12 , C07D413/12 , C07D417/12
摘要： An N-phenylarylsulfonylamide compound of formula (I) (R1 is COOH etc.; R2 is hydrogen, methyl, etc.; R3 and R4 are a combination of methyl and methyl, etc.; R5 is isopropyl etc.; Ar is thiazolyl, pyridyl, 5-methyl-2-furyl each optionally substituted with methyl; n is zero or 1), a synthetic intermediate for the compound and a process for its preparation. The compound of formula (I) binds to a prostaglandin E2 receptor, especially an EP1 subtype receptor, and antagonizes it. It is less affected by protein binding, so it has a satisfactory in vivo activity. Therefore, it is considered to be useful as an analgesic, an antipyretic agent, an agent for the treatment of pollakiuria (frequent urination) and/or lower urinary tract disease syndrome or an antineoplastic agent.
摘要翻译：式（I）的N-苯基芳基磺酰胺化合物（R 1）是COOH等; R 2是氢，甲基等; R 3 O >和R 4是甲基和甲基等的组合; R 5是异丙基等; Ar是噻唑基，吡啶基，5-甲基-2-呋喃基任选被甲基取代; n为0或1），化合物的合成中间体及其制备方法。式（I）化合物与前列腺素E 2受体结合，特别是EP 1亚型受体，并拮抗它。蛋白质结合的影响较小，因此具有令人满意的体内活性。因此，认为可用作止痛剂，解热剂，治疗尿频（尿频）和/或下尿路疾病综合征或抗肿瘤药物的药剂。

7. 发明申请

US20060030713A1 N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for its preparation 失效
标题翻译： N-苯基芳基磺酰胺化合物，包含该化合物作为活性成分的药物组合物，该化合物的合成中间体及其制备方法
公开(公告)号：US20060030713A1
公开(公告)日：2006-02-09
申请号：US11239406
申请日：2005-09-30
申请人： Atsushi Naganawa , Tetsuji Saito , Kaoru Kobayashi , Takayuki Maruyama , Yoshihiko Nakai , Shinsuke Hashimoto
发明人： Atsushi Naganawa , Tetsuji Saito , Kaoru Kobayashi , Takayuki Maruyama , Yoshihiko Nakai , Shinsuke Hashimoto
IPC分类号： A61K31/44 , C07C309/28 , C07D277/36 , C07D285/18
CPC分类号： C07D213/70 , C07D277/36 , C07D307/64 , C07D401/12 , C07D405/12 , C07D413/12 , C07D417/12
摘要： An N-phenylarylsulfonylamide compound of formula (I) (R1 is COOH etc.; R2 is hydrogen, methyl, etc.; R3 and R4 are a combination of methyl and methyl, etc.; R5 is isopropyl etc.; Ar is thiazolyl, pyridyl, 5-methyl-2-furyl each optionally substituted with methyl; n is zero or 1), a synthetic intermediate for the compound and a process for its preparation. The compound of formula (I) binds to a prostaglandin E2 receptor, especially an EP1 subtype receptor, and antagonizes it. It is less affected by protein binding, so it has a satisfactory in vivo activity. Therefore, it is considered to be useful as an analgesic, an antipyretic agent, an agent for the treatment of pollakiuria (frequent urination) and/or lower urinary tract disease syndrome or an antineoplastic agent.
摘要翻译：式（I）的N-苯基芳基磺酰胺化合物（R 1）是COOH等; R 2是氢，甲基等; R 3 O >和R 4是甲基和甲基等的组合; R 5是异丙基等; Ar是噻唑基，吡啶基，5-甲基-2-呋喃基任选被甲基取代; n为0或1），化合物的合成中间体及其制备方法。式（I）化合物与前列腺素E 2受体结合，特别是EP 1亚型受体，并拮抗它。蛋白质结合的影响较小，因此具有令人满意的体内活性。因此，认为可用作止痛剂，解热剂，治疗尿频（尿频）和/或下尿路疾病综合征或抗肿瘤药物的药剂。

8. 发明授权

US08649597B2 Image processing apparatus and control method thereof detecting from a histogram a gradation level whose frequency is a peak value 有权
标题翻译：图像处理装置及其控制方法从直方图检测其频率为峰值的灰度级
公开(公告)号：US08649597B2
公开(公告)日：2014-02-11
申请号：US12821699
申请日：2010-06-23
申请人： Yuuki Shindo , Izumi Kanai , Tetsuji Saito
发明人： Yuuki Shindo , Izumi Kanai , Tetsuji Saito
IPC分类号： G06K9/00 , G09G5/02 , G09G5/10 , H04N1/40
CPC分类号： G06T5/009 , G06T5/40
摘要： An image processing apparatus includes a histogram creation unit that creates a histogram from an input image, a detection unit that detects a gradation level of interest from the histogram, a gradation correction parameter generation unit that generates a gradation correction parameter to improve a gradation characteristic in a gradation range around the gradation level of interest, and a correction unit that corrects the gradation of the image using the gradation correction parameter. The detection unit detects, as the gradation level of interest, a gradation level whose frequency is a peak value equal to or more than a predetermined threshold, and which has variation width of frequencies in a predetermined range including this gradation level to be smaller than a predetermined width in the histogram.
摘要翻译：图像处理装置包括从输入图像生成直方图的直方图创建单元，从直方图检测感兴趣的灰度级的检测单元，生成灰度校正参数以提高灰度等级特性的灰度校正参数生成单元围绕感兴趣的灰度等级的灰度范围;以及校正单元，其使用灰度校正参数校正图像的灰度。检测单元检测作为感兴趣的灰度级的频率是等于或大于预定阈值的峰值的灰度级，并且具有包括该灰度级的预定范围内的频率的变化宽度小于直方图中的预定宽度。

9. 发明授权

US08380043B2 Reproducing apparatus and reproducing method 失效
标题翻译：再现装置和再现方法
公开(公告)号：US08380043B2
公开(公告)日：2013-02-19
申请号：US12694590
申请日：2010-01-27
申请人： Tetsuji Saito
发明人： Tetsuji Saito
IPC分类号： H04N9/80
CPC分类号： H04N5/265 , H04N5/225 , H04N5/23293 , H04N5/2355 , H04N5/57 , H04N5/76 , H04N9/80 , H04N21/4318 , H04N21/44008
摘要： Moving image data, obtained by capturing a plurality of frames within the period of a single frame of display output while changing the exposure condition, can be more flexibly produced. For example, such moving image data is stored in a recording portion. When the moving image data is reproduced from the recording portion, a single frame is selected and output by a reproduced frame selecting portion for each period of a single frame of display output. In response to a user operation instructing to make the displayed image darker, a frame having an exposure condition of underexposure is selected and output from the moving image data to be reproduced from the recording portion for each period of a single frame of display output.
摘要翻译：可以更灵活地产生通过在显示输出的单个帧的周期内捕获多个帧而获得的移动图像数据，同时改变曝光条件。例如，这样的运动图像数据被存储在记录部分中。当从记录部分再现运动图像数据时，对于单帧显示输出的每个周期，由再现的帧选择部分选择并输出单个帧。响应于指示使显示图像变暗的用户操作，选择具有曝光不足的曝光条件的帧并且从单帧显示输出的每个周期的从记录部分再现的运动图像数据中输出。

10. 发明申请

US20100329559A1 IMAGE PROCESSING APPARATUS AND CONTROL METHOD THEREOF 有权
标题翻译：图像处理装置及其控制方法
公开(公告)号：US20100329559A1
公开(公告)日：2010-12-30
申请号：US12821699
申请日：2010-06-23
申请人： Yuuki Shindo , Izumi Kanai , Tetsuji Saito
发明人： Yuuki Shindo , Izumi Kanai , Tetsuji Saito
IPC分类号： G06K9/38
CPC分类号： G06T5/009 , G06T5/40
摘要： An image processing apparatus according to the present invention, comprises a histogram creation unit creates a histogram from an input image, a detection unit detects a gradation level of interest from the histogram, a gradation correction parameter generation unit generates a gradation correction parameter to improve a gradation characteristic in a gradation range around the gradation level of interest, and a correction unit corrects the gradation of the image using the gradation correction parameter, wherein the detection unit detects, as the gradation level of interest, a gradation level of which frequency is a peak value equal to or more than a predetermined threshold, and which has variation width of frequencies in a predetermined range including this gradation level to be smaller than a predetermined width in the histogram.
摘要翻译：根据本发明的图像处理装置包括直方图创建单元，从输入图像生成直方图，检测单元从直方图检测感兴趣的灰度等级，灰度校正参数生成单元生成灰度校正参数，以改善校正单元使用灰度校正参数对图像的灰度进行校正，其中检测单元检测出感兴趣的灰度等级为灰度等级的灰度等级峰值等于或大于预定阈值，并且其在包括该灰度级的预定范围内的频率的变化宽度小于直方图中的预定宽度。

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