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    • 9. 发明授权
    • Calcium receptor activator
    • 钙受体活化剂
    • US08106020B2
    • 2012-01-31
    • US12117041
    • 2008-05-08
    • Takeaki OhsuSen TakeshitaYuzuru EtoYusuke Amino
    • Takeaki OhsuSen TakeshitaYuzuru EtoYusuke Amino
    • C07K5/06
    • A61K38/06A61K38/05
    • A calcium receptor activator and compositions containing at least one of the following: γ-Glu-Cys-Gly, γ-Glu-Cys(SNO)-Gly, γ-Glu-Ala, γ-Glu-Gly, γ-Glu-Cys, γ-Glu-Met, γ-Glu-Thr, γ-Glu-Val, γ-Glu-Orn, Asp-Gly, Cys-Gly, Cys-Met, Glu-Cys, Gly-Cys, Leu-Asp, D-Cys, γ-Glu-Met(O), γ-Glu-Val-Val, γ-Glu-Val-Glu, γ-Glu-Val-Lys, γ-Glu-γ-Glu-Val, γ-Glu-Val-NH2, γ-Glu-Val-ol, γ-Glu-Ser, γ-Glu-Tau, γ-Glu-Cys(S-Me)(O), γ-Glu-Leu, γ-Glu-Ile, γ-Glu-t-Leu, γ-Glu-Cys(S-allyl)-Gly, γ-Glu-Gly-Gly, γ-Glu-Val-Phe, γ-Glu-Val-Ser, γ-Glu-Val-Pro, γ-Glu-Val-Arg, γ-Glu-Val-Asp, γ-Glu-Val-Met, γ-Glu-Val-Thr, γ-Glu-Val-His, γ-Glu-Val-Asn, γ-Glu-Val-Gln, γ-Glu-Val-Cys, γ-Glu-Val-Orn, γ-Glu-Ser-Gly, γ-Glu-Cys(S-Me), γ-Glu-Abu-Gly, γ-Glu-Cys(S-Me)-Gly, and γ-Glu-Val-Gly.
    • 钙受体激活剂和含有以下至少一种的组合物:γ-Glu-Cys-Gly,γ-Glu-Cys(SNO)-Gly,γ-Glu-Ala,γ-Glu-Gly,γ-Glu-Cys ,γ-Glu-Met,γ-Glu-Thr,γ-Glu-Val,γ-Glu-Orn,Asp-Gly,Cys-Gly,Cys-Met,Glu-Cys,Gly-Cys,Leu-Asp,D -Cys,γ-Glu-Met(O),γ-Glu-Val-Val,γ-Glu-Val-Glu,γ-Glu-Val-Lys,γ-Glu-γ-Glu-Val, Val-NH 2,γ-Glu-Val-ol,γ-Glu-Ser,γ-Glu-Tau,γ-Glu-Cys(S-Me)(O) γ-Glu-t-Leu,γ-Glu-Cys(S-烯丙基)-Gly,γ-Glu-Gly-Gly,γ-Glu-Val-Phe,γ-Glu-Val-Ser, -Pro,γ-Glu-Val-Arg,γ-Glu-Val-Asp,γ-Glu-Val-Asp,γ-Glu-Val-Met,γ-Glu-Val-Thr, ,γ-Glu-Val-Gln,γ-Glu-Val-Cys,γ-Glu-Val-Orn,γ-Glu-Ser-Gly,γ-Glu-Cys(S-Me) Gly,γ-Glu-Cys(S-Me)-Gly和γ-Glu-Val-Gly。
    • 10. 发明申请
    • CALCIUM RECEPTOR ACTIVATOR
    • 钙受体激活剂
    • US20090239808A1
    • 2009-09-24
    • US12117041
    • 2008-05-08
    • Takeaki OhsuSen TakeshitaYuzuru EtoYusuke Amino
    • Takeaki OhsuSen TakeshitaYuzuru EtoYusuke Amino
    • A61K38/06C07K5/093C07C55/02
    • A61K38/06A61K38/05
    • A calcium receptor activator and compositions containing at least one of the following: γ-Glu-Cys-Gly, γ-Glu-Cys(SNO)-Gly, γ-Glu-Ala, γ-Glu-Gly, γ-Glu-Cys, γ-Glu-Met, γ-Glu-Thr, γ-Glu-Val, γ-Glu-Orn, Asp-Gly, Cys-Gly, Cys-Met, Glu-Cys, Gly-Cys, Leu-Asp, D-Cys, γ-Glu-Met(O), γ-Glu-Val-Val, γ-Glu-Val-Glu, γ-Glu-Val-Lys, γ-Glu-γ-Glu-Val, γ-Glu-Val-NH2, γ-Glu-Val-ol, γ-Glu-Ser, γ-Glu-Tau, γ-Glu-Cys(S-Me)(O), γ-Glu-Leu, γ-Glu-Ile, γ-Glu-t-Leu, γ-Glu-Cys(S-allyl)-Gly, γ-Glu-Gly-Gly, γ-Glu-Val-Phe, γ-Glu-Val-Ser, γ-Glu-Val-Pro, γ-Glu-Val-Arg, γ-Glu-Val-Asp, γ-Glu-Val-Met, γ-Glu-Val-Thr, γ-Glu-Val-His, γ-Glu-Val-Asn, γ-Glu-Val-Gln, γ-Glu-Val-Cys, γ-Glu-Val-Orn, γ-Glu-Ser-Gly, γ-Glu-Cys(S-Me), γ-Glu-Abu-Gly, γ-Glu-Cys(S-Me)-Gly, and γ-Glu-Val-Gly.
    • 钙受体激活剂和含有以下至少一种的组合物:γ-Glu-Cys-Gly,γ-Glu-Cys(SNO)-Gly,γ-Glu-Ala,γ-Glu-Gly,γ-Glu-Cys ,γ-Glu-Met,γ-Glu-Thr,γ-Glu-Val,γ-Glu-Orn,Asp-Gly,Cys-Gly,Cys-Met,Glu-Cys,Gly-Cys,Leu-Asp,D -Cys,γ-Glu-Met(O),γ-Glu-Val-Val,γ-Glu-Val-Glu,γ-Glu-Val-Lys,γ-Glu-γ-Glu-Val, Val-NH2,γ-Glu-Val-ol,γ-Glu-Ser,γ-Glu-Tau,γ-Glu-Cys(S-Me)(O),γ-Glu-Leu, γ-Glu-t-Leu,γ-Glu-Cys(S-烯丙基)-Gly,γ-Glu-Gly-Gly,γ-Glu-Val-Phe,γ-Glu-Val-Ser, -Pro,γ-Glu-Val-Arg,γ-Glu-Val-Asp,γ-Glu-Val-Met,γ-Glu-Val-Thr,γ-Glu-Val-His, ,γ-Glu-Val-Gln,γ-Glu-Val-Cys,γ-Glu-Val-Orn,γ-Glu-Ser-Gly,γ-Glu-Cys(S-Me) Gly,γ-Glu-Cys(S-Me)-Gly和γ-Glu-Val-Gly。