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1. 发明授权

US06511975B1 Spiropiperidine derivatives 失效
标题翻译：螺哌啶衍生物
公开(公告)号：US06511975B1
公开(公告)日：2003-01-28
申请号：US09616092
申请日：2000-07-13
申请人： Takahide Nishi , Takeshi Yamaguchi , Yukiko Iio , Toshiyasu Takemoto , Katsuyoshi Nakajima
发明人： Takahide Nishi , Takeshi Yamaguchi , Yukiko Iio , Toshiyasu Takemoto , Katsuyoshi Nakajima
IPC分类号： C07D41306
CPC分类号： C07D413/06
摘要： A compound of the formula (I) wherein R1 and R2 is a substituted or unsubstituted aryl group, or a substituted or unsubstituted heteroaryl group. A is CH2, CO or SO2. B is a single bond, alkylene or alkenylene. D is O or S. E is alkylene or alkenylene. wherein G is a substituted or unsubstituted cycloalkene ring, or a substituted cycloalkane ring. Ar is a substituted or unsubstituted aryl ring, or a substituted or unsubstituted heteroaryl ring. R3 is alkyl. n is 1-3. The invention includes a pharmacologically acceptable salt, ester or other derivative of a compound of the formula (I). The invention also provides pharmaceutical compositions and methods of treating specified diseases utilizing a compound of formula (I).
摘要翻译：式（I）的化合物，其中R 1和R 2是取代或未取代的芳基，或取代或未取代的杂芳基。 A是CH 2，CO或SO 2。 B是单键，亚烷基或亚烯基。 D是O或S.E是亚烷基或亚烯基，其中G是取代或未取代的环烯烃环或取代的环烷烃环。 Ar是取代或未取代的芳基环，或取代或未取代的杂芳基环。 R3是烷基。 n为1-3。本发明包括式（I）化合物的药学上可接受的盐，酯或其它衍生物。本发明还提供了利用式（I）化合物治疗特定疾病的药物组合物和方法。

2. 发明授权

US6159967A Heterocyclic compounds having tachykinin receptor antagonist activity their preparation and their use 失效
标题翻译：具有速激肽受体拮抗剂活性的杂环化合物的制备及其用途
公开(公告)号：US6159967A
公开(公告)日：2000-12-12
申请号：US758421
申请日：1996-12-02
申请人： Takahide Nishi , Koki Ishibashi , Katsuyoshi Nakajima , Tetsuya Fukazawa , Hitoshi Kurata , Takeshi Yamaguchi , Kazuhiro Ito
发明人： Takahide Nishi , Koki Ishibashi , Katsuyoshi Nakajima , Tetsuya Fukazawa , Hitoshi Kurata , Takeshi Yamaguchi , Kazuhiro Ito
IPC分类号： A61K31/44 , A61K31/4523 , A61K31/4709 , A61K31/495 , A61K31/535 , A61K31/5377 , A61K31/55 , A61K31/553 , A61P17/00 , A61P19/00 , A61P25/00 , C07D263/04 , C07D413/06 , C07D413/14 , C07D417/06 , C07D471/10 , C07D487/10 , C07D491/10 , C07D495/10 , C07D498/10 , C07D265/00 , C07D265/30 , C07D295/00
CPC分类号： C07D263/04 , C07D413/06 , C07D413/14 , C07D471/10 , C07D491/10 , C07D495/10
摘要： Compounds of the formula and quaternary ammonium ions thereof, wherein R.sup.1 and R.sup.2 are the same or different and are carbocyclic aryl or aromatic heterocyclic; A is methylene, carbonyl or sulfonyl; B is a single bond, C.sub.1 -C.sub.4 alkylene or C.sub.2 -C.sub.4, alkenylene; D is oxygen; E is C.sub.2 alkylene; G is C.sub.1 -C.sub.4 alkylene or C.sub.2 -C.sub.4 alkenylene; and L is --C(R.sup.4)(R.sup.5), wherein R.sup.4 and R.sup.5 together with the carbon atom to which they are attached represent a C.sub.5 -C.sub.10 cycloalkyl or a C.sub.5 -C.sub.10 heterocyclic. Especially preferred are compounds wherein L represents ##STR1## wherein J is a C.sub.1 -C.sub.6 alkylene; Ar is a ring carbocyclic or aromatic heterocyclic and S*.fwdarw.O is a sulfoxide in which the sulfur atom is in the 5-configuration. The compounds have tachykinin receptor antagonist activity and exhibit an activity against both the NK.sub.1 and NK.sub.2 receptors.
摘要翻译：式及其季铵离子的化合物，其中R 1和R 2相同或不同，为碳环芳基或芳族杂环; A是亚甲基，羰基或磺酰基; B是单键，C 1 -C 4亚烷基或C 2 -C 4亚烯基; D是氧; E为C2亚烷基; G是C 1 -C 4亚烷基或C 2 -C 4亚烯基; 并且L是-C（R 4）（R 5），其中R 4和R 5与它们所连接的碳原子一起代表C5-C10环烷基或C5-C10杂环。特别优选的是其中L表示其中J为C1-C6亚烷基的化合物; Ar是环碳环或芳族杂环，并且S * - > O是其中硫原子为5构型的亚砜。该化合物具有速激肽受体拮抗剂活性，并表现出对NK1和NK2受体的活性。

3. 发明授权

US06448247B1 Method for treating an inflammatory disease 失效
标题翻译：治疗炎性疾病的方法
公开(公告)号：US06448247B1
公开(公告)日：2002-09-10
申请号：US09533061
申请日：2000-03-22
申请人： Takahide Nishi , Koki Ishibashi , Katsuyoshi Nakajima , Tetsuya Fukazawa , Hitoshi Kurata , Takeshi Yamaguchi , Kazuhiro Ito
发明人： Takahide Nishi , Koki Ishibashi , Katsuyoshi Nakajima , Tetsuya Fukazawa , Hitoshi Kurata , Takeshi Yamaguchi , Kazuhiro Ito
IPC分类号： A61K315375
CPC分类号： C07D263/04 , C07D413/06 , C07D413/14 , C07D471/10 , C07D491/10 , C07D495/10
摘要： Compounds of the formula and quaternary ammonium ions thereof, wherein R1 and R2 are the same or different and are carbocyclic aryl or aromatic heterocyclic; A is methylene, carbonyl or sulfonyl; B is a single bond, C1-C4 alkylene or C2-C4 alkenylene; D is oxygen or sulfur; E is C2-C6 alkylene, C1-C6 haloalkylene, C3-C6 cycloalkane-1,1-diyl or C3-C6-cycloalkane-1,1-diylmethyl; G is C1-C4 alkylene or C2-C4 alkenylene; and L is —NR3 or —C(R4)(R5), wherein R3 is a carbocyclic aryl or an aromatic heterocyclic; R4 is hydrogen, carbocyclic aryl or aromatic heterocyclic; R5 is —COR6, C1-C6 alkyl, C1-C6 alkoxy, amino, or acylamino, wherein R6 is C1-C6 alkyl or C1-C6 alkoxy, or R4 and R5 together with the carbon atom to which they are attached represent a C5-C10 cycloalkyl or a C5-C10 heterocyclic. The compounds have tachykinin receptor antagonist activity and exhibit an activity against both the NK1 and NK2 receptors.
摘要翻译：其中式和季铵离子的化合物，其中R 1和R 2相同或不同，为碳环芳基或芳族杂环; A是亚甲基，羰基或磺酰基; B是单键，C1-C4亚烷基或C2-C4亚烯基; D是氧或硫; E为C2-C6亚烷基，C1-C6卤代亚烷基，C3-C6环烷烃-1,1-二基或C3-C6-环烷烃-1,1-二基甲基; G是C 1 -C 4亚烷基或C 2 -C 4亚烯基; 并且L是-NR 3或-C（R 4）（R 5），其中R 3是碳环芳基或芳族杂环; R4是氢，碳环芳基或芳族杂环; R 5是-COR 6，C 1 -C 6烷基，C 1 -C 6烷氧基，氨基或酰氨基，其中R 6是C 1 -C 6烷基或C 1 -C 6烷氧基，或者R 4和R 5与它们所连接的碳原子一起代表C5 -C 10环烷基或C 5 -C 10杂环。该化合物具有速激肽受体拮抗剂活性，并表现出对NK1和NK2受体的活性。

4. 发明授权

US06362179B1 Salts of an optically-active sulfoxide derivative 失效
标题翻译：光学活性亚砜衍生物的盐
公开(公告)号：US06362179B1
公开(公告)日：2002-03-26
申请号：US09447401
申请日：1999-11-23
申请人： Takahide Nishi , Takeshi Yamaguchi
发明人： Takahide Nishi , Takeshi Yamaguchi
IPC分类号： A61K315377
CPC分类号： C07D495/10
摘要： Hydrochloride of fumarate of 1-{2-[(2R)-(3,4-dichlorophenyl)-4-(3,4,5-trimethyoxybenzoyl)morpholin-2-yl]ethyl}spiro[benzo(c)thiophene-1(3H),4′-piperidin]-(2S)-oxide. These compounds have good oral adsorption and exhibit markedly excellent antagonistic action against both NK1 receptors and NK2 receptors. These compounds are useful as an active ingredient in pharmaceutical compositions for administering to patients for treatment of tachykinin-medicated diseases.
摘要翻译：富马酸盐的1- {2 - [（2R） - （3,4-二氯苯基）-4-（3,4,5-三甲氧基苯甲酰基）吗啉-2-基]乙基}螺[苯并[c]噻吩-1 （3H），4'-哌啶] - （2S） - 氧化物。这些化合物具有良好的口服吸附，并且对NK1受体和NK2受体均表现出显着优异的拮抗作用。这些化合物可用作药物组合物中的活性成分，用于给予患者治疗速激肽药物疾病。

5. 发明授权

US06288059B1 Acylated hetero-alicyclic derivatives 失效
标题翻译：酰化的杂脂环衍生物
公开(公告)号：US06288059B1
公开(公告)日：2001-09-11
申请号：US09586728
申请日：2000-06-05
申请人： Takahide Nishi , Takeshi Yamaguchi
发明人： Takahide Nishi , Takeshi Yamaguchi
IPC分类号： A61K315377
CPC分类号： C07D265/30 , C07D405/06 , C07D413/06 , C07D417/14 , C07D495/10
摘要： A compound of formula (I), a pharmaceutically acceptable salt or ester or other derivative thereof: R1 is optionally substituted cycloalkyl or optionally substituted saturated heterocyclic group. R2 is optionally substituted aryl or optionally substituted heteroaryl. A is methylene, carbonyl or sulfonyl. B is a single bond, alkylene or alkenylene. D is oxygen or sulfur. G is alkylene or alkenylene. L is —N(R3)— or —C(R4)(R5)—. R3 is optionally substituted aryl or optionally substituted heteroaryl. R4 is H, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted cycloalkyl or optionally substituted saturated heterocyclic group. R5 is alkyl optionally substituted with amino, amino, optionally substituted acylamino, OH, optionally substituted hydroxyalkyl, alkoxy or —CO—R6. R6 is alkyl, alkoxy or amine residue. R4 together with R5 forms a cycloalkane ring, cycloalkene ring, or saturated heterocyclic ring. R7 is alkyl. Z is two hydrogens or oxygen. n is 0. 1 or 2. These compounds have selective antagonistic activity against the NK2 receptor.
摘要翻译：式（I）的化合物，其药学上可接受的盐或酯或其它衍生物：R1是任选取代的环烷基或任选取代的饱和杂环基。 R2是任选取代的芳基或任选取代的杂芳基。 A是亚甲基，羰基或磺酰基。 B是单键，亚烷基或亚烯基。 D是氧或硫。 G是亚烷基或亚烯基。 L是-N（R 3） - 或-C（R 4）（R 5） - 。 R3是任选取代的芳基或任选取代的杂芳基。 R 4是H，任选取代的芳基，任选取代的杂芳基，任选取代的环烷基或任选取代的饱和杂环基。 R5是任选被氨基，氨基，任选取代的酰基氨基，OH，任选取代的羟烷基，烷氧基或-CO-R 6取代的烷基。 R6是烷基，烷氧基或胺残基。 R4与R5一起形成环烷烃环，环烯烃环或饱和杂环。 R7是烷基。 Z是两个氢或氧。 n为0.1或2.这些化合物对NK2受体具有选择性拮抗活性。

6. 发明授权

US11159030B2 Battery pack, secondary battery protecting integrated circuit, battery monitoring module, and data reading method 有权
公开(公告)号：US11159030B2
公开(公告)日：2021-10-26
申请号：US15911308
申请日：2018-03-05
申请人： Takeshi Yamaguchi
发明人： Takeshi Yamaguchi
IPC分类号： H02J7/00 , H01M10/02 , H01M10/42 , H01M10/48 , H01M50/20 , H01M50/209
摘要： A battery pack includes a secondary battery, a secondary battery protecting integrated circuit configured to protect the secondary battery, at least one sensor configured to output a fault signal indicating sensing of a fault in the battery pack or an electronic apparatus including the battery pack, a detecting circuit configured to output a fault detection signal indicating a detection of the fault signal, a delay circuit configured to output a pulse delaying from the fault detection signal, and a counter configured to count a number of generating the pulse, the counter having at least N bits (N is an integer greater than 1), wherein the counter stops an operation until a count of 2(N-1).

7. 发明授权

US08842335B2 Apparatus, method, and non-transitory computer readable medium to achieve appropriate color reproduction characteristics 有权
标题翻译：装置，方法和非暂时的计算机可读介质，以实现适当的色彩再现特性
公开(公告)号：US08842335B2
公开(公告)日：2014-09-23
申请号：US12831653
申请日：2010-07-07
申请人： Takeshi Yamaguchi
发明人： Takeshi Yamaguchi
IPC分类号： H04N1/60
CPC分类号： H04N1/6088 , H04N1/6097
摘要： Disclosed is an information processing apparatus including: a control section to obtain output condition information to show an output condition when a color chart is output, to obtain colorimetric data obtained by measuring the color chart, to create a color conversion profile based on the obtained colorimetric data, and to embed the output condition information in the created color conversion profile according to an order determined in advance.
摘要翻译：公开了一种信息处理设备，包括：控制部分，用于获得输出条件信息，以便在输出彩色图表时显示输出条件，以获得通过测量色彩图得到的色度数据，以便根据获得的色度产生颜色转换曲线数据，并且根据预先确定的顺序将输出条件信息嵌入到所创建的颜色转换简档中。

8. 发明授权

US08797614B2 Creating a color conversion table by performing color conversion using a 3D and 1D table after limiting total color material amount 有权
标题翻译：通过在限制总颜色材料量之后使用3D和1D表执行颜色转换来创建颜色转换表
公开(公告)号：US08797614B2
公开(公告)日：2014-08-05
申请号：US13713195
申请日：2012-12-13
申请人： Takeshi Yamaguchi
发明人： Takeshi Yamaguchi
IPC分类号： H04N1/60
CPC分类号： H04N1/60 , H04N1/6019
摘要： Disclosed are a device, a method, and a storage medium to create a color conversion table. According to one implementation, a color conversion table creating device includes, a color material amount limiting processing section; a first color conversion processing section; a second color conversion processing section; a combining section; a color material amount limiting inverse conversion processing section; and an output value determining section. The color material amount limiting processing section performs color material amount limiting of an input value in the color conversion table. The color material limiting inverse conversion processing section performs inverse conversion of the color material amount limiting after color conversion and combining the CMYK components. The output value determining section sets the inverted CMYK color components as an output value in the color conversion table.
摘要翻译：公开了一种用于创建颜色转换表的设备，方法和存储介质。根据一个实施方案，一种颜色转换表创建装置包括：色材量限制处理部分; 第一颜色转换处理部; 第二颜色转换处理部; 组合部分; 色材量限制逆变换处理部; 和输出值确定部分。颜色材料量限制处理部分对颜色转换表中的输入值进行颜色量限制。色材限制逆变换处理部对颜色转换后的色材量限制进行逆变换，并组合CMYK成分。输出值确定部分将反转的CMYK颜色分量设置为颜色转换表中的输出值。

9. 发明授权

US08487345B2 Information recording and reproducing device 失效
标题翻译：信息记录和再现装置
公开(公告)号：US08487345B2
公开(公告)日：2013-07-16
申请号：US12885952
申请日：2010-09-20
申请人： Takayuki Tsukamoto , Tsukasa Nakai , Akira Kikitsu , Takeshi Yamaguchi , Sumio Ashida
发明人： Takayuki Tsukamoto , Tsukasa Nakai , Akira Kikitsu , Takeshi Yamaguchi , Sumio Ashida
IPC分类号： H01L21/02
CPC分类号： G11B11/002 , B82Y10/00 , G11B9/04 , G11B9/149 , G11B11/08 , G11C11/56 , G11C11/5678 , G11C13/0004 , G11C13/003 , G11C16/0483 , G11C2211/565 , G11C2213/53 , G11C2213/56 , G11C2213/71 , G11C2213/72 , G11C2213/75 , G11C2213/78 , G11C2213/79 , H01L27/2409 , H01L27/2481 , H01L45/06 , H01L45/1233 , H01L45/1246 , H01L45/1286 , H01L45/144 , H01L45/1683
摘要： According to one embodiment, an information recording and reproducing device includes a stacked body. The stacked body includes a first layer, a second layer and a recording layer provided between the first layer and the second layer. The recording layer includes a phase-change material and a crystal nucleus. The phase-change material is capable of reversely changing between a crystal state and an amorphous state by a current supplied via the first layer and the second layer. The crystal nucleus is provided in contact with the phase-change material and includes a crystal nucleus material having a crystal structure identical to a crystal structure of the crystal state of the phase-change material, and a crystal nucleus coating provided on a surface of the crystal nucleus material and having a composition different from a composition of the crystal nucleus material.
摘要翻译：根据一个实施例，信息记录和再现装置包括堆叠体。层叠体包括设置在第一层和第二层之间的第一层，第二层和记录层。记录层包括相变材料和晶核。相变材料能够通过经由第一层和第二层提供的电流在晶体状态和非晶状态之间反向变化。提供与相变材料接触的晶核，并且包括具有与相变材料的晶体状态的晶体结构相同的晶体结构的晶核材料，以及设置在相变材料的表面上的晶核涂层并且具有与晶核材料的组成不同的组成的晶核材料。

10. 发明授权

US08416606B2 Information recording and reproducing device 有权
标题翻译：信息记录和再现装置
公开(公告)号：US08416606B2
公开(公告)日：2013-04-09
申请号：US13040823
申请日：2011-03-04
申请人： Takayuki Tsukamoto , Tsukasa Nakai , Chikayoshi Kamata , Mariko Hayashi , Fumihiko Aiga , Takeshi Yamaguchi
发明人： Takayuki Tsukamoto , Tsukasa Nakai , Chikayoshi Kamata , Mariko Hayashi , Fumihiko Aiga , Takeshi Yamaguchi
IPC分类号： G11C11/00
CPC分类号： G11B9/04 , G11C13/0004 , G11C13/0007 , G11C13/003 , G11C2213/51 , G11C2213/56 , G11C2213/71 , G11C2213/72 , G11C2213/75 , G11C2213/79 , H01L27/101 , H01L27/2409 , H01L27/2481 , H01L45/04 , H01L45/1233 , H01L45/126 , H01L45/147
摘要： According to one embodiment, an information recording and reproducing device includes a recording layer and a driving unit. The recording layer includes a first layer containing a first compound. The first compound includes a first positive ion element. The first positive ion element is made of a transition metal element and serves as a first positive ion. The second positive ion element serves as a second positive ion. The driving unit is configured to generate a phase change in the recording layer and to record information by at least one of application of a voltage and application of a current to the recording layer. The coordination number of the first positive ion element at a position of a second coordination of the second positive ion element is 80% or more and less than 100% of the coordination number when the first compound is assumed to be a perfect crystal.
摘要翻译：根据一个实施例，信息记录和再现装置包括记录层和驱动单元。记录层包括含有第一化合物的第一层。第一化合物包括第一正离子元素。第一正离子元件由过渡金属元素制成并用作第一正离子。第二正离子元素用作第二正离子。驱动单元被配置为在记录层中产生相变，并且通过施加电压和施加电流到记录层中的至少一个来记录信息。当假设第一化合物为完美晶体时，第二正离子元件的第二配位位置处的第一正离子元素的配位数为配位数的80％以上且小于配位数的100％。

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