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1. 发明授权

US06590102B1 Process for producing piperidinecarbinols 有权
公开(公告)号：US06590102B1
公开(公告)日：2003-07-08
申请号：US09721762
申请日：2000-11-27
申请人： Shu-zhong Wang , Takashi Okazoe , Yasushi Matsumura , Nobuaki Mori , Jiro Nishino , Kazuhiro Ookura
发明人： Shu-zhong Wang , Takashi Okazoe , Yasushi Matsumura , Nobuaki Mori , Jiro Nishino , Kazuhiro Ookura
IPC分类号： C07D21140
CPC分类号： C07D211/22 , C07C255/41 , C07D211/78
摘要： A process for producing a piperidinecarbinol represented by the general formula (2), which comprises reducing the trans isomer of a compound represented by the general formula (1): wherein R1 is a hydrogen atom, a lower alkyl group or an aralkyl group, R2 is a hydrogen atom, a lower alkyl group, an aryl group or an aralkyl group, and X is a hydrogen atom, a halogen atom, an alkyl group, an aryl group, an aralkyl group, an alkoxy group, a dialkylamino group, an alkylthio group, an arylthio group or CmF2m+1— wherein m is an integer of from 1 to 20.

2. 发明授权

US06433179B1 Process for producing paroxetine 失效
标题翻译：帕罗西汀生产工艺
公开(公告)号：US06433179B1
公开(公告)日：2002-08-13
申请号：US08861393
申请日：1997-05-21
申请人： Shu-zhong Wang , Yasushi Matsumura
发明人： Shu-zhong Wang , Yasushi Matsumura
IPC分类号： C07D40512
CPC分类号： C07D405/12
摘要： A process for producing a paroxetine represented by the following formula (4), which comprises reacting an N-alkylpiperidine represented by the following general formula (1) with a haloformic acid ester represented by the general formula (2) to prepare an alkoxycarbonylpiperidine represented by the general formula (3), and hydrolyzing the alkoxycarbonylpiperidine under alkaline conditions: wherein each of R1 and R2 is a lower alkyl group, a lower cycloalkyl group, an aralkyl group or CmF2m+1 (wherein m is an integer of from 1 to 6), and X is a halogen atom.
摘要翻译：一种由下述通式（4）表示的帕罗西汀生产方法，其特征在于：将下述通式（1）表示的N-烷基哌啶与通式（2）表示的卤代甲酸酯反应，制备由通式（3），在碱性条件下水解烷氧基羰基哌啶：其中R1和R2分别为低级烷基，低级环烷基，芳烷基或CmF2m + 1（其中m为1〜6的整数）），X为卤素原子。

3. 发明授权

US06476228B1 Process for producing piperidinecarbinols 有权
标题翻译：制备哌啶甲醇的方法
公开(公告)号：US06476228B1
公开(公告)日：2002-11-05
申请号：US09666585
申请日：2000-09-20
申请人： Shu-zhong Wang , Takashi Okazoe , Yasushi Matsumura , Nobuaki Mori , Jiro Nishino , Kazuhiro Ookura
发明人： Shu-zhong Wang , Takashi Okazoe , Yasushi Matsumura , Nobuaki Mori , Jiro Nishino , Kazuhiro Ookura
IPC分类号： C07D21140
CPC分类号： C07D211/22 , C07C255/41 , C07D211/78
摘要： A process for producing a piperidinecarbinol represented by the general formula (2), which comprises reducing the trans isomer of a compound represented by the general formula (1): wherein R1 is a hydrogen atom, a lower alkyl group or an aralkyl group, R2 is a hydrogen atom, a lower alkyl group, an aryl group or an aralkyl group, and X is a hydrogen atom, a halogen atom, an alkyl group, an aryl group, an aralkyl group, an alkoxy group, a dialkylamino group, an alkylthio group, an arylthio group or CmF2m+1— wherein m is an integer of from 1 to 20.
摘要翻译：一种制备由通式（2）表示的哌啶甲醇的方法，其包括降低由通式（1）表示的化合物的反式异构体：其中R1是氢原子，低级烷基或芳烷基，R2 是氢原子，低级烷基，芳基或芳烷基，X是氢原子，卤素原子，烷基，芳基，芳烷基，烷氧基，二烷基氨基，烷硫基，芳硫基或CmF2m + 1-，其中m为1〜20的整数。

4. 发明授权

US06197960B1 Process for producing piperidinecarbinols 失效
标题翻译：制备哌啶甲醇的方法
公开(公告)号：US06197960B1
公开(公告)日：2001-03-06
申请号：US08835646
申请日：1997-04-11
申请人： Shu-zhong Wang , Takashi Okazoe , Yasushi Matsumura , Nobuaki Mori , Jiro Nishino , Kazuhiro Ookura
发明人： Shu-zhong Wang , Takashi Okazoe , Yasushi Matsumura , Nobuaki Mori , Jiro Nishino , Kazuhiro Ookura
IPC分类号： C07D21140
CPC分类号： C07D211/22 , C07C255/41 , C07D211/78
摘要： A process for producing a piperidinecarbinol represented by the general formula (2), which comprises reducing the trans isomer of a compound represented by the general formula (1): wherein R1 is a hydrogen atom, a lower alkyl group or an aralkyl group, R2 is a hydrogen atom, a lower alkyl group, an aryl group or an aralkyl group, and X is a hydrogen atom, a halogen atom, an alkyl group, an aryl group, an aralkyl group, an alkoxy group, a dialkylamino group, an alkylthio group, an arylthio group or CmF2m+1— wherein m is an integer of from 1 to 20.
摘要翻译：一种制备由通式（2）表示的哌啶甲醇的方法，其包括降低由通式（1）表示的化合物的反式异构体：其中R1是氢原子，低级烷基或芳烷基，R2 是氢原子，低级烷基，芳基或芳烷基，X是氢原子，卤素原子，烷基，芳基，芳烷基，烷氧基，二烷基氨基，烷硫基，芳硫基或CmF2m + 1-，其中m为1〜20的整数。

5. 发明授权

US08557376B2 Polishing pad 有权
标题翻译：抛光垫
公开(公告)号：US08557376B2
公开(公告)日：2013-10-15
申请号：US12678207
申请日：2008-09-24
申请人： Yasushi Matsumura , Masataka Takagi
发明人： Yasushi Matsumura , Masataka Takagi
IPC分类号： B32B3/26 , B24D11/02
CPC分类号： B24B37/24 , B24B37/22 , Y10T428/249981 , Y10T428/249989 , Y10T428/249991
摘要： A polishing pad which suppresses occurrence of a scratch or a roll-off on an object to be polished so that flatness is improved is provided. A polishing pad 1 is comprised a polyurethane sheet 2 having a polishing surface P for performing polishing processing to an object to be polished and an elastic sheet 3 having elasticity joined on a surface of the polyurethane sheet 2 on the opposite side to the polishing surface P. The polyurethane sheet 2 is set higher in compressibility than the elastic sheet 3, and is set lower in A hardness than the elastic sheet 3. The elastic sheet 3 is set at 1% or more in compressibility, and is set at 90 degrees or less in A hardness. Further, both of the polyurethane sheet 2 and the elastic sheet 3 are formed to have a thickness of 0.2 mm or more. The flexibility of the polyurethane sheet 2 is exerted during polishing processing so that the polyurethane sheet 2 deforms to press the polishing surface P approximately evenly on the object to be polished.
摘要翻译：提供一种抛光垫，其可以抑制抛光对象上的刮擦或滚降的发生，从而提高平坦度。抛光垫1包括：聚氨酯片材2，其具有用于对待抛光物体进行抛光处理的抛光面P和在与抛光面P相反的一侧的聚氨酯片材2的表面上具有弹性的弹性片材3 聚氨酯片材2的压缩性比弹性片材3高，并且设定为低于弹性片材3的A硬度。弹性片材3的压缩率设定为1％以上，设定为90度， A硬度较低。此外，聚氨酯片材2和弹性片材3都形成为具有0.2mm以上的厚度。在抛光加工过程中，发挥聚氨酯片材2的柔软性，使得聚氨酯片材2发生变形，将抛光面P大致均匀地压在待研磨物上。

6. 发明申请

US20120265405A1 VEHICULAR ELECTRONIC CONTROL APPARATUS 有权
标题翻译：车用电子控制装置
公开(公告)号：US20120265405A1
公开(公告)日：2012-10-18
申请号：US13426700
申请日：2012-03-22
申请人： Yasushi Matsumura , Eiichi Kamei
发明人： Yasushi Matsumura , Eiichi Kamei
IPC分类号： G06F7/00 , B60R21/00
CPC分类号： B60R16/0238 , B60W50/0225 , B60W50/04 , B60W2050/0006 , B60W2050/041
摘要： A vehicular electronic control apparatus includes a mother unit having a microcomputer, a plurality of ECU modules connected to the mother unit detachably and configured to execute respective vehicle controls, an operation data communication section for communicating with the microcomputer operation data used by the plurality of ECU modules in executing respective control operation processing, and alternative operation execution section for causing at least one of the other ECU modules and the microcomputer to execute, as an alternative operation, at least a part of the arithmetic operation processing, which is to be executed by at least one of the plurality of the ECU modules.
摘要翻译：一种车载电子控制装置，包括：具有微电脑的母单元，可拆卸地连接到母单元的多个ECU模块，用于执行各自的车辆控制;操作数据通信部，用于与多个ECU使用的微机操作数据进行通信; 执行相应的控制操作处理的模块以及替代操作执行部分，用于使其他ECU模块和微计算机中的至少一个作为替代操作执行至少一部分算术运算处理，该运算处理将由所述多个ECU模块中的至少一个。

7. 发明授权

US07530310B2 Metal holder with electrode pin, method of manufacturing the metal holder, and gas generator 失效
标题翻译：具有电极针的金属支架，金属支架的制造方法和气体发生器
公开(公告)号：US07530310B2
公开(公告)日：2009-05-12
申请号：US10594271
申请日：2005-03-30
申请人： Akitoshi Hironaka , Yasushi Matsumura , Dairi Kubo
发明人： Akitoshi Hironaka , Yasushi Matsumura , Dairi Kubo
IPC分类号： F42B3/10 , F42B3/103
CPC分类号： F42B3/198 , B60R2021/26029
摘要： A metal holder, and a method of producing the same, with electrode pins suitably used for a gas generator having a structure that can prevent electrode pins from being burst forth easily even when the gas generator is brought into action under high temperature. The metal holder with electrode pins includes a metal holder and at least two electrode pins for allowing passage of electrical current. Each electrode pin is larger in diameter at its head portion than at its terminal portion. Plastic members are arranged to surround a part of the respective electrode pins circumferentially. Holes for the respective electrode pins to pass through the holder are formed in the holder, and the electrode pins are fixed to the holes via the plastic members, each hole having a diameter-reduction portion at a part thereof.
摘要翻译：金属保持器及其制造方法，具有适合用于具有能够容易地防止电极针突出的结构的气体发生器的电极针，即使当气体发生器在高温下起作用时。具有电极引脚的金属保持器包括金属保持器和用于允许电流通过的至少两个电极引脚。每个电极引脚在其头部处的直径比在其端部处的直径大。塑料构件被布置成围绕各个电极销的一部分周向包围。用于各电极针穿过保持器的孔形成在保持器中，并且电极销通过塑料构件固定到孔，每个孔的一部分具有直径减小部分。

8. 发明申请

US20080255385A1 METHOD FOR PRODUCING OPTICALLY ACTIVE (4E)-5-CHLORO-2-ISOPROPYL-4-PENTENOIC ACID OR BASIC AMINO ACID SALT THEREOF 审中-公开
标题翻译：生产光学活性（4E）-5-氯-2-异丙基-4-苯基丙酸或其碱性氨基酸盐的方法
公开(公告)号：US20080255385A1
公开(公告)日：2008-10-16
申请号：US12139553
申请日：2008-06-16
申请人： Mayumi Makino , Kazuhisa Sakata , Yasushi Matsumura
发明人： Mayumi Makino , Kazuhisa Sakata , Yasushi Matsumura
IPC分类号： C07C69/65 , C07C209/68 , C07C57/03
CPC分类号： C07C229/26 , C07B57/00 , C07B2200/07 , C07C51/487 , C07C57/52
摘要： To provide a method for producing an optically active (4E)-5-chloro-2-isopropyl-4-pentenoic acid, a basic amino acid salt thereof or an optically active (4E)-5-chloro-2-isopropyl-4-pentenoic acid ester with high yield and high optical purity by simple operation.An optically active (4E)-5-chloro-2-isopropyl-4-pentenoic acid is obtained by precipitating a basic amino acid salt of optically active (4E)-5-chloro-2-isopropyl-4-pentenoic acid from a solvent solution containing an optical isomer mixture of (4E)-5-chloro-2-isopropyl-4-pentenoic acid and an optically active basic amino acid or a salt thereof, and then the basic amino acid salt of optically active (4E)-5-chloro-2-isopropyl-4-pentenoic acid is subjected to a desalting reaction. Further, an esterification reaction is carried out to obtain an optically active (4E)-5-chloro-2-isopropyl-4-pentenoic acid ester.
摘要翻译：为了提供一种制备光学活性（4E）-5-氯-2-异丙基-4-戊烯酸，其碱性氨基酸盐或光学活性（4E）-5-氯-2-异丙基-4-戊烯酸的方法，戊烯酸酯，产率高，光学纯度高。通过从溶剂中沉淀光学活性（4E）-5-氯-2-异丙基-4-戊烯酸的碱性氨基酸盐获得光学活性（4E）-5-氯-2-异丙基-4-戊烯酸（4E）-5-氯-2-异丙基-4-戊烯酸和光学活性碱性氨基酸或其盐的光学异构体混合物，然后将光学活性（4E）-5的碱性氨基酸盐 - 氯-2-异丙基-4-戊烯酸进行脱盐反应。此外，进行酯化反应以获得光学活性（4E）-5-氯-2-异丙基-4-戊烯酸酯。

9. 发明申请

US20070163457A1 Igniter and gas generator having the same 审中-公开
标题翻译：点火器和气体发生器具有相同的功能
公开(公告)号：US20070163457A1
公开(公告)日：2007-07-19
申请号：US11578110
申请日：2005-04-15
申请人： Yasushi Matsumura , Junya Maruyama , Akitoshi Hironaka , Kazumasa Kurita , Kenjiro Ikeda
发明人： Yasushi Matsumura , Junya Maruyama , Akitoshi Hironaka , Kazumasa Kurita , Kenjiro Ikeda
IPC分类号： F42C11/00 , F42C19/02
CPC分类号： F42B3/103 , B60R2021/26029 , F42B3/124 , F42B3/195
摘要： Provided is a squib for attaining a normal ignition of gas generants even when an adhesion state of the plug with enhancers is released by vibration or impact and a gas generator having the squib. A squib including a plug 13, two or more electrode pins 14 which pass through the plug 13 and respectively provided with a head 25, a bridge wire 16 connecting spaces between the respective heads 25 on at least two electrode pins 14 among the electrode pins 14, and ignition charge 10 which are ignited by the bridge wire 16 electrified via the electrode pins 14, wherein the plug 13 is a cured composition of thermosetting resins, the electrode pin 14 in which the bridge wire 16 is connected to the head 25 passes through the plug 13, with a predetermined distance A kept between the head 25 and the plug 13, and at least the head 25 and the bridge wire 16 are enclosed by the ignition charge 10, which is a solid, and fixed to the plug 13.
摘要翻译：即使当通过振动或冲击释放具有增强剂的塞子的粘附状态以及具有爆管的气体发生器时，也提供用于获得气体发生剂的正常点火的爆管。包括插头13的点火器，穿过插头13并分别设置有头部25的两个或更多个电极引脚14，连接电极引脚14中的至少两个电极引脚14上的各个头部25之间的空间的桥接线16 ，以及点火电荷10，其被桥接线16点燃，经由电极销14通电，其中插头13是热固性树脂的固化组合物，桥接电线16连接到头部25的电极销14穿过具有保持在头部25和插头13之间的预定距离A的插头13，并且至少头部25和桥接线16被固体的点火充电器10包围并固定到插头13。

10. 发明申请

US20060058529A1 Method for producing 3-substituted 2-chloro-5-fluoro-pyridine or its salt 失效
标题翻译：制备3-取代的2-氯-5-氟 - 吡啶或其盐的方法
公开(公告)号：US20060058529A1
公开(公告)日：2006-03-16
申请号：US11265179
申请日：2005-11-03
申请人： Yasushi Matsumura , Nobuaki Mori , Yasuhiro Yamada
发明人： Yasushi Matsumura , Nobuaki Mori , Yasuhiro Yamada
IPC分类号： C07D213/84 , C07D213/46
CPC分类号： C07D213/80
摘要： To provide a method for producing a 3-substituted 2-chloro-5-fluoro-pyridine or its salt in high yield from a readily available material through a short process under mild reaction conditions using a reagent which is easy for handling and simple in the reaction operation. Namely, a method for producing the following compound (2) or its salt which comprises selectively reducing a chlorine atom at the 6-position of the following compound (1) or its salt, is provided. Further, a method for producing the following compound (4) or its salt which comprises substituting a Z1 group of the following compound (2) or its salt obtained by the reduction reaction, by a Z2 group, is provided. Here, Z1 is —CO2R1, etc., and R1 is a hydrogen atom, an alkyl group, an alkenyl group, an aryl group, an aralkyl group or a cycloalkyl group. Z2 is a group different from Z1 and is —CO2R5, etc., and R5 is an alkyl group, an alkenyl group, an aryl group, an aralkyl group or a cycloalkyl group.
摘要翻译：提供一种通过使用容易处理的试剂在温和的反应条件下通过短时间过程从容易获得的材料以高产率制备3-取代的2-氯-5-氟 - 吡啶或其盐的方法，反应操作。即，提供了下述化合物（1）或其盐选择性还原6-位的氯原子的下述化合物（2）或其盐的制造方法。此外，制备下列化合物（4）或其盐的方法，该方法包括用下列化合物（2）或其还原反应得到的盐代替Z ^{2 组。这里，Z 1是-CO 2 R 1等，R 1是氢原子，烷基，烯基，芳基，芳烷基或环烷基。 Z 2是与Z 1不同的基团，并且是-CO 2 R 5等，R 2 5是烷基，烯基，芳基，芳烷基或环烷基环}

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