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1. 发明申请

US20060106221A1 Process for the preparation of thiazolidinedione derivatives 审中-公开
标题翻译：噻唑烷二酮衍生物的制备方法
公开(公告)号：US20060106221A1
公开(公告)日：2006-05-18
申请号：US11326003
申请日：2006-01-05
申请人： Robert Giles , Norman Lewis , John Quick
发明人： Robert Giles , Norman Lewis , John Quick
IPC分类号： A61K31/4439 , C07D417/02
CPC分类号： C07D417/12
摘要： A process for preparing a compound of formula (I): or a tautomeric form thereof or a pharmaceutically acceptable salt thereof, or a pharmaceutically acceptable solvate thereof, wherein: A1 represents a substituted or unsubstituted aromatic heterocyclyl group; R1 represents a hydrogen atom, an alkyl group, an acyl group, an aralkyl group, wherein the aryl moiety may be substituted or unsubstituted, or a substituted or unsubstituted aryl group; A2 represents a benzene ring having in total up to five substituents; and n represents an integer in the range of from 2 to 6, which process comprises catalytically reducing a compound of formula (II): wherein A1, R1, A2 and n are as defined in relation to formula (I), characterised in that the reduction reaction is carried out using a hydrogen pressure above 20 psi; and thereafter if required forming a pharmaceutically acceptable salt and/or a pharmaceutically acceptable solvate of the compound of formula (I).
摘要翻译：制备式（I）化合物或其互变异构体或其药学上可接受的盐或其药学上可接受的溶剂合物的方法，其中：A 1表示取代或未取代的芳族杂环基 ; R 1表示氢原子，烷基，酰基，芳烷基，其中芳基部分可以是取代或未取代的，或取代或未取代的芳基; 代表一个总共有五个取代基的苯环; 并且n表示2至6的整数，该方法包括催化还原式（II）的化合物：其中A 1，R 2， SUP> 2和n如关于式（I）所定义，其特征在于还原反应使用高于20psi的氢气压力进行; 然后如果需要，形成式（I）化合物的药学上可接受的盐和/或药学上可接受的溶剂化物。

2. 发明申请

US20070066662A1 PROCESS FOR THE PREPARATION OF THIAZOLIDINEDIONE DERIVATIVES 失效
标题翻译：制备噻唑啉衍生物的方法
公开(公告)号：US20070066662A1
公开(公告)日：2007-03-22
申请号：US11550506
申请日：2006-10-18
申请人： Robert Giles , Norman Lewis , John Quick
发明人： Robert Giles , Norman Lewis , John Quick
IPC分类号： A61K31/4439 , C07D417/02
CPC分类号： C07D417/12
摘要： A process for preparing a compound of formula (I): or a tautomeric form thereof or a pharmaceutically acceptable salt thereof, or a pharmaceutically acceptable solvate thereof, wherein: A1 represents a substituted or unsubstituted aromatic heterocyclyl group; R1 represents a hydrogen atom, an alkyl group, an acyl group, an aralkyl group, wherein the aryl moiety may be substituted or unsubstituted, or a substituted or unsubstituted aryl group; A2 represents a benzene ring having in total up to five substituents; and n represents an integer in the range of from 2 to 6, which process comprises catalytically reducing a compound of formula (II): wherein A1, R1, A2 and n are as defined in relation to formula (I), characterised in that the reduction reaction is carried out using a hydrogen pressure above 20 psi; and thereafter if required forming a pharmaceutically acceptable salt and/or a pharmaceutically acceptable solvate of the compound of formula (I).
摘要翻译：制备式（I）化合物或其互变异构体或其药学上可接受的盐或其药学上可接受的溶剂合物的方法，其中：A 1表示取代或未取代的芳族杂环基 ; R 1表示氢原子，烷基，酰基，芳烷基，其中芳基部分可以是取代或未取代的，或取代或未取代的芳基; 代表一个总共有五个取代基的苯环; 并且n表示2至6的整数，该方法包括催化还原式（II）的化合物：其中A 1，R 2， SUP> 2和n如关于式（I）所定义，其特征在于还原反应使用高于20psi的氢气压力进行; 然后如果需要，形成式（I）化合物的药学上可接受的盐和/或药学上可接受的溶剂化物。

3. 发明申请

US20070021470A1 Crystalline N-(2-((4-Hydroxyphenyl)amino)pyridin-3-yl)-4-methoxybenzenesulfonamide methanolates 审中-公开
标题翻译：结晶N-（2 - （（4-羟基苯基）氨基）吡啶-3-基）-4-甲氧基苯磺酰胺甲醇化物
公开(公告)号：US20070021470A1
公开(公告)日：2007-01-25
申请号：US11331535
申请日：2006-01-13
申请人： Jorge Gandarilla , Kathryn Schardt , John Quick
发明人： Jorge Gandarilla , Kathryn Schardt , John Quick
IPC分类号： A61K31/44 , C07D213/78
CPC分类号： C07D213/76
摘要： Methanolates of N-(2-((4-Hydroxyphenyl)amino)pyridin-3-yl)-4-methoxybenzenesulfonamide, ways to make them, compositions containing them or made with them, and methods of treating diseases using them or drugs made from them are disclosed.
摘要翻译： N-（2 - （（4-羟基苯基）氨基）吡啶-3-基）-4-甲氧基苯磺酰胺，制备它们的方法，含有它们或用它们制备的组合物的甲醇盐，以及使用它们治疗疾病的方法或由他们被披露。

4. 再颁专利

USRE36539E Seal and installation improvements 失效
标题翻译：密封和安装改进
公开(公告)号：USRE36539E
公开(公告)日：2000-02-01
申请号：US908722
申请日：1997-08-08
申请人： John Quick
发明人： John Quick
IPC分类号： F16J15/10 , F16L5/02 , F24C3/00 , F24H9/12
CPC分类号： F16L5/10 , Y10T16/063
摘要： A direct vent gas baseboard heater has field installable concentric air intake tube and exhaust pipe. The intake pipe and exhaust tube can be cut separately from the remainder of the heater, improving the efficiency of installation. They can also be transported aligned with the remainder of the heater, reducing packaging size. The manufacturer can provide a single size of tube and pipe for a variety of installation situations. The tube connects to a base cabinet through a key hole configuration of tabs and cuts, and is twisted until the tabs meet stops in the base cabinet. An extrusion in an air box in the base cabinet is brought against a gasket on a flange on the tube, fixing the tube and sealing it with the air box. The exhaust tube has a threaded end and is threaded into an exhaust outlet in the air box, sealing is to a heat exchanger. A vent seal kit creates a seal assembly having a resiliently deformable ring seal extending into a wall sleeve with straps. The assembly is inserted ring first into a hole in a structure which deforms the seal by bending it back. When the seal engages through the structure, it rebounds to its original position and the straps are pulled. This brings the seal into contact with the exterior wall, sealing it. Insulation is sprayed from the interior about the wall sleeve, sealing the internal cavity. An O-ring is slipped over the intake tube previously installed on the heater. The intake tube and exhaust pipe are inserted through the wall sleeve, sealed to the wall sleeve by the O-ring. The seal assembly allows the entire installation process to take place from the interior and is particularly advantageous for high-rise installations.
摘要翻译：直排式气体底板加热器具有现场安装的同心进气管和排气管。进气管和排气管可以与加热器的其余部分分开切割，提高安装效率。它们也可以与加热器的其余部分一起运输，减少包装尺寸。制造商可以为各种安装情况提供单一尺寸的管和管道。管通过突出部和切口的键孔配置连接到基座，并被扭转，直到接头与基座中的止挡件相接。将基座机柜中的空气箱中的挤出件压靠在管上的凸缘上的垫圈上，固定管并用空气箱密封。排气管具有螺纹端并且拧入空气箱中的排气出口，密封是热交换器。排气密封套件产生密封组件，该密封组件具有可弹性变形的环形密封件，其延伸到具有带的壁套筒中。组件首先插入到通过弯曲使密封件变形的结构中的孔中。当密封件通过结构接合时，它反弹到其原始位置并且拉紧带。这使得密封件与外壁接触，密封。绝缘材料是从内壁围绕壁套筒进行喷涂，密封内腔。 O型圈滑过预先安装在加热器上的进气管。进气管和排气管穿过壁套筒，通过O型圈密封到壁套筒上。密封组件允许整个安装过程从内部进行，并且对于高层安装是特别有利的。

5. 发明申请

US20070140621A1 Connector assembly with integrated electromagnetic shield 失效
标题翻译：带集成电磁屏蔽的连接器总成
公开(公告)号：US20070140621A1
公开(公告)日：2007-06-21
申请号：US11314665
申请日：2005-12-21
申请人： Casimer DeCusatis , John Quick
发明人： Casimer DeCusatis , John Quick
IPC分类号： G02B6/36
CPC分类号： G02B6/4248 , G02B6/3817 , G02B6/3887 , G02B6/4292
摘要： A conductive, compliant, deformable boot for a fiber optic or other cable assembly is described, which both provides traditional cable strain relief functions and extends over the body of the connector to form an electrically conductive shield over the cable receptacle aperture when the cable assembly is plugged into the aperture. The boot deforms slightly upon insertion of the cable assembly and compresses against a mating component to form a shield against electrostatic discharge which can accumulate on the cable or card and also to shield against electromagnetic emissions entering or leaving the circuit card package. The boot also shields against emissions when two cable assemblies are mated together by deforming slightly upon mating and then returning to its original state when the assemblies are disconnected.
摘要翻译：描述了用于光纤或其他电缆组件的导电的，柔性的可变形的靴子，其提供传统的电缆应变消除功能，并且在连接器的主体上延伸以在电缆组件为插入光圈。当插入电缆组件时，护罩会轻微变形，并压缩配合部件，以形成防止静电放电的屏蔽物，从而可以积聚在电缆或卡上，并且还可防止进入或离开电路卡封装的电磁辐射。当两个电缆组件通过在配合时稍微变形而配合在一起，然后当组件断开时返回到其初始状态，该引导罩也可防止排放。

6. 发明申请

US20070021471A1 Crystalline N-(2-((4-Hydroxyphenyl)amino)pyridin-3-yl)-4-methoxybenzenesulfonamide ethanolates 审中-公开
标题翻译：结晶N-（2 - （（4-羟基苯基）氨基）吡啶-3-基）-4-甲氧基苯磺酰胺乙醇化物
公开(公告)号：US20070021471A1
公开(公告)日：2007-01-25
申请号：US11332274
申请日：2006-01-13
申请人： Jorge Gandarilla , Karthryn Schardt , John Quick
发明人： Jorge Gandarilla , Karthryn Schardt , John Quick
IPC分类号： A61K31/44 , C07D213/72
CPC分类号： C07D213/76
摘要： Ethanolates of N-(2-((4-Hydroxyphenyl)amino)pyridin-3-yl)-4-methoxybenzenesulfonamide, ways to make them, compositions containing them or made with them, and methods of treating diseases using them or drugs made from them. are disclosed.
摘要翻译： N-（2 - （（4-羟基苯基）氨基）吡啶-3-基）-4-甲氧基苯磺酰胺的制备方法，含有它们或用它们制备的组合物，以及使用它们治疗疾病的方法或由他们。被披露。

7. 发明授权

US5551414A Seal and installation improvements 失效
标题翻译：密封和安装改进
公开(公告)号：US5551414A
公开(公告)日：1996-09-03
申请号：US396710
申请日：1995-03-01
申请人： John Quick
发明人： John Quick
IPC分类号： F16J15/10 , F16L5/02 , F24C3/00 , F24H9/12
CPC分类号： F16L5/10 , Y10T16/063
摘要： A direct vent gas baseboard heater has field installable concentric air intake tube and exhaust pipe. The intake pipe and exhaust tube can be cut separately from the remainder of the heater, improving the efficiency of installation. They can also be transported aligned with the remainder of the heater, reducing packaging size. The manufacturer can provide a single size of tube and pipe for a variety of installation situations. The tube connects to a base cabinet through a key hole configuration of tabs and cuts, and is twisted until the tabs meet stops in the base cabinet. An extrusion in an air box in the base cabinet is brought against a gasket on a flange of the tube, fixing the tube and sealing it with the air box. The exhaust tube has a threaded end and is threaded into an exhaust outlet in the air box, sealing it to a heat exchanger. A vent seal kit creates a seal assembly having a resiliently deformable ring seal extending into a wall sleeve with straps. The assembly is inserted ring first into a hole in a structure which deforms the seal by bending it back. When the seal emerges through the structure, it rebounds to its original position and the straps are pulled. This brings the seal into contact with the exterior wall, sealing it. Insulation is sprayed from the interior about the wall sleeve, sealing the internal cavity. An O-ring is slipped over the intake tube previously installed on the heater. The intake tube and exhaust pipe are inserted through the wall sleeve, sealed to the wall sleeve by the O-ring. The seal assembly allows the entire installation process to take place from the interior and is particularly advantageous for high-rise installations.
摘要翻译：直排式气体底板加热器具有现场安装的同心进气管和排气管。进气管和排气管可以与加热器的其余部分分开切割，提高安装效率。它们也可以与加热器的其余部分一起运输，减少包装尺寸。制造商可以为各种安装情况提供单一尺寸的管和管道。管通过突出部和切口的键孔配置连接到基座，并被扭转，直到接头与基座中的止挡件相接。将基座机柜中的空气箱中的挤压件压靠在管的凸缘上的垫圈上，固定管并用空气箱密封。排气管具有螺纹端并且拧入空气箱中的排气出口，将其密封到热交换器。排气密封套件产生密封组件，该密封组件具有可弹性变形的环形密封件，其延伸到具有带的壁套筒中。组件首先插入到通过弯曲使密封件变形的结构中的孔中。当密封件通过结构出现时，它将弹回到其原始位置并拉紧带子。这使得密封件与外壁接触，密封。绝缘材料是从内壁围绕壁套筒进行喷涂，密封内腔。 O型圈滑过预先安装在加热器上的进气管。进气管和排气管穿过壁套筒，通过O型圈密封到壁套筒上。密封组件允许整个安装过程从内部进行，并且对于高层安装是特别有利的。

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